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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • Elobixibat hydrate

    CAS:
    <p>Elobixibat hydrate, an IBAT inhibitor, IC50: 0.53 nM (human), 0.13 nM (mouse), 5.8 nM (canine); for CIC research.</p>
    Formula:C36H47N3O8S2
    Color and Shape:Solid
    Molecular weight:713.9
  • Loreclezole

    CAS:
    <p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>
    Formula:C10H6Cl3N3
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:274.53
  • Anthracene-9-carboxylic acid

    CAS:
    <p>Anthracene-9-carboxylic acid is an inhibitor of chloride transport with a moderate to strong inhibitory action on PKA activated cardiac IcI.</p>
    Formula:C15H10O2
    Purity:99.05%
    Color and Shape:Yellow Cystalline Powder
    Molecular weight:222.24
  • FGH10019

    CAS:
    <p>FGH10019 is a novel inhibitor of sterol regulatory element-binding protein (SREBP) ( IC50 :1 μM).</p>
    Formula:C18H19N3O2S2
    Purity:98.93%
    Color and Shape:Solid
    Molecular weight:373.49
  • Evenamide

    CAS:
    <p>Evenamide (NW-3509) is a sodium channel blocker. Which shows efficacy in a broad spectrum of rodent models of psychosis, mania, depression, and aggressiveness.</p>
    Formula:C16H26N2O2
    Purity:96.74% - 99.15%
    Color and Shape:Solid
    Molecular weight:278.39
  • (S)-(-)-5-Fluorowillardiine

    CAS:
    (S)-(-)-5-Fluorowillardiine ((S)-5-Fluorowillardiine) is an AMPA receptor-specific agonist
    Formula:C7H8FN3O4
    Purity:99.69%
    Color and Shape:Off-White Solid
    Molecular weight:217.15
  • A-967079

    CAS:
    <p>A 967079 is a potent, selective, and bioavailable inhibitor of the TRPA1 channel, with IC50 values of 67 and 289 nM for the human and rat isoforms, respectively</p>
    Formula:C12H14FNO
    Purity:98.34% - 99.75%
    Color and Shape:Solid
    Molecular weight:207.24
  • Prilocaine

    CAS:
    <p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>
    Formula:C13H20N2O
    Purity:98.49%
    Color and Shape:Needles Solid
    Molecular weight:220.31
  • Transdermal Peptide Disulfide Acetate


    <p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>
    Formula:C42H68N14O18S2
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:1121.2
  • β-Pompilidotoxin Acetate


    <p>β-Pompilidotoxin Acetate is a wasp venom peptide.</p>
    Formula:C73H128N22O19
    Purity:98.64%
    Color and Shape:Solid
    Molecular weight:1617.93
  • 4-Chlorophenylguanidine hydrochloride

    CAS:
    <p>4-Chlorophenylguanidine hydrochloride is a potent inhibitor of urokinase selectivity.  </p>
    Formula:C7H9Cl2N3
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:206.07
  • HC-030031

    CAS:
    <p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>
    Formula:C18H21N5O3
    Purity:99.69% - ≥95%
    Color and Shape:Solid
    Molecular weight:355.39
  • rac-BHFF

    CAS:
    <p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency &gt;15x, efficacy &gt;149%, has anxiolytic effects, and is orally active.</p>
    Formula:C17H21F3O3
    Purity:99.69% - >99.99%
    Color and Shape:Solid
    Molecular weight:330.34
  • VU6036720 hydrochloride


    <p>VU6036720 hydrochloride inhibits Kir4.1/5.1. channels with 0.24 μM IC50; used in brain and kidney research.</p>
    Formula:C20H23Cl2FN4O2S
    Color and Shape:Solid
    Molecular weight:473.39
  • Flupirtine

    CAS:
    <p>Flupirtine(D 9998) is a selective neuronal potassium channel opener as well as shows properties of NMDA receptor antagonist.</p>
    Formula:C15H17FN4O2
    Color and Shape:Solid
    Molecular weight:304.32
  • Esomeprazole

