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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • Valsartan-d9

    CAS:
    <p>Valsartan D9: deuterium-labeled, angiotensin II receptor antagonist, treats hypertension &amp; heart failure.</p>
    Formula:C24H29N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.57
  • Valsartan Ethyl Ester

    CAS:
    <p>Valsartan Ethyl Ester, an impurity in Valsartan, treats hypertension and heart failure by blocking angiotensin II receptors.</p>
    Formula:C26H33N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.57
  • Azilsartan-d5

    CAS:
    <p>Azilsartan (TAK-536) D5 is the deuterium-labeled Azilsartan. Azilsartan is a specific antagonist of the angiotensin II type 1 receptor.</p>
    Formula:C25H20N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.48
  • 5β-Dihydroprogesterone

    CAS:
    <p>5β-Dihydroprogesterone (5β-DHP) is a progesterone receptor agonist and metabolite of progesterone .1,2It is formed from progesterone by 5β-reductase.25β-DHP</p>
    Formula:C21H32O2
    Color and Shape:Solid
    Molecular weight:316.485
  • ML334

    CAS:
    <p>ML334 (LH601A) is an NRF2 activator that inhibits cardiac fibroblast activation and proliferation ameliorating myocardial infarction-induced cardiac fibrosis.</p>
    Formula:C26H26N2O5
    Purity:98.06% - 98.06%
    Color and Shape:Solid
    Molecular weight:446.49
  • NQO1 substrate

    CAS:
    <p>NQO1 substrate is a highly potent NQO1 substrate with potential antitumor activity for leukemia research.</p>
    Formula:C13H2F2N4O
    Purity:98.02% - 98.02%
    Color and Shape:Solid
    Molecular weight:268.18
  • Hydrocortisone cypionate

    CAS:
    <p>Hydrocortisone cypionate is a corticosteroid ester and synthetic glucocorticoid corticosteroid.</p>
    Formula:C29H42O6
    Color and Shape:Solid
    Molecular weight:486.64
  • AVE 0991 sodium salt

    CAS:
    <p>AVE 0991, a nonpeptide, oral Mas agonist, binds [125I]-Ang-(1-7) with IC50 of 21±35 nM.</p>
    Formula:C29H31N4NaO5S2
    Color and Shape:Solid
    Molecular weight:602.7
  • Vanilpyruvic acid

    CAS:
    <p>Vanillylpyruvic acid is a phenylpyruvic acid derivative applicable in biochemical experiments and drug synthesis research.</p>
    Formula:C10H10O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:210.18
  • GW-1100

    CAS:
    <p>GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic diseases.</p>
    Formula:C27H25FN4O4S
    Purity:97.01%
    Color and Shape:Solid
    Molecular weight:520.58
  • (Rac)-PF-998425

    CAS:
    <p>(Rac)-PF-998425: nonsteroidal AR antagonist, potent &amp; selective, IC50: 26 nM (binding), 90 nM (cellular), potential for androgenetic alopecia study.</p>
    Formula:C14H14F3NO
    Color and Shape:Solid
    Molecular weight:269.267
  • Betamethasone acetate

    CAS:
    <p>Betamethasone acetate, the 21-acetate ester of betamethasone, is a synthetic glucocorticoid corticosteroid and a corticosteroid ester.</p>
    Formula:C24H31FO6
    Color and Shape:Solid
    Molecular weight:434.50
  • Leelamine hydrochloride

    CAS:
    <p>Leelamine hydrochloride, a pine bark extract, inhibits androgen receptor and CB1, reducing lipid synthesis in prostate cancer.</p>
    Formula:C20H32ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.93
  • Fenarimol

    CAS:
    <p>Fenarimol, a pyrimidine-type fungicide, exhibits potent inhibitory activity against BR biosynthesis.</p>
    Formula:C17H12Cl2N2O
    Color and Shape:Solid
    Molecular weight:331.2
  • TA 0910 acid-type

    CAS:
    <p>TA 0910 acid-type is a metabolite of TA 0910. TA-0910 is a metabolically stable analog of thyrotropin-releasing hormone.</p>
    Formula:C17H22N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.39
  • Hydrocortisone buteprate

    CAS:
    <p>Hydrocortisone buteprate is a medium-potent, non-halogenated double-ester of hydrocortisone with a highly favorable benefit-to-risk ratio for inflammatory skin disorders.</p>
    Formula:C28H40O7
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:488.61
  • Loperamide phenyl

    CAS:
    <p>Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.</p>
    Formula:C35H37ClN2O2
    Color and Shape:Solid
    Molecular weight:553.14
  • AMG7703

    CAS:
    <p>AMG7703 is a bioactive chemical.</p>
    Formula:C14H15ClN2OS
    Color and Shape:Solid
    Molecular weight:294.8
  • Diflorasone Diacetate

    CAS:
    <p>Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.</p>
    Formula:C26H32F2O7
    Color and Shape:Crystals
    Molecular weight:494.53
  • Dihydromunduletone

    CAS:
    <p>Dihydromunduletone (DHM) is an adhesion G protein-coupled receptor (aGPCR) antagonist inhibits GPR56 and GPR114/ADGRG5, which have similar tethered agonists.</p>
    Formula:C25H28O6
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:424.49
  • VTP-27999 Hydrochloride

    CAS:
    <p>VTP-27999 Hcl is an alkyl amine Renin inhibitor; VTP-27999 is useful for Hypertension and End-Organ Diseases.<br><br>IC50 value:<br><br>Target: Renin</p>
    Formula:C26H42Cl2N4O5
    Color and Shape:Solid
    Molecular weight:561.55
  • Olmesartan lactone impurity

