CymitQuimica logo
Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

Show 6 more subcategories

Found 3183 products of "Endocrinology/Hormones"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • VPC-13163

    CAS:
    <p>VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.</p>
    Formula:C16H14N2
    Purity:98.02%
    Color and Shape:Solid
    Molecular weight:234.3
  • α-Zearalenol

    CAS:
    <p>α-Zearalenol is one of the major metabolites of Zearalenone.</p>
    Formula:C18H24O5
    Purity:90% - 99.72%
    Color and Shape:Solid
    Molecular weight:320.38
  • Nafoxidine

    CAS:
    <p>Nafoxidine is an estrogen antagonist that has been used in the treatment of breast cancer.</p>
    Formula:C29H31NO2
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:425.56
  • Enclomiphene hydrochloride

    CAS:
    <p>Enclomiphene hydrochloride is an oral non-steroidal anti-estrogen for ovarian dysfunction and hypogonadism.</p>
    Formula:C26H29Cl2NO
    Color and Shape:Solid
    Molecular weight:442.42
  • Deltorphin 2

    CAS:
    <p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>
    Formula:C38H54N8O10
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:782.88
  • TUG-1375

    CAS:
    <p>TUG-1375 is an Agonist of Thiazolidine Free Fatty Acid Receptor 2</p>
    Formula:C22H19ClN2O4S
    Purity:99.41% - 99.55%
    Color and Shape:Solid
    Molecular weight:442.92
  • Estradiol dipropionate

    CAS:
    <p>Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.</p>
    Formula:C24H32O4
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:384.51
  • Desoximetasone

    CAS:
    <p>Desoximetasone (Topicort) is a topical corticosteroid for treating skin conditions like rashes.</p>
    Formula:C22H29FO4
    Purity:99.06% - 99.89%
    Color and Shape:Solid
    Molecular weight:376.46
  • Harman hydrochloride

    CAS:
    <p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>
    Formula:C12H11ClN2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:218.68
  • Antide acetate


    <p>Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. </p>
    Formula:C84H112ClN17O16
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:1651.34
  • Halobetasol propionate

    CAS:
    <p>Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.</p>
    Formula:C25H31ClF2O5
    Purity:99.89%
    Color and Shape:Distributed As 0 05% Ointment
    Molecular weight:484.96
  • PSN 375963 hydrochloride(388575-52-8 Free base)

    CAS:
    <p>PSN 375963 hydrochloride, a potent GPR119 agonist, demonstrates EC50 values of 8.4 μM and 7.9 μM for human and mouse GPR119, respectively.</p>
    Formula:C17H24ClN3O
    Color and Shape:Solid
    Molecular weight:321.85
  • 2,4'-Dihydroxybenzophenone

    CAS:
    <p>2,4'-Dihydroxybenzophenone can effectively protect C57BL/6J mice from APAP-induced hepatotoxicity.</p>
    Formula:C13H10O3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:214.22
  • Pipendoxifene

    CAS:
    <p>Pipendoxifene (ERA-923) is an antiestrogen that blocks ER-alpha and inhibits MCF-7 breast cancer cell growth, effective even when tamoxifen-resistant.</p>
    Formula:C29H32N2O3
    Color and Shape:Solid
    Molecular weight:456.58
  • (Sar¹)-Angiotensin II acetate


    <p>(Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor.</p>
    Formula:C51H75N13O12
    Purity:99.89%
    Color and Shape:Soild
    Molecular weight:1062.22
  • Leucylarginylproline

    CAS:
    <p>Leucylarginylproline is an inhibitor of angiotensin-converting enzyme (ACE) (IC50 : 0.27μM).</p>
    Formula:C17H32N6O4
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:384.47
  • Teriparatide acetate

    CAS:
    <p>Teriparatide acetate (Forteo), a synthetic parathyroid hormone, treats osteoporosis by favoring bone growth with a 2 nM IC50.</p>
    Formula:C183H295N55O53S2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:4177.83
  • Zaprinast

    CAS:
    <p>Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist.</p>
    Formula:C13H13N5O2
    Purity:99.73% - 99.77%
    Color and Shape:White To Off White Powder
    Molecular weight:271.27
  • Norgestrel

    CAS:
    <p>Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.</p>
    Formula:C21H28O2
    Purity:99.71% - 99.72%
    Color and Shape:Crystals From Methanol White Crystalline Powder
    Molecular weight:312.45
  • ARD-2128

