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Cell Cycle/Checkpoint

Cell Cycle/Checkpoint

Cell cycle/checkpoint inhibitors are compounds that disrupt the normal progression of the cell cycle, particularly at key regulatory checkpoints. These inhibitors are crucial for studying cell division, understanding cancer cell proliferation, and developing anti-cancer therapies. By targeting specific phases of the cell cycle, these inhibitors can induce cell cycle arrest, leading to apoptosis or senescence in rapidly dividing cells. At CymitQuimica, we offer a diverse range of high-quality cell cycle/checkpoint inhibitors to support your research in cancer biology, cell biology, and drug development.

Subcategories of "Cell Cycle/Checkpoint"

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Found 3485 products of "Cell Cycle/Checkpoint"

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  • XL-188

    CAS:
    <p>XL-188: Potent, selective USP7 inhibitor, IC50 = 193 nM (domain), 90 nM (full). Boosts p53, p21; degrades HDM2. Unique among DUB inhibitors.</p>
    Formula:C32H42N6O4
    Color and Shape:Solid
    Molecular weight:574.71
  • FRα-IN-1

    CAS:
    <p>FRα-IN-1 (Compound 4) is a tumour targeting agent. FRα-IN-1 exhibits selective anti-cancer effects on FRα and FRβ expressing cells.</p>
    Formula:C21H24N6O6
    Color and Shape:Solid
    Molecular weight:456.45
  • Nucleoside-Analog-1

    CAS:
    <p>Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.</p>
    Formula:C9H9N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.2
  • L-Fd4A

    CAS:
    <p>L-Fd4A (compound 36) is an adenine derivative with anti-HIV (EC50=1.5μM) and anti-HBV (EC50=1.7μM) effects, low cytotoxicity.</p>
    Formula:C10H10FN5O2
    Color and Shape:Solid
    Molecular weight:251.22
  • CLK1-IN-2


    <p>CLK1-IN-2: Metabolically stable, Clk1-selective inhibitor; IC50=1.7nM; useful in tumor, Duchenne MD, HIV-1, influenza research.</p>
    Formula:C16H12Cl2N2O2S
    Color and Shape:Solid
    Molecular weight:367.25
  • TDRL-X80

    CAS:
    <p>TDRL-X80 inhibits XPA DNA binding; effective on single, double, and cisplatin-damaged DNA; IC50: 18-29 μM (FP), 21-39 μM (ELISA).</p>
    Formula:C23H15ClN2O6
    Color and Shape:Solid
    Molecular weight:450.83
  • Metioprim

    CAS:
    <p>Metioprim is a competitive bacterial dihydrofolate reductases inhibitor.</p>
    Formula:C14H18N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:306.38
  • CCT068127

    CAS:
    <p>CCT068127 is a potent CDK2 and CDK9 inhibitor.</p>
    Formula:C19H27N7O
    Color and Shape:Solid
    Molecular weight:369.46
  • L-Cytidine

    CAS:
    <p>L-Cytidine, pyrimidine nucleoside in RNA, regulates glial glutamate, brain lipids, catecholamines, and mitochondria.</p>
    Formula:C9H13N3O5
    Color and Shape:Solid
    Molecular weight:243.22
  • hDHODH-IN-5

    CAS:
    <p>hDHODH-IN-5 is an inhibitor of human dihydroorotate dehydrogenase (hDHODH, IC50 = 0.91 μM).</p>
    Formula:C21H21F3N2O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:390.4
  • DHODH-IN-13

    CAS:
    <p>DHODH-IN-13 is an inhibitor of DHODH with IC50 of 4.3 μM for rat liver. DHODH-IN-13 can be used in studies about rheumatoid arthritis.</p>
    Formula:C10H6F3N3O3
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:273.17
  • (S)-CR8

    CAS:
    <p>(S)-CR8 is an effective second-generation cyclin-dependent kinase inhibitor.</p>
    Formula:C24H29N7O
    Color and Shape:Solid
    Molecular weight:431.53
  • Eg5 Inhibitor V, trans-24

    CAS:
    <p>Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.</p>
    Formula:C26H21N3O3
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:423.46
  • BPKDi

    CAS:
    <p>BPKDi is a potent and selective inhibitor of PKD (protein kinase D).</p>
    Formula:C21H28N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:380.49
  • hDHODH-IN-3