    CAS:
    <p>Olmesartan lactone impurity, a cyclic ester from Olmesartan, aids in hypertension research as an AT1R blocker.</p>
    Formula:C24H24N6O2
    Color and Shape:Solid
    Molecular weight:428.496
  • Enalaprilat

    CAS:
    <p>Enalaprilat (Enalapril acid) is an ACE inhibitor used in the study of cardiovascular disease.</p>
    Formula:C18H24N2O5
    Purity:97.28%
    Color and Shape:Solid
    Molecular weight:348.39
  • Losartan (D4 Carboxylic Acid)

    CAS:
    <p>Losartan D4 Carboxylic Acid is the deuterium labeled Losartan, which is an angiotensin II receptor antagonist.</p>
    Formula:C22H21ClN6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.92
  • Dienestrol diacetate

    CAS:
    <p>Dienestrol diacetate, a derivative of the synthetic non-steroid phenolic compound, DIENESTROL, exhibits estrogenic activities.</p>
    Formula:C22H22O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.41
  • Pamoic acid disodium

    CAS:
    <p>Pamoic acid disodium is a GPR35 agonist.</p>
    Formula:C23H16NaO6
    Purity:99.73%
    Color and Shape:Yellow Powder
    Molecular weight:411.36
  • 2-Bromoestradiol

    CAS:
    <p>2-Bromoestradiol, an estrogen 2-hydroxylase inhibitor, reduces the irreversible binding of radiolabeled estradiol metabolite(s) to microsomal proteins [1].</p>
    Formula:C18H23BrO2
    Color and Shape:Solid
    Molecular weight:351.28
  • DL-Cystine

    CAS:
    <p>DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .</p>
    Formula:C6H12N2O4S2
    Color and Shape:Solid
    Molecular weight:240.3
  • Desoxycorticosterone pivalate

    CAS:
    <p>DOCP, a mineralocorticoid, treats dogs with adrenal insufficiency.</p>
    Formula:C26H38O4
    Color and Shape:Solid
    Molecular weight:414.58
  • AC-186

    CAS:
    <p>AC-186 is an ERβ agonist with neuroprotective activity for the study of Parkinson's disease.</p>
    Formula:C18H17F3O
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:306.32
  • Monomethyl fumarate-d3

    CAS:
    <p>Monomethyl fumarate D3 is a deuterium labeled Monomethyl fumarate.</p>
    Formula:C5H6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:133.12
  • Trans-Diethyl-1,1,1',1'-Stilbestrol-3,3',5,5'-d8

    CAS:
    <p>Trans-Diethyl-1,1,1',1'-Stilbestrol-3,3',5,5'-d8 is a deuterated compound of Trans-Diethyl-Stilbestrol. Trans-Diethyl-Stilbestrol has a CAS number of 56-53-1. Diethylstilbestrol is used in the treatment of menopausal and postmenopausal disorders.</p>
    Formula:C18H12D8O2
    Color and Shape:Solid
    Molecular weight:276.40
  • Dehydroepiandrosterone-d2

    CAS:
    <p>Dehydroepiandrosterone-d2 is a deuterated compound of Dehydroepiandrosterone.</p>
    Formula:C19H26D2O2
    Color and Shape:Solid
    Molecular weight:290.44
  • MK-0773

    CAS:
    <p>MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.</p>
    Formula:C27H34FN5O2
    Purity:98.38% - 99.14%
    Color and Shape:Solid
    Molecular weight:479.59
  • 17β-Estradiol-2,4-d2

    CAS:
    <p>17β-Estradiol-2,4-d2 is a deuterated compound of 17β-Estradiol. 17β-Estradiol has a CAS number of 50-28-2. Estradiol is an Estrogen. The mechanism of action of estradiol is as an Estrogen Receptor Agonist.</p>
    Formula:C18H22D2O2
    Color and Shape:Solid
    Molecular weight:274.39
  • (R,S)-Ivosidenib

    CAS:
    <p>(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .</p>
    Formula:C28H22ClF3N6O3
    Color and Shape:Solid
    Molecular weight:582.96
  • BAN ORL 24 dihydrochloride

    CAS:
    <p>BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.</p>
    Formula:C27H37Cl2N3O2
    Purity:95.03%
    Color and Shape:Solid
    Molecular weight:506.51
  • Azilsartan mepixetil

    CAS:
    <p>Azilsartan mepixetil: potent, long-acting angiotensin II blocker, safely lowers blood pressure, protects heart and kidneys.</p>
    Formula:C36H34N6O8
    Color and Shape:Solid
    Molecular weight:678.702
  • BMS-986121

    CAS:
    <p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>
    Formula:C15H9Cl2N3O2S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:366.22
  • Bazedoxifene

    CAS:
    <p>Bazedoxifene is an orally active SERM against ERα and ERβ and inhibits IL-6/GP130, applied in postmenopausal osteoporosis and pancreatic cancer research.</p>
    Formula:C30H34N2O3
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:470.61
  • Atosiban

    CAS:
    <p>Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.</p>
    Formula:C43H67N11O12S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:994.19
  • CGP-42112

    CAS:
    <p>CGP-42112 is an agonist of the Angiotensin-II subtype 2 receptor (AT2 R).</p>
    Formula:C52H69N13O11
    Color and Shape:White Solid
    Molecular weight:1052.18
  • YE 120

    CAS:
    <p>YE 120 is a GPR35 agonist.</p>
    Formula:C16H9Cl2N3O
    Purity:99.59% - 99.81%
    Color and Shape:Solid
    Molecular weight:330.17
  • GDC-0927