    CAS:
    <p>ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.</p>
    Formula:C45H50ClN7O6
    Purity:98.8%
    Color and Shape:Solid
    Molecular weight:820.37
  • Alvimopan monohydrate

    CAS:
    <p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>
    Formula:C25H34N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.55
  • ADL-5747 (HCl)

    CAS:
    <p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>
    Formula:C24H29ClN2O3
    Color and Shape:Solid
    Molecular weight:428.95
  • Sparsentan

    CAS:
    <p>Sparsentan (DARA-a) is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM,</p>
    Formula:C32H40N4O5S
    Purity:97.94% - 98.69%
    Color and Shape:Solid
    Molecular weight:592.75
  • MCOPPB

    CAS:
    <p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>
    Formula:C26H40N4
    Color and Shape:Solid
    Molecular weight:408.62
  • EST73502 hydrochloride

    CAS:
    <p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>
    Formula:C19H27ClF2N2O2
    Color and Shape:Solid
    Molecular weight:388.88
  • ARV-471

    CAS:
    <p>ARV-471 (Vepdegestrant) is a orally active Cereblon -based estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer.</p>
    Formula:C45H49N5O4
    Purity:97.15% - >99.99%
    Color and Shape:Solid
    Molecular weight:723.9
  • MCOPPB triHydrochloride

    CAS:
    <p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>
    Formula:C26H43Cl3N4
    Purity:99.89% - 99.91%
    Color and Shape:Solid
    Molecular weight:518.01
  • Chlorotrianisene

    CAS:
    <p>Chlorotrianisene, a synthetic SERM, is orally active, lipophilic, and has estrogenic and antiestrogenic effects.</p>
    Formula:C23H21ClO3
    Purity:98.88% - 99.03%
    Color and Shape:Crystals From Methanol Physical Description Small White Crystals Or White Powder Softens At 226°F Odorless (Ntp 1992)
    Molecular weight:380.86
  • PZM21

    CAS:
    <p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>
    Formula:C19H27N3O2S
    Purity:99.93% - >99.99%
    Color and Shape:Solid
    Molecular weight:361.5
  • 1-methoxycyclopropanecarboxylic acid

    CAS:
    <p>1-methoxycyclopropanecarboxylic acid is an agonist of free fatty acid receptor 3 (FFAR3, human).</p>
    Formula:C5H8O3
    Purity:99.44%
    Color and Shape:Light-Yellow To Yellow Solid Or Liquid
    Molecular weight:116.12
  • Ulipristal

    CAS:
    <p>Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.</p>
    Formula:C28H35NO3
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:433.58
  • SNAP 94847 hydrochloride

    CAS:
    <p>SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)</p>
    Formula:C29H33ClF2N2O2
    Purity:99.85% - >99.99%
    Color and Shape:Solid
    Molecular weight:515.03
  • Fevipiprant

    CAS:
    <p>Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.</p>
    Formula:C19H17F3N2O4S
    Purity:99.32% - 99.59%
    Color and Shape:Solid
    Molecular weight:426.41
  • Enalapril Maleate

    CAS:
    <p>Enalapril Maleate (MK-421 Maleate), an ACE inhibitor, is utilized in the treatment of hypertension, chronic heart failure, and diabetic nephropathy.</p>
    Formula:C20H28N2O5·C4H4O4
    Purity:99.02% - ≥95%
    Color and Shape:White To Off-White Crystalline Powder Solid
    Molecular weight:492.52
  • N-Desmethylclozapine

    CAS:
    <p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>
    Formula:C17H17ClN4
    Purity:97.25% - 99.83%
    Color and Shape:Yellow Crystalline Solid
    Molecular weight:312.8
  • Broparestrol (E)-

    CAS:
    <p>Broparestrol (E)- has antifertility activity and is a potent inhibitor of rodent mammary tumorigenesis.</p>
    Formula:C22H19Br
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:363.29
  • N-Acetyl-Ser-Asp-Lys-Pro

    CAS:
    <p>Acetyl Ser-Asp-Lys-Pro, derived from thymosin β4 in bone marrow, blocks stem cell cycle progression and shields mice from Ara-C toxicity.</p>
    Formula:C20H33N5O9
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:487.5
  • (D-Ser2)-Leu-Enkephalin-Thr