    CAS:
    <p>hDHODH-IN-3 is an inhibitor of human dihydroorotate dehydrogenase with a pMIC50 value of 8.6. hDHODH-IN-3 can inhibit measles virus replication.</p>
    Formula:C18H19BrN4O2
    Purity:99.871%
    Color and Shape:Solid
    Molecular weight:403.27
  • BMVC

    CAS:
    <p>BMVC is a potent G-quadruplex (G4) stabilizer and a selective telomerase inhibitor (IC50: ~0.2 μM) with anticancer activities.</p>
    Formula:C28H25I2N3
    Color and Shape:Solid
    Molecular weight:657.33
  • Aloisine A

    CAS:
    <p>Aloisine A, a CDK/GSK-3 inhibitor with IC50: Cdk1/B-150nM, Cdk2/A-120nM, Cdk2/E-400nM, Cdk5/25-200nM, Cdk5/35-160nM, GSK-3α-500nM, GSK-3β-650nM, JNK-3-10μM.</p>
    Formula:C16H17N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.33
  • CDK2-IN-11

    CAS:
    <p>CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.</p>
    Formula:C18H14ClN7O2S
    Color and Shape:Solid
    Molecular weight:427.87
  • TP1287

    CAS:
    <p>TP-1287 is an oral phosphate prodrug of the CDK9 inhibitor, alvocidib.</p>
    Formula:C21H21ClNO8P
    Color and Shape:Solid
    Molecular weight:481.82
  • (S)-LY3177833 hydrate

    CAS:
    <p>(S)-LY3177833 ((S)-Example 2) hydrate, an orally active CDC7 kinase inhibitor, exhibits extensive in vitro anticancer efficacy.</p>
    Formula:C16H14FN5O2
    Color and Shape:Solid
    Molecular weight:327.31
  • Bofumustine

    CAS:
    <p>Bofumustine is a chloroethyl nitrosourea with anti tumor properties.</p>
    Formula:C18H21ClN4O9
    Color and Shape:Solid
    Molecular weight:472.83
  • AS-136A

    CAS:
    <p>AS-136A is an orally active MV RdRp inhibitor with antiviral activity that inhibits measles virus and blocks viral RNA synthesis.</p>
    Formula:C17H19F3N4O3S
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:416.42
  • Levoleucovorin disodium

    CAS:
    <p>Levoleucovorin disodium is the sodium salt of the enantiomerically active form of Folinic Acid.</p>
    Formula:C20H21N7Na2O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:517.41
  • Nitracrine

    CAS:
    <p>Nitracrine: a 1-nitroacridine, hypoxia-selective, anti-tumor agent; inhibits RNA synthesis, binds DNA reversibly and forms covalent adducts.</p>
    Formula:C18H20N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.38
  • ProTAME

    CAS:
    <p>ProTAME inhibits APC/CFzr &amp; APC/CCdc20, enhances cell death with doxorubicin/etoposide in primary/MM cells, especially after TOPIIα upregulation.</p>
    Formula:C34H38N4O12S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:726.75
  • Braco-19 trihydrochloride

    CAS:
    <p>BRACO19 3HCl inhibits telomerase, blocking its capping function, and prevents HAdV viral replication.</p>
    Formula:C35H46Cl3N7O2
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:703.14
  • DDD100097

    CAS:
    <p>DDD100097 is a N-myristoyltransferase inhibitor with potential inhibitory effects on Trypanosoma brucei, which can be used to study neurological disorders.</p>
    Formula:C22H30Cl2F2N4O2S
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:523.47
  • DHODH-IN-8

    CAS:
    <p>DHODH-IN-8 is a DHODH inhibitor with antimalarial properties, IC50: 0.13 μM (human), 47.4 μM (P. falciparum); Ki: 0.016 μM (human), 5.6 μM (P. falciparum).</p>
    Formula:C17H13ClN2O2
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:312.75
  • LY 222306

    CAS:
    <p>LY 222306 is a glycinamide ribonucleotide formyltransferase (GARFT) inhibitor with a Ki of 0.77 nM.</p>
    Formula:C19H23N5O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.42
  • CDK5 inhibitor 20-223

    CAS:
    <p>CDK5 inhibitor 20-223 is a potent CDK2/CDK5 inhibitor,anti-Colorectal Cancer (CRC), inhibiting cell migration and inducing cell cycle arrest.</p>
    Formula:C19H19N3O
    Color and Shape:Solid
    Molecular weight:305.37
  • 2-Fluoroadenine

