Apoptosi
Gli inibitori dell'apoptosi sono composti che prevengono o ritardano il processo di morte cellulare programmata, noto come apoptosi. Questi inibitori sono fondamentali per lo studio dei meccanismi di sopravvivenza cellulare e vengono utilizzati per indagare sulle malattie in cui l'apoptosi è disregolata, come il cancro, i disturbi neurodegenerativi e le malattie autoimmuni. Modulando l'apoptosi, questi inibitori possono aiutare nello sviluppo di terapie mirate a controllare la morte cellulare. Presso CymitQuimica, offriamo una vasta selezione di inibitori dell'apoptosi di alta qualità per supportare le tue ricerche in biologia cellulare, oncologia e campi correlati.
Sottocategorie di "Apoptosi"
- ASK(6 prodotti)
- BCL(11 prodotti)
- Caspasi(127 prodotti)
- FOXO1(3 prodotti)
- IAP(66 prodotti)
- Mdm2(12 prodotti)
- PD-1/PD-L1(126 prodotti)
- PDK(9 prodotti)
- PERK(23 prodotti)
- Chinasi di serina/treonina(15 prodotti)
- Survivin(13 prodotti)
- TNF(91 prodotti)
- c-RET(51 prodotti)
- p53(62 prodotti)
Mostrare 6 più sottocategorie
Trovati 5618 prodotti di "Apoptosi"
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Chelerythrine chloride
CAS:<p>Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the phosphate acceptor and non-competitive with respect to</p>Formula:C21H18ClNO4Purezza:95% - 99.19%Colore e forma:Yellow To Orange SolidPeso molecolare:383.83M50054
CAS:<p>Apoptosis Inhibitor was a novel inhibitor of programmed cell death associate with caspase-3 inhibition.</p>Formula:C13H16O4Purezza:97.8%Colore e forma:SolidPeso molecolare:236.26BI-847325
CAS:<p>BI-847325 is a selective dual inhibitor of MEK and aurora kinases (AK) with IC50 values of 4 and 15 nM for human MEK2 and AK-C, respectively.</p>Formula:C29H28N4O2Purezza:97.13% - 97.54%Colore e forma:SolidPeso molecolare:464.56BI 2536
CAS:<p>BI2536 is an effective Plk1 inhibitor (IC50: 0.83 nM). It has 4- and 11-fold greater selectivity than Plk2 and Plk3.</p>Formula:C28H39N7O3Purezza:98% - 99.88%Colore e forma:SolidPeso molecolare:521.65Amuvatinib
CAS:Amuvatinib (MP470) is an orally bioavailable synthetic carbothioamide with potential antineoplastic activity.Formula:C23H21N5O3SPurezza:99.38% - >99.99%Colore e forma:SolidPeso molecolare:447.51DAPK Substrate Peptide acetate
<p>DAPK Substrate Peptide acetate is a death-associated protein kinase (DAPK, Km = 9 μM) peptide substrate.</p>Formula:C70H115N25O17Purezza:98.12%Colore e forma:SolidPeso molecolare:1578.82Copanlisib
CAS:<p>Copanlisib (BAY 80-6946), a PI3K inhibitor, may block tumor growth and improve cancer treatment efficacy.</p>Formula:C23H28N8O4Purezza:99% - 99.88%Colore e forma:SolidPeso molecolare:480.52Concanavalin A
CAS:<p>Concanavalin A is a natural product, a phytoalexin. Concanavalin A has antitumor activity and can also induce acute liver injury. Cost effective and quality assured.</p>Formula:C23H32N6O8SPurezza:98%Colore e forma:SolidPeso molecolare:104-112 kDaAvicularin
CAS:<p>Avicularin reduces inflammation via ERK pathway in RAW 264.7 cells and hinders lipid buildup in adipocytes by limiting glucose uptake and fatty acid synthesis.</p>Formula:C20H18O11Purezza:97.02% - 99.94%Colore e forma:White PowderPeso molecolare:434.35PHA-665752
CAS:<p>PHA-665752 is an effective, specific and ATP-competitive c-Met inhibitor (IC50: 9 nM), >50-fold selectivity for c-Met than STKs or RTKs.</p>Formula:C32H34Cl2N4O4SPurezza:97.05% - 98.82%Colore e forma:SolidPeso molecolare:641.61PD146176
CAS:<p>PD146176 (NSC-168807) is an inhibitor of 15-Lipoxygenase (15-LO) , it inhibits rabbit reticulocyte 15-LO with Ki of 197 nM and IC50 of 0.54 μM.</p>Formula:C15H11NSPurezza:98.00%Colore e forma:SolidPeso molecolare:237.32Terrestrosin D
CAS:<p>Terrestrosin D triggers apoptosis, halts cell cycles, and blocks angiogenesis in tumor cells, displaying anti-cancer effects.</p>Formula:C50H80O23Purezza:99.92% - 99.96%Colore e forma:SolidPeso molecolare:1049.16Ganetespib
CAS:<p>Ganetespib (STA-9090) is a synthetic small-molecule inhibitor of heat shock protein 90 (Hsp90) with potential antineoplastic activity.</p>Formula:C20H20N4O3Purezza:98% - 99.95%Colore e forma:SolidPeso molecolare:364.4Aminopurvalanol A
CAS:<p>Aminopurvalanol A is a competitive, selective and cell-permeable inhibitor of cyclin-dependent kinase (CDK) that potently inhibits Cyclin A/cdk2, Cyclin B/cdk1</p>Formula:C19H26ClN7OPurezza:99.73%Colore e forma:SolidPeso molecolare:403.91Notopterol
CAS:<p>1. Notopterol induces apoptosis and inhibits cell cycle-specific.</p>Formula:C21H22O5Purezza:97.57% - 99.82%Colore e forma:SolidPeso molecolare:354.4Apomine
CAS:<p>Apomine (SR-9223i) 是一种 HMG-CoA-还原酶抑制剂，可在体外促进骨髓瘤细胞的凋亡，并与体内骨髓瘤的调节有关。 Apomine 加速 3-羟基-3-甲基戊二酰-CoA 还原酶的降解并刺激低密度脂蛋白受体活性。 Apomine 通过下调 3-羟基-3-甲基戊二酰-CoA 还原酶来增强洛伐他汀对骨髓瘤细胞的抗肿瘤作用。</p>Formula:C28H52O7P2Purezza:>99.99%Colore e forma:SolidPeso molecolare:562.66VR23
CAS:<p>VR23: Potent proteasome inhibitor; IC50: 1 nM trypsin, 50-100 nM chymotrypsin, 3 μM caspase-like.</p>Formula:C19H16ClN5O6SPurezza:98.99% - 99.22%Colore e forma:SolidPeso molecolare:477.88Caffeic Acid Phenethyl Ester
CAS:<p>CAPE, in propolis, blocks NF-kappa B, suppresses p70S6K/Akt pathways, and inhibits PDGF, aiding in cancer protection and immune modulation.</p>Formula:C17H16O4Purezza:99.18% - 99.35%Colore e forma:Less Transparent Liquid Colorless Transparent LiquidPeso molecolare:284.31TBHQ
CAS:TBHQ (tert-Butylhydroquinone) is an antioxidant that induces an antioxidant response through the redox-sensitive transcription factor Nrf2.Formula:C10H14O2Purezza:99.17% - 99.53%Colore e forma:White Solid PowderPeso molecolare:166.22HBX 41108
CAS:<p>HBX 41108: non-competitive, reversible USP7 inhibitor; IC50: 424nM; blocks USP7-p53 deubiquitination; IC50: 0.8μM.</p>Formula:C13H3ClN4OPurezza:95.63%Colore e forma:SolidPeso molecolare:266.64Ginsenoside Rh2
