
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(939 produtos)
- ACK(1 produtos)
- AChR(575 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.945 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(561 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor GABA(336 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(358 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(28 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5400 produtos de "Neurociência"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
SAHM1
CAS:<p>Notch pathway inhibitor - stabilized hydrocarbon-stapled alpha helical peptide. Targets the protein-protein interface and prevents Notch complex assembly.</p>Fórmula:C94H162N36O23SPureza:98%Cor e Forma:SolidPeso molecular:2196.58Dicloromezotiaz
CAS:<p>Dicloromezotiaz: Potent insecticide targeting nAChRs, controls various lepidoptera.</p>Fórmula:C19H12Cl3N3O2SCor e Forma:SolidPeso molecular:452.74Deoxynojirimycin Tetrabenzyl Ether
CAS:<p>Deoxynojirimycin tetrabenzyl ether aids in making 1-dNM, a strong α-glucosidase I & II blocker.</p>Fórmula:C34H37NO4Cor e Forma:SolidPeso molecular:523.673Laniquidar TFA
<p>Laniquidar TFA (R101933), a non-competitive P-gp inhibitor, has an IC50 of 0.51 μM; used to study AML and MDS, but with limited bioavailability.</p>Fórmula:C39H37F3N4O5Pureza:99.85%Cor e Forma:SoildPeso molecular:698.73Cyclodrine
CAS:<p>Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.</p>Fórmula:C19H29NO3Pureza:97.62%Cor e Forma:SoildPeso molecular:319.443-Aminopropylphosphinic acid
CAS:<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Fórmula:C3H10NO2PCor e Forma:SolidPeso molecular:123.0922-Hydroxyalbrassitriol
CAS:<p>2-Hydroxyalbrassitriol (Compound 6) is an AChE inhibitor with an IC 50 of 35.97 μM [1] .</p>Fórmula:C15H26O4Cor e Forma:SolidPeso molecular:270.36COX-2-IN-49
<p>COX-2-IN-49 (compound 6c) is a potent inhibitor of cyclooxygenase-2 (COX-2), displaying an IC50 value of 2.671 µM. This compound exhibits anti-proliferative properties and holds potential for use in cancer research.</p>Cor e Forma:Odour SolidFeralolide
CAS:<p>Feralolide, a dihydroisocoumarin from the methanolic extract of aloe vera resin, functions as a dual inhibitor of acetylcholinesterase (AChE) and</p>Fórmula:C18H16O7Cor e Forma:SolidPeso molecular:344.32AChE-IN-87
<p>AChE-IN-87 is an AChE inhibitor with an IC50 of 0.05 μM and a Ki of 16.93 nM. It exhibits no cytotoxicity toward 3T3 cells and is suitable for Alzheimer's disease (AD) research.</p>Fórmula:C32H39N3O12S2Cor e Forma:SolidPeso molecular:721.19752LU-32-176B
CAS:<p>LU32-176B is a bioactive chemical.</p>Fórmula:C23H24F2N2O2Cor e Forma:SolidPeso molecular:398.45MK-0969
CAS:<p>MK-0969 (J-104135) is a possible M3 antagonist for the treatment of chronic obstructive pulmonary disease.</p>Fórmula:C24H30F2N4O2Cor e Forma:SolidPeso molecular:444.52TZ4M
<p>TZ4M, a 2,4-thiazolidinedione (TZD)-based anti-ADV agent, exhibits neuroprotective effects and acetylcholinesterase (AChE) inhibition in human plasma.</p>Fórmula:C19H15NO4SCor e Forma:SolidPeso molecular:353.392-Methyl-N,N-dimethyltryptamine
CAS:<p>2-Methyl-N,N-dimethyltryptamine (2,N,N-TMT, compound 15) exhibits binding affinity for the serotonin (5-HT) receptor, with a pA2 value of 6.04. It plays a significant role in neurological disease research.</p>Fórmula:C13H18N2Cor e Forma:SolidPeso molecular:202.3β-Amyloid (1-34)
CAS:<p>This is a fragment of beta-amyloid peptide. It has amino acids 1 through 34.</p>Fórmula:C170H253N47O52Pureza:98%Cor e Forma:SolidPeso molecular:3787.2Methyl ganoderate A acetonide
CAS:<p>Methyl ganoderate A from Ganoderma lucidum is a natural AChE inhibitor (IC50=18.35 μM) for Alzheimer's research.</p>Fórmula:C34H50O7Cor e Forma:SolidPeso molecular:570.76Antidepressant agent 4
<p>Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.</p>Fórmula:C19H38ClN5O2SCor e Forma:SolidPeso molecular:436.06Lesogaberan napadisylate
CAS:<p>Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.</p>Fórmula:C13H17FNO5PSCor e Forma:SolidPeso molecular:349.31Antipsychotic agent-2
<p>Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.</p>Fórmula:C22H26FN5OCor e Forma:SolidPeso molecular:395.47Withasomniferolide B
CAS:<p>Withasomniferolide B, a withanolide from Withania somnifera root, activates GABAA receptors.</p>Fórmula:C28H36O4Cor e Forma:SolidPeso molecular:436.58(R,R)-Palonosetron Hydrochloride
CAS:<p>(R,R)-Palonosetron Hydrochloride is the active enantiomer of Palonosetron</p>Fórmula:C19H25ClN2OPureza:98%Cor e Forma:SolidPeso molecular:332.87β-Amyloid (4-10)
CAS:<p>Antibodies corresponding to beta-amyloid (4-10) are effective in vivo inhibitors of cytotoxicity, amyloid plaque formation and special memory disturbances in</p>Fórmula:C39H52N12O12Pureza:98%Cor e Forma:SolidPeso molecular:880.9hAChE/hBuChE-IN-1