    CAS:
    <p>2-Fluoroadenine (NSC-27364) has toxicity in nonproliferating and proliferating tumor cells. 2-Fluoroadenine can be used for anticancer studies.</p>
    Formula:C5H4FN5
    Purity:98.84% - 99.62%
    Color and Shape:White To Light Yellow Crystal Powder
    Molecular weight:153.12
  • Ipivivint

    CAS:
    <p>Ipivivint: orally active, potent CLK inhibitor; hinders CLK1, CLK2, &amp; CLK3; curbs Wnt signaling &amp; SRSF phosphorylation for cancer research.</p>
    Formula:C26H21FN8
    Color and Shape:Solid
    Molecular weight:464.5
  • OM-137

    CAS:
    <p>OM137 inhibits Aurora kinases, impedes cell growth at high doses, and enhances low-dose paclitaxel effects.</p>
    Formula:C13H14N4O3S
    Color and Shape:Solid
    Molecular weight:306.34
  • VRX-0466617

    CAS:
    <p>VRX-0466617 is a novel selective Chk2 inhibitor.</p>
    Formula:C19H20BrN5O2S
    Color and Shape:Solid
    Molecular weight:462.36
  • CDK2-IN-12

    CAS:
    <p>CDK2-IN-12 (10b), potent CDK2 inhibitor, IC50: 11.6 μM; inhibits hCA I/II/IX/XII, KI: 3534/638.4/44.3/48.8 nM; anti-cancer properties.</p>
    Formula:C20H17N9O2S
    Color and Shape:Solid
    Molecular weight:447.47
  • CDK8-IN-6

    CAS:
    <p>CDK8-IN-6 (compound 9) is a potent inhibitor of cyclin-dependent kinase 8 (CDK8) (Kd: 13 nM), CDK8-IN-6 showed potential research value in AML cancers.</p>
    Formula:C26H37ClN2
    Color and Shape:Solid
    Molecular weight:413.04
  • KH-CB19

    CAS:
    <p>KH-CB19 is an effective and highly specific inhibitor of the CDC2-like kinase isoforms 1 and 4 (CLK1/CLK4).</p>
    Formula:C15H13Cl2N3O2
    Color and Shape:Solid
    Molecular weight:338.19
  • Litronesib Racemate

    CAS:
    <p>Litronesib is a selective, allosteric inhibitor of kinesin Eg5.Litronesib (Racemate) is the racemate of litronesib.</p>
    Formula:C23H37N5O4S2
    Color and Shape:Solid
    Molecular weight:511.7
  • Dyrk1A-IN-3

    CAS:
    <p>Dyrk1A-IN-3 is a selective DYRK1A inhibitor with an IC50 of 76 nM, useful for neurodegenerative disease research.</p>
    Formula:C18H16N6
    Color and Shape:Solid
    Molecular weight:316.36
  • 3,6-DMAD dihydrochloride

    CAS:
    <p>3,6-DMAD dihydrochloride: Potent IRE1α-XBP1s inhibitor, affects IL-6 secretion and RNase activity, used in cancer research.</p>
    Formula:C22H33Cl2N5
    Color and Shape:Solid
    Molecular weight:438.44
  • Synucleozid

    CAS:
    <p>Synucleozid is a potent the SNCA mRNA inhibitor that encodes α-synuclein protein (IC50=1.5 μM), has the potential for the investigation of Parkinson’s disease.</p>
    Formula:C22H20N6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.43
  • PF-4950834

    CAS:
    <p>PF-4950834, a ATP-competitive, selective Rho kinase inhibitor, provides therapeutic benefits in chronic inflammatory diseases.</p>
    Formula:C21H19N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.39
  • GP29

    CAS:
    <p>GP29 is a Type II kinase inhibitor of the IRE1α endoribonuclease that acts by targeting the ATP-binding pocket of IRE1α.</p>
    Formula:C33H28F3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:599.6
  • PV-1115

    CAS:
    <p>PV-1115 is an effective and highly selective inhibitor of the Chk2.</p>
    Formula:C20H19N7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.41
  • HIV-1 inhibitor-43

    CAS:
    <p>HIV-1 Inhibitor-43 suppresses HIV-1, with EC50: 21.3 nM (Y188L), 6.2 nM (K103N-Y181C), &lt;0.7 nM (K103N/Y181C), and lowers HIV RNA/p24 protein.</p>
    Formula:C24H21ClN2O4S
    Color and Shape:Solid
    Molecular weight:468.95
  • BMVC2