CAS:<p>Ginsenoside Rh2 (20(S)-Ginsenoside Rh2), an extract of red Panax ginseng, is a potent anti-inflammatory and anticancer drug.</p>Formula:C36H62O8Purezza:99.20% - 99.76%Colore e forma:White PowderPeso molecolare:622.87CGP 57380
CAS:<p>CGP 57380 (MNK1 Inhibitor) is a potent MNK1 inhibitor with IC50 of 2.2 μM, exhibiting no inhibitory activity on p38, JNK1, ERK1 and -2, PKC, or c-Src-like</p>Formula:C11H9FN6Purezza:98.49%Colore e forma:SolidPeso molecolare:244.23(Z)-Guggulsterone
CAS:<p>(Z)-Guggulsterone triggers apoptosis in prostate cancer cells and blocks angiogenesis by inhibiting VEGF pathways.</p>Formula:C21H28O2Purezza:98.93% - 99.72%Colore e forma:SolidPeso molecolare:312.45NSC348884
CAS:<p>NSC348884, a nucleophosmin inhibitor, disrupts oligomers, induces apoptosis, and inhibits cancer cell growth (IC50: 1.7-4.0 μM).</p>Formula:C38H40N10Purezza:98.69% - 99.91%Colore e forma:SolidPeso molecolare:636.79Berbamine dihydrochloride
CAS:<p>Berbamine dihydrochloride (Berbamine), a natural compound derived from the Berberis amurensis plant, has been shown to exhibit antitumor activity in several Ys.</p>Formula:C37H42Cl2N2O6Purezza:95% - 99.99%Colore e forma:SolidPeso molecolare:681.65Scoulerine
CAS:<p>Scoulerine is an inhibitor of ß-site amyloid precursor protein cleaving enzyme 1(BACE1).</p>Formula:C19H21NO4Purezza:98.62%Colore e forma:SolidPeso molecolare:327.37SP-141
CAS:<p>SP 141 is a MDM2 inhibitor.SP-141 promotes MDM2 auto-ubiquitination and degradation, with anticancer activity.</p>Formula:C22H16N2OPurezza:98.01%Colore e forma:SolidPeso molecolare:324.38BIO-acetoxime
CAS:<p>BIO-acetoxime (GSK-3 Inhibitor X) is a potent dual GSK3α/β inhibitor with IC50 of 10 nM, >240-fold selectivity over CDK5/p25, CDK2/cyclin A and CDK1/cyclin B.</p>Formula:C18H12BrN3O3Purezza:97.15%Colore e forma:SolidPeso molecolare:398.215,7,4'-Trimethoxyflavone
CAS:<p>5,7,4'-Trimethoxyflavone (4',5,7-Trimethoxyflavone) is isolated from Kaempferia parviflora (KP) which is a medicinal plant from Thailand.</p>Formula:C18H16O5Purezza:97.53%Colore e forma:SolidPeso molecolare:312.32Dehydroeffusol
CAS:<p>Dehydroeffusol: anti-cancer, anxiolytic, sedative; halts gastric cancer growth via ER stress and apoptosis.</p>Formula:C17H14O2Purezza:99.35%Colore e forma:SolidPeso molecolare:250.29Domatinostat tosylate
CAS:<p>4SC-202 is a class I HDAC inhibitor targeting HDAC1/2/3; shows activity against LSD1. IC50: HDAC1 (1.20 μM), HDAC2 (1.12 μM), HDAC3 (0.57 μM).</p>Formula:C30H29N5O6S2Purezza:97.35% - >99.99%Colore e forma:Solid PowderPeso molecolare:619.71Spautin-1
CAS:<p>Spautin-1 is an autophagy inhibitor that can suppress the deubiquitination activity of ubiquitin-specific peptidase USP10 and USP13. Cost-effective and quality-assured.</p>Formula:C15H11F2N3Purezza:97.69% - 98.99%Colore e forma:SolidPeso molecolare:271.26AKT inhibitor VIII
CAS:<p>AKT inhibitor VIII (AKTi-1/2) is a highly specific Akt1/2 inhibitor (IC50: 58/210 nM). The selectivity for Akt1 is higher about 36-fold than Akt3.</p>Formula:C34H29N7OPurezza:98.31% - 98.65%Colore e forma:Pale Yellow SolidPeso molecolare:551.64LJH685
CAS:<p>LJH685 is an effective pan-RSK inhibitor for RSK1/2/3 (IC50: 6/5/4 nM).</p>Formula:C22H21F2N3OPurezza:99.13% - 99.78%Colore e forma:SolidPeso molecolare:381.42PF-543 hydrochloride
CAS:<p>PF-543 hydrochloride (PF-543) inhibits SphK1 with a K(i) of 3.6 nM, is sphingosine-competitive and is more than 100-fold selective for SphK1 over the SphK2</p>Formula:C27H32ClNO4SPurezza:98.9% - 99.93%Colore e forma:SolidPeso molecolare:502.1Sesamol
CAS:<p>Sesamol (1,3-Benzodioxol-5-ol) could decrease lung inflammation and lipopolysaccharide (LPS)-induced lung injury in rats.</p>Formula:C7H6O3Purezza:99.67% - 99.76%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:138.12Ginsenoside F5
CAS:<p>Ginsenoside F5 is a natural product from Panax ginseng C. A. Mey, remarkably inhibits the growth of HL-60 cells by the apoptosis pathway</p>Formula:C41H70O13Purezza:99.78% - 99.86%Colore e forma:SolidPeso molecolare:770.99Paris saponin VII
CAS:<p>Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.</p>Formula:C51H82O21Purezza:99.51% - 99.63%Colore e forma:SolidPeso molecolare:1031.18Sophoridine
CAS:Sophoridine, a natural Chinese anticancer drug, has a potent derivative 6b targeting DNA topoisomerase I in tumor cells, inducing apoptosis.Formula:C15H24N2OPurezza:97.33% - 99.28%Colore e forma:SolidPeso molecolare:248.36DBEQ
CAS:<p>DBEQ (JRF 12) is a selective, potent, reversible, and ATP-competitive p97 inhibitor.</p>Formula:C22H20N4Purezza:98.93% - ≥95%Colore e forma:SolidPeso molecolare:340.42AZD5582 acetate (1258392-53-8 free base)
<p>AZD5582 acetate is an inhibitor of IAPs, which binds to the BIR3 domains cIAP1, cIAP2, and XIAP with IC50s of 15, 21, and 15 nM, respectively.</p>Formula:C60H82N8O10Purezza:97.76%Colore e forma:SolidPeso molecolare:1075.36Dipyrithione
CAS:<p>Dipyrithione appears to have novel cytotoxicity and potent broad-spectrum antitumor activity</p>Formula:C10H8N2O2S2Purezza:99.9%Colore e forma:Beige Crystalline PowderPeso molecolare:252.31Phenoxodiol
CAS:Phenoxodiol (Idronoxil) activates the mitochondrial caspase system, inhibits X-linked inhibitor of apoptosis(XIAP), disrupts FLICE inhibitory protein(FLIP)Formula:C15H12O3Purezza:98.07% - 99.18%Colore e forma:SolidPeso molecolare:240.25Anisomycin
CAS:<p>Anisomycin (NSC-76712), an antibiotic from Streptomyces, blocks protein/DNA synthesis by targeting peptidyl transferase/80S ribosomes.</p>Formula:C14H19NO4Purezza:98.33% - 99.81%Colore e forma:White Crystalline SolidPeso molecolare:265.3ARS-853
