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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5516 produtos de "Neurociência"

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  • Legumain inhibitor 1

    CAS:
    Legumain inhibitor 1 is a highly potent and specific Legumain inhibitor with potential anticancer activity for cancer research.
    Fórmula:C23H25N5O4S
    Pureza:98.14%
    Cor e Forma:Solid
    Peso molecular:467.54
  • Furosemide-d5

    CAS:
    Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.
    Fórmula:C12H11ClN2O5S
    Cor e Forma:Solid
    Peso molecular:335.78
  • SU 5416

    CAS:
    Fórmula:C15H14N2O
    Pureza:>98.0%(T)(HPLC)
    Cor e Forma:White to Yellow to Orange powder to crystal
    Peso molecular:238.29

    Ref: 3B-E1494

    100mg
    227,00€
  • SB 202190

    CAS:
    Fórmula:C20H14FN3O
    Pureza:>95.0%(HPLC)
    Cor e Forma:White to Light yellow to Light orange powder to crystal
    Peso molecular:331.35

    Ref: 3B-F0870

    5mg
    264,00€
  • Quetiapine-d8 Hemifumarate

    CAS:
    Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
    Fórmula:C25H21D8N3O6S
    Cor e Forma:Solid
    Peso molecular:507.63
  • Anti-NGF Antibody (6U823)


    Anti-NGF Antibody (6U823) is an antibody targeting NGF. Anti-NGF Antibody (6U823) can be used in ELISA, FCM.
    Cor e Forma:Odour Liquid
  • Colivelin

    CAS:
    <p>Colivelin is a neuroprotective peptide and activator of STAT3. Colivelin is a hybrid peptide synthesized to enhance the neuroprotective effects of humanin (HN).</p>
    Fórmula:C119H206N32O35
    Pureza:96.56%
    Cor e Forma:Solid
    Peso molecular:2645.1
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Fórmula:C11H11N3O
    Pureza:99.03%
    Cor e Forma:Solid
    Peso molecular:201.22
  • Ursulcholic acid

    CAS:
    Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
    Fórmula:C24H40O10S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:552.7
  • DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Fórmula:C19H23Cl2N3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:364.31
  • Ro0711401

    CAS:
    <p>Ro0711401 is an agonist of mGlu1 receptor.</p>
    Fórmula:C18H11F3N2O3
    Pureza:97.57%
    Cor e Forma:Solid
    Peso molecular:360.29
  • 6-Methylflavone

    CAS:
    6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
    Fórmula:C16H12O2
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:236.27
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Fórmula:C17H16FN3
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:281.33
  • Pardoprunox hydrochloride

    CAS:
    Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)
    Fórmula:C12H16ClN3O2
    Pureza:98.95% - 99.13%
    Cor e Forma:Solid
    Peso molecular:269.73
  • mAChR-IN-1 hydrochloride

    CAS:
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.
    Fórmula:C23H26ClIN2O2
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:524.82
  • Autocamtide-2-related inhibitory peptide

    CAS:
    <p>Autocamtide-2-related inhibitory peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>
    Fórmula:C64H116N22O19
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1497.74
  • VU 0364439

    CAS:
    VU 0364439 is a mGlu4 positive allosteric modulator (C50: 19.8 nM).
    Fórmula:C18H13Cl2N3O3S
    Pureza:97.9%
    Cor e Forma:Solid
    Peso molecular:422.29
  • Propyphenazone

    CAS:
    <p>Propyphenazone: an anti-inflammatory, analgesic, antipyretic pyrazolone; prodrug; COX-2 inhibitor.</p>
    Fórmula:C14H18N2O
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:230.31
  • FK 3311

    CAS:
    <p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>
    Fórmula:C15H13F2NO4S
    Pureza:97.98%
    Cor e Forma:Solid
    Peso molecular:341.33
  • Ondansetron hydrochloride

    CAS:
    <p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>
    Fórmula:C18H19N3O·HCl
    Pureza:99.78%
    Cor e Forma:White Powder
    Peso molecular:329.82
  • CALP1 acetate


    <p>CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.</p>
    Fórmula:C42H79N9O12
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:902.13
  • pep2-EVKI acetate(1315378-67-6 free base)


    Pep2-EVKI acetate, a cell-permeable peptide, disrupts PICK1-GluR2 AMPA receptor binding.
    Fórmula:C64H99N13O21
    Pureza:97.63%
    Cor e Forma:Solid
    Peso molecular:1386.55
  • ML 10302

    CAS:
    ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.
    Fórmula:C15H21ClN2O3
    Cor e Forma:Solid
    Peso molecular:312.79
  • Teriflunomide impurity 3

    CAS:
    <p>Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) is a selective COX-1 inhibitor(IC50 of 30 μM).</p>
    Fórmula:C14H11F3N2O
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:280.25
  • Quipazine maleate

