Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(51 products)
- Calcium Channel(494 products)
- Chloride channel(49 products)
- GABA Receptor(336 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(276 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2280 products of "Membrane Transporter/Ion Channel"
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ZM 226600
CAS:<p>ZM 226600 is an ATP-sensitive potassium channel opener with an EC50 value of 500 nM. ZM226600 has an inhibitory effect on spontaneous bladder activity.</p>Formula:C16H14F3NO4SPurity:99.87%Color and Shape:SolidMolecular weight:373.35NC-1300-B
CAS:<p>NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.</p>Formula:C17H19N3OSPurity:99.50%Color and Shape:SolidMolecular weight:313.42Silperisone HCl
CAS:<p>Silperisone HCl is a muscle relaxant and vasodilator, treating myoclonus, hypertonia, dystonia, and myospasm by blocking Na+ and Ca2+ channels.</p>Formula:C15H25ClFNSiPurity:99.62%Color and Shape:SolidMolecular weight:301.9NS-2710
CAS:<p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>Formula:C22H20N4OPurity:99.7% - 99.82%Color and Shape:SolidMolecular weight:356.42CNS-5161 hydrochloride
CAS:<p>CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel.</p>Formula:C16H19Cl2N3S2Purity:99.53%Color and Shape:SolidMolecular weight:388.38RL648_81
CAS:<p>RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be used in studies about neuronal hyperexcitability neurologic disorders.</p>Formula:C17H17F4N3O2Purity:99.82%Color and Shape:SolidMolecular weight:371.33Abeprazan hydrochloride
CAS:<p>Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting H+, K+ -atPase</p>Formula:C19H18ClF3N2O3SPurity:98.57%Color and Shape:SolidMolecular weight:446.87Sipatrigine
CAS:<p>Sipatrigine (619C89) is an inhibitor of glutamate release, TREK ion channels, TRESK channels, sodium channels, and calcium channels.</p>Formula:C15H16Cl3N5Purity:98.64% - 99.77%Color and Shape:SolidMolecular weight:372.68HC-070
CAS:<p>HC-070 is a TRPC5 and TRPC4 antagonist (IC50 = 9.3 nM and 46 nM).</p>Formula:C22H20Cl2N4O4Purity:98.48%Color and Shape:SolidMolecular weight:475.32Ro 25-6981
CAS:<p>Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.</p>Formula:C22H29NO2Purity:99.88%Color and Shape:SolidMolecular weight:339.47KT-362 fumarate
CAS:<p>KT-362 fumarate, a novel antagonist of Ca, K, and Na channels, induces vasodilation and relaxes rabbit arterial strips.</p>Formula:C26H32N2O7SPurity:99.75% - 99.98%Color and Shape:SolidMolecular weight:516.61AGN-201904
CAS:AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.Formula:C25H25N3O8S2Purity:97.32%Color and Shape:SolidMolecular weight:559.61L-838417
CAS:<p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>Formula:C19H19F2N7OPurity:98.12% - 99.70%Color and Shape:SolidMolecular weight:399.4PD-118057
CAS:<p>PD-118057, a potent hERG activator, may treat long QT syndrome and heart failure without hERG activity inhibition.</p>Formula:C21H17Cl2NO2Purity:99.16% - 99.97%Color and Shape:SolidMolecular weight:386.27JNJ-26489112
CAS:<p>JNJ-26489112 is a CNS-active agent and an inhibitor of voltage-gated Na+ channels and N-type Ca2+ channels.</p>Formula:C9H11ClN2O4SPurity:99.31%Color and Shape:SolidMolecular weight:278.71Protonstatin-1
CAS:<p>Protonstatin-1: treats hypoglycemia & Alzheimer's, inhibits IGFIR kinase, used in cancer studies.</p>Formula:C8H5NO2S2Purity:99.77%Color and Shape:SolidMolecular weight:211.26Dasolampanel
CAS:<p>Dasolampanel (NGX-426) is an ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study of chronic pain disorders.</p>Formula:C17H20ClN5O3Purity:98.70%Color and Shape:SolidMolecular weight:377.83Alpidem
CAS:<p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>Formula:C21H23Cl2N3OPurity:99.56% - 99.97%Color and Shape:White To Off-White SolidMolecular weight:404.33FR183998 free base
CAS:<p>FR183998 free base is an inhibitor of Na+/Ca2+ Exchanger.</p>Formula:C17H19Cl2N5O2SPurity:99.61%Color and Shape:SolidMolecular weight:428.34(+)-KCC2 blocker 1
CAS:<p>(+)-KCC2 blocker 1 is a selective blocker of KCC2 (IC50 = 0.4 μM).</p>Formula:C22H25NO5SPurity:99.88%Color and Shape:SolidMolecular weight:415.5SET 2
CAS:<p>SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 of 0.46 μM. SET 2 shows selectivity over TRPV1, TRPV3 and TRPV4.</p>Formula:C17H21F3N4O2SPurity:99.77%Color and Shape:SolidMolecular weight:402.438-Bromo-cGