
Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(209 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(120 products)
- RAAS(87 products)
- Reductase(52 products)
- Somatostatin(49 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3183 products of "Endocrinology/Hormones"
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VPC-13163
CAS:<p>VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.</p>Formula:C16H14N2Purity:98.02%Color and Shape:SolidMolecular weight:234.3α-Zearalenol
CAS:<p>α-Zearalenol is one of the major metabolites of Zearalenone.</p>Formula:C18H24O5Purity:90% - 99.72%Color and Shape:SolidMolecular weight:320.38Nafoxidine
CAS:<p>Nafoxidine is an estrogen antagonist that has been used in the treatment of breast cancer.</p>Formula:C29H31NO2Purity:99.93%Color and Shape:SolidMolecular weight:425.56Enclomiphene hydrochloride
CAS:<p>Enclomiphene hydrochloride is an oral non-steroidal anti-estrogen for ovarian dysfunction and hypogonadism.</p>Formula:C26H29Cl2NOColor and Shape:SolidMolecular weight:442.42Deltorphin 2
CAS:<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Formula:C38H54N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:782.88TUG-1375
CAS:<p>TUG-1375 is an Agonist of Thiazolidine Free Fatty Acid Receptor 2</p>Formula:C22H19ClN2O4SPurity:99.41% - 99.55%Color and Shape:SolidMolecular weight:442.92Estradiol dipropionate
CAS:<p>Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.</p>Formula:C24H32O4Purity:99.68%Color and Shape:SolidMolecular weight:384.51Desoximetasone
CAS:<p>Desoximetasone (Topicort) is a topical corticosteroid for treating skin conditions like rashes.</p>Formula:C22H29FO4Purity:99.06% - 99.89%Color and Shape:SolidMolecular weight:376.46Harman hydrochloride
CAS:<p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>Formula:C12H11ClN2Purity:99.35%Color and Shape:SolidMolecular weight:218.68Antide acetate
<p>Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. </p>Formula:C84H112ClN17O16Purity:99.57%Color and Shape:SolidMolecular weight:1651.34Halobetasol propionate
CAS:<p>Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.</p>Formula:C25H31ClF2O5Purity:99.89%Color and Shape:Distributed As 0 05% OintmentMolecular weight:484.96PSN 375963 hydrochloride(388575-52-8 Free base)
CAS:<p>PSN 375963 hydrochloride, a potent GPR119 agonist, demonstrates EC50 values of 8.4 μM and 7.9 μM for human and mouse GPR119, respectively.</p>Formula:C17H24ClN3OColor and Shape:SolidMolecular weight:321.852,4'-Dihydroxybenzophenone
CAS:<p>2,4'-Dihydroxybenzophenone can effectively protect C57BL/6J mice from APAP-induced hepatotoxicity.</p>Formula:C13H10O3Purity:99.85%Color and Shape:SolidMolecular weight:214.22Pipendoxifene
CAS:<p>Pipendoxifene (ERA-923) is an antiestrogen that blocks ER-alpha and inhibits MCF-7 breast cancer cell growth, effective even when tamoxifen-resistant.</p>Formula:C29H32N2O3Color and Shape:SolidMolecular weight:456.58(Sar¹)-Angiotensin II acetate
<p>(Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor.</p>Formula:C51H75N13O12Purity:99.89%Color and Shape:SoildMolecular weight:1062.22Leucylarginylproline
CAS:<p>Leucylarginylproline is an inhibitor of angiotensin-converting enzyme (ACE) (IC50 : 0.27μM).</p>Formula:C17H32N6O4Purity:99.58%Color and Shape:SolidMolecular weight:384.47Teriparatide acetate
CAS:<p>Teriparatide acetate (Forteo), a synthetic parathyroid hormone, treats osteoporosis by favoring bone growth with a 2 nM IC50.</p>Formula:C183H295N55O53S2Purity:99.86%Color and Shape:SolidMolecular weight:4177.83Zaprinast
CAS:<p>Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist.</p>Formula:C13H13N5O2Purity:99.73% - 99.77%Color and Shape:White To Off White PowderMolecular weight:271.27Norgestrel
CAS:<p>Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.</p>Formula:C21H28O2Purity:99.71% - 99.72%Color and Shape:Crystals From Methanol White Crystalline PowderMolecular weight:312.45ARD-2128
CAS:<p>ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.</p>Formula:C45H50ClN7O6Purity:98.8%Color and Shape:SolidMolecular weight:820.37Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formula:C25H34N2O5Purity:98%Color and Shape:SolidMolecular weight:442.55ADL-5747 (HCl)
CAS:<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Formula:C24H29ClN2O3Color and Shape:SolidMolecular weight:428.95Sparsentan
CAS:<p>Sparsentan (DARA-a) is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM,</p>Formula:C32H40N4O5SPurity:97.94% - 98.69%Color and Shape:SolidMolecular weight:592.75MCOPPB