CAS:<p>ARS-853 is an inhibitor of K-RASG12C(IC50 : 2.5 μM), a mutant form of K-RAS that accumulates in the active GTP-bound state in certain cancer cells</p>Formula:C22H29ClN4O3Purezza:97.43% - 98.4%Colore e forma:SolidPeso molecolare:432.94Lorlatinib
CAS:<p>Lorlatinib (PF-6463922) is an orally available, ATP-competitive inhibitor of the receptor tyrosine kinases, anaplastic lymphoma kinase (ALK) and C-ros oncogene</p>Formula:C21H19FN6O2Purezza:99.77% - 99.95%Colore e forma:SolidPeso molecolare:406.41Ginsenoside F2
CAS:<p>Ginsenoside F2 halts breast CSCs growth, induces apoptosis via intrinsic pathway and impairs mitochondria.</p>Formula:C42H72O13Purezza:99.04% - 99.3%Colore e forma:SolidPeso molecolare:785.01Carvacrol
CAS:<p>1.</p>Formula:C10H14OPurezza:99.05%Colore e forma:Needles LiquidPeso molecolare:150.22MFCD01917484
CAS:<p>MFCD01917484: A thiophene derivative with ligand, catalyst, and photosensitizer roles, used in biochemical research and drug development.</p>Formula:C14H15NO3SPurezza:98.09%Colore e forma:SolidPeso molecolare:277.34Taccalonolide A
CAS:<p>Taccalonolide A is the first microtubule stabilizing agent to be discovered from a plant since identification of the mechanism of action of paclitaxel and it is</p>Formula:C36H46O14Purezza:98.16% - 99.4%Colore e forma:SolidPeso molecolare:702.74Onatasertib
CAS:<p>Onatasertib (CC223) is an orally available mTOR inhibitor with potential antitumor activity.</p>Formula:C21H27N5O3Purezza:99.14% - 99.97%Colore e forma:SolidPeso molecolare:397.47β-Elemonic Acid
CAS:<p>β-Elemonic Acid (3-Oxotirucallenoic Acid) exhibits anti-inflammatory effects, which inhibits proliferation by inducing hypoploid cells and cell apoptosis.</p>Formula:C30H46O3Purezza:99.61% - 99.8%Colore e forma:SolidPeso molecolare:454.68BAY 11-7082
CAS:BAY 11-7082 (BAY 11-7821) is an NF-κB inhibitor that inhibits TNFα-induced IκBα phosphorylation (IC50=10 μM).Formula:C10H9NO2SPurezza:98% - 99.92%Colore e forma:SolidPeso molecolare:207.25(6R)-FR054
CAS:<p>(6R)-FR054 is an inhibitor of the Hexosamine Biosynthetic Pathway (HBP) enzyme PGM3, with a remarkable anti-breast cancer effect.</p>Formula:C14H19NO8Purezza:99.61%Colore e forma:SolidPeso molecolare:329.3(-)-Epipodophyllotoxin
CAS:(-)-Epipodophyllotoxin: anticancer, GI50=0.36μM (HeLa), 0.24μM (MCF-7), inhibits spindle assembly.Formula:C22H22O8Purezza:99.72% - 99.97%Colore e forma:SolidPeso molecolare:414.41PD173074
CAS:<p>PD173074 inhibits FGFR1 (IC50: 25 nM) and VEGFR2 (100-200 nM); ~1000x more selective for FGFR1 over PDGFR/c-Src.</p>Formula:C28H41N7O3Purezza:98.15% - 98.21%Colore e forma:Yellow SolidPeso molecolare:523.67HA14-1
CAS:<p>HA14-1, a Bcl-2/Bcl-XL antagonist, is a non-peptidic ligand of a Bcl-2 surface pocket (IC50: ~9 μM).</p>Formula:C17H17BrN2O5Purezza:95.07% - 98%Colore e forma:SolidPeso molecolare:409.23JNJ-7706621
CAS:<p>JNJ-7706621 is a potent aurora kinase inhibitor, and also inhibits CDK1 and CDK2.</p>Formula:C15H12F2N6O3SPurezza:99.1% - 99.85%Colore e forma:SolidPeso molecolare:394.36WP1066
CAS:<p>WP1066 is a inhibitor of JAK2 (IC50: 2.30 μM) and STAT3 (IC50: 2.43 μM) in HEL cells; shows activity to JAK2, STAT3/5, and ERK1/2, not JAK1 and JAK3.</p>Formula:C17H14BrN3OPurezza:98.92% - 99.73%Colore e forma:SolidPeso molecolare:356.22Gemcitabine hydrochloride
CAS:Gemcitabine hydrochloride (LY 188011 hydrochloride) is a synthetic cytosine nucleoside derivative and an inhibitor of DNA synthesis.Formula:C9H11F2N3O4·HClPurezza:99.28% - 99.98%Colore e forma:White Crystalline Granular OdorlessPeso molecolare:299.66AZ960
CAS:<p>AZ960 is an effective ATP competitive JAK2 inhibitor (IC50/Ki: <3 nM and0.45 nM).</p>Formula:C18H16F2N6Purezza:96.02% - 98.51%Colore e forma:SolidPeso molecolare:354.36AEE788
CAS:<p>AEE788 (NVP-AEE 788) has been used in trials studying the treatment of Cancer, Glioblastoma Multiforme, and Brain and Central Nervous System Tumors.</p>Formula:C27H32N6Purezza:98% - >99.99%Colore e forma:SolidPeso molecolare:440.5818α-Glycyrrhetinic acid
CAS:<p>18α-Glycyrrhetinic acid (Enoxolone) is a pentacyclic triterpenoid derivative of the beta-amyrin type obtained from the hydrolysis of glycyrrhizic acid.</p>Formula:C30H46O4Purezza:98.54% - 99.68%Colore e forma:SolidPeso molecolare:470.68Antineoplaston A10
CAS:Antineoplaston A10 (NSC-648539) is a Ras inhibitor potentially for the treatment of glioma, lymphoma, astrocytoma and breast cancer.Formula:C13H14N2O3Purezza:99.42%Colore e forma:SolidPeso molecolare:246.26Valepotriate
CAS:<p>Valepotriates are sedative, enhance memory, have anti-cancer properties, and may reduce anxiety.</p>Formula:C22H30O8Purezza:97.29% - 99.90%Colore e forma:SolidPeso molecolare:422.47(E)-Flavokawain A
CAS:<p>(E)-Flavokawain A, a novel chalcone from kava extract, induces apoptosis by involvement of Bax protein-dependent and mitochondria-dependent apoptotic pathway.</p>Formula:C18H18O5Purezza:98% - 99.75%Colore e forma:SolidPeso molecolare:314.332Atractylenolide III
CAS:<p>Atractylenolide III could treat cognitive issues and lung cancer by modulating apoptosis factors.</p>Formula:C15H20O3Purezza:99.53% - 99.82%Colore e forma:SolidPeso molecolare:248.32Oleuropein
CAS:<p>Oleuropein is an antioxidant polyphenol isolated from olive leaf.</p>Formula:C25H32O13Purezza:98% - 99.95%Colore e forma:Brown PowderPeso molecolare:540.51Columbianadin
CAS:Columbianadin (Zosimin), one of the main bioactive constituents of the roots of Angelica pubescens Maxim.Formula:C19H20O5Purezza:98.44% - 99.48%Colore e forma:SolidPeso molecolare:328.36Flavokawain C
CAS:<p>Flavokawain C: natural chalcone from Kava with potential as a colon cancer drug.</p>Formula:C17H16O5Purezza:99.94% - ≥95%Colore e forma:SolidPeso molecolare:300.31GSK2606414