<p>hAChE/hBuChE-IN-1 (compound C2) acts as a dual inhibitor of cholinesterases, exhibiting IC50 values of 514 nM for hAChE and 358 nM for hBuChE. It is orally active and capable of enhancing cognitive function and spatial memory.</p>Fórmula:C30H31FN2O3Cor e Forma:SolidPeso molecular:486.577nAChR agonist 2
CAS:<p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>Fórmula:C11H16N2Cor e Forma:SolidPeso molecular:176.263Dehydro Aripiprazole (hydrochloride)
CAS:<p>Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.</p>Fórmula:C23H26Cl3N3O2Cor e Forma:SolidPeso molecular:482.83Aloveroside A
CAS:<p>Aloveroside A, a triglucosylnaphthalene derivative extracted from Aloe vera using ethanol, exhibits modest inhibitory activity against bACE, demonstrating</p>Fórmula:C30H40O17Cor e Forma:SolidPeso molecular:672.63SQ-3
<p>SQ-3, a quinoline analogue, prefers α-syn (Ki=39.3nM) to Aβ (Ki=230nM), and [18F]SQ3 is a lead for α-syn probes. [1]</p>Fórmula:C21H21FN2OCor e Forma:SolidPeso molecular:336.4Naratriptan D3 Hydrochloride
CAS:<p>Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.</p>Fórmula:C17H26ClN3O2SPureza:98%Cor e Forma:SolidPeso molecular:374.94δ-secretase inhibitor 11
CAS:<p>δ-secretase inhibitor 11 is an inhibitor of δ-secretase and can be used as a lead compound for translational development of AD treatment.</p>Fórmula:C10H12N4O2Pureza:99.84%Cor e Forma:SolidPeso molecular:220.23(±)-Acetylcarnitine chloride
CAS:<p>(±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can be used in studies of neuritis.</p>Fórmula:C9H18ClNO4Pureza:99.98%Cor e Forma:White Crystalline PowderPeso molecular:239.7Orexin B, rat, mouse
CAS:<p>Orexin B, rat, mouse is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.</p>Fórmula:C126H215N45O34SPureza:98%Cor e Forma:SolidPeso molecular:2936.45BuChE-IN-13
<p>BuChE-IN-13 (compound 3) is a BuChE inhibitor that exhibits anti-Alzheimers activity. It is utilized in the research of neurodegenerative diseases.</p>Cor e Forma:Odour SolidDexetimide
CAS:<p>Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.</p>Fórmula:C23H26N2O2Cor e Forma:SolidPeso molecular:362.46Ladostigil hemitartrate
CAS:<p>Ladostigil hemitartrate (TV-3326) inhibits cholinesterase & MAO-B, has neuroprotective traits, and is used in depression & Alzheimer's research.</p>Fórmula:C20H26N2O8Cor e Forma:SolidPeso molecular:422.434VU0364770 hydrochloride
CAS:<p>VU0364770 hydrochloride: potent, selective mGlu4 PAM; EC50=290 nM (rat), 1.1 μM (human).</p>Fórmula:C12H10Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:269.13SL 327
CAS:Fórmula:C16H12F3N3SPureza:>97.0%(HPLC)Cor e Forma:White to Light yellow powder to crystalPeso molecular:335.35Sumatriptan
CAS:<p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>Fórmula:C14H21N3O2SPureza:99.93%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:295.4SSR180711 hydrochloride
CAS:<p>SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.</p>Fórmula:C14H18BrClN2O2Pureza:99.22%Cor e Forma:SolidPeso molecular:361.66Mofegiline hydrochloride
CAS:<p>Mofegiline hydrochloride is a potent and selective enzyme-activated irreversible MAO-B inhibitor.</p>Fórmula:C11H14ClF2NPureza:98%Cor e Forma:SolidPeso molecular:233.69Altanserin
CAS:<p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>Fórmula:C22H22FN3O2SCor e Forma:SolidPeso molecular:411.49Isoprocarb
CAS:<p>Isoprocarb is a metabolite of the pesticide.</p>Fórmula:C11H15NO2Cor e Forma:SolidPeso molecular:193.24K 02288
CAS:Fórmula:C20H20N2O4Pureza:>98.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:352.39Anti-APP Antibody (8U619)
<p>Anti-APP Antibody (8U619) is an antibody targeting APP. Anti-APP Antibody (8U619) can be used in ELISA, WB, IF.</p>Cor e Forma:Odour LiquidL-655708
CAS:<p>L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.</p>Fórmula:C18H19N3O4Pureza:98.41%Cor e Forma:PowderPeso molecular:341.36Fluvoxamine
CAS:<p>Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.</p>Fórmula:C15H21F3N2O2Cor e Forma:SolidPeso molecular:318.33Trihexyphenidyl Hydrochloride
CAS:Fórmula:C20H31NO·HClPureza:>98.0%(T)(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:337.93Cisatracurium Besylate
CAS:Fórmula:C65H82N2O18S2Pureza:>98.0%(HPLC)(qNMR)Cor e Forma:White to Light yellow powder to crystalPeso molecular:1,243.49Anti-APP Antibody (3L659)
<p>Anti-APP Antibody (3L659) is a Mouse antibody targeting APP. Anti-APP Antibody (3L659) can be used in ELISA, WB, IHC, IF.</p>Pureza:>95%Cor e Forma:Odour LiquidAnti-APP Antibody (5W753)
<p>Anti-APP Antibody (5W753) is an antibody targeting APP. Anti-APP Antibody (5W753) can be used in ELISA, IF, FCM.</p>Cor e Forma:Odour LiquidSaracatinib
CAS:Fórmula:C27H32ClN5O5Pureza:>95.0%(HPLC)(qNMR)Cor e Forma:White to Light yellow to Light orange powder to crystalPeso molecular:542.03