    <p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>
    Formula:C33H46N6O10
    Purity:94.17%
    Color and Shape:Soild
    Molecular weight:686.75
  • BigLEN (mouse) acetate


    <p>BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 (GPR171), with a Kd of ∼0.5 nM.</p>
    Formula:C80H134N24O24
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1816.07
  • BW-180C

    CAS:
    <p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>
    Formula:C29H39N5O7
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:569.65
  • Temocapril hydrochloride

    CAS:
    <p>Temocapril hydrochloride (CS-622 HCl), the hydrochloride of Temocapril, is a long-acting ACE inhibitor used for the therapy of hypertension.</p>
    Formula:C23H28N2O5S2·HCl
    Purity:99.26% - 99.48%
    Color and Shape:White Solid Powder
    Molecular weight:513.07
  • Alamandine TFA


    <p>Alamandine TFA, a RAS peptide, binds MrgD receptors, has anti-hypertensive effects, and protects heart and kidneys.</p>
    Formula:C42H63F3N12O11
    Purity:99.62%
    Color and Shape:Soild
    Molecular weight:969.02
  • Acein acetate


    <p>ACE ligand with Kd 2.79 nM, inactive on ACE up to 500 nM. Boosts NMDA/D-serine-induced dopamine release in striatum.</p>
    Formula:C45H72N10O15
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:993.11
  • FH1

    CAS:
    <p>FH1 (NSC-12407) (BRD-K4477), a small molecule, enhances the functions of hepatocytes and promotes differentiation hepatocytes derived by iPS.</p>
    Formula:C17H18N2O2
    Purity:98% - 99.64%
    Color and Shape:Solid
    Molecular weight:282.34
  • Azilsartan Medoxomil

    CAS:
    <p>Azilsartan Medoxomil (TAK-491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults</p>
    Formula:C30H24N4O8
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:568.53
  • BNP (1-32), human

    CAS:
    <p>BNP (1-32), human is a brain natriuretic peptide</p>
    Formula:C143H244N50O42S4
    Purity:98.52%
    Color and Shape:White Powder
    Molecular weight:3464.04
  • Osilodrostat phosphate

    CAS:
    <p>Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.</p>
    Formula:C13H13FN3O4P
    Color and Shape:Solid
    Molecular weight:325.23
  • Bavdegalutamide

    CAS:
    <p>Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).</p>
    Formula:C41H43ClFN9O6
    Purity:97.17% - 99.04%
    Color and Shape:Solid
    Molecular weight:812.29
  • AR 231453

    CAS:
    <p>Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.</p>
    Formula:C21H24FN7O5S
    Purity:99.31% - 99.34%
    Color and Shape:Solid
    Molecular weight:505.52
  • Resmetirom

    CAS:
    <p>Resmetirom (MGL-3196) is a THR-β agonist (EC50=0.21 μM), with high selectivity and oral activity. High-Quality, Low-Cost!</p>
    Formula:C17H12Cl2N6O4
    Purity:99.05% - >99.99%
    Color and Shape:Solid
    Molecular weight:435.22
  • Deltorphin I

    CAS:
    <p>Deltorphin I is an agonist of δ-opioid receptor.</p>
    Formula:C37H52N8O10
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:768.86
  • MK-6892

    CAS:
    <p>MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM).</p>
    Formula:C19H22N4O5
    Purity:99.01% - 99.67%
    Color and Shape:Solid
    Molecular weight:386.4
  • Sobetirome

    CAS:
    <p>Sobetirome (IACS-010759) is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).</p>
    Formula:C20H24O4
    Purity:98.08% - 98.25%
    Color and Shape:Solid
    Molecular weight:328.4
  • Fasiglifam

    CAS:
    <p>Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.</p>
    Formula:C29H32O7S
    Purity:99.82% - 99.9%
    Color and Shape:Solid
    Molecular weight:524.63
  • GW9508

    CAS:
    <p>GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.</p>
    Formula:C22H21NO3
    Purity:97.89% - 99.19%
    Color and Shape:Solid
    Molecular weight:347.41
  • Nalmefene hydrochloride

    CAS:
    <p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>
    Formula:C21H26ClNO3
    Purity:98% - 99.85%
    Color and Shape:Solid
    Molecular weight:375.89
  • VPC-13566