CAS:<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Formula:C26H40N4Color and Shape:SolidMolecular weight:408.62EST73502 hydrochloride
CAS:<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Formula:C19H27ClF2N2O2Color and Shape:SolidMolecular weight:388.88ARV-471
CAS:<p>ARV-471 (Vepdegestrant) is a orally active Cereblon -based estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer.</p>Formula:C45H49N5O4Purity:97.15% - >99.99%Color and Shape:SolidMolecular weight:723.9MCOPPB triHydrochloride
CAS:<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Formula:C26H43Cl3N4Purity:99.89% - 99.91%Color and Shape:SolidMolecular weight:518.01Chlorotrianisene
CAS:<p>Chlorotrianisene, a synthetic SERM, is orally active, lipophilic, and has estrogenic and antiestrogenic effects.</p>Formula:C23H21ClO3Purity:98.88% - 99.03%Color and Shape:Crystals From Methanol Physical Description Small White Crystals Or White Powder Softens At 226°F Odorless (Ntp 1992)Molecular weight:380.86PZM21
CAS:<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formula:C19H27N3O2SPurity:99.93% - >99.99%Color and Shape:SolidMolecular weight:361.51-methoxycyclopropanecarboxylic acid
CAS:<p>1-methoxycyclopropanecarboxylic acid is an agonist of free fatty acid receptor 3 (FFAR3, human).</p>Formula:C5H8O3Purity:99.44%Color and Shape:Light-Yellow To Yellow Solid Or LiquidMolecular weight:116.12Ulipristal
CAS:<p>Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.</p>Formula:C28H35NO3Purity:99.82%Color and Shape:SolidMolecular weight:433.58SNAP 94847 hydrochloride
CAS:<p>SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)</p>Formula:C29H33ClF2N2O2Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:515.03Fevipiprant
CAS:<p>Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.</p>Formula:C19H17F3N2O4SPurity:99.32% - 99.59%Color and Shape:SolidMolecular weight:426.41Enalapril Maleate
CAS:<p>Enalapril Maleate (MK-421 Maleate), an ACE inhibitor, is utilized in the treatment of hypertension, chronic heart failure, and diabetic nephropathy.</p>Formula:C20H28N2O5·C4H4O4Purity:99.02% - ≥95%Color and Shape:White To Off-White Crystalline Powder SolidMolecular weight:492.52N-Desmethylclozapine
CAS:<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Formula:C17H17ClN4Purity:97.25% - 99.83%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8Broparestrol (E)-
CAS:<p>Broparestrol (E)- has antifertility activity and is a potent inhibitor of rodent mammary tumorigenesis.</p>Formula:C22H19BrPurity:>99.99%Color and Shape:SolidMolecular weight:363.29N-Acetyl-Ser-Asp-Lys-Pro
CAS:<p>Acetyl Ser-Asp-Lys-Pro, derived from thymosin β4 in bone marrow, blocks stem cell cycle progression and shields mice from Ara-C toxicity.</p>Formula:C20H33N5O9Purity:99.85%Color and Shape:SolidMolecular weight:487.5(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Formula:C33H46N6O10Purity:94.17%Color and Shape:SoildMolecular weight:686.75BigLEN (mouse) acetate
<p>BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 (GPR171), with a Kd of ∼0.5 nM.</p>Formula:C80H134N24O24Purity:>99.99%Color and Shape:SolidMolecular weight:1816.07BW-180C
CAS:<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Formula:C29H39N5O7Purity:>99.99%Color and Shape:SolidMolecular weight:569.65Temocapril hydrochloride
CAS:<p>Temocapril hydrochloride (CS-622 HCl), the hydrochloride of Temocapril, is a long-acting ACE inhibitor used for the therapy of hypertension.</p>Formula:C23H28N2O5S2·HClPurity:99.26% - 99.48%Color and Shape:White Solid PowderMolecular weight:513.07Alamandine TFA
<p>Alamandine TFA, a RAS peptide, binds MrgD receptors, has anti-hypertensive effects, and protects heart and kidneys.</p>Formula:C42H63F3N12O11Purity:99.62%Color and Shape:SoildMolecular weight:969.02Acein acetate
<p>ACE ligand with Kd 2.79 nM, inactive on ACE up to 500 nM. Boosts NMDA/D-serine-induced dopamine release in striatum.</p>Formula:C45H72N10O15Purity:99.43%Color and Shape:SolidMolecular weight:993.11FH1
CAS:<p>FH1 (NSC-12407) (BRD-K4477), a small molecule, enhances the functions of hepatocytes and promotes differentiation hepatocytes derived by iPS.</p>Formula:C17H18N2O2Purity:98% - 99.64%Color and Shape:SolidMolecular weight:282.34Azilsartan Medoxomil
CAS:<p>Azilsartan Medoxomil (TAK-491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults</p>Formula:C30H24N4O8Purity:99.83%Color and Shape:SolidMolecular weight:568.53BNP (1-32), human
