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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5389 produtos de "Neurociência"

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  • FK 3311

    CAS:
    <p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>
    Fórmula:C15H13F2NO4S
    Pureza:97.98%
    Cor e Forma:Solid
    Peso molecular:341.33
  • Ondansetron hydrochloride

    CAS:
    <p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>
    Fórmula:C18H19N3O·HCl
    Pureza:99.78%
    Cor e Forma:White Powder
    Peso molecular:329.82
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Fórmula:C22H26ClNO2
    Pureza:98.02%
    Cor e Forma:Solid
    Peso molecular:371.9
  • Revefenacin

    CAS:
    <p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>
    Fórmula:C35H43N5O4
    Pureza:98.12%
    Cor e Forma:Solid
    Peso molecular:597.75
  • TAT-GluA2 3Y acetate(1404188-93-7 free base)


    <p>TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis.Systemic administration of Tat-GluA2(3Y) during the induction phase of d-amphetamine blocked</p>
    Fórmula:C115H185N43O29
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:2634.02
  • Ziprasidone mesylate

    CAS:
    <p>Ziprasidone mesylate (CP-88059), an oral 5-HT &amp; dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>
    Fórmula:C22H25ClN4O4S2
    Cor e Forma:Solid
    Peso molecular:509.04
  • Trihexyphenidyl hydrochloride

    CAS:
    <p>Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.</p>
    Fórmula:C20H32ClNO
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:337.927
  • Acamprosate calcium

    CAS:
    Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
    Fórmula:C10H20CaN2O8S2
    Pureza:98% - 99.93%
    Cor e Forma:White Odorless Or Nearly Odorless Powder
    Peso molecular:400.48
  • CALP1 acetate


    <p>CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.</p>
    Fórmula:C42H79N9O12
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:902.13
  • NMDAR antagonist 1

    CAS:
    <p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>
    Fórmula:C20H20BrN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:414.3
  • Omberacetam

    CAS:
    <p>Omberacetam (Noopept), a synthetic dipeptide, enhances cognition similarly to racetams.</p>
    Fórmula:C17H22N2O4
    Pureza:≥95%
    Cor e Forma:White Powder
    Peso molecular:318.37
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Fórmula:C19H26ClNOS
    Pureza:99.53% - 99.56%
    Cor e Forma:Almost White To White Crystalline Powder
    Peso molecular:351.93
  • Hemicholinium 3

    CAS:
    <p>Hemicholinium 3 is a potent and selective choline uptake blocker.</p>
    Fórmula:C24H34Br2N2O4
    Pureza:98% - 99.95%
    Cor e Forma:Solid
    Peso molecular:574.35
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Cor e Forma:Solid
    Peso molecular:386.37
  • Pempidine

    CAS:
    <p>Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.</p>
    Fórmula:C10H21N
    Pureza:98.18% - 99.28%
    Cor e Forma:Colorless - Light Yellow Clear Liquid
    Peso molecular:155.28
  • ADX88178

    CAS:
    <p>ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 of 4 nM for human mGluR4.</p>
    Fórmula:C12H12N6S
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:272.33
  • VU10010

    CAS:
    <p>VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.</p>
    Fórmula:C17H16ClN3OS
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:345.85
  • RU 24969 free base

    CAS:
    <p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>
    Fórmula:C14H16N2O
    Pureza:97.38%
    Cor e Forma:Solid
    Peso molecular:228.29
  • ZL006

    CAS:
    <p>ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.</p>
    Fórmula:C14H11Cl2NO4
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:328.15
  • Cinitapride

    CAS:
    <p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>
    Fórmula:C21H30N4O4
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:402.49
  • Sepimostat

    CAS:
    <p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>
    Fórmula:C21H19N5O2
    Pureza:97.75%
    Cor e Forma:Solid
    Peso molecular:373.41
  • SEN12333

    CAS:
    <p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>
    Fórmula:C20H25N3O2
    Pureza:99.02%
    Cor e Forma:Solid
    Peso molecular:339.43
  • Nor-benzetimide

    CAS:
    <p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>
    Fórmula:C16H20N2O2
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:272.34
  • 7-Amino-4-(trifluoromethyl)coumarin

    CAS:
    7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.
    Fórmula:C10H6F3NO2
    Pureza:97.31% - 97.84%
    Cor e Forma:Yellow Powder
    Peso molecular:229.16
  • α-Conotoxin PIA acetate


    α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.
    Pureza:98%
    Cor e Forma:Liquid
    Peso molecular:N/A
  • VU0119498

    CAS:
    <p>VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.</p>
    Fórmula:C15H10BrNO2
    Pureza:97.56%
    Cor e Forma:Solid
    Peso molecular:316.15
  • Acamprosate