    CAS:
    Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.
    Formula:C17H19N3O3S
    Purity:97.3%
    Color and Shape:Solid
    Molecular weight:345.42
  • TCN 201

    CAS:
    TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.
    Formula:C21H17ClFN3O4S
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:461.89
  • Epaminurad

    CAS:
    <p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>
    Formula:C14H10Br2N2O3
    Color and Shape:Solid
    Molecular weight:414.05
  • ML335

    CAS:
    <p>ML335 is a selective activator of TREK-1 and TREK-2.</p>
    Formula:C15H14Cl2N2O3S
    Purity:99.73% - 99.79%
    Color and Shape:Solid
    Molecular weight:373.25
  • JNJ-26990990

    CAS:
    "JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."
    Formula:C9H10N2O2S2
    Purity:97.37%
    Color and Shape:Solid
    Molecular weight:242.32
  • Levcromakalim

    CAS:
    <p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>
    Formula:C16H18N2O3
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:286.33
  • Aptiganel hydrochloride

    CAS:
    <p>Aptiganel hydrochloride(Cerestat) is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.</p>
    Formula:C20H22ClN3
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:339.86
  • Felbamate

    CAS:
    Felbamate (W-554) is an Anti-epileptic Agent.
    Formula:C11H14N2O4
    Purity:99% - >99.99%
    Color and Shape:White Powder Solid
    Molecular weight:238.24
  • Ipidacrine

    CAS:
    Ipidacrine (NIK‐247) (NIK‐247) is an Antidementia Agent
    Formula:C12H16N2
    Purity:97.73% - 99.99%
    Color and Shape:Solid
    Molecular weight:188.27
  • PAP-1

    CAS:
    <p>PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).</p>
    Formula:C21H18O5
    Purity:99.35% - 99.75%
    Color and Shape:White Solid
    Molecular weight:350.36
  • ML213

    CAS:
    <p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>
    Formula:C17H23NO
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:257.37
  • Licarbazepine

    CAS:
    <p>Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial</p>
    Formula:C15H14N2O2
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:254.28
  • Phenibut (hydrochloride)

    CAS:
    <p>Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.</p>
    Formula:C10H14ClNO2
    Purity:99.93%
    Color and Shape:White Crystalline Powder
    Molecular weight:215.68
  • Enflurane

    CAS:
    Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.
    Formula:C3H2ClF5O
    Purity:99.64%
    Color and Shape:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As An
    Molecular weight:184.49
  • UBP710

    CAS:
    <p>UBP710 is an effective and selective NMDA receptor modulator.</p>
    Formula:C18H14O2
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:262.3
  • Tiludronate

    CAS:
    <p>Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.</p>
    Formula:C7H9ClO6P2S
    Color and Shape:Solid
    Molecular weight:318.61
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Formula:C22H26ClNO2
    Purity:98.02%
    Color and Shape:Solid
    Molecular weight:371.9
  • Methyl homoveratrate

    CAS:
    <p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>
    Formula:C11H14O4
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:210.23
  • Tricaine methanesulfonate

    CAS:
    <p>Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.</p>
    Formula:C10H15NO5S
    Purity:99.259% - 99.86%
    Color and Shape:White Powder
    Molecular weight:261.30
  • Neramexane HCl

    CAS:
    PAC is a cyclic amine used as a chiral auxiliary in various asymmetric syntheses.
    Formula:C11H24ClN
    Purity:95.00%
    Color and Shape:Solid
    Molecular weight:205.768
  • Pipequaline hydrochloride

    CAS:
    <p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict &amp; anticonvulsant quinoline derivative.</p>
    Formula:C22H25ClN2
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:352.9
  • Tezacaftor

    CAS:
    <p>Tezacaftor (VX661) is a small molecule that can be used as a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) gene function.</p>
    Formula:C26H27F3N2O6
    Purity:98.84% - >99.99%
    Color and Shape:Solid
    Molecular weight:520.5
  • Memantine

