
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(942 produtos)
- ACK(1 produtos)
- AChR(576 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.949 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(565 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor GABA(337 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(359 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(26 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5389 produtos de "Neurociência"
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FK 3311
CAS:<p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>Fórmula:C15H13F2NO4SPureza:97.98%Cor e Forma:SolidPeso molecular:341.33Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Fórmula:C18H19N3O·HClPureza:99.78%Cor e Forma:White PowderPeso molecular:329.82SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Fórmula:C22H26ClNO2Pureza:98.02%Cor e Forma:SolidPeso molecular:371.9Revefenacin
CAS:<p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>Fórmula:C35H43N5O4Pureza:98.12%Cor e Forma:SolidPeso molecular:597.75TAT-GluA2 3Y acetate(1404188-93-7 free base)
<p>TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis.Systemic administration of Tat-GluA2(3Y) during the induction phase of d-amphetamine blocked</p>Fórmula:C115H185N43O29Pureza:99.43%Cor e Forma:SolidPeso molecular:2634.02Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Fórmula:C22H25ClN4O4S2Cor e Forma:SolidPeso molecular:509.04Trihexyphenidyl hydrochloride
CAS:<p>Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.</p>Fórmula:C20H32ClNOPureza:99.65%Cor e Forma:SolidPeso molecular:337.927Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Fórmula:C10H20CaN2O8S2Pureza:98% - 99.93%Cor e Forma:White Odorless Or Nearly Odorless PowderPeso molecular:400.48CALP1 acetate
<p>CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.</p>Fórmula:C42H79N9O12Pureza:99.63%Cor e Forma:SolidPeso molecular:902.13NMDAR antagonist 1
CAS:<p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>Fórmula:C20H20BrN3O2Pureza:98%Cor e Forma:SolidPeso molecular:414.3Omberacetam
CAS:<p>Omberacetam (Noopept), a synthetic dipeptide, enhances cognition similarly to racetams.</p>Fórmula:C17H22N2O4Pureza:≥95%Cor e Forma:White PowderPeso molecular:318.37Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Cor e Forma:Almost White To White Crystalline PowderPeso molecular:351.93Hemicholinium 3
CAS:<p>Hemicholinium 3 is a potent and selective choline uptake blocker.</p>Fórmula:C24H34Br2N2O4Pureza:98% - 99.95%Cor e Forma:SolidPeso molecular:574.35Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Cor e Forma:SolidPeso molecular:386.37Pempidine
CAS:<p>Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.</p>Fórmula:C10H21NPureza:98.18% - 99.28%Cor e Forma:Colorless - Light Yellow Clear LiquidPeso molecular:155.28ADX88178
CAS:<p>ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 of 4 nM for human mGluR4.</p>Fórmula:C12H12N6SPureza:99.55%Cor e Forma:SolidPeso molecular:272.33VU10010
CAS:<p>VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.</p>Fórmula:C17H16ClN3OSPureza:99.36%Cor e Forma:SolidPeso molecular:345.85RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Fórmula:C14H16N2OPureza:97.38%Cor e Forma:SolidPeso molecular:228.29ZL006
CAS:<p>ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.</p>Fórmula:C14H11Cl2NO4Pureza:98.29%Cor e Forma:SolidPeso molecular:328.15Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Fórmula:C21H30N4O4Pureza:99.52%Cor e Forma:SolidPeso molecular:402.49Sepimostat
CAS:<p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>Fórmula:C21H19N5O2Pureza:97.75%Cor e Forma:SolidPeso molecular:373.41SEN12333
CAS:<p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>Fórmula:C20H25N3O2Pureza:99.02%Cor e Forma:SolidPeso molecular:339.43Nor-benzetimide
CAS:<p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>Fórmula:C16H20N2O2Pureza:98.63%Cor e Forma:SolidPeso molecular:272.347-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Cor e Forma:Yellow PowderPeso molecular:229.16α-Conotoxin PIA acetate