CAS:GSK2606414 is a cell-permeable and orally active protein kinase R-like endoplasmic reticulum kinase（PERK）inhibitor.Cost-effective and quality-assured.Formula:C24H20F3N5OPurezza:98% - >99.99%Colore e forma:SolidPeso molecolare:451.44PK11007
CAS:<p>PK11007 is an anti-p53 drug.</p>Formula:C15H11ClFN5O3S2Purezza:97.55%Colore e forma:SolidPeso molecolare:427.86Masitinib mesylate
CAS:<p>Masitinib mesylate (AB-1010 mesylate) is a selective and orally bioavailable c-Kit inhibitor (IC50 of 200 nM,540/800 nM,510 nM for human recombinant c-Kit;</p>Formula:C29H34N6O4S2Purezza:97.67% - 98.44%Colore e forma:SolidPeso molecolare:594.75Sulforaphene
CAS:<p>Sulforaphene, from radish seeds, aids cancer cell apoptosis and inhibits migration; has an ED50 for velvetleaf at ~2x10^-4 M.</p>Formula:C6H9NOS2Purezza:97.55% - 99.19%Colore e forma:Slightly Yellowish LiquidPeso molecolare:175.27Didanosine
CAS:<p>Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).</p>Formula:C10H12N4O3Purezza:99.64%Colore e forma:White Crystalline PowderPeso molecolare:236.23Neogambogic acid
CAS:<p>Neogambogic acid, an active ingredient in garcinia, can inhibit the growth of some solid tumors and result in an anticancer effect.</p>Formula:C38H46O9Purezza:97.74% - 99.38%Colore e forma:SolidPeso molecolare:646.77SB 415286
CAS:SB 415286 is a potent GSK3α inhibitor with IC50/Ki of 78 nM/31 nM with equally effective inhibition of GSK-3β.Formula:C16H10ClN3O5Purezza:99.55%Colore e forma:SolidPeso molecolare:359.72SR-4835
CAS:<p>SR-4835 is a highly selective dual inhibitor of CDK12 and CDK13(CDK12: IC50=99 nM, Kd=98 nM; CDK13: Kd=4.9 nM), which disables triple-negative breast cancer (</p>Formula:C21H20Cl2N10OPurezza:98.09% - >99.99%Colore e forma:SolidPeso molecolare:499.36Indirubin
CAS:<p>Indirubin (Couroupitine B) is a potent cyclin-dependent kinases and GSK-3β inhibitor with IC50 of about 5 uM and 0.6 uM.</p>Formula:C16H10N2O2Purezza:97.21% - 99.74%Colore e forma:Reddish-Violet PowderPeso molecolare:262.26UC2288
CAS:<p>UC2288, a Sorafenib-based p21 attenuator, reduces p21 levels without affecting its stability.</p>Formula:C20H18ClF6N3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:481.82dBET6
CAS:<p>dBET6 is a selective and cell-permeable degrader of BET based on PROTAC (IC50: 14 nM). It has antitumor activity.</p>Formula:C42H45ClN8O7SPurezza:97.57% - 99.12%Colore e forma:SolidPeso molecolare:841.37Carnosic acid
CAS:Carnosic acid is a lipid absorption inhibitor, endowed with antioxidative, antimicrobial, photoprotective potential, and antiproliferative properties.Formula:C20H28O4Purezza:98.31% - 99.5%Colore e forma:Yellow PowderPeso molecolare:332.43MG-132
CAS:<p>MG-132 (Z-Leu-Leu-Leu-al) is a 26S proteasome inhibitor, cell-permeable and reversible,an autophagy activator, induces apoptosis. High-Quality, Low-Cost!</p>Formula:C26H41N3O5Purezza:95% - 99.99%Colore e forma:White To Off-White PowderPeso molecolare:475.62Taurodeoxycholic acid sodium hydrate
CAS:<p>Taurodeoxycholic acid sodium hydrate (Sodium taurodeoxycholate monohydrate), a hydrophilic bile salt, on bile salt and biliary lipid secretion in the rat.</p>Formula:C26H46NNaO7SPurezza:99.95%Colore e forma:SolidPeso molecolare:539.70Triglycidyl isocyanurate
CAS:<p>Triglycidyl isocyanurate (Teroxirone) is a cancer-research chemical with DNA-altering properties, also used in metal finishing.</p>Formula:C12H15N3O6Purezza:99.01%Colore e forma:White Solid ParticulatesPeso molecolare:297.26GSK4112
CAS:<p>GSK4112 (SR6452) is a Rev-erbα agonist with EC50 of 0.4 μM, also is a small molecule chemical probe for the cell biology of the nuclear heme receptor Rev-erbα.</p>Formula:C18H21ClN2O4SPurezza:99.69%Colore e forma:SolidPeso molecolare:396.89CCF642
CAS:<p>CCF642 (AC1LYELL) is a novel PDI-inhibiting compound with antimyeloma activity.</p>Formula:C15H10N2O4S3Purezza:97.12% - 98.82%Colore e forma:SolidPeso molecolare:378.45PFI-90
CAS:<p>PFI-90, a selective histone demethylase (KDM3B) inhibitor, targets PAX3-FOXO1 action and demonstrates potential antitumor activity.</p>Formula:C11H10N4OPurezza:99.46%Colore e forma:SolidPeso molecolare:214.22Triptonide
CAS:<p>Triptonide treats autoimmune diseases, has antileukemic/tumor effects, is anti-inflammatory, and boosts IL-37.</p>Formula:C20H22O6Purezza:99.11% - 99.64%Colore e forma:White Crystalline PowderPeso molecolare:358.39Nelarabine
CAS:<p>Nelarabine (GW 506U78) is a purine nucleoside analog and DNA synthesis inhibitor with IC50 from 0.067-2.15 μM in tumor cells.</p>Formula:C11H15N5O5Purezza:98.10% - 99.6%Colore e forma:White SolidPeso molecolare:297.27Abacavir sulfate
CAS:<p>Abacavir sulfate (Ziagen) , a nucleoside analogue, effectively utilize its antiviral activity</p>Formula:C14H18N6OH2O4SPurezza:99.79% - 99.85%Colore e forma:White To Off-White SolidPeso molecolare:335.38Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formula:C18H26ClN3O3·C4H6O4Purezza:99.24%Colore e forma:SolidPeso molecolare:485.96Bromosporine
CAS:<p>Bromosporine is a broad spectrum inhibitor for bromodomains for BRD2/4/9 and CECR2 (IC50: 0.41/0.29/0.122/0.017 μM), respectively.</p>Formula:C17H20N6O4SPurezza:99.65% - 99.79%Colore e forma:SolidPeso molecolare:404.44Hispidol
CAS:<p>Hispidol ((Z)-Hispidol) ((Z)-Hispidol) is a potential therapeutic for inflammatory bowel disease; inhibits TNF-α induced adhesion of monocytes to colon</p>Formula:C15H10O4Purezza:97.86% - 98.45%Colore e forma:SolidPeso molecolare:254.24LCL161
CAS:LCL161 is a SMAC mimetic, an IAP antagonist with oral activity that inhibits XIAP and cIAP1. LCL161 has potential antitumor activity. Cost-effective and quality-assured.Formula:C26H33FN4O3SPurezza:99.13% - 99.87%Colore e forma:SolidPeso molecolare:500.63Mocetinostat