    CAS:
    <p>GDC-0927 is a novel,non-steroidal, potent, orally bioavailable, selective estrogen receptor antagonist.</p>
    Formula:C28H28FNO4
    Color and Shape:Solid
    Molecular weight:461.52
  • Alvimopan dihydrate (LY246736 dihydrate)

    CAS:
    <p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>
    Formula:C25H36N2O6
    Color and Shape:Solid
    Molecular weight:460.56
  • TUG-770

    CAS:
    <p>TUG-770 is a highly potent agonist of free fatty acid receptor 1 (FFA1/GPR40, EC50: 6 nM for hFFA1).</p>
    Formula:C19H14FNO2
    Purity:97.6%
    Color and Shape:Solid
    Molecular weight:307.32
  • Prednisolone valerate acetate

    CAS:
    <p>Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.</p>
    Formula:C28H38O7
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:486.6
  • Candesartan-d4

    CAS:
    <p>Candesartan D4 is the deuterium labeled Candesartan. Candesartan is an antagonist of angiotensin II receptor.</p>
    Formula:C24H20N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.48
  • ARD-1676

    CAS:
    <p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>
    Formula:C44H46ClN7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:788.33
  • Olmesartan-d4

    CAS:
    <p>Olmesartan D4 is the deuterium labeled Olmesartan. Olmesartan is an antagonist of angiotensin II receptor (AT1R) used to treat high blood pressure.</p>
    Formula:C24H26N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:450.53
  • MS 15203

    CAS:
    <p>MS 15203 is a GPR171 agonist that reduces chronic neuropathic and inflammatory pain in male mice.</p>
    Formula:C12H11NO5
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:249.22
  • Beclomethasone 17-propionate

    CAS:
    <p>Beclomethasone 17-propionate is the active metabolite of BDP. As a GR agonist, 17-BMP inhibits the production of pro-inflammatory cytokines.</p>
    Formula:C25H33ClO6
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:464.98
  • Estradiol valerate

    CAS:
    <p>β-estradiol 17-valerate (EV) is a synthetic estrogen. In hormone replacement therapy drugs, it is widely used in combination with other steroid hormones.</p>
    Formula:C23H32O3
    Purity:99.11% - 99.9%
    Color and Shape:Na
    Molecular weight:356.51
  • Endomorphin 2 TFA

    CAS:
    <p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>
    Formula:C34H38F3N5O7
    Color and Shape:Solid
    Molecular weight:685.69
  • PD 123319 ditrifluoroacetate

    CAS:
    <p>PD 123319 ditrifluoroacetate is a selective non-peptide AT2 receptor antagonist with IC50 of 34 nM.</p>
    Formula:C35H34F6N4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:736.66
  • Taltirelin

    CAS:
    <p>Taltirelin (TA-0910) is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in</p>
    Formula:C17H23N7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.41
  • Angiotensin II (3-8), human

    CAS:
    <p>Angiotensin II (3-8), human is a less effective agonist at the angiotensin AT1 receptor.</p>
    Color and Shape:Solid
  • Rezvilutamide

    CAS:
    <p>Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and has antitumor activity.</p>
    Formula:C22H20F3N3O4S
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:479.47
  • D4-abiraterone

    CAS:
    <p>D4-abiraterone is the active metabolite of abiraterone.Δ4-Abiraterone is a inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.</p>
    Formula:C24H29NO
    Purity:99.75% - 99.8%
    Color and Shape:Solid
    Molecular weight:347.49
  • Endoxifen Z-isomer hydrochloride

    CAS:
    <p>Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.</p>
    Formula:C25H28ClNO2
    Color and Shape:Solid
    Molecular weight:409.95
  • Protirelin

    CAS:
    <p>Protirelin (Thyroliberin) is a tripeptide that stimulates the release of thyrotropin and prolactin.</p>
    Formula:C16H22N6O4
    Purity:99.76%
    Color and Shape:White Or Almost White Powder
    Molecular weight:362.38
  • Asimadoline

    CAS:
    <p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>
    Formula:C27H30N2O2
    Color and Shape:Solid
    Molecular weight:414.54
  • AZD1979

    CAS:
    <p>AZD1979 is a highly potent MCHR1 (Melanin-concentrating hormone receptor 1) antagonist , CNS exposure and insulin sensitivity in steady-state model assessments,</p>
    Formula:C25H26N4O5
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:462.5
  • Apalutamide-13C-d3


    <p>Apalutamide-13C-d3 is a 13C and 2H labeled Apalutamide. Apalutamide is an androgen receptor (AR) antagonist, used in research on prostate diseases.</p>
    Formula:CC20H12F4N5O2SD3
    Color and Shape:Solid
    Molecular weight:481.45
  • Zearalanone

    CAS:
    <p>Zearalenone is a nonsteroidal estrogenic mycotoxin produced by Fusarium species, which colonizes several grains.</p>
    Formula:C18H24O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.38
  • GPR40 agonist 6

    CAS:
    <p>GPR40 agonist 6 (Compound 7a) is a potent and selective agonist of free fatty acid receptor 1 ( FFAR1 or GPR40 ) with an EC 50 of 0.058 μM against GPR40 [1].</p>
    Formula:C20H19NO4
    Color and Shape:Solid
    Molecular weight:337.37
  • ERα degrader-2

    CAS:
    <p>ERα degrader-2 is an estrogen receptor (SERD) degrader with anticancer activity that inhibits ERα for the prevention and treatment of HER-positive breast canc</p>
    Formula:C29H27F3N2O2
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:492.53
  • ZQ-16

