PKC
PKC (Protein Kinase C) inhibitors target the PKC family of serine/threonine kinases, which are involved in a wide range of cellular processes, including cell cycle regulation, apoptosis, and differentiation. PKC plays a key role in signal transduction pathways that influence cell proliferation and survival. Inhibiting PKC can lead to changes in cell cycle progression, making these inhibitors valuable in research related to cancer, neurobiology, and cardiovascular diseases. At CymitQuimica, we provide a diverse selection of high-quality PKC inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
Read more
Rottlerin
CAS:82-08-6
Rottlerin (NSC-56346), a Mallotus Philippinensis extract, inhibits PKC (3-100 μM IC50); triggers apoptosis by activating …
Formula:
C30H28O8
Purity:
97.41% - 99.44%
Color and Shape:
Orange To Brown Powder
Molecular weight:
516.54
Ref: TM-T16791
| 5mg | 41.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 114.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
D-ERYTHRO-SPHINGOSINE
CAS:123-78-4
D-erythro-Sphingosine (trans-4-Sphingenine) is a protein kinase C (PKC) inhibitor. D-erythro-Sphingosine (Erythrosphingosine) is also a PP2A …
Formula:
C18H37NO2
Purity:
98% - ≥98%
Color and Shape:
Solid
Molecular weight:
299.49
Ref: TM-T5891
| 10mg | 46.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 166.00 € | ||
| 500mg | 398.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Procyanidin A1
CAS:103883-03-0
Procyanidin A1 (Proanthocyanidin A1) has antiallergic effects, it inhibits degranulation downstream of protein kinase C …
Formula:
C30H24O12
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
576.5
Ref: TM-TN1136
| 1mg | 87.00 € | ||
| 5mg | 155.00 € | ||
| 10mg | 241.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 590.00 € | ||
| 1mL*10mM (DMSO) | 182.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Afuresertib
CAS:1047644-62-1
Afuresertib (GSK2110183) is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase …
Formula:
C18H17Cl2FN4OS
Purity:
97.51% - 99.17%
Color and Shape:
Solid
Molecular weight:
427.32
Ref: TM-T1911
| 1mg | 39.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 467.00 € | ||
| 500mg | 1,013.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bisindolylmaleimide IV
CAS:119139-23-0
Bisindolylmaleimide IV is a protein kinase C (PKC) cell permeable inhibitor( IC50 : 0.10 - …
Formula:
C20H13N3O2
Purity:
98.2%
Color and Shape:
Dark Red Solid
Molecular weight:
327.34
Ref: TM-T7659
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 294.00 € | ||
| 50mg | 372.00 € | ||
| 100mg | 553.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Daphnoretin
CAS:2034-69-7
1.
Formula:
C19H12O7
Purity:
98% - 99.85%
Color and Shape:
Solid
Molecular weight:
352.29
Ref: TM-T4S1335
| 5mg | 55.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 227.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
TPPB
CAS:497259-23-1
TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).
Formula:
C27H30F3N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
501.54
Ref: TM-T17148
| 1mg | 158.00 € | ||
| 5mg | 512.00 € | ||
| 1mL*10mM (DMSO) | 552.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ro 31-8220 Mesylate
CAS:138489-18-6
Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor, and also shows potent inhibition …
Formula:
C25H23N5O2S·CH4O3S
Purity:
99.02% - 99.18%
Color and Shape:
Solid
Molecular weight:
553.65
Ref: TM-T6643
| 1mg | 52.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 238.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 489.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ingenol
CAS:30220-46-3
Ingenol mebutate treats actinic keratosis, has anticancer properties, and may reactivate latent HIV.