CAS:<p>Mocetinostat (MG0103) is an orally available HDAC inhibitor with most potency for HDAC1 (IC50: 0.15 μM), 2- to 10- fold selectivity against HDAC2/3/11.</p>Formula:C23H20N6OPurezza:99% - 99.21%Colore e forma:SolidPeso molecolare:396.44AG1024
CAS:<p>AG1024 (Tyrphostin) suppresses IGF-1R autophosphorylation(IC50=7 μM), and is less potent for IR(IC50=57 μM).</p>Formula:C14H13BrN2OPurezza:98% - 99.37%Colore e forma:SolidPeso molecolare:305.174-Methyldaphnetin
CAS:4-Methyldaphnetin (DHMC) is a potent inhibitor of lipid peroxidation and scavengers of superoxide anion radicals and of aqueous alkylperoxyl radicals.Formula:C10H8O4Purezza:99.73%Colore e forma:SolidPeso molecolare:192.17Brevilin A
CAS:<p>Brevilin A, a sesquiterpene from Centipeda minima, hinders JAK and blocks STAT3 (IC50=10.6μM), inducing apoptosis and autophagy in cancer cells.</p>Formula:C20H26O5Purezza:99.97% - >99.99%Colore e forma:SolidPeso molecolare:346.42Methotrexate disodium
CAS:<p>Methotrexate disodium is an tetrahydrofolate dehydrogenase inhibitor</p>Formula:C20H20N8Na2O5Purezza:99.77% - 99.96%Colore e forma:SolidPeso molecolare:498.4Actein
CAS:<p>Actein stimulates bone formation, counters osteoporosis and oxidative damage, and may treat lipid disorders and cancer, inhibiting breast cancer cell growth.</p>Formula:C37H56O11Purezza:≥98%Colore e forma:Brown PowderPeso molecolare:676.83UCF 101
CAS:<p>UCF 101 is a specific inhibitor of HtrA2 and reduces apoptosis in PC12 cells.</p>Formula:C27H17N3O5SPurezza:99.64%Colore e forma:SolidPeso molecolare:495.51Gomisin N
CAS:<p>Gomisin N from Schisandra chinensis offers sedative effects, allergy relief, and cancer cell inhibition/apoptosis.</p>Formula:C23H28O6Purezza:99.97% - >99.99%Colore e forma:SolidPeso molecolare:400.46PHYTOSPHINGOSINE
CAS:<p>Phytosphingosine: anticancer phospholipid; triggers apoptosis in cancer cells via caspase 8 activation and Bax translocation.</p>Formula:C18H39NO3Purezza:99.81%Colore e forma:SolidPeso molecolare:317.51Barasertib-HQPA
CAS:<p>Barasertib-HQPA (AZD2811) is a highly selective Aurora B inhibitor (IC50: 0.37 nM) and demonstrates ~3,700-fold greater selectivity than Aurora A.</p>Formula:C26H30FN7O3Purezza:98.43% - 99.29%Colore e forma:SolidPeso molecolare:507.56AZD-7648
CAS:<p>AZD-7648 is an inhibitor of DNA-dependent protein kinase (DNA-PK) with the IC50 of 0.63 nM in an enzyme assay,has anti-tumor activity.</p>Formula:C18H20N8O2Purezza:99.03% - 99.85%Colore e forma:SolidPeso molecolare:380.4Verbascoside
CAS:<p>Verbascoside (Kusaginin) is a protein kinase C inhibitor with antimicrobial, anti-inflammatory activities.</p>Formula:C29H36O15Purezza:97.46% - 99.55%Colore e forma:SolidPeso molecolare:624.59CAY10404
CAS:<p>CAY10404: potent COX-1/2 inhibitor; blocks PKB/Akt, MAPK pathways; triggers NSC-LC apoptosis; analgesic, anti-inflammatory, anti-cancer.</p>Formula:C17H12F3NO3SPurezza:99.02%Colore e forma:SolidPeso molecolare:367.34Picroside II
CAS:<p>Picroside II (Vanilloyl catalpol) is the main active ingredient in iridoid glycosides.</p>Formula:C23H28O13Purezza:98% - 99.83%Colore e forma:SolidPeso molecolare:512.46Desmethylanethol trithione
CAS:<p>Desmethylanethol trithione (ADT-OH), a synthetic H2S donor, modulates tPA effects, reduces stroke damage, and improves recovery in mice.</p>Formula:C9H6OS3Purezza:98.05% - 98.41%Colore e forma:SolidPeso molecolare:226.34ONC212
CAS:<p>ONC212, a fluorinated-ONC201 analogue, is a selective agonist of GPR132.</p>Formula:C24H23F3N4OPurezza:99.79%Colore e forma:SolidPeso molecolare:440.46β-Ionone
CAS:<p>β-Ionone (β-lonone) is an end-ring analog of β-carotenoids which widely distributed in fruit and vegetables,with anti-proliferative, anti-metastatic</p>Formula:C13H20OPurezza:98.52%Colore e forma:Colourless Liquid OilyPeso molecolare:192.3GS-444217
CAS:<p>GS-444217 is a selective ATP-competitive inhibitor of apoptosis signal-regulating kinase 1 (ASK1, IC50: 2.87 nM).</p>Formula:C23H21N7OPurezza:99.08%Colore e forma:SolidPeso molecolare:411.46OUL35
CAS:<p>OUL35 (NSC-39047) is a selective PARP-10 inhibitor, and small-molecule ARTD10 inhibitor. OUL35 has been shown to rescue cells from ARTD10-induced cell death.</p>Formula:C14H12N2O3Purezza:99.2%Colore e forma:SolidPeso molecolare:256.26TCPOBOP
CAS:<p>TCPOBOP is a constitutive androstane receptor agonist that induces robust hepatocyte proliferation and hepatomegaly.</p>Formula:C16H8Cl4N2O2Purezza:99.7%Colore e forma:SolidPeso molecolare:402.06UTL-5g
CAS:<p>UTL-5g is a chemoprotective TNF-α inhibitor reducing cisplatin side effects and toxicity in liver, kidneys, and blood.</p>Formula:C11H8Cl2N2O2Purezza:99.83%Colore e forma:SolidPeso molecolare:271.1OTS514
CAS:OTS514 (OTS514 Hydrochloride) is a potent TOPK inhibitor.Formula:C21H20N2O2SPurezza:99.62%Colore e forma:SolidPeso molecolare:364.46UAMC-3203
CAS:<p>UAMC-3203 is a potent and selective Ferroptosis inhibitor (IC50: 12 nM).</p>Formula:C25H37N5O2SPurezza:97.052% - 99.72%Colore e forma:SolidPeso molecolare:471.66Isocurcumenol
CAS:1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).Formula:C15H22O2Purezza:99.29% - ≥95%Colore e forma:SolidPeso molecolare:234.33CCT007093
CAS:<p>CCT007093 is an effective PPM1D (WIP1) inhibitor (IC50: 8.4 μM).</p>Formula:C15H12OS2Purezza:98% - 99.88%Colore e forma:SolidPeso molecolare:272.39Obatoclax Mesylate
CAS:Obatoclax Mesylate (GX15-070) is a Bcl-2 antagonist (Ki: 0.22 μM) and can induce apoptosis with up-regulation of Bim, induced cytochrome c release, andFormula:C20H19N3O·CH4O3SPurezza:99.58% - 99.88%Colore e forma:SolidPeso molecolare:413.49CHR-6494 TFA
CAS:<p>CHR-6494 TFA: potent haspin inhibitor (IC50=2 nM), blocks H3T3 phosphorylation, triggers apoptosis in cancer cells. Used for cancer research.</p>Formula:C18H17F3N6O2Purezza:99.50%Colore e forma:SolidPeso molecolare:406.36MPTP hydrochloride