    CAS:
    <p>ZQ-16 is a potent GPR84 agonist (EC50=0.213 μM) activating multiple signaling pathways.</p>
    Formula:C10H16N2O2S
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:228.31
  • GPR41 agonist-1

    CAS:
    <p>GPR41 agonist-1 is a GPR41 agonist, used for studying metabolic diseases such as diabetes and obesity.</p>
    Formula:C24H23N3O4
    Purity:98.40%
    Color and Shape:Solid
    Molecular weight:417.46
  • Porcine dynorphin A(1-13)

    CAS:
    <p>Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.</p>
    Formula:C75H126N24O15
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1603.95
  • GPR30 agonist-1

    CAS:
    <p>GPR30 agonist-1 is a compound that acts as an agonist for G protein-coupled receptor 30 (GPR30), inducing vasorelaxation.</p>
    Formula:C19H17BrFNO
    Color and Shape:Solid
    Molecular weight:374.253
  • Desoximetasone

    CAS:
    <p>Desoximetasone (Topicort) is a topical corticosteroid for treating skin conditions like rashes.</p>
    Formula:C22H29FO4
    Purity:99.06% - 99.89%
    Color and Shape:Solid
    Molecular weight:376.46
  • Halobetasol propionate

    CAS:
    <p>Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.</p>
    Formula:C25H31ClF2O5
    Purity:99.89%
    Color and Shape:Distributed As 0 05% Ointment
    Molecular weight:484.96
  • Saralasin acetate(34273-10-4 free base)

    CAS:
    <p>Saralasin acetate is a Non-selective angiotensin II antagonist.</p>
    Formula:C44H71N13O13
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:990.11
  • Nafoxidine HCl(1845-11-0 Free base)

    CAS:
    <p>Nafoxidine is a partial estrogen antagonist.</p>
    Formula:C29H32ClNO2
    Color and Shape:Solid
    Molecular weight:462.03
  • Harman hydrochloride

    CAS:
    <p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>
    Formula:C12H11ClN2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:218.68
  • A 779 TFA(159432-28-7 free base)


    <p>A 779 TFA is a potent antagonist of angiotensin-(1-7) receptor.</p>
    Formula:C41H61F3N12O13
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:987.01
  • AL 082D06

    CAS:
    <p>AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.</p>
    Formula:C23H24ClN3O2
    Purity:99.05% - 99.06%
    Color and Shape:Solid
    Molecular weight:409.91
  • 2,4'-Dihydroxybenzophenone

    CAS:
    <p>2,4'-Dihydroxybenzophenone can effectively protect C57BL/6J mice from APAP-induced hepatotoxicity.</p>
    Formula:C13H10O3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:214.22
  • Novokinin acetate


    <p>Novokinin acetate binds AT2 receptor (Ki=7 nM); antihypertensive effect blocked by PD123319.</p>
    Formula:C41H65N11O9
    Purity:99.37%
    Color and Shape:Soild
    Molecular weight:856.02
  • Elacestrant dihydrochloride

    CAS:
    <p>Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for</p>
    Formula:C30H40Cl2N2O2
    Purity:99.59% - >99.99%
    Color and Shape:Solid
    Molecular weight:531.56
  • Eprotirome

    CAS:
    <p>Eprotirome (KB2115), a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.</p>
    Formula:C18H17Br2NO5
    Purity:98.42% - 98.56%
    Color and Shape:Solid
    Molecular weight:487.14
  • SNG-1153

    CAS:
    <p>SNG-1153 is a estrogen receptor ER-alpha36 modulator.</p>
    Formula:C21H17F3O5
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:406.35
  • EST73502 hydrochloride

    CAS:
    <p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>
    Formula:C19H27ClF2N2O2
    Color and Shape:Solid
    Molecular weight:388.88
  • S-23

    CAS:
    <p>S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (</p>
    Formula:C18H13ClF4N2O3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:416.75
  • Abaloparatide TFA


    <p>Abaloparatide TFA (BIM 44058 TFA) is a parathyroid hormone-related protein (PTHrP) analog drug used to treat osteoporosis like the related drug teriparatide.</p>
    Formula:C176H301N56F3O51
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:4074.61
  • Teriparatide acetate

    CAS:
    <p>Teriparatide acetate (Forteo), a synthetic parathyroid hormone, treats osteoporosis by favoring bone growth with a 2 nM IC50.</p>
    Formula:C183H295N55O53S2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:4177.83
  • Spinorphin

    CAS:
    <p>Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.</p>
    Formula:C45H64N8O10
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:877
  • Ciclesonide

    CAS:
    <p>Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.</p>
    Formula:C32H44O7
    Purity:99.89% - >99.99%
    Color and Shape:Solid
    Molecular weight:540.69
  • Chlorotrianisene

    CAS:
    <p>Chlorotrianisene, a synthetic SERM, is orally active, lipophilic, and has estrogenic and antiestrogenic effects.</p>
    Formula:C23H21ClO3
    Purity:98.88% - 99.03%
    Color and Shape:Crystals From Methanol Physical Description Small White Crystals Or White Powder Softens At 226°F Odorless (Ntp 1992)
    Molecular weight:380.86
  • VTP-27999 TFA

    CAS:
    <p>VTP-27999 TFA is an inhibitor of Renin (IC50 : 0.47 nM).</p>
    Formula:C28H42ClF3N4O7
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:639.1
  • Fevipiprant

    CAS:
    <p>Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.</p>
    Formula:C19H17F3N2O4S
    Purity:99.32% - 99.59%
    Color and Shape:Solid
    Molecular weight:426.41
  • Beclometasone dipropionate monohydrate