    CAS:
    <p>BMVC2 (o-BMVC), a carbazole derivative of BMVC, is a G-quadruplex (G4) stabilizer.</p>
    Formula:C28H25I2N3
    Color and Shape:Solid
    Molecular weight:657.33
  • BMH-22

    CAS:
    <p>BMH-22 is an RNA polymerase I inhibitor that acts by causing nucleolar stress and showing potent anticancer activity across many tumor types.</p>
    Formula:C16H17N3
    Color and Shape:Solid
    Molecular weight:251.33
  • MSC-1186

    CAS:
    <p>MSC-1186 selectively inhibits SRPKs—IC50: 2.7nM (SRPK1), 81nM (SRPK2), 0.6nM (SRPK3)—for cancer research.</p>
    Formula:C19H17ClFN7O2S
    Color and Shape:Solid
    Molecular weight:461.9
  • Bis-Pro-5FU

    CAS:
    <p>Bis-Pro-5FU enhances oral uptake and safety of 5-FU, an anti-cancer drug for colorectal and pancreatic tumors.</p>
    Formula:C10H7FN2O2
    Color and Shape:Solid
    Molecular weight:206.17
  • Carbonic anhydrase inhibitor 14

    CAS:
    <p>CA inhibitor 14 blocks hCA I/II/IX/XII (K i of 1203/99.7/9.4/27.7 nM) and CDK2 (IC50: 20.3 μM), showing antitumor effects.</p>
    Formula:C18H17N7O2S
    Color and Shape:Solid
    Molecular weight:395.44
  • 2-Keto-D-galactose

    CAS:
    <p>2-Keto-D-galactose inhibits DNA synthesis and inhibits the proliferation of in vitro grown Ehrlich ascites tumor cells.</p>
    Formula:C6H10O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:178.14
  • Fozivudine tidoxil

    CAS:
    <p>Fozivudine tidoxil, a reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>
    Formula:C35H64N5O8PS
    Color and Shape:Solid
    Molecular weight:745.95
  • (Rac)-Managlinat dialanetil

    CAS:
    <p>Managlinat dialanetil, an orally available and potent inhibitor of fructose 1,6-bisphosphatase (FBPase) used in research 2 type diabetes.</p>
    Formula:C21H33N4O6PS
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:500.55
  • DHODH-IN-12

    CAS:
    <p>DHODH-IN-12 is a leflunomide derivative and a weak dihydrorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.07.</p>
    Formula:C10H9N3O2
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:203.2
  • CAP-53194

    CAS:
    <p>CAP-53194 is a selective Plk1 inhibitor.</p>
    Formula:C21H14N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.37
  • CGP 53353

    CAS:
    <p>CGP 53353 (DAPH-7) is a PKC inhibitor with inhibitory effects on PKCβII and PKCβI and can be used to study atherosclerosis.</p>
    Formula:C20H13F2N3O2
    Purity:98.11%
    Color and Shape:Solid
    Molecular weight:365.33
  • Aditoprime

    CAS:
    <p>Aditoprime inhibits bacterial growth by blocking DHFR, effective against L.casei and E.coli with IC50 of 520/47 nM.</p>
    Formula:C15H21N5O2
    Color and Shape:Solid
    Molecular weight:303.36
  • GSK-3008348

    CAS:
    <p>GSK-3008348 is an antagonist of integrin alpha(v)beta6.</p>
    Formula:C29H37N5O2
    Purity:99.547%
    Color and Shape:Solid
    Molecular weight:487.64
  • Mivobulin Isethionate

    CAS:
    <p>Mivobulin, a tubulin inhibitor (CI-980), may treat glioma, melanoma, prostate, and ovarian cancer, targeting colchicine-binding site.</p>
    Formula:C19H25N5O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:451.5
  • PKC-9

    CAS:
    <p>PKC-9 is a PKC-zeta inhibitor 9.</p>
    Formula:C25H25N7
    Color and Shape:Solid
    Molecular weight:423.51
  • DHODH-IN-20

    CAS:
    <p>Dhodh-in-20 (Compound 133), a potent DHODH inhibitor, may help study acute myeloid leukemia and inhibit tumor growth.</p>
    Formula:C24H25F4N3O3
    Color and Shape:Solid
    Molecular weight:479.47
  • Picoplatin