CAS:<p>MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.</p>Formula:C12H16ClNPurezza:96.35% - >99.99%Colore e forma:SolidPeso molecolare:209.72B355252
CAS:<p>B355252 prevents glutamate-induced cell death and boosts NGF's nerve growth effects.</p>Formula:C25H24ClN3O3S2Purezza:98.73% - 99.92%Colore e forma:SolidPeso molecolare:514.06Choline
CAS:<p>Choline is a ubiquitous water soluble nutrient, often associated with the B vitamins</p>Formula:C5H15NO2Purezza:99.97% - ≥98%Colore e forma:LiquidPeso molecolare:121.18Salubrinal
CAS:<p>Salubrinal, a phosphatases (PP1) inhibitor(IC50=1.7 μM), exhibits function on the eukaryotic translation initiation factor 2 subunit (eIF2α).</p>Formula:C21H17Cl3N4OSPurezza:97.25% - >99.99%Colore e forma:SolidPeso molecolare:479.81Polygalacin D
CAS:<p>Polygalacin D shows anti- proliferation, anti-inflammary, and hepatoprotective activities, it can inhibit the expression of lipopolysaccharide (LPS)-induced</p>Formula:C57H92O27Purezza:98.95% - ≥98%Colore e forma:SolidPeso molecolare:1209.4m-3M3FBS
CAS:<p>m-3M3FBS is a phospholipase C (PLC) activator.</p>Formula:C16H16F3NO2SPurezza:99.66%Colore e forma:SolidPeso molecolare:343.36ENMD-2076
CAS:<p>ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.</p>Formula:C21H25N7Purezza:97.63% - ≥95%Colore e forma:SolidPeso molecolare:375.47(E/Z)-TG003
CAS:<p>(E/Z)-TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor.</p>Formula:C13H15NO2SPurezza:98% - 99.04%Colore e forma:SolidPeso molecolare:249.33Malabaricone B
CAS:<p>Malabaricone B is a Spice-derived phenolic, it induces mitochondrial damage in lung cancer cells via a p53-independent pathway.</p>Formula:C21H26O4Purezza:99.84% - 99.91%Colore e forma:SolidPeso molecolare:342.43PD0166285
CAS:<p>PD0166285 is a potent Wee1 and Chk1 inhibitor with activity at nanomolar concentrations.PD0166285 is a novel G2 checkpoint abrogator.</p>Formula:C26H27Cl2N5O2Purezza:99.23%Colore e forma:SolidPeso molecolare:512.43AT7519
CAS:<p>AT7519 is a CDK1/2/4/6/9 inhibitor (IC50: 10-210 nM). It is less effective to CDK3 and little active to CDK7.</p>Formula:C16H17Cl2N5O2Purezza:98.88% - 99.65%Colore e forma:SolidPeso molecolare:382.24Telekin
CAS:<p>Telekin, a sesquiterpene lactone from Carpesium divaricatum, strongly inhibits cancer cell growth.</p>Formula:C15H20O3Purezza:99.86% - 99.97%Colore e forma:SolidPeso molecolare:248.32Delanzomib
CAS:<p>Delanzomib (CEP-18770) is an oral proteasome inhibitor with an IC50 of 3.8 nM, targeting chymotrypsin-like activity with minimal effect on other activities.</p>Formula:C21H28BN3O5Purezza:95.52% - 99.46%Colore e forma:SolidPeso molecolare:413.28Gardenin B
CAS:<p>Gardenin B exhibits superior antiproliferative activity against lung, breast, colon, hepatic and leukaemia cell lines as well as in keratinocytes .</p>Formula:C19H18O7Purezza:98.80% - 99.74%Colore e forma:SolidPeso molecolare:358.34Salvigenin
CAS:<p>Salvigenin is a potent hMAO-A inhibitor, has neuroprotective, antitumor and immunomodulatory effects.</p>Formula:C18H16O6Purezza:99.17% - 99.78%Colore e forma:SolidPeso molecolare:328.32Toddaculin
CAS:<p>Toddaculine may be beneficial for the prevention and treatment of osteoporosis, it can not only inhibit the differentiation of osteoclasts via activation of the</p>Formula:C16H18O4Purezza:99.91%Colore e forma:SolidPeso molecolare:274.31Zoledronic acid monohydrate
CAS:<p>Zoledronic acid monohydrate (CGP 42446) is a synthetic imidazole bisphosphonate analog with anti-bone-resorption activity.</p>Formula:C5H12N2O8P2Purezza:99.91%Colore e forma:White To Off-White PowderPeso molecolare:290.1Isoalantolactone
CAS:<p>Isoalantolactone (Isohelenin), isolated from Inula spp., can inhibit the growth of several types of Y cells.</p>Formula:C15H20O2Purezza:99.75% - 99.94%Colore e forma:SolidPeso molecolare:232.32Momordin Ic
CAS:<p>Momordin Ic (Momordin 1c) might represent a potential anticancer activity, by inducing apoptosis through oxidative stress-regulated mitochondrial dysfunction</p>Formula:C41H64O13Purezza:98% - 99.69%Colore e forma:SolidPeso molecolare:764.94Neferine
CAS:<p>Neferine: anti-tumor, enhances DOX efficacy, prevents diabetic vasculopathy; mediates via CYP3A4, GSH depletion, blocks ROS/Akt/NF-κB.</p>Formula:C38H44N2O6Purezza:98.81% - 99.65%Colore e forma:SolidPeso molecolare:624.77PKR-IN-C16
CAS:<p>PKR-IN-C16: inhibits PKR autophosphorylation and translation blockade; binds ATP site; IC50 of 186-210 nM; protects cells from ER stress damage.</p>Formula:C13H8N4OSPurezza:97.8%Colore e forma:SolidPeso molecolare:268.29AC1NS4RE
CAS:<p>It is a tyrosine kinase inhibitor.</p>Formula:C15H13ClN2OPurezza:99.53%Colore e forma:SolidPeso molecolare:272.73Acacetin
CAS:<p>Acacetin (5,7-Dihydroxy-4'-methoxyflavone) is an O-methylated flavone found in various plants, shows antinociceptive, anti-inflammatory, and antioxidant</p>Formula:C16H12O5Purezza:96.26% - ≥95%Colore e forma:Pale-Yellow NeedlesPeso molecolare:284.26VK3-OCH3
CAS:VK3-OCH3 (2-[(2-Methoxy)ethylthio]-3-methyl-1,4-na) is a selective antitumor agent via heme oxygenase (HO-1) related mechanisms; Vitamine K3 analogue.Formula:C14H14O3SPurezza:99.71%Colore e forma:SolidPeso molecolare:262.32CAY10505
CAS:<p>CAY10505, a form of dehydroxyl of AS-252424, is a PI3Kγ inhibitor (IC50: 33 nM).</p>Formula:C14H8FNO3SPurezza:99.69% - 99.74%Colore e forma:SolidPeso molecolare:289.28MRS 2578
CAS:MRS2578, an effective P2Y6 receptor antagonist with IC50 of 37 nM, shows insignificant inhibition at P2Y1, P2Y2, P2Y4, and P2Y11 receptors.Formula:C20H20N6S4Purezza:97.58% - 99.73%Colore e forma:White SolidPeso molecolare:472.67Levomenol