    CAS:
    <p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>
    Formula:C18H14N2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:258.32
  • Estradiol hemihydrate

    CAS:
    <p>Estradiol hemihydrate: major female hormone, boosts neural differentiation, studied for cancer and neurodegenerative disease.</p>
    Formula:C18H26O3
    Color and Shape:Solid
    Molecular weight:281.39
  • Angiotensin I/II (1-6)

    CAS:
    <p>Angiotensin I/II (1-6) is a peptide (ASP-ARG-VAL-TYR-ILE-HIS) that contains the amino acids 1-6 and is converted from Angiotensin I/II peptide.</p>
    Formula:C36H55N11O10
    Purity:99.44%
    Color and Shape:Solid
    Molecular weight:801.89
  • 3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile

    CAS:
    <p>3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.</p>
    Formula:C18H14N4O
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:302.33
  • CID1231538

    CAS:
    <p>CID1231538 is a potent GPR35 antagonist.</p>
    Formula:C26H22ClN3O3S2
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:524.05
  • Lasofoxifene

    CAS:
    <p>Lasofoxifene (CP-336156) is a selective oestrogen receptor modulator/antagonist that reduces serum IL-6 levels and inhibits joint inflammation and osteoporosis.</p>
    Formula:C28H31NO2
    Purity:99.6%
    Color and Shape:Solid
    Molecular weight:413.55
  • CTK8A3536

    CAS:
    <p>CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.</p>
    Formula:C14H16N2O2S
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:276.35
  • Finerenone

    CAS:
    <p>Finerenone (BAY-948862) is a selective and orally nonsteroidal antagonist of the mineralocorticoid receptor (MR). Cost effective and quality assured.</p>
    Formula:C21H22N4O3
    Purity:99.45% - 99.91%
    Color and Shape:Solid
    Molecular weight:378.42
  • H3B-5942

    CAS:
    <p>H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).</p>
    Formula:C31H34N4O2
    Purity:99.21% - ≥95%
    Color and Shape:Solid
    Molecular weight:494.63
  • N-terminally acetylated Leu-enkephalin


    <p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>
    Formula:C30H39N5O8
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:597.66
  • Ferrous Bisglycinate

    CAS:
    <p>Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.</p>
    Formula:C4H8FeN2O4
    Purity:≥95%
    Color and Shape:Solid
    Molecular weight:203.96
  • 6-OAU

    CAS:
    <p>6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.</p>
    Formula:C12H21N3O2
    Purity:98.14% - 99.01%
    Color and Shape:Solid
    Molecular weight:239.31
  • Sufugolix

    CAS:
    <p>Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.</p>
    Formula:C36H31F2N5O4S
    Purity:97.78%
    Color and Shape:Solid
    Molecular weight:667.72
  • Velsecorat

    CAS:
    <p>Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).</p>
    Formula:C32H32F2N4O6
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:606.62
  • Boldenone Undecylenate

    CAS:
    <p>Boldenone Undecylenate (Parenabol) is a synthetic steroid.</p>
    Formula:C30H44O3
    Purity:99.39%
    Color and Shape:Light Yellow Oily Matter
    Molecular weight:452.67
  • Nociceptin (1-7) acetate


    <p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>
    Formula:C31H41N7O9
    Purity:98.92%
    Color and Shape:Soild
    Molecular weight:655.7
  • Angiotensin II 5-valine TFA


    <p>Angiotensin II 5-valine TFA is an agonist of angiotensin receptor.</p>
    Formula:C51H70F3N13O14
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:1146.18
  • Angiotensin 1/2 (5-7) acetate


    <p>Angiotensin 1/2 (5-7) acetate: a dipsogenic hormone peptide, sequence H2N-Ile-His-Pro-OH, from liver-produced angiotensinogen.</p>
    Formula:C19H31N5O6
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:425.49
  • [Leu5]-Enkephalin, amide acetate


    <p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>
    Formula:C30H42N6O8
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:614.69
  • Urotensin II, mouse acetate (9047-55-6 free base)


    <p>Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.</p>
    Formula:C64H88N14O19S2
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:1421.61
  • Iprodione

    CAS:
    <p>Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.</p>
    Formula:C13H13Cl2N3O3
    Purity:98.82%
    Color and Shape:Colorless Crystals Cream To Colorless Odorless Powder
    Molecular weight:330.17
  • JNJ-63576253