    CAS:
    <p>Picoplatin, an anti-cancer agent overcoming platinum resistance, alkylates DNA to block replication, transcription, and induce apoptosis.</p>
    Formula:C6H10Cl2N2Pt
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.14
  • HHL-6

    CAS:
    <p>HHL-6 is a c-Fos and BDNF protein expression modulator.</p>
    Formula:C19H26N2O3
    Color and Shape:Solid
    Molecular weight:330.42
  • Metralindole HCl

    CAS:
    <p>Metralindole is a reversible monoamine oxidase A (RIMA) inhibitor, it was investigated as a potential antidepressant.</p>
    Formula:C15H18ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.78
  • HR22C16

    CAS:
    <p>HR22C16 is an effective, selective, and cell-permeable mitotic kinesin Eg5 inhibitor.</p>
    Formula:C23H23N3O3
    Color and Shape:Solid
    Molecular weight:389.45
  • JFN05510

    CAS:
    <p>Compound: 3'-O-tert-BDMS-5'-O-DMT-N2-IBG 2'-CE phosphoramidite; has anticancer properties and activates enzymes.</p>
    Formula:C50H68N7O9PSi
    Color and Shape:Solid
    Molecular weight:970.18
  • HIPP

    CAS:
    <p>HIPP is a highly selective inhibitor of antineoplastic CtBP.</p>
    Formula:C9H9NO3
    Color and Shape:Solid
    Molecular weight:179.17
  • NPD9948

    CAS:
    <p>NPD9948 is a competitive inhibitor of MTH1.</p>
    Formula:C13H14N6
    Color and Shape:Solid
    Molecular weight:254.29
  • LDN-209929

    CAS:
    <p>LDN-209929 2HCl is a potent and selective inhibitor of haspin kinase.</p>
    Formula:C17H17ClN2OS
    Color and Shape:Solid
    Molecular weight:332.85
  • DYRKi

    CAS:
    <p>DYRKi is a nontoxic, DYRK1-selective inhibitor.</p>
    Formula:C20H13F3N4O2S
    Color and Shape:Solid
    Molecular weight:430.4
  • BIPM

    CAS:
    <p>BIPM inhibits ROCK2, alters SH-SY5Y cell migration, actin fibers, neurite length, and reduces cofilin phosphorylation.</p>
    Formula:C23H22N2O3
    Color and Shape:Solid
    Molecular weight:374.43
  • REV7/REV3L-IN-1

    CAS:
    <p>REV7/REV3L-IN-1 is a inhibitor of REV7/REV3L interaction(IC50 of 78 μM),</p>
    Formula:C19H21N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.45
  • NSC47924

    CAS:
    <p>NSC47924 is a laminin receptor (LR) inhibitor.</p>
    Formula:C18H17NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.33
  • AB-182

    CAS:
    <p>AB-182 is an aziridine derivative with antitumor activity.</p>
    Formula:C11H22N3O4P
    Color and Shape:Solid
    Molecular weight:291.28
  • Ro 43-5054

    CAS:
    <p>Ro 43-5054 is a small molecular, noncyclic peptidomimetic inhibitor.</p>
    Formula:C24H27N5O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.5
  • ROCK-IN-D1

    CAS:
    <p>ROCK-IN-D1 is an effective and selective inhibitor of ROCK.</p>
    Formula:C22H27N5O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.55
  • SNX2-1-108

    CAS:
    <p>SNX2-1-108 is a selective CDK8 and CDK19 inhibitor.</p>
    Formula:C21H16N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.38
  • L-Guanosine

    CAS:
    <p>L-Guanosine is the L-configuration of Guanosine. Guanosine is a purine nucleoside that has anti-herpesvirus activity [1] [2].</p>
    Formula:C10H13N5O5
    Color and Shape:Solid
    Molecular weight:283.24
  • LIMK-IN-14

    CAS:
    <p>LIMK-IN-14 is an effective and selective inhibitor of LIMK.</p>
    Formula:C22H27N7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:437.49
  • Fosteabine

    CAS:
    <p>Fosteabine is an oral and prodrug analog of cytarabine. It is resistant to deoxycytidine deaminase.</p>
    Formula:C27H50N3O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:575.67
  • Denopterin

    CAS:
    <p>Denopterin is an antineoplastic agent.</p>
    Formula:C21H23N7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.45
  • UIAA-II-232