CAS:<p>Levomenol, or (-)-α-Bisabolol, is a sesquiterpene in aromatic plant oils with antioxidant, anti-inflammatory, and anti-apoptotic properties.</p>Formula:C15H26OPurezza:96.01%Colore e forma:Clear To Yellowish LiquidPeso molecolare:222.37Polyphyllin I
CAS:<p>Polyphyllin D induces apoptosis via the mitochondrial apoptotic pathway as evidenced by decreased Bcl-2 expression levels, disruption of MMP and increased Bax,</p>Formula:C44H70O16Purezza:98% - 99.5%Colore e forma:SolidPeso molecolare:855.02PIK-75
CAS:<p>PIK-75, a DNA-PK and PI3K inhibitor, suppresses DNA-PK(IC50=2 nM), p110α(IC50=5.8 nM) and p110γ(IC50=76 nM).</p>Formula:C16H14BrN5O4SPurezza:98.52% - >99.99%Colore e forma:SolidPeso molecolare:452.28Epothilone A
CAS:<p>Epothilone A (Epo A) is a microtubule-stabilizing agent with EC0.01 of 2 μM.</p>Formula:C26H39NO6SPurezza:99.89% - 99.92%Colore e forma:SolidPeso molecolare:493.66Fedratinib hydrochloride hydrate
CAS:<p>Fedratinib hydrochloride hydrate (SAR 302503 hydrochloride hydrate) is a potent, selective, ATP-competitive and orally active JAK2 inhibitor.</p>Formula:C27H40Cl2N6O4SPurezza:98.96% - 99.87%Colore e forma:SolidPeso molecolare:615.61G5-7
CAS:<p>G5-7 is an oral JAK2 inhibitor targeting EGFR/STAT3 phosphorylation with potential for glioma research.</p>Formula:C22H19F2NO3Purezza:97.3%Colore e forma:SolidPeso molecolare:383.39Goserelin acetate
CAS:<p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>Formula:C61H88N18O16Purezza:99.77% - >99.99%Colore e forma:White Crystalline PowderPeso molecolare:1329.46Alginic acid
CAS:<p>Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.</p>Formula:C14H22O13Purezza:≥98%Colore e forma:SolidPeso molecolare:398.317OTS514 hydrochloride
CAS:OTS514 hydrochloride is a highly effective TOPK(T-LAK cell-originated protein kinase) inhibitor (IC50: 2.6 nM).Formula:C21H20N2O2S·HClPurezza:99.67% - 99.84%Colore e forma:SolidPeso molecolare:400.92Kynurenic acid sodium
CAS:Kynurenic acid sodium salt is an endogenous tryptophan metabolite. It antagonizes NMDA, glutamate, and α7 nicotinic receptors, and agonizes GPR35.Formula:C10H6NNaO3Purezza:99.47%Colore e forma:SolidPeso molecolare:211.15MK-886
CAS:MK-886 (L 663536) is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP).Formula:C27H34ClNO2SPurezza:99.23% - 99.84%Colore e forma:SolidPeso molecolare:472.08Xanthatin
CAS:Xanthatin exhibits cytotoxic, antibacterial, antifungal properties, may treat NSCLC, and inhibits melanoma by targeting Wnt/β-catenin and angiogenesis.Formula:C15H18O3Purezza:98.48% - 99.96%Colore e forma:SolidPeso molecolare:246.3CASIN
CAS:CASIN (Pirl1-related Compound 2) is a specific inhibitor of GTPase Cdc42 (IC50: 2 uM).Formula:C20H22N2OPurezza:98.18% - >99.99%Colore e forma:SolidPeso molecolare:306.4NU 7026
CAS:<p>NU 7026 (DNA-PK Inhibitor II) is an effective DNA-PK inhibitor (IC50: 0.23 μM, in cell-free assays), 60-fold selective for DNA-PK than PI3K and no inhibition</p>Formula:C17H15NO3Purezza:99.51% - >99.99%Colore e forma:SolidPeso molecolare:281.314EGI-1
CAS:<p>4EGI-1, a competitive eIF4E/eIF4 g interaction inhibitor, binds to eIF4E(KD=25 μM).</p>Formula:C18H12Cl2N4O4SPurezza:96.8% - 99.12%Colore e forma:SolidPeso molecolare:451.28Lithocholic acid
CAS:Lithocholic acid (3α-Hydroxy-5β-cholanic acid) is a toxic secondary bile acid, They were FXR antagonists (IC50=0.7, 1.4 μM). High-Quality, Low-Cost!Formula:C24H40O3Purezza:98% - 99.93%Colore e forma:Hexagonal Leaflets From Alc Prisms From Acetic Acid Powder (Ntp 1992)Peso molecolare:376.57SKF-96365 hydrochloride
CAS:<p>SKF-96365 hydrochloride (SKF96365) , a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal Y</p>Formula:C22H27ClN2O3Purezza:99.47% - 99.92%Colore e forma:SolidPeso molecolare:402.91Xanthohumol
CAS:<p>Xanthohumol, also known as 2', 4, 4'-trihydroxy-6'-methoxy-3'-prenylchalcone or desmethylxanthohumol, is a member of the class of compounds known as 3-</p>Formula:C21H22O5Purezza:98.19% - 99.67%Colore e forma:Orange PowderPeso molecolare:354.4NSC 66811
CAS:<p>NSC 66811 inhibits MDM2-p53 interaction with 120 nM affinity, activating p53 in cancer cells.</p>Formula:C23H20N2OPurezza:96.94%Colore e forma:SolidPeso molecolare:340.42Palmatine
CAS:<p>Palmatine, also known as Burasaine, inhibits dopamine production and may treat flavivirus, jaundice, dysentery, hypertension, and liver issues.</p>Formula:C21H22NO4Purezza:96.28% - 99.49%Colore e forma:SolidPeso molecolare:352.4Midostaurin
CAS:<p>PKC412(Midostaurin (PKC412); CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor.</p>Formula:C35H30N4O4Purezza:97.61% - >99.99%Colore e forma:SolidPeso molecolare:570.64Suramin Sodium Salt
CAS:<p>Suramin Sodium Salt (BAY-205) is a polysulphonated naphthylurea with potential antineoplastic activity. Suramin blocks the binding of various growth factors.</p>Formula:C51H34N6Na6O23S6Purezza:97.47% - 99.97%Colore e forma:WhitePeso molecolare:1429.15(S)-10-Hydroxycamptothecin
CAS:<p>(S)-10-Hydroxycamptothecin (10-HCPT) is a DNA topoisomerase I inhibitor, utilized as a clinical therapy agent against hepatoma.</p>Formula:C20H16N2O5Purezza:99.09% - 99.81%Colore e forma:SolidPeso molecolare:364.35AZD0156
CAS:<p>AZD0156 , an effective and specific inhibitors of ATM kinase, is potential antineoplastic activities and chemo-/radio-sensitizing.</p>Formula:C26H31N5O3Purezza:99.13% - 99.87%Colore e forma:SolidPeso molecolare:461.56TG101209
CAS:<p>TG101209 is a selective JAK2 inhibitor with IC50 of 6 nM.</p>Formula:C26H35N7O2SPurezza:99% - >99.99%Colore e forma:SolidPeso molecolare:509.67MGCD-265 analog
CAS:<p>Glesatinib, an oral tyrosine kinase inhibitor, targets c-Met and VEGFR2 with IC50s of 29 nM and 10 nM, may treat cancer.</p>Formula:C26H20FN5O2S2Purezza:98.06% - 98.68%Colore e forma:SolidPeso molecolare:517.6Ginsenoside Rg1