CAS:<p>BNP (1-32), human is a brain natriuretic peptide</p>Formula:C143H244N50O42S4Purity:98.52%Color and Shape:White PowderMolecular weight:3464.04Osilodrostat phosphate
CAS:<p>Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.</p>Formula:C13H13FN3O4PColor and Shape:SolidMolecular weight:325.23Bavdegalutamide
CAS:<p>Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).</p>Formula:C41H43ClFN9O6Purity:97.17% - 99.04%Color and Shape:SolidMolecular weight:812.29AR 231453
CAS:<p>Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.</p>Formula:C21H24FN7O5SPurity:99.31% - 99.34%Color and Shape:SolidMolecular weight:505.52Resmetirom
CAS:<p>Resmetirom (MGL-3196) is a THR-β agonist (EC50=0.21 μM), with high selectivity and oral activity. High-Quality, Low-Cost!</p>Formula:C17H12Cl2N6O4Purity:99.05% - >99.99%Color and Shape:SolidMolecular weight:435.22Deltorphin I
CAS:<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Formula:C37H52N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:768.86MK-6892
CAS:<p>MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM).</p>Formula:C19H22N4O5Purity:99.01% - 99.67%Color and Shape:SolidMolecular weight:386.4Sobetirome
CAS:<p>Sobetirome (IACS-010759) is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).</p>Formula:C20H24O4Purity:98.08% - 98.25%Color and Shape:SolidMolecular weight:328.4Fasiglifam
CAS:<p>Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.</p>Formula:C29H32O7SPurity:99.82% - 99.9%Color and Shape:SolidMolecular weight:524.63GW9508
CAS:<p>GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.</p>Formula:C22H21NO3Purity:97.89% - 99.19%Color and Shape:SolidMolecular weight:347.41Nalmefene hydrochloride
CAS:<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Formula:C21H26ClNO3Purity:98% - 99.85%Color and Shape:SolidMolecular weight:375.89VPC-13566
CAS:<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Formula:C18H14N2Purity:99.55%Color and Shape:SolidMolecular weight:258.32Estradiol hemihydrate
CAS:<p>Estradiol hemihydrate: major female hormone, boosts neural differentiation, studied for cancer and neurodegenerative disease.</p>Formula:C18H26O3Color and Shape:SolidMolecular weight:281.39Angiotensin I/II (1-6)
CAS:<p>Angiotensin I/II (1-6) is a peptide (ASP-ARG-VAL-TYR-ILE-HIS) that contains the amino acids 1-6 and is converted from Angiotensin I/II peptide.</p>Formula:C36H55N11O10Purity:99.44%Color and Shape:SolidMolecular weight:801.893-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:<p>3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.</p>Formula:C18H14N4OPurity:98.41%Color and Shape:SolidMolecular weight:302.33CID1231538
CAS:<p>CID1231538 is a potent GPR35 antagonist.</p>Formula:C26H22ClN3O3S2Purity:98.79%Color and Shape:SolidMolecular weight:524.05Lasofoxifene
CAS:<p>Lasofoxifene (CP-336156) is a selective oestrogen receptor modulator/antagonist that reduces serum IL-6 levels and inhibits joint inflammation and osteoporosis.</p>Formula:C28H31NO2Purity:99.6%Color and Shape:SolidMolecular weight:413.55CTK8A3536
CAS:<p>CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.</p>Formula:C14H16N2O2SPurity:99.62%Color and Shape:SolidMolecular weight:276.35Finerenone
CAS:<p>Finerenone (BAY-948862) is a selective and orally nonsteroidal antagonist of the mineralocorticoid receptor (MR). Cost effective and quality assured.</p>Formula:C21H22N4O3Purity:99.45% - 99.91%Color and Shape:SolidMolecular weight:378.42H3B-5942
CAS:<p>H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).</p>Formula:C31H34N4O2Purity:99.21% - ≥95%Color and Shape:SolidMolecular weight:494.63N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Formula:C30H39N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:597.66Ferrous Bisglycinate
CAS:<p>Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.</p>Formula:C4H8FeN2O4Purity:≥95%Color and Shape:SolidMolecular weight:203.966-OAU
CAS:<p>6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.</p>Formula:C12H21N3O2Purity:98.14% - 99.01%Color and Shape:SolidMolecular weight:239.31Sufugolix
CAS:<p>Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.</p>Formula:C36H31F2N5O4SPurity:97.78%Color and Shape:SolidMolecular weight:667.72Velsecorat
CAS:<p>Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).</p>Formula:C32H32F2N4O6Purity:99.35%Color and Shape:SolidMolecular weight:606.62Boldenone Undecylenate