    CAS:
    <p>UIAA-II-232 (compound 19b) is a potent inhibitor of DNA gyrase catalytic (IC 50= 3.5 μM).</p>
    Formula:C20H24FN5O3
    Color and Shape:Solid
    Molecular weight:401.43
  • Protein kinase D inhibitor 1

    CAS:
    <p>Protein kinase D inhibitor 1 (17m) is a potent pan-PKD suppressant with IC50 of 17-35 nM, targeting cortactin phosphorylation.</p>
    Formula:C19H21N7
    Color and Shape:Solid
    Molecular weight:347.42
  • BAY-707

    CAS:
    <p>BAY-707: tolerable in mice, no anticancer efficacy; potent, selective MTH1 inhibitor, IC50 = 2.3 nM; good PK profile.</p>
    Formula:C15H20N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:288.34
  • Cdc7-IN-14

    CAS:
    <p>Cdc7-IN-14 (compound 82) is a potent CDC7 inhibitor with an IC50 &lt; 1 nM, promising for cancer research.</p>
    Formula:C18H20N4O2S
    Color and Shape:Solid
    Molecular weight:356.44
  • 1-Acetyl-3-o-toluyl-5-fluorouracil

    CAS:
    <p>1-Acetyl-3-o-toluyl-5-fluorouracil is a potent antineoplastic agent.</p>
    Formula:C14H11FN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:290.25
  • Rho-Kinase-IN-2

    CAS:
    <p>Rho-Kinase-IN-2, an oral ROCK inhibitor (IC50=3nM), penetrates the CNS; potential in Huntington's research.</p>
    Formula:C20H25FN4O2
    Color and Shape:Solid
    Molecular weight:372.44
  • Rabacfosadine succinate

    CAS:
    <p>Rabacfosadine succinate is the acyclic nucleoside phosphonate PMEG double prodrug.</p>
    Formula:C25H41N8O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:644.623
  • Thiamiprine

    CAS:
    <p>Thiamiprine is an agent with the activity of antineoplastic.</p>
    Formula:C9H8N8O2S
    Color and Shape:Solid
    Molecular weight:292.28
  • Meturedepa

    CAS:
    <p>Meturedepa is an antineoplastic agent.</p>
    Formula:C11H22N3O3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:275.28
  • RK-9123016

    CAS:
    <p>RK-9123016 is a SIRT2 inhibitor.</p>
    Formula:C16H18N6O3S
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:374.42
  • MK-0668

    CAS:
    <p>MK-0668 is a very potent and orally active very late antigen-4 antagonist.</p>
    Formula:C31H30Cl2N6O6S
    Color and Shape:Solid
    Molecular weight:685.58
  • BI-831266

    CAS:
    <p>BI-831266 is a potent and selective Aurora kinase B inhibitor.</p>
    Formula:C27H38ClN7O2
    Color and Shape:Solid
    Molecular weight:528.09
  • BzDANP

    CAS:
    <p>BzDANP is a modulator of pre-miR-29a maturation by Dicer.</p>
    Formula:C18H24N6
    Color and Shape:Solid
    Molecular weight:324.42
  • L 703014

    CAS:
    <p>L 703014 is an antagonist of the fibrinogen receptor.</p>
    Formula:C24H34N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.55
  • SEC inhibitor KL-2

    CAS:
    <p>KL-2: potent SEC inhibitor, selectively disrupts AFF4-CCNT1, dose-dependent, Ki: 1.50 μM.</p>
    Formula:C17H13ClFNO3
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:333.74
  • BMH-23

    CAS:
    <p>BMH-23 is an RNA polymerase I inhibitor that acts by causing nucleolar stress and showing potent anticancer activity across many tumor types.</p>
    Formula:C15H15N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:237.3
  • (R)-DRF053 dihydrochloride

    CAS:
    <p>cdk/CK1 inhibitor,potent and ATP-competitive</p>
    Formula:C23H29Cl2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:490.43
  • AM-TS23

    CAS:
    <p>AM-TS23 is used as a DNA polymerase lambda and beta inhibitor.</p>
    Formula:C17H12N2O3S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:388.48
  • Scaff10-8

    CAS:
    <p>Scaff10-8 blocks AKAP-Lbc-RhoA, aiding aquaporin-2 movement in kidney cells.</p>
    Formula:C22H18O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.37