    CAS:
    Memantine treats moderate to severe Alzheimer's; it's an amantadine derivative blocking NMDA receptors.
    Formula:C12H21N
    Purity:≥98%
    Color and Shape:White Powder
    Molecular weight:179.3
  • Trans-ACBD

    CAS:
    <p>Trans-ACBD (Trans-1-aminocyclobutane-1,3-dicarboxylic acid) is an effective and specific N-methyl-D-aspartate receptor agonist.</p>
    Formula:C6H9NO4
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:159.14
  • 9-Phenanthrol

    CAS:
    <p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>
    Formula:C14H10O
    Purity:98.48%
    Color and Shape:Solid
    Molecular weight:194.23
  • O4I1

    CAS:
    <p>O4I1 is an effective Oct3/4 inducer.</p>
    Formula:C16H15NO2
    Purity:96.25% - 99.47%
    Color and Shape:Solid
    Molecular weight:253.3
  • AM92016

    CAS:
    <p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>
    Formula:C26H30Cl2N2O6S
    Color and Shape:Solid
    Molecular weight:569.49
  • MK6-83

    CAS:
    <p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>
    Formula:C16H20N2O2S2
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:336.47
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Formula:C18H21ClF3N3O
    Purity:99.03% - 99.95%
    Color and Shape:Solid
    Molecular weight:387.83
  • (S)-(-)-5-Fluorowillardiine hydrochloride

    CAS:
    <p>(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.</p>
    Formula:C7H9ClFN3O4
    Color and Shape:Solid
    Molecular weight:253.62
  • BzATP triethylammonium salt

    CAS:
    <p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>
    Formula:C30H39N6O15P3
    Purity:95% - 99.57%
    Color and Shape:Solid
    Molecular weight:816.59
  • Caroverine hydrochloride

    CAS:
    Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.
    Formula:C22H28ClN3O2
    Purity:98.37% - 98.75%
    Color and Shape:Solid
    Molecular weight:401.9
  • GNE-131

    CAS:
    <p>GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).</p>
    Formula:C23H30N4O3S
    Purity:98.54% - 99.59%
    Color and Shape:Solid
    Molecular weight:442.57
  • XEN907

    CAS:
    <p>XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).</p>
    Formula:C21H21NO4
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:351.4
  • TRPM4-IN-1

    CAS:
    <p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>
    Formula:C15H11Cl2NO4
    Purity:97.22%
    Color and Shape:Solid
    Molecular weight:340.16
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Formula:C4H10N2
    Color and Shape:Solid
    Molecular weight:86.14
  • Esomeprazole magnesium salt

    CAS:
    <p>Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.</p>
    Formula:C17H21MgN3O3S
    Color and Shape:Solid
    Molecular weight:371.74
  • PF 05089771

    CAS:
    <p>PF 05089771 is a Selective inhibitor of Nav1.7 (IC50 = 11 nM) that interacts with the voltage-sensor domain of domain IV.</p>
    Formula:C18H12Cl2FN5O3S2
    Purity:99.03% - 99.42%
    Color and Shape:Solid
    Molecular weight:500.35
  • YHO-13351

    CAS:
    YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.
    Formula:C27H37N3O7S2
    Purity:97.88%
    Color and Shape:Solid
    Molecular weight:579.73
  • Cinacalcet metabolite M4

    CAS:
    <p>Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.</p>
    Formula:C10H12F3N
    Purity:97.13%
    Color and Shape:Solid
    Molecular weight:203.2
  • Pico145

    CAS:
    <p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>
    Formula:C23H20ClF3N4O5
    Purity:99.06%
    Color and Shape:Solid
    Molecular weight:524.88
  • Acecainide hydrochloride

    CAS:
    <p>Acecainide hydrochloride (NAPA) is the major hepatic metabolite of procainamide.Cost-effective and quality-assured.</p>
    Formula:C15H24ClN3O2
    Purity:98.023% - 99.81%
    Color and Shape:Solid
    Molecular weight:313.83
  • Tegoprazan

