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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5400 produtos de "Neurociência"

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  • BSB

    CAS:
    <p>BSB is a Congo red-derived fluorescent probe, an amyloid protein imaging agent, interacting with amyloid fibrils formed by Aβ (1-40) peptides in rodents.</p>
    Fórmula:C24H17BrO6
    Pureza:95.53%
    Cor e Forma:Solid
    Peso molecular:481.29
  • Amyloid β-Protein (3-42)

    CAS:
    <p>Amyloid β-Protein (3-42), the precursor of Pyr peptide, serves as the foundation of the amyloid template block in Alzheimer's disease when modified to</p>
    Cor e Forma:Solid
  • Desfesoterodine

    CAS:
    <p>Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.</p>
    Fórmula:C22H31NO2
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:341.49
  • Biotin-β-Amyloid (1-42), human TFA


    <p>Biotin-β-Amyloid (1-42), human TFA, also known as Biotin-Amyloid β-Peptide (1-42) (human) TFA, is a biotin-labeled 42-amino acid peptide implicated in the</p>
    Fórmula:C215H326F3N57O64S2
    Cor e Forma:Solid
    Peso molecular:4854.36
  • AChE/Aβ-IN-6


    <p>BACE1-IN-15 (compound 4j) serves as an effective inhibitor of BACE1 (β-secretase), efficiently mitigating the copper-induced toxicity of Aβ, with an EC50 value of 0.68 μM.</p>
    Cor e Forma:Odour Solid
  • ZZL-7

    CAS:
    <p>ZZL-7 is a rapid antidepressant targeting nNOS &amp; SERT in DRN, crosses blood-brain barrier, with MDD research potential.</p>
    Fórmula:C11H20N2O4
    Pureza:99.79%
    Cor e Forma:Soild
    Peso molecular:244.29
  • Lu AF27139

    CAS:
    <p>Lu AF27139: P2X7 receptor antagonist; IC50: 12 nM (human), 2.4 nM (rat); Ki: 22 (mouse), 54 (human), 13 nM (rat); for CNS research.</p>
    Fórmula:C21H19ClF3N5O2S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:497.92
  • KRP-199 sodium


    <p>KRP-199 sodium sodium is highly potent and selective for AMPA-R in vitro and exhibits good neuroprotection in vivo.</p>
    Fórmula:C22H12F3N5Na2O7
    Pureza:97.27%
    Cor e Forma:Soild
    Peso molecular:561.33
  • mGluR3 modulator-1

    CAS:
    <p>1-ethyl-3-morpholin-4-yl tetrahydroisoquinoline: mGluR3 modulator, potential for Parkinson's.</p>
    Fórmula:C16H21N3O
    Pureza:98.99%
    Cor e Forma:Solid
    Peso molecular:271.36
  • (±)-Acetylcarnitine chloride

    CAS:
    <p>(±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can be used in studies of neuritis.</p>
    Fórmula:C9H18ClNO4
    Pureza:99.98%
    Cor e Forma:White Crystalline Powder
    Peso molecular:239.7
  • SB656104

    CAS:
    <p>SB656104 is a bioactive chemical.</p>
    Fórmula:C25H30ClN3O3S
    Cor e Forma:Solid
    Peso molecular:488.04
  • Dalidnetug

    CAS:
    <p>Dalidnetug is a humanized monoclonal antibody that targets human β-amyloid precursor protein (APP). By specifically binding to APP, Dalidnetug reduces the production of β-amyloid (Aβ), thereby demonstrating activity in clearing β-amyloid. This compound holds potential for research in Alzheimer's disease.</p>
    Cor e Forma:Liquid
  • Pomaglumetad methionil anhydrous

    CAS:
    <p>LY2140023, potential schizophrenia treatment, is an oral prodrug of LY404039, a selective mGlu2/3 agonist.</p>
    Fórmula:C12H18N2O7S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:366.41
  • Brexpiprazole S-oxide D8

    CAS:
    <p>Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled metabolite of Brexpiprazole, a partial agonist at 5-HT1A and dopamine receptors.</p>
    Fórmula:C25H19D8N3O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:457.61
  • β-Amyloid (35-42)

    CAS:
    <p>β-Amyloid (35-42) is a peptide derived from the beta-amyloid protein, encompassing amino acids 35 through 42.</p>
    Fórmula:C33H60N8O9S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:744.94
  • Encecalinol

    CAS:
    <p>Encecalinol, a compound isolated from the aerial parts of Ageratina grandifolia, acts as a potent inhibitor of calmodulin [1].</p>
    Fórmula:C14H18O3
    Cor e Forma:Solid
    Peso molecular:234.29
  • SB 216641

    CAS:
    <p>SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety disorders and depression.</p>
    Fórmula:C28H30N4O4
    Pureza:98.09%
    Cor e Forma:Solid
    Peso molecular:486.56
  • TIM-098a


    <p>TIM-098a is a selective AAK1 inhibitor with an IC50 of 0.24 µM. It does not inhibit CaMKK isoforms. By inhibiting AAK1 kinase activity, TIM-098a disrupts AAK1-regulated endocytosis.</p>
    Fórmula:C18H11N3O2
    Peso molecular:301.08513
  • AChE-IN-49


    <p>AChE-IN-49 (Compd (S)-7g) is an acetylcholinesterase (AChE) inhibitor with an IC50 value of 0.0003 μM.</p>
    Fórmula:C31H28BrClN2O3
    Peso molecular:590.09718
  • AChE-IN-60


    <p>AChE-IN-60 (compound 6k) is a potent inhibitor of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), with IC50 values of 27 nM and 43 nM, respectively. It also inhibits monoamine oxidase MAO-A and MAO-B, with IC50 values of 353 nM and 716 nM, respectively.</p>
    Fórmula:C24H29N3O4S3
    Peso molecular:519.13202