CAS:<p>Ginsenoside Rg1 (Panaxoside Rg1) is a class of steroid glycosides, and triterpene saponins found exclusively in the plant genus Panax (ginseng).</p>Formula:C42H72O14Purezza:99% - 99.74%Colore e forma:White Crystalline PowderPeso molecolare:801.01Valinomycin
CAS:<p>Valinomycin (NSC-122023) is a cyclic depsipeptide antibiotic and a potassium-specific ionophore.Valinomycin induces PINK1 activation and promotes Parkin</p>Formula:C54H90N6O18Purezza:95.37% - 97.16%Colore e forma:White SolidPeso molecolare:1111.32Boc-Asp(OMe)-fluoromethyl ketone
CAS:<p>Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.</p>Formula:C11H18FNO5Purezza:≥98%Colore e forma:SolidPeso molecolare:263.26LYN-1604
CAS:<p>LYN-1604 is a novel activator of ULK1, inducing cell death involved in ATF3, RAD21, and caspase3, accompanied by autophagy and apoptosis.</p>Formula:C33H43Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:584.62BMS-202
CAS:<p>BMS-202 (PD1-PDL1 inhibitor 2) is an inhibitor of the PD-1 (Programmed death- 1) /PD-Ll (Programmed death-ligand 1) protein/protein interaction.</p>Formula:C25H29N3O3Purezza:97.92% - 99.66%Colore e forma:SolidPeso molecolare:419.52Tasisulam
CAS:<p>Tasisulam (LY573636) is an apoptosis inducer and an antitumor agent via the intrinsic pathway.</p>Formula:C11H6BrCl2NO3S2Purezza:99% - >99.99%Colore e forma:SolidPeso molecolare:415.11SP2509
CAS:<p>SP2509 is a specific histone demethylase LSD1 inhibitor(IC50 =13 nM).</p>Formula:C19H20ClN3O5SPurezza:98.82% - 99.53%Colore e forma:SolidPeso molecolare:437.9RO8994
CAS:<p>RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).</p>Formula:C31H31Cl2FN4O4Purezza:99.31% - 99.44%Colore e forma:SolidPeso molecolare:613.51PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formula:C16H12N4SPurezza:99.35%Colore e forma:SolidPeso molecolare:292.36Kaempferol
CAS:<p>Kaempferol (Robigenin) is a natural flavonoid and an inverse agonist of ERRα and ERRγ.</p>Formula:C15H10O6Purezza:98% - 99.41%Colore e forma:Yellow Needles From Alcohol And Water SolidPeso molecolare:286.24physalin F
CAS:<p>Physalin F is a natural blocker of CaV2.3 (R-type) and CaV2.2 (N-type) voltage-gated calcium channels.Cost-effective and quality-assured.</p>Formula:C28H30O10Purezza:99.5% - 99.61%Colore e forma:SolidPeso molecolare:526.53Apitolisib
CAS:<p>Apitolisib (RG 7422) is a PI3K inhibitor, used in cancer trials, targeting PI3Kα, β, δ, γ (IC50= 5, 27, 7, 14 nM).</p>Formula:C23H30N8O3SPurezza:98.28% - 99.64%Colore e forma:SolidPeso molecolare:498.6Kobe0065
CAS:<p>Kobe0065: novel small-molecule, inhibits Ras–Raf, Ki=46±13 μM, blocks H-Ras·GTP/c-Raf-1 RBD binding.</p>Formula:C15H11ClF3N5O4SPurezza:98% - >99.99%Colore e forma:SolidPeso molecolare:449.79α-Mangostin
CAS:alpha-Mangostin (Mangostin) is a natural xanthonoid, a type of organic compound isolated from various parts of the mangosteen tree.Formula:C24H26O6Purezza:98.22% - 99.49%Colore e forma:Yellow PowderPeso molecolare:410.46DPN
CAS:<p>DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .</p>Formula:C15H13NO2Purezza:99.01%Colore e forma:Off-White SolidPeso molecolare:239.27Selumetinib
CAS:<p>Selumetinib (AZD6244) is a selectivity and non-ATP-competitive MEK1/2 inhibitor. Selumetinib has antitumor activity. Cost-effective and quality-assured.</p>Formula:C17H15BrClFN4O3Purezza:98.1% - 99.90%Colore e forma:White Or Pale White SolidPeso molecolare:457.68SM-164
CAS:<p>SM-164 binds to XIAP protein containing both the BIR2 and BIR3 domains (IC50: 1.39 nM). It acts as an extremely potent antagonist of XIAP.</p>Formula:C62H84N14O6Purezza:98.53% - 99.92%Colore e forma:SolidPeso molecolare:1121.42SGI-1027
CAS:<p>SGI-1027 (DNA Methyltransferase Inhibitor II) is an effective and selective inhibitor of DNA methyltransferase (DNMT).</p>Formula:C27H23N7OPurezza:99.45% - 99.78%Colore e forma:SolidPeso molecolare:461.52FTI-277 hydrochloride
CAS:<p>FTI-277 HCl: potent FTase inhibitor, IC50 500 pM, 100x more selective than GGTase I.</p>Formula:C22H30ClN3O3S2Purezza:97.57% - 97.61%Colore e forma:SolidPeso molecolare:484.07CID5721353
CAS:<p>CID5721353 disrupts BCL6/corepressor complexes, binds critical BTB groove site in vitro/vivo.</p>Formula:C15H9BrN2O6S2Purezza:98.90%Colore e forma:SolidPeso molecolare:457.28Nutlin-3a
CAS:<p>Nutlin-3a is the active enantiomer of Nutlin-3, an MDM2 antagonist that inhibits MDM2-p53 interaction. Nutlin-3a has antitumor activity. Cost-effective and quality-assured.</p>Formula:C30H30Cl2N4O4Purezza:95.62% - 99.71%Colore e forma:SolidPeso molecolare:581.49Apoptozole
CAS:<p>Apoptozole (Apoptosis Activator VII) is an inhibitor of the ATPase domain of Hsc70 and Hsp70, and can induce apoptosis.</p>Formula:C33H25F6N3O3Purezza:99.75%Colore e forma:SolidPeso molecolare:625.56Quisinostat dihydrochloride
CAS:<p>Quisinostat dihydrochloride (JNJ26854165(Quisinostat) 2HCl) 是一种有口服活性，高效的 pan-HDAC 抑制剂，具有广泛的抗肿瘤活性。它对 HDAC1、HDAC2、HDAC4、HDAC10和HDAC11 的IC50值分别为 0.11 nM、0.33 nM、0.64 nM、0.46 nM 和 0.37 nM。</p>Formula:C21H28Cl2N6O2Purezza:97.13%Colore e forma:SolidPeso molecolare:467.39Pifithrin-α hydrobromide
CAS:Pifithrin-α hydrobromide (Pifithrin-α hydrobromide) is a p53 inhibitor, inhibiting p53-dependent transactivation of p53-responsive genes.Formula:C16H18N2OS·HBrPurezza:97.71% - >99.99%Colore e forma:SolidPeso molecolare:367.3Atopaxar hydrochloride
CAS:<p>Atopaxar hydrochloride is used in the Treatment of Cardiovascular Disorders.</p>Formula:C29H39ClFN3O5Colore e forma:SolidPeso molecolare:564.1R1530
CAS:<p>R1530 is a multikinase inhibitor with antineoplastic and antiangiogenesis activities.</p>Formula:C18H14ClFN4OPurezza:98.422%Colore e forma:SolidPeso molecolare:356.78