Formula:
C20H28O5
Purity:
97.53% - 99.87%
Color and Shape:
Solid
Molecular weight:
348.43
Ref: TM-T5S2017
| 1mg | 52.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 242.00 € | ||
| 50mg | 457.00 € | ||
| 100mg | 628.00 € | ||
| 500mg | 1,333.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PKCβ inhibitor 1
CAS:257879-35-9
PKCβ inhibitor 1 (KUN79359)(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of …
Formula:
C24H21N5O2
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
411.46
Ref: TM-T8376
| 1mg | 153.00 € | ||
| 5mg | 421.00 € | ||
| 10mg | 601.00 € | ||
| 25mg | 914.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,633.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Protein Kinase C 19-31 acetate
PKC 19-31 acetate, a serine-altered PKCa-derived PKC inhibitor, tests PKC activity.
Formula:
C69H122N26O18
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1603.9
Ref: TM-TP1053L
| 1mg | 36.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 338.00 € | ||
| 200mg | 480.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Hypericin
CAS:548-04-9
Hypericin (Cyclosan) is a natural anthraquinone compound. Hypericin exhibits antimicrobial, antiviral, antitumor, and antidepressant effects. …
Formula:
C30H16O8
Purity:
99.05% - ≥98%
Color and Shape:
Red-Coloured Anthraquinone-Derivative
Molecular weight:
504.44
Ref: TM-T6S0923
| 1mg | 61.00 € | ||
| 5mg | 129.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 731.00 € | ||
| 500mg | 1,483.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Enzastaurin
CAS:170364-57-5
Enzastaurin (LY317615) (LY317615) is an effective PKCβ selective inhibitor (IC50: 6 nM), 6- to 20-fold …
Formula:
C32H29N5O2
Purity:
100% - 99.24%
Color and Shape:
Solid
Molecular weight:
515.6
Ref: TM-T6280
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 121.00 € | ||
| 100mg | 184.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ionomycin calcium
CAS:56092-82-1
Ionomycin calcium (SQ23377 calcium) is an effective and selective calcium ionophore, exhibiting high specificity for …
Formula:
C41H70CaO9
Purity:
98% - 98.11%
Color and Shape:
Solid
Molecular weight:
747.07
Ref: TM-T11665
| 1mg | 123.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
NSC668394
CAS:382605-72-3
NSC668394 is an ezrin phosphorylation inhibitor.NSC668394 has antitumor activity and increases ezrin cleavage.NSC668394 can be …
Formula:
C17H12Br2N2O3
Purity:
99.29% - 99.29%
Color and Shape:
Solid
Molecular weight:
452.1
Ref: TM-T28212
| 1mg | 49.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 21 Jan 2025
DCP-LA
CAS:28399-31-7
DCP-LA (FR236924), linoleic acid derivatives, selective and direct activation of PKCε.
Formula:
C20H36O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
308.5
Ref: TM-T13637
| 1mg | 141.00 € | ||
| 5mg | 230.00 € | ||
| 500µg | To inquire |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CGP 53353
CAS:145915-60-2
CGP 53353 (DAPH-7) is a PKC inhibitor with inhibitory effects on PKCβII and PKCβI and …
Formula:
C20H13F2N3O2
Purity:
98.11%
Color and Shape:
Solid
Molecular weight:
365.33
Ref: TM-T22650
| 5mg | 124.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 423.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 1,194.00 € | ||
| 1mL*10mM (DMSO) | 138.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
PS315
CAS:1221964-50-6
PS315, a PS48 derivative, allosterically inhibits PKCζ/η (IC50: 10/30 μM), targeting aPKC's PIF-pocket, with anti-cancer …
Formula:
C23H19ClO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
362.85
Ref: TM-T16671
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
AJH-836
CAS:388621-67-8
AJH-836 is a compound that activates Munc13-1 and PKC ε/α, demonstrating a dissociation constant (Kd) …
Formula:
C22H38O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
382.53
Ref: TM-T78833
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
BJE6-106
CAS:1564249-38-2
BJE6-106 (B106) is a potent, selective PKCδ inhibitor (IC50: 0.05 μM) and targets selectivity over …
Formula:
C26H23NO2
Color and Shape:
Solid
Molecular weight:
381.47
Ref: TM-T10555
| 25mg | 1,058.00 € | ||
| 50mg | 1,395.00 € | ||
| 100mg | 2,172.00 € | ||
| 1mL*10mM (DMSO) | 345.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
