
Ciclo celular / Checkpoint
Los inhibidores del ciclo celular/puntos de control son compuestos que interrumpen la progresión normal del ciclo celular, particularmente en puntos de control regulatorios clave. Estos inhibidores son cruciales para estudiar la división celular, comprender la proliferación de células cancerosas y desarrollar terapias anticancerígenas. Al dirigirse a fases específicas del ciclo celular, estos inhibidores pueden inducir la detención del ciclo celular, lo que lleva a apoptosis o senescencia en células de división rápida. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad del ciclo celular/puntos de control para apoyar su investigación en biología del cáncer, biología celular y desarrollo de fármacos.
Subcategorías de "Ciclo celular / Checkpoint"
- Aurora quinasa(120 productos)
- CDK(561 productos)
- Detención del ciclo celular(8 productos)
- Chk(49 productos)
- DYRK(47 productos)
- Dynamin(28 productos)
- Ferroptosis(229 productos)
- HSP(184 productos)
- Integrin(288 productos)
- Kinesina(88 productos)
- LIM quinasa(22 productos)
- Asociado a microtúbulos(286 productos)
- PKC(130 productos)
- PLK(25 productos)
- ROCK(62 productos)
- Rho(7 productos)
- Wee1(19 productos)
- c-Myc(80 productos)
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Se han encontrado 2894 productos para "Ciclo celular / Checkpoint".
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Cinoxacin
CAS:Cinoxacin (Compound 64716), an older synthetic antimicrobial, was related to the quinolone class of antibiotics.Fórmula:C12H10N2O5Pureza:99.62% - 99.98%Forma y color:White SolidPeso molecular:262.22Cyclin K degrader 1
Cyclin K degrader 1 is a Cyclin K degrader.Cyclin K degrader 1 is a degrader converted from AT-7519.Cyclin K degrader 1 has weak degrading activity against Cyclin K but does not result in a sustained decrease in degradation affinity.Cyclin K degrader 1 is a degrader converted from AT-7519.Fórmula:C23H17Cl2N5O2Pureza:99.91%Forma y color:SolidPeso molecular:466.32hSMG-1 inhibitor 11j
CAS:hSMG-1 inhibitor 11j: pyrimidine, IC50=0.11 nM, >455x selective vs. mTOR/PI3Kα/γ/CDK1/CDK2; cancer research use.Fórmula:C27H28ClN7O3SPureza:99.22% - 99.65%Forma y color:Yellow SolidPeso molecular:566.07K34c hydrochloride
CAS:K34c hydrochloride is an alpha5β1 integrin antagonist for glioblastoma study.Fórmula:C26H30ClN3O4Pureza:99.76% - 99.89%Forma y color:White SolidPeso molecular:483.99PTBP1-RNA-binding inhibitor P6 TFA
PTBP1-RNA-binding inhibitor P6 TFA is a stapled peptide inhibitor of PTBP1, used to inhibit RNA alternative splicing events regulated by PTBP1.Forma y color:Odour SolidLedoxantrone trihydrochloride
CAS:Ledoxantrone trihydrochloride is a Top II inhibitor with anticancer activity and is used in the study of digestive disorders and urologic disorders.Fórmula:C21H30Cl3N5OSPureza:97.02%Forma y color:Yellow SolidPeso molecular:506.92R-10015
CAS:R-10015, potent LIMK inhibitor with 38 nM IC50 for LIMK1, targets ATP pocket, and serves as a broad-spectrum HIV antiviral.Fórmula:C20H19ClN6O2Pureza:98.68%Forma y color:SolidPeso molecular:410.86Ref: TM-T12609
1mg50,00€5mg112,00€1mL*10mM (DMSO)124,00€10mg170,00€25mg280,00€50mg371,00€100mg525,00€200mg712,00€TAME hydrochloride