CAS:<p>Boldenone Undecylenate (Parenabol) is a synthetic steroid.</p>Formula:C30H44O3Purity:99.39%Color and Shape:Light Yellow Oily MatterMolecular weight:452.67Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Formula:C31H41N7O9Purity:98.92%Color and Shape:SoildMolecular weight:655.7Angiotensin II 5-valine TFA
<p>Angiotensin II 5-valine TFA is an agonist of angiotensin receptor.</p>Formula:C51H70F3N13O14Purity:99.69%Color and Shape:SolidMolecular weight:1146.18Angiotensin 1/2 (5-7) acetate
<p>Angiotensin 1/2 (5-7) acetate: a dipsogenic hormone peptide, sequence H2N-Ile-His-Pro-OH, from liver-produced angiotensinogen.</p>Formula:C19H31N5O6Purity:99.13%Color and Shape:SolidMolecular weight:425.49[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Formula:C30H42N6O8Purity:99.36%Color and Shape:SolidMolecular weight:614.69Urotensin II, mouse acetate (9047-55-6 free base)
<p>Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.</p>Formula:C64H88N14O19S2Purity:97.86%Color and Shape:SolidMolecular weight:1421.61Iprodione
CAS:<p>Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.</p>Formula:C13H13Cl2N3O3Purity:98.82%Color and Shape:Colorless Crystals Cream To Colorless Odorless PowderMolecular weight:330.17JNJ-63576253
CAS:<p>JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).</p>Formula:C23H22ClF3N6O2SPurity:98.71%Color and Shape:SolidMolecular weight:538.97Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Formula:C51H73N15O11Purity:98.59%Color and Shape:SolidMolecular weight:1072.22Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Formula:C51H68N12O13Purity:99.66%Color and Shape:SolidMolecular weight:1057.16AH-7614
CAS:<p>AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.</p>Formula:C20H17NO3SPurity:98.05%Color and Shape:SolidMolecular weight:351.42REVERSE T3
CAS:<p>Reverse T3 (3,3',5'-triiodo-L-thyronine) inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.</p>Formula:C15H12I3NO4Purity:95.99% - 97.89%Color and Shape:PowderMolecular weight:650.97Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Formula:C59H95N19O14Purity:99.88%Color and Shape:SolidMolecular weight:1294.53[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Formula:C29H39N5O7Purity:98.06%Color and Shape:SolidMolecular weight:569.65Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35STF-62247
CAS:<p>STF-62247 is TGN inhibitor with IC50 of 0.625 μM and 16 μM in RCC4 and RCC4/VHL cells, respectively.</p>Formula:C15H13N3SPurity:99.6% - 99.67%Color and Shape:SolidMolecular weight:267.35MBX-2982
CAS:<p>MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.</p>Formula:C22H24N8OSPurity:98% - 99.96%Color and Shape:SolidMolecular weight:448.54cangrelor tetrasodium
CAS:<p>Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent antiplatelet effects.</p>Formula:C17H21Cl2F3N5Na4O12P3S2Purity:98.51% - 98.6%Color and Shape:SolidMolecular weight:864.29Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formula:C50H72N15O15SPurity:>99.99%Color and Shape:SolidMolecular weight:1326.26Nestoron
CAS:<p>Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).</p>Formula:C23H30O4Purity:99.48% - 99.83%Color and Shape:SolidMolecular weight:370.48Isoflupredone Acetate
CAS:<p>Isoflupredone Acetate is a corticosteroid with the activity of topical anti-inflammatory.</p>Formula:C23H29FO6Purity:99.43%Color and Shape:SolidMolecular weight:420.47Eprosartan Mesylate
CAS:<p>Eprosartan Mesylate (SKF-108566J) is a competitive and reversible Angiotensin II Receptor Blocker.</p>Formula:C23H24N2O4S·CH4O3SPurity:99.72% - 99.93%Color and Shape:A White To Off- White PowderMolecular weight:520.62PW0787
CAS:<p>PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).</p>Formula:C23H20F4N4O2Purity:98.42%Color and Shape:SolidMolecular weight:460.42EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Formula:C19H27ClF2N2O2Purity:99.96%Color and Shape:SolidMolecular weight:388.88Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26BMS986188
CAS:<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Formula:C30H31BrO4Purity:98.76%Color and Shape:SolidMolecular weight:535.47MS21570
CAS:<p>MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 Nm,that reduces anxiety-like behavior and fear conditioning in mice.</p>Formula:C10H11N3S2Purity:97.79%Color and Shape:SolidMolecular weight:237.34b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
CAS:<p>Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.</p>Formula:C18H18O3Purity:99.85% - 99.96%Color and Shape:SolidMolecular weight:282.33DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59