    CAS:
    <p>Tegoprazan is an orally active, highly selective gastric H+/K+-ATPase inhibitor.Cost-effective and quality-assured.</p>
    Formula:C20H19F2N3O3
    Purity:98.22%
    Color and Shape:Solid
    Molecular weight:387.38
  • HC067047 Hydrochloride(883031-03-6 free base)

    CAS:
    HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.
    Formula:C26H29ClF3N3O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:507.98
  • Dotinurad

    CAS:
    Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).
    Formula:C14H9Cl2NO4S
    Purity:97.43% - 98.04%
    Color and Shape:Solid
    Molecular weight:358.2
  • DL-Willardiine

    CAS:
    <p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>
    Formula:C7H9N3O4
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:199.16
  • ML277

    CAS:
    <p>ML277 (CID-53347902) was identified as a potent activator of KCNQ1 channels (EC(50)=260 nM).</p>
    Formula:C23H25N3O4S2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:471.59
  • A2793

    CAS:
    <p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>
    Formula:C13H12ClNO3
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:265.69
  • CX614

    CAS:
    <p>CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.</p>
    Formula:C13H13NO4
    Purity:97.37%
    Color and Shape:Solid
    Molecular weight:247.25
  • 5,7-Dichlorokynurenic acid

    CAS:
    5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.
    Formula:C10H5Cl2NO3
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:258.06
  • TC-I2000

    CAS:
    <p>TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.</p>
    Formula:C23H18F4N2O
    Purity:99.778%
    Color and Shape:Solid
    Molecular weight:414.4
  • S107

    CAS:
    <p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>
    Formula:C11H15NOS
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:209.31
  • PF-01247324

    CAS:
    <p>PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).</p>
    Formula:C13H10Cl3N3O
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:330.6
  • Quadrol

    CAS:
    <p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>
    Formula:C14H32N2O4
    Purity:99.91% - 99.92%
    Color and Shape:Viscous Liquid Liquid Viscous
    Molecular weight:292.41
  • Vanillyl butyl ether

    CAS:
    <p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>
    Formula:C12H18O3
    Purity:99.57%
    Color and Shape:Yellowish Liquid Liquid
    Molecular weight:210.27
  • VU0071063

    CAS:
    VU0071063 is a Kir6.2/SUR1 activator.
    Formula:C18H22N4O2
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:326.39
  • (2S)-6-Prenylnaringenin

    CAS:
    <p>(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.</p>
    Formula:C20H20O5
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:340.37
  • Amifampridine phosphate

    CAS:
    <p>Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.</p>
    Formula:C5H10N3O4P
    Color and Shape:Solid
    Molecular weight:207.12
  • IDRA-21

    CAS:
    IDRA-21 is a positive AMPA receptor modulator.
    Formula:C8H9ClN2O2S
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:232.69
  • Guan-fu base A hydrochloride(1394-48-5 free base)

    CAS:
    <p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>
    Formula:C24H32NO6Cl
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:465.97
  • Pyr10

    CAS:
    <p>Pyr10, a pyrazole derivative, selectively inhibits TRPC3, not STIM1/Orai1, with IC50 of 0.72 μM in TRPC3-HEK293, and 13.08 μM in BRL-2H3 cells.</p>
    Formula:C18H13F6N3O2S
    Purity:99.69% - 99.7%
    Color and Shape:Solid
    Molecular weight:449.37
  • VX-150

    CAS:
    <p>VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (&gt;400-fold).</p>
    Formula:C21H17F4N2O7P
    Purity:97.58%
    Color and Shape:Solid
    Molecular weight:516.34
  • Cis-ACBD

    CAS:
    <p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>
    Formula:C6H9NO4
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:159.14
  • Parimifasor

    CAS:
    <p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>
    Formula:C18H11Cl2F4N5O
    Purity:96.77% - 98.97%
    Color and Shape:Solid
    Molecular weight:460.21
  • α-Thujone

    CAS:
    <p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>
    Formula:C10H16O
    Purity:97.02% - 98.41%
    Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)
    Molecular weight:152.23
  • Eperisone hydrochloride