    CAS:
    <p>Beclometasone dipropionate monohydrate, precursor to oral glucocorticoid for inflammation and asthma research.</p>
    Formula:C28H39ClO8
    Color and Shape:Solid
    Molecular weight:539.06
  • Ospemifene

    CAS:
    <p>Ospemifene (FC-1271a) is a new selective non-hormonal estrogen receptor modulator (SERM) that is used for the treatment of moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause. FDA approved on February 26, 2013.</p>
    Formula:C24H23ClO2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:378.89
  • PZM21

    CAS:
    <p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>
    Formula:C19H27N3O2S
    Purity:99.93% - >99.99%
    Color and Shape:Solid
    Molecular weight:361.5
  • BW-180C

    CAS:
    <p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>
    Formula:C29H39N5O7
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:569.65
  • Nociceptin

    CAS:
    <p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>
    Formula:C79H129N27O22
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:1809.04
  • Fluorometholone Acetate

    CAS:
    <p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>
    Formula:C24H31FO5
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:418.50
  • Nandrolone phenylpropionate

    CAS:
    <p>Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis</p>
    Formula:C27H34O3
    Purity:99.2% - 99.46%
    Color and Shape:White Or Milky Crystalline Powder
    Molecular weight:406.56
  • ADL-5747 (HCl)

    CAS:
    <p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>
    Formula:C24H29ClN2O3
    Color and Shape:Solid
    Molecular weight:428.95
  • SNAP 94847 hydrochloride

    CAS:
    <p>SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)</p>
    Formula:C29H33ClF2N2O2
    Purity:99.85% - >99.99%
    Color and Shape:Solid
    Molecular weight:515.03
  • Brilanestrant

    CAS:
    <p>Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).</p>
    Formula:C26H20ClFN2O2
    Purity:99.07% - 99.17%
    Color and Shape:Solid Powder
    Molecular weight:446.9
  • PHTPP

    CAS:
    <p>PHTPP is a selective ERβ antagonist.</p>
    Formula:C20H11F6N3O
    Purity:98.81% - 99.57%
    Color and Shape:Solid
    Molecular weight:423.31
  • AR 231453

    CAS:
    <p>Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.</p>
    Formula:C21H24FN7O5S
    Purity:99.31% - 99.34%
    Color and Shape:Solid
    Molecular weight:505.52
  • Iprodione

    CAS:
    <p>Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.</p>
    Formula:C13H13Cl2N3O3
    Purity:98.82%
    Color and Shape:Colorless Crystals Cream To Colorless Odorless Powder
    Molecular weight:330.17
  • BNP (1-32), human

    CAS:
    <p>BNP (1-32), human is a brain natriuretic peptide</p>
    Formula:C143H244N50O42S4
    Purity:98.52%
    Color and Shape:White Powder
    Molecular weight:3464.04
  • Deltorphin I

    CAS:
    <p>Deltorphin I is an agonist of δ-opioid receptor.</p>
    Formula:C37H52N8O10
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:768.86
  • Diflorasone

    CAS:
    <p>Diflorasone is a synthetic glucocorticoid. It has anti-inflammatory and immunosuppressive effects by acting on gene expression.</p>
    Formula:C22H28F2O5
    Purity:99.02% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.45
  • BTB06584

    CAS:
    <p>BTB06584: IF1-dependent F1 Fo-ATPase inhibitor; novel AHAS inhibitor targeting MTB.</p>
    Formula:C19H12ClNO6S
    Purity:97.63% - ≥95%
    Color and Shape:Solid
    Molecular weight:417.82
  • Ulipristal acetate

    CAS:
    <p>Ulipristal acetate (CDB-2914) is an oral selective progesterone modulator used for emergency contraception and suppressing uterine growths.</p>
    Formula:C30H37NO4
    Purity:98.83% - 99.94%
    Color and Shape:Solid
    Molecular weight:475.62
  • FH1

    CAS:
    <p>FH1 (NSC-12407) (BRD-K4477), a small molecule, enhances the functions of hepatocytes and promotes differentiation hepatocytes derived by iPS.</p>
    Formula:C17H18N2O2
    Purity:98% - 99.64%
    Color and Shape:Solid
    Molecular weight:282.34
  • Angiotensin III, human, mouse

    CAS:
    <p>Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA))(3TFA) is an endogenous angiotensin II receptor (AT2R) agonist(IC50s of 0.648 nM).</p>
    Formula:C46H66N12O9
    Purity:98.44%
    Color and Shape:Solid
    Molecular weight:931.09
  • Broparestrol (E)-

    CAS:
    <p>Broparestrol (E)- has antifertility activity and is a potent inhibitor of rodent mammary tumorigenesis.</p>
    Formula:C22H19Br
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:363.29
  • MK-6892

    CAS:
    <p>MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM).</p>
    Formula:C19H22N4O5
    Purity:99.01% - 99.67%
    Color and Shape:Solid
    Molecular weight:386.4
  • Fasiglifam

    CAS:
    <p>Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.</p>
    Formula:C29H32O7S
    Purity:99.82% - 99.9%
    Color and Shape:Solid
    Molecular weight:524.63
  • L-Thyroxine sodium

    CAS:
    <p>L-Thyroxine sodium (LT4 sodium), the major hormone derived from the thyroid gland, is the agonist of Thyroid hormone receptor alpha and beta.</p>
    Formula:C15H10I4NO4·Na
    Purity:98.74%
    Color and Shape:Yellowish To Buff-Colored Amorphous Powder Solid
    Molecular weight:798.85
  • β-Estradiol 17-hemisuccinate

    CAS:
    <p>beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells.</p>
    Formula:C22H28O5
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:372.45
  • GW9508