CAS:TAME hydrochloride (Tos-Arg-OMe HCl) is a kind od amino acid derivatives.Fórmula:C14H23ClN4O4SPureza:99.11% - 99.21%Forma y color:SolidPeso molecular:378.87ROCK inhibitor-2
CAS:ROCK inhibitor-2 is a selective dual inhibitor of ROCK1 and ROCK2 (IC50s of 17 nM and 2 nM, respectively).Fórmula:C21H20N2O2Pureza:99.85%Forma y color:SolidPeso molecular:332.4Ref: TM-T12746
1mg63,00€1mL*10mM (DMSO)101,00€5mg137,00€10mg205,00€25mg409,00€50mg612,00€100mg858,00€ZN-c3
CAS:Azenosertib (ZN-c3) is a potent and selective Wee1 inhibitor with balanced potency, ADME, and pharmacokinetic properties. Cost-effective and quality-assured.Fórmula:C29H34N8O2Pureza:99.98%Forma y color:SolidPeso molecular:526.63Ref: TM-T9643
1mg90,00€5mg215,00€1mL*10mM (DMSO)250,00€10mg334,00€25mg620,00€50mg982,00€100mg1.468,00€200mg1.972,00€HBX 19818
CAS:HBX 19818 is a specific ubiquitin-specific protease 7 (USP7) inhibitor (IC50: 28.1 μM).Fórmula:C25H28ClN3OPureza:97.71%Forma y color:SolidPeso molecular:421.96Ref: TM-T15464
1mg35,00€5mg80,00€1mL*10mM (DMSO)89,00€10mg111,00€25mg177,00€50mg253,00€100mg353,00€200mg502,00€Folinic acid calcium
CAS:Folinic acid calcium (Leucovorin Calcium) is the active metabolite of folic acid. Leucovorin is used principally as an antidote to folic acid antagonists.Fórmula:C20H21CaN7O7Pureza:98.72% - >99.99%Forma y color:Yellow SolidPeso molecular:511.51CHK1-IN-4 hydrochloride
CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1).Fórmula:C18H19BrClN7O2Pureza:99.29%Forma y color:SolidPeso molecular:480.75ATN-161 trifluoroacetate salt
CAS:ATN-161 TFA salt, a new integrin α5β1 inhibitor, curbs angiogenesis, liver metastases growth, enhances survival in mice.Fórmula:C25H36F3N9O10SPureza:98% - 99.98%Forma y color:White SolidPeso molecular:711.67Pefloxacin Mesylate Dihydrate
CAS:Pefloxacin Mesylate Dihydrate (1589 RB) , an antibacterial agent, restrains bacterial DNA replication by inhibiting DNA gyrase (topoisomerase).Fórmula:C17H20FN3O3·CH4O3S·2H2OPureza:99.79%Forma y color:SolidPeso molecular:465.49Upamostat
CAS:Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.Fórmula:C32H47N5O6SPureza:99.41%Forma y color:White SolidPeso molecular:629.81Ref: TM-T13257
1mg60,00€2mg89,00€5mg138,00€1mL*10mM (DMSO)155,00€10mg215,00€25mg359,00€50mg510,00€100mg692,00€AZ-Dyrk1B-33
CAS:AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.Fórmula:C19H16N4Pureza:99.91%Forma y color:SolidPeso molecular:300.36Ref: TM-T14364
1mg44,00€5mg92,00€1mL*10mM (DMSO)100,00€10mg147,00€25mg289,00€50mg419,00€100mg583,00€200mg787,00€Tadocizumab
CAS:Tadocizumab (C4G1) is a humanized monoclonal antibody targeting integrin αIIbβ3 with antiplatelet and antithrombotic effects.Pureza:97.1% (SDS-PAGE); 97.2% (SEC-HPLC) - 97.1% (SDS-PAGE); 97.2% (SEC-HPLC)Forma y color:Transparent LiquidPeso molecular:47.59 kDaBersanlimab
CAS:Bersanlimab (BI-505) is a fully human monoclonal antibody targeting Intercellular Adhesion Molecule-1 (ICAM-1).Bersanlimab has anticancer properties.Pureza:> 95% - > 95%Forma y color:Transparent LiquidPeso molecular:144.22 kDaFolinic Acid Calcium Salt Pentahydrate
CAS:Folinic Acid Calcium Salt Pentahydrate (Leucovorin Calcium Pentahydrate), a reduced folic acid, is used in combination with other chemotherapeutics.Fórmula:C20H21CaN7O7·5H2OPureza:99.17% - >99.99%Forma y color:Yellow SolidPeso molecular:601.58