    CAS:
    <p>JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).</p>
    Formula:C23H22ClF3N6O2S
    Purity:98.71%
    Color and Shape:Solid
    Molecular weight:538.97
  • Ac-RYYRWK-NH2 acetate


    <p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>
    Formula:C51H73N15O11
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:1072.22
  • Hemorphin-7 acetate(152685-85-3 free base)


    <p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>
    Formula:C51H68N12O13
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:1057.16
  • AH-7614

    CAS:
    <p>AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.</p>
    Formula:C20H17NO3S
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:351.42
  • REVERSE T3

    CAS:
    <p>Reverse T3 (3,3',5'-triiodo-L-thyronine) inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.</p>
    Formula:C15H12I3NO4
    Purity:95.99% - 97.89%
    Color and Shape:Powder
    Molecular weight:650.97
  • Dynorphin A 1-10 acetate(79994-24-4 free base)


    <p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>
    Formula:C59H95N19O14
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:1294.53
  • [D-Ala2]leucine-enkephalin

    CAS:
    <p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>
    Formula:C29H39N5O7
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:569.65
  • Methylnaltrexone bromide

    CAS:
    Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.
    Formula:C21H26BrNO4
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:436.35
  • STF-62247

    CAS:
    <p>STF-62247 is TGN inhibitor with IC50 of 0.625 μM and 16 μM in RCC4 and RCC4/VHL cells, respectively.</p>
    Formula:C15H13N3S
    Purity:99.6% - 99.67%
    Color and Shape:Solid
    Molecular weight:267.35
  • MBX-2982

    CAS:
    <p>MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.</p>
    Formula:C22H24N8OS
    Purity:98% - 99.96%
    Color and Shape:Solid
    Molecular weight:448.54
  • cangrelor tetrasodium

    CAS:
    <p>Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent antiplatelet effects.</p>
    Formula:C17H21Cl2F3N5Na4O12P3S2
    Purity:98.51% - 98.6%
    Color and Shape:Solid
    Molecular weight:864.29
  • Adrenorphin 3TFA(88377-68-8(free base))


    <p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>
    Formula:C50H72N15O15S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1326.26
  • Nestoron

    CAS:
    <p>Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).</p>
    Formula:C23H30O4
    Purity:99.48% - 99.83%
    Color and Shape:Solid
    Molecular weight:370.48
  • Isoflupredone Acetate

    CAS:
    <p>Isoflupredone Acetate is a corticosteroid with the activity of topical anti-inflammatory.</p>
    Formula:C23H29FO6
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:420.47
  • Eprosartan Mesylate

    CAS:
    <p>Eprosartan Mesylate (SKF-108566J) is a competitive and reversible Angiotensin II Receptor Blocker.</p>
    Formula:C23H24N2O4S·CH4O3S
    Purity:99.72% - 99.93%
    Color and Shape:A White To Off- White Powder
    Molecular weight:520.62
  • PW0787

    CAS:
    <p>PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).</p>
    Formula:C23H20F4N4O2
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:460.42
  • EST73502 HCl

    CAS:
    <p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>
    Formula:C19H27ClF2N2O2
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:388.88
  • Orphanin FQ(1-11) acetate(178249-41-7 free base)


    <p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>
    Formula:C51H79N15O16
    Purity:95.54%
    Color and Shape:Solid
    Molecular weight:1158.26
  • BMS986188

    CAS:
    <p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>
    Formula:C30H31BrO4
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:535.47
  • MS21570

    CAS:
    <p>MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 Nm,that reduces anxiety-like behavior and fear conditioning in mice.</p>
    Formula:C10H11N3S2
    Purity:97.79%
    Color and Shape:Solid
    Molecular weight:237.34
  • b-Casomorphin (1-3) Acetate


    <p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>
    Formula:C25H31N3O7
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:485.53
  • Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-

    CAS:
    <p>Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.</p>
    Formula:C18H18O3
    Purity:99.85% - 99.96%
    Color and Shape:Solid
    Molecular weight:282.33
  • DAMGO

    CAS:
    <p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>
    Formula:C26H35N5O6
    Purity:98.83% - 99.92%
    Color and Shape:Solid
    Molecular weight:513.59