    CAS:
    <p>GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.</p>
    Formula:C22H21NO3
    Purity:97.89% - 99.19%
    Color and Shape:Solid
    Molecular weight:347.41
  • VPC-13566

    CAS:
    <p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>
    Formula:C18H14N2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:258.32
  • Temocapril hydrochloride

    CAS:
    <p>Temocapril hydrochloride (CS-622 HCl), the hydrochloride of Temocapril, is a long-acting ACE inhibitor used for the therapy of hypertension.</p>
    Formula:C23H28N2O5S2·HCl
    Purity:99.26% - 99.48%
    Color and Shape:White Solid Powder
    Molecular weight:513.07
  • Aviptadil Acetate

    CAS:
    <p>Aviptadil Acetate (Vasoactive Intestinal Peptide acetate salt) induces pulmonary vasodilation and inhibits the proliferation of vascular SMCs.</p>
    Formula:C147H238N44O42S·C2H4O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:3385.9
  • DIM-C-pPhOCH3

    CAS:
    <p>DIM-C-pPhOCH3 (C-DIM5) is a Nerve Growth Factor-Induced Bα (NGFI-Bα, Nur77) agonist</p>
    Formula:C24H20N2O
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:352.43
  • Naloxegol (NKTR-118)

    CAS:
    <p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>
    Formula:C34H53NO11
    Color and Shape:Solid
    Molecular weight:651.78
  • Olmesartan

    CAS:
    <p>Olmesartan (RNH 6270) is an Angiotensin II Type I receptor antagonist.</p>
    Formula:C24H26N6O3
    Purity:91.89% - 99.81%
    Color and Shape:White To Beige Solid Solid
    Molecular weight:446.5
  • GR 89696 free base

    CAS:
    <p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>
    Formula:C19H25Cl2N3O3
    Color and Shape:Solid
    Molecular weight:414.33
  • 4-Hydroxytamoxifen

    CAS:
    <p>4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency.</p>
    Formula:C26H29NO2
    Purity:99.37% - 99.93%
    Color and Shape:Solid
    Molecular weight:387.51
  • BMS986188

    CAS:
    <p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>
    Formula:C30H31BrO4
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:535.47
  • Estradiol hemihydrate

    CAS:
    <p>Estradiol hemihydrate: major female hormone, boosts neural differentiation, studied for cancer and neurodegenerative disease.</p>
    Formula:C18H26O3
    Color and Shape:Solid
    Molecular weight:281.39
  • Nociceptin (1-7) acetate


    <p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>
    Formula:C31H41N7O9
    Purity:98.92%
    Color and Shape:Soild
    Molecular weight:655.7
  • [Leu5]-Enkephalin, amide acetate


    <p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>
    Formula:C30H42N6O8
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:614.69
  • Isoflupredone Acetate

    CAS:
    <p>Isoflupredone Acetate is a corticosteroid with the activity of topical anti-inflammatory.</p>
    Formula:C23H29FO6
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:420.47
  • WAY-200070

    CAS:
    <p>WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).</p>
    Formula:C13H8BrNO3
    Purity:99.45% - 99.75%
    Color and Shape:Solid
    Molecular weight:306.11
  • Dynorphin A 1-10 acetate(79994-24-4 free base)


    <p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>
    Formula:C59H95N19O14
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:1294.53
  • DPC AJ1951 acetate


    <p>DPC-AJ1951 acetate: 14-amino acid peptide, potent PTH/PPR agonist, tested for bone resorption activity ex vivo/in vivo.</p>
    Formula:C78H131N23O21
    Purity:96.63%
    Color and Shape:Solid
    Molecular weight:1727.02
  • Pipendoxifene

    CAS:
    <p>Pipendoxifene (ERA-923) is an antiestrogen that blocks ER-alpha and inhibits MCF-7 breast cancer cell growth, effective even when tamoxifen-resistant.</p>
    Formula:C29H32N2O3
    Color and Shape:Solid
    Molecular weight:456.58
  • Orphanin FQ(1-11) acetate(178249-41-7 free base)


    <p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>
    Formula:C51H79N15O16
    Purity:95.54%
    Color and Shape:Solid
    Molecular weight:1158.26
  • Hemorphin-7 acetate(152685-85-3 free base)


    <p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>
    Formula:C51H68N12O13
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:1057.16
  • Urotensin II, mouse acetate (9047-55-6 free base)


    <p>Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.</p>
    Formula:C64H88N14O19S2
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:1421.61
  • Alacepril

    CAS:
    <p>Alacepril (DU-1219) is a relatively novel angiotensin-converting enzyme inhibitor, used as an antihypertensive</p>
    Formula:C20H26N2O5S
    Purity:97.78%
    Color and Shape:Solid
    Molecular weight:406.5
  • N-terminally acetylated Leu-enkephalin


    <p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>
    Formula:C30H39N5O8
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:597.66
  • Methylnaltrexone bromide

    CAS:
    <p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>
    Formula:C21H26BrNO4
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:436.35
  • EST73502 HCl

    CAS:
    <p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>
    Formula:C19H27ClF2N2O2
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:388.88
  • PF3274167

    CAS:
    <p>PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.</p>
    Formula:C19H19ClFN5O3
    Purity:99.67% - 99.88%
    Color and Shape:Solid
    Molecular weight:419.84
  • AH-7614

    CAS:
    <p>AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.</p>
    Formula:C20H17NO3S
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:351.42
  • ms48107

    CAS:
    <p>MS48107 enhances GPR68, crosses BBB in mice, and is selective over related proton GPCRs, transporters, and hERG channels.</p>
    Formula:C23H20FN5O2
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:417.44
  • Eprosartan Mesylate