    CAS:
    <p>Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust</p>
    Fórmula:C5H11NO4S
    Pureza:98.30%
    Cor e Forma:Solid
    Peso molecular:181.21
  • ML380

    CAS:
    <p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>
    Fórmula:C23H25F3N4O3S
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:494.53
  • Risperidone hydrochloride

    CAS:
    <p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>
    Fórmula:C23H28ClFN4O2
    Cor e Forma:Solid
    Peso molecular:446.95
  • PNU-282987

    CAS:
    <p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>
    Fórmula:C14H18Cl2N2O
    Pureza:99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:301.21
  • PFE-360

    CAS:
    <p>PFE-360 (PF-06685360) is a potent and selective inhibitor of LRRK2 kinase (IC50: 2.3 nM in vivo).</p>
    Fórmula:C16H16N6O
    Pureza:98.14% - 99.73%
    Cor e Forma:Solid
    Peso molecular:308.34
  • Isopropamide Iodide

    CAS:
    <p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>
    Fórmula:C23H33IN2O
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:480.43
  • Semagacestat

    CAS:
    <p>Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).</p>
    Fórmula:C19H27N3O4
    Pureza:97.1% - 99.9%
    Cor e Forma:Solid
    Peso molecular:361.44
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Fórmula:C6H6N2O2
    Pureza:99.94%
    Cor e Forma:Soild
    Peso molecular:138.1238
  • VU0155041

    CAS:
    <p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>
    Fórmula:C14H15Cl2NO3
    Pureza:99.52% - 99.56%
    Cor e Forma:Solid
    Peso molecular:316.18
  • Losartan Carboxaldehyde

    CAS:
    <p>Losartan Carboxaldehyde is an endothelial cyclooxygenase (COX)-2 inhibitor.</p>
    Fórmula:C22H21ClN6O
    Pureza:99.1%
    Cor e Forma:Solid
    Peso molecular:420.89
  • BRL 54443

    CAS:
    <p>BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).</p>
    Fórmula:C14H18N2O
    Pureza:98.07%
    Cor e Forma:Solid
    Peso molecular:230.31
  • AZ 11645373

    CAS:
    <p>AZ 11645373 (3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE) is a highly selective and potent human P2X7 receptor</p>
    Fórmula:C24H21N3O5S
    Pureza:99.47%
    Cor e Forma:Solid
    Peso molecular:463.51
  • Hypidone hydrochloride

    CAS:
    <p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>
    Fórmula:C18H23ClN2O2
    Pureza:99.82% - 99.93%
    Cor e Forma:Solid
    Peso molecular:334.84
  • Myristicin

    CAS:
    <p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>
    Fórmula:C11H12O3
    Pureza:99.828%
    Cor e Forma:Liquid
    Peso molecular:192.21
  • Pikamilone

    CAS:
    Pikamilone (Picamilon) is an intelligent medicine.
    Fórmula:C10H12N2O3
    Pureza:99.38%
    Cor e Forma:White Crystalline Powder
    Peso molecular:208.21
  • SB 242084 dihydrochloride

    CAS:
    SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.
    Fórmula:C21H21Cl3N4O2
    Cor e Forma:Solid
    Peso molecular:467.78
  • MK 212 hydrochloride

    CAS:
    <p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>
    Fórmula:C8H11ClN4·HCl
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:235.12
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Fórmula:C14H17ClN2
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:248.75
  • Lu AF21934

    CAS:
    <p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>
    Fórmula:C14H16Cl2N2O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:315.2
  • Orexin 2 Receptor Agonist

    CAS:
    Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.
    Fórmula:C32H34N4O5S
    Pureza:98.26% - 99.43%
    Cor e Forma:Solid
    Peso molecular:586.7
  • Naluzotan

    CAS:
    <p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>
    Fórmula:C23H38N4O3S
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:450.64
  • S 14506 HCl

    CAS:
    <p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), &lt;6.0 (5-HT3).</p>
    Fórmula:C24H26FN3O2
    Cor e Forma:Solid
    Peso molecular:407.48
  • FLI-06

    CAS:
    FLI-06 is a Notch signaling inhibitor (EC50: 2.3 μM).
    Fórmula:C25H30N2O5
    Pureza:99.81% - ≥98%
    Cor e Forma:Solid
    Peso molecular:438.52
  • Acephate

    CAS:
    <p>Acephate (Orthene) is an anticholinesterase insecticide with a weak inhibitory effect on AChE in rats, but it can effectively inhibit AChE in cockroaches.</p>
    Fórmula:C4H10NO3PS
    Pureza:≥98%
    Cor e Forma:Colorless Crystals Acephate Is A White Solid Used As A Contact And Systemic Insecticide
    Peso molecular:183.17