    CAS:
    <p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>
    Formula:C17H26ClNO
    Purity:99.80%
    Color and Shape:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter Taste
    Molecular weight:295.85
  • Benzamil

    CAS:
    <p>Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.</p>
    Formula:C13H14ClN7O
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:319.75
  • KB-R7943 mesylate

    CAS:
    <p>KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.</p>
    Formula:C17H21N3O6S2
    Purity:99.88% - ≥95%
    Color and Shape:Solid
    Molecular weight:427.5
  • Benzocaine xHCl(94-09-7(free base))


    <p>Benzocaine shares a common receptor with all othe rLAs in the voltage-gated Na+ channel(IC50 of 0.8 mM tested with a potential of +30 mV).</p>
    Formula:C9H11NO2·xHCl
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:N/A
  • Mitiglinide calcium hydrate

    CAS:
    <p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>
    Formula:C38H52CaN2O8
    Purity:98.97% - 99.96%
    Color and Shape:White Solid
    Molecular weight:704.91
  • Argireline

    CAS:
    <p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>
    Formula:C34H60N14O12S
    Purity:96.79% - 99.65%
    Color and Shape:White Powder
    Molecular weight:888.99
  • DAAO inhibitor-1

    CAS:
    <p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>
    Formula:C7H5FN2O
    Purity:97.84%
    Color and Shape:Solid
    Molecular weight:152.13
  • Cholesterol myristate

    CAS:
    <p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>
    Formula:C41H72O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:597.01
  • BRITE-338733

    CAS:
    <p>BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.</p>
    Formula:C27H35N3O2
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:433.59
  • Lumacaftor

    CAS:
    <p>Lumacaftor (VRT 826809) is a CFTR modulator that corrects the folding and trafficking of CFTR protein.</p>
    Formula:C24H18F2N2O5
    Purity:99.48% - 99.68%
    Color and Shape:Solid
    Molecular weight:452.41
  • SG-209

    CAS:
    <p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>
    Formula:C10H12N2O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:208.21
  • DQP 1105

    CAS:
    <p>DQP 1105 is a NMDA receptor antagonist.</p>
    Formula:C29H24BrN3O4
    Purity:98.6%
    Color and Shape:Solid
    Molecular weight:558.42
  • Drotaverine hydrochloride

    CAS:
    Drotaverine hydrochloride is a type 4 cyclic nucleotide phosphodiesterase (PDE4) inhibitor,and is an antispasmodic drug, used to enhance cervical dilation
    Formula:C24H32ClNO4
    Purity:99.81%
    Color and Shape:Pale-Yellow Crystalline Solid
    Molecular weight:433.968
  • Chembridge-5861528

    CAS:
    <p>Chembridge-5861528 (TCS 5861528) is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx with IC50 values of 14.3 and 18.7 μM.</p>
    Formula:C19H23N5O3
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:369.42
  • JNJ-17203212

    CAS:
    JNJ-17203212 is a potent and selective antagonist of TRPV1 (human TRPV1 and rat TRPV1, IC50 of 65 nM and 102 nM).
    Formula:C17H15F6N5O
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:419.32
  • Imidazenil

    CAS:
    <p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>
    Formula:C18H12BrFN4O
    Purity:98.4%
    Color and Shape:Solid
    Molecular weight:399.22
  • GMQ hydrochloride

    CAS:
    <p>GMQ hydrochloride, a potent ASIC modulator, activates ASIC3 at neutral pH and inhibits acid-induced peak current.</p>
    Formula:C10H12ClN5
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:237.69
  • Gabazine free base

    CAS:
    <p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>
    Formula:C15H17N3O3
    Color and Shape:Solid
    Molecular weight:287.31
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Formula:C34H31F2N3O3
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:567.62
  • Piperazine citrate

    CAS:
    <p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>
    Formula:C24H46N6O14
    Purity:99.8%
    Color and Shape:Crystals Indication
    Molecular weight:642.65