    CAS:
    <p>Eprosartan Mesylate (SKF-108566J) is a competitive and reversible Angiotensin II Receptor Blocker.</p>
    Formula:C23H24N2O4S·CH4O3S
    Purity:99.72% - 99.93%
    Color and Shape:A White To Off- White Powder
    Molecular weight:520.62
  • DY131

    CAS:
    <p>DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.</p>
    Formula:C18H21N3O2
    Purity:98.65% - 99.66%
    Color and Shape:Solid
    Molecular weight:311.38
  • panomifene

    CAS:
    <p>Panomiphene (Gyki-13504, EGIS-5650) is an anti-estrogen drug that is a tamoxifen (TMX) analogue.</p>
    Formula:C25H24F3NO2
    Color and Shape:Solid
    Molecular weight:427.46
  • CLP-3094

    CAS:
    <p>CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.</p>
    Formula:C15H13ClN2OS
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:304.79
  • VPC-13163

    CAS:
    <p>VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.</p>
    Formula:C16H14N2
    Purity:98.02%
    Color and Shape:Solid
    Molecular weight:234.3
  • α-Zearalenol

    CAS:
    <p>α-Zearalenol is one of the major metabolites of Zearalenone.</p>
    Formula:C18H24O5
    Purity:90% - 99.72%
    Color and Shape:Solid
    Molecular weight:320.38
  • Apararenone

    CAS:
    <p>Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy.</p>
    Formula:C17H17FN2O4S
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:364.39
  • G15

    CAS:
    <p>G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)</p>
    Formula:C19H16BrNO2
    Purity:98.46% - 98.59%
    Color and Shape:Solid
    Molecular weight:370.24
  • [D-Ala2]leucine-enkephalin

    CAS:
    <p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>
    Formula:C29H39N5O7
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:569.65
  • Ac-RYYRWK-NH2 acetate


    <p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>
    Formula:C51H73N15O11
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:1072.22
  • 6-OAU

    CAS:
    <p>6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.</p>
    Formula:C12H21N3O2
    Purity:98.14% - 99.01%
    Color and Shape:Solid
    Molecular weight:239.31
  • BigLEN (mouse) acetate


    <p>BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 (GPR171), with a Kd of ∼0.5 nM.</p>
    Formula:C80H134N24O24
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1816.07
  • Bisphenol B

    CAS:
    <p>Bisphenol B has a binding affinity for estrogen receptors.</p>
    Formula:C16H18O2
    Purity:97.35% - 99.62%
    Color and Shape:Crystal Or Tan Granules Odorless Slightly Brown Solid
    Molecular weight:242.31
  • H-Val-Pro-Pro-OH

    CAS:
    <p>H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).</p>
    Formula:C15H25N3O4
    Purity:98.23%
    Color and Shape:Solid
    Molecular weight:311.38
  • Palosuran hydrochloride 540769-28-6(free base)


    <p>Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.</p>
    Formula:C25H31ClN4O2
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:454.99
  • Urotensin II (114-124), human acetate


    <p>Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor and agonist for the orphan receptor GPR14.</p>
    Formula:C66H89N13O20S2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1448.63
  • Antide acetate


    <p>Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. </p>
    Formula:C84H112ClN17O16
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:1651.34
  • DAMGO

    CAS:
    <p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>
    Formula:C26H35N5O6
    Purity:98.83% - 99.92%
    Color and Shape:Solid
    Molecular weight:513.59
  • MCOPPB

    CAS:
    <p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>
    Formula:C26H40N4
    Color and Shape:Solid
    Molecular weight:408.62
  • MS21570

    CAS:
    <p>MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 Nm,that reduces anxiety-like behavior and fear conditioning in mice.</p>
    Formula:C10H11N3S2
    Purity:97.79%
    Color and Shape:Solid
    Molecular weight:237.34
  • AS1269574

    CAS:
    <p>AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes.</p>
    Formula:C13H14BrN3O
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:308.17
  • Nafoxidine

    CAS:
    <p>Nafoxidine is an estrogen antagonist that has been used in the treatment of breast cancer.</p>
    Formula:C29H31NO2
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:425.56
  • Apalutamide

    CAS:
    <p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>
    Formula:C21H15F4N5O2S
    Purity:99.03% - 99.91%
    Color and Shape:Solid
    Molecular weight:477.43
  • TC-O 9311

    CAS:
    <p>TC-O 9311 (TCO-9311) is an effective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing human GPR139).</p>
    Formula:C20H19N3O4
    Purity:99.24% - 99.84%
    Color and Shape:Solid
    Molecular weight:365.38
  • 4-CMTB

    CAS:
    <p>4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).</p>
    Formula:C14H15ClN2OS
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:294.8
  • Timapiprant

    CAS:
    <p>Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).</p>
    Formula:C21H17FN2O2
    Purity:97.44% - 99.51%
    Color and Shape:Solid
    Molecular weight:348.37
  • Norgestrel

    CAS:
    <p>Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.</p>
    Formula:C21H28O2
    Purity:99.71% - 99.72%
    Color and Shape:Crystals From Methanol White Crystalline Powder
    Molecular weight:312.45
  • AZD1981

    CAS:
    <p>AZD1981: selective CRTh2 antagonist, IC50 4 nM, 1000x specificity over 340+ enzymes/receptors, tested in asthma and other trials.</p>
    Formula:C19H17ClN2O3S
    Purity:98.87% - 99.67%
    Color and Shape:Solid
    Molecular weight:388.87
  • b-Casomorphin (1-3) Acetate