    CAS:
    Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.
    Fórmula:C17H19N3O4
    Cor e Forma:Solid
    Peso molecular:329.356
  • CL 218872

    CAS:
    CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.
    Fórmula:C13H9F3N4
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:278.23
  • BRL-15572 dihydrochloride

    CAS:
    BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.
    Fórmula:C25H27ClN2O·2HCl
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:479.87
  • Tiprenolol

    CAS:
    Tiprenolol is a beta adrenergic receptor antagonist.[1]
    Fórmula:C13H21NO2S
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:255.38
  • PHA 543613 hydrochloride

    CAS:
    PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.
    Fórmula:C15H18ClN3O2
    Cor e Forma:Solid
    Peso molecular:307.78
  • Quipazine

    CAS:
    <p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>
    Fórmula:C13H15N3
    Cor e Forma:Solid
    Peso molecular:213.28
  • Eltoprazine dihydrochloride

    CAS:
    <p>Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.</p>
    Fórmula:C12H18Cl2N2O2
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:293.19
  • 6-fluoro-DL-Tryptophan

    CAS:
    <p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>
    Fórmula:C11H11FN2O2
    Pureza:99.25%
    Cor e Forma:Off-White Powder
    Peso molecular:222.22
  • LOX-IN-3 dihydrochloride monohydrate

    CAS:
    LOX-IN-3 dihydrochloride monohydrate is an oral lysyl oxidase inhibitor for research in fibrosis, cancer, and angiogenesis.
    Fórmula:C13H17Cl2FN2O3S
    Cor e Forma:Solid
    Peso molecular:371.25
  • ARC-239

    CAS:
    <p>ARC-239 is an agonist of α2-adrenergic receptor.</p>
    Fórmula:C24H29N3O3
    Cor e Forma:Solid
    Peso molecular:407.51
  • LP-922761 hydrate


    LP-922761 hydrate: selective AAK1 inhibitor; IC50: 4.8 nM (enzyme), 7.6 nM (cellular); also inhibits BIKE (IC50: 24 nM); inert to GAK, opioids, α2, GABAa.
    Fórmula:C21H28N6O4
    Cor e Forma:Solid
    Peso molecular:414.98
  • Milnacipran

    CAS:
    <p>Milnacipran, an SNRI with 85% bioavailability, treats fibromyalgia and is well absorbed orally.</p>
    Fórmula:C15H22N2O
    Cor e Forma:Solid
    Peso molecular:246.35
  • (S)-Amisulpride

    CAS:
    (S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.
    Fórmula:C17H27N3O4S
    Pureza:98.38%
    Cor e Forma:Solid
    Peso molecular:369.48
  • TCN238

    CAS:
    <p>TCN238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 (mGluR4with an EC50 of 1 μM).</p>
    Fórmula:C12H11N3
    Pureza:99.9% - 99.92%
    Cor e Forma:Solid
    Peso molecular:197.24
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Cor e Forma:Solid
    Peso molecular:386.37
  • Alosetron (Hydrochloride(1:X))

    CAS:
    <p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>
    Fórmula:C17H18ClN4O
    Cor e Forma:Solid
    Peso molecular:329.11691
  • S 14506 HCl

    CAS:
    S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).
    Fórmula:C24H26FN3O2
    Cor e Forma:Solid
    Peso molecular:407.48
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Fórmula:C17H25N3O2S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:335.47
  • Arecaidine hydrochloride

    CAS:
    Arecaidine hydrochloride may have carcinogenesis.
    Fórmula:C7H12ClNO2
    Pureza:99.69% - ≥95%
    Cor e Forma:Solid
    Peso molecular:177.63
  • CNQX

    CAS:
    <p>CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C9H4N4O4
    Pureza:99.70%
    Cor e Forma:Pale Yellow Solid
    Peso molecular:232.15
  • (R)-baclofen

    CAS:
    <p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>
    Fórmula:C10H12ClNO2
    Pureza:97.20% - 98.94%
    Cor e Forma:Solid
    Peso molecular:213.66
  • SC-560

    CAS:
    <p>SC-560 is a member of the diaryl heterocycle class of cyclooxygenase (COX) inhibitors.</p>
    Fórmula:C17H12ClF3N2O
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:352.74
  • WAY-100635 Monomaleate

    CAS:
    WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Cor e Forma:Solid
    Peso molecular:538.64
  • Ocinaplon

    CAS:
    <p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>
    Fórmula:C17H11N5O
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:301.3
  • Ro 67-7476

    CAS:
    Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors.
    Fórmula:C17H18FNO2S
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:319.39
  • Epinastine hydrochloride

    CAS:
    Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
    Fórmula:C16H15N3·HCl
    Pureza:99.26% - 99.62%
    Cor e Forma:White Solid
    Peso molecular:285.77