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.Pureza:98%Cor e Forma:LiquidPeso molecular:N/AVU0119498
CAS:<p>VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.</p>Fórmula:C15H10BrNO2Pureza:97.56%Cor e Forma:SolidPeso molecular:316.15Acamprosate
CAS:<p>Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust</p>Fórmula:C5H11NO4SPureza:98.30%Cor e Forma:SolidPeso molecular:181.21ML380
CAS:<p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>Fórmula:C23H25F3N4O3SPureza:99.69%Cor e Forma:SolidPeso molecular:494.53Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Cor e Forma:SolidPeso molecular:446.95PNU-282987
CAS:<p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>Fórmula:C14H18Cl2N2OPureza:99% - >99.99%Cor e Forma:SolidPeso molecular:301.21PFE-360
CAS:<p>PFE-360 (PF-06685360) is a potent and selective inhibitor of LRRK2 kinase (IC50: 2.3 nM in vivo).</p>Fórmula:C16H16N6OPureza:98.14% - 99.73%Cor e Forma:SolidPeso molecular:308.34Isopropamide Iodide
CAS:<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Fórmula:C23H33IN2OPureza:99.67%Cor e Forma:SolidPeso molecular:480.43Semagacestat
CAS:<p>Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).</p>Fórmula:C19H27N3O4Pureza:97.1% - 99.9%Cor e Forma:SolidPeso molecular:361.446-Aminonicotinic acid
CAS:<p>6-Aminonicotinic acid is a natural product.</p>Fórmula:C6H6N2O2Pureza:99.94%Cor e Forma:SoildPeso molecular:138.1238VU0155041
CAS:<p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>Fórmula:C14H15Cl2NO3Pureza:99.52% - 99.56%Cor e Forma:SolidPeso molecular:316.18Losartan Carboxaldehyde
CAS:<p>Losartan Carboxaldehyde is an endothelial cyclooxygenase (COX)-2 inhibitor.</p>Fórmula:C22H21ClN6OPureza:99.1%Cor e Forma:SolidPeso molecular:420.89BRL 54443
CAS:<p>BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).</p>Fórmula:C14H18N2OPureza:98.07%Cor e Forma:SolidPeso molecular:230.31AZ 11645373
CAS:<p>AZ 11645373 (3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE) is a highly selective and potent human P2X7 receptor</p>Fórmula:C24H21N3O5SPureza:99.47%Cor e Forma:SolidPeso molecular:463.51Hypidone hydrochloride
CAS:<p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>Fórmula:C18H23ClN2O2Pureza:99.82% - 99.93%Cor e Forma:SolidPeso molecular:334.84Myristicin
CAS:<p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>Fórmula:C11H12O3Pureza:99.828%Cor e Forma:LiquidPeso molecular:192.21Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Fórmula:C10H12N2O3Pureza:99.38%Cor e Forma:White Crystalline PowderPeso molecular:208.21SB 242084 dihydrochloride
CAS:SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Fórmula:C21H21Cl3N4O2Cor e Forma:SolidPeso molecular:467.78MK 212 hydrochloride
CAS:<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Fórmula:C8H11ClN4·HClPureza:99.88%Cor e Forma:SolidPeso molecular:235.121-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Fórmula:C14H17ClN2Pureza:98.27%Cor e Forma:SolidPeso molecular:248.75Lu AF21934
CAS:<p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>Fórmula:C14H16Cl2N2O2Pureza:99.79%Cor e Forma:SolidPeso molecular:315.2Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Fórmula:C32H34N4O5SPureza:98.26% - 99.43%Cor e Forma:SolidPeso molecular:586.7Naluzotan
CAS:<p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>Fórmula:C23H38N4O3SPureza:>99.99%Cor e Forma:SolidPeso molecular:450.64S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Fórmula:C24H26FN3O2Cor e Forma:SolidPeso molecular:407.48FLI-06
CAS:FLI-06 is a Notch signaling inhibitor (EC50: 2.3 μM).Fórmula:C25H30N2O5Pureza:99.81% - ≥98%Cor e Forma:SolidPeso molecular:438.52Acephate
CAS:<p>Acephate (Orthene) is an anticholinesterase insecticide with a weak inhibitory effect on AChE in rats, but it can effectively inhibit AChE in cockroaches.</p>Fórmula:C4H10NO3PSPureza:≥98%Cor e Forma:Colorless Crystals Acephate Is A White Solid Used As A Contact And Systemic InsecticidePeso molecular:183.17