    <p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>
    Formula:C25H31N3O7
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:485.53
  • MBX-2982

    CAS:
    <p>MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.</p>
    Formula:C22H24N8OS
    Purity:98% - 99.96%
    Color and Shape:Solid
    Molecular weight:448.54
  • Sparsentan

    CAS:
    <p>Sparsentan (DARA-a) is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM,</p>
    Formula:C32H40N4O5S
    Purity:97.94% - 98.69%
    Color and Shape:Solid
    Molecular weight:592.75
  • (Sar¹)-Angiotensin II acetate


    <p>(Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor.</p>
    Formula:C51H75N13O12
    Purity:99.89%
    Color and Shape:Soild
    Molecular weight:1062.22
  • JTC-801

    CAS:
    <p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>
    Formula:C26H25N3O2·HCl
    Purity:99.27% - 99.59%
    Color and Shape:Solid
    Molecular weight:447.96
  • 2-(pentylsulfanyl)pyrimidine-4,6-diol

    CAS:
    <p>2-(pentylsulfanyl)pyrimidine-4,6-diol 是一种新型 GRP84 激动剂。</p>
    Formula:C9H14N2O2S
    Purity:97.58%
    Color and Shape:Solid
    Molecular weight:214.28
  • CVN424

    CAS:
    <p>CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.</p>
    Formula:C24H29F2N5O3
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:473.52
  • Leucylarginylproline

    CAS:
    <p>Leucylarginylproline is an inhibitor of angiotensin-converting enzyme (ACE) (IC50 : 0.27μM).</p>
    Formula:C17H32N6O4
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:384.47
  • [Leu5]-Enkephalin TFA(58822-25-6(free bas))

    CAS:
    <p>[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago</p>
    Formula:C30H38F3N5O9
    Purity:97.03% - 99.78%
    Color and Shape:Solid
    Molecular weight:669.64
  • Gluten Exorphin C

    CAS:
    <p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>
    Formula:C29H45N5O8
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:591.7
  • Tyr-Gly-Gly-Phe-Met-OH

    CAS:
    <p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>
    Formula:C27H35N5O7S
    Purity:≥95%
    Color and Shape:White Lyophilised Solid
    Molecular weight:573.66
  • Osilodrostat phosphate

    CAS:
    <p>Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.</p>
    Formula:C13H13FN3O4P
    Color and Shape:Solid
    Molecular weight:325.23
  • Carbetocin acetate

    CAS:
    <p>Carbetocin acetate is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.</p>
    Formula:C47H73N11O14S
    Purity:98.16% - 99.22%
    Color and Shape:Solid
    Molecular weight:1048.22
  • PSN 375963

    CAS:
    <p>PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.</p>
    Formula:C17H23N3O
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:285.38
  • GSK1292263

    CAS:
    <p>GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.</p>
    Formula:C23H28N4O4S
    Purity:98.34% - 99.53%
    Color and Shape:Solid
    Molecular weight:456.56
  • JNJ-63533054

    CAS:
    <p>JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.</p>
    Formula:C17H17ClN2O2
    Purity:99.71% - 99.88%
    Color and Shape:Solid
    Molecular weight:316.78
  • Zaprinast

    CAS:
    <p>Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist.</p>
    Formula:C13H13N5O2
    Purity:99.73% - 99.77%
    Color and Shape:White To Off White Powder
    Molecular weight:271.27
  • Methylprednisolone succinate

    CAS:
    <p>Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent.</p>
    Formula:C26H34O8
    Purity:98.41% - 99.82%
    Color and Shape:White Or Almost-White Solid Powder
    Molecular weight:474.54
  • XCT790

    CAS:
    <p>XCT790 is a potent, selective and inverse agonist of estrogen-related receptor alpha(ERRα).</p>
    Formula:C23H13F9N4O3S
    Purity:99% - 99.61%
    Color and Shape:Solid
    Molecular weight:596.42
  • Myristyl nicotinate

    CAS:
    <p>Myristyl nicotinate (Tetradecyl nicotinate) is an ester prodrug being developed for delivery of nicotinic acid (NIC) into the skin for prevention of actinic</p>
    Formula:C20H33NO2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:319.48
  • Alvimopan monohydrate

    CAS:
    <p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>
    Formula:C25H34N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.55
  • Delapril hydrochloride

    CAS:
    <p>Delapril HCl (indalapril) is a prodrug forming two ACE inhibitors, blocking angiotensin I-II conversion.</p>
    Formula:C26H33ClN2O5
    Purity:97.18% - 97.45%
    Color and Shape:White Crystalline Powder
    Molecular weight:489.01
  • DJ-V-159

    CAS:
    <p>DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A).</p>
    Formula:C24H12F6N4O2
    Purity:99.85% - 99.96%
    Color and Shape:Solid
    Molecular weight:502.37
  • Kisspeptin-10, human (TFA)(374675-21-5,FREE)


    <p>Kisspeptin-10 TFA: vasoconstrictor, inhibits angiogenesis &amp; metastasis; key in kidney development &amp; osteoblast differentiation via GPR54 &amp; NFATc4/BMP2.</p>
    Formula:C63H83N17O14·C2HF3O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1416.46
  • Adrenorphin 3TFA(88377-68-8(free base))


    <p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>
    Formula:C50H72N15O15S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1326.26
  • AZD9977

    CAS:
    <p>AZD9977 is a novel, selective modulator of mineralocorticoid receptor .</p>
    Formula:C20H18FN3O5
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:399.37
  • Ac-RYYRIK-NH2 acetate


    <p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>
    Formula:C46H74N14O11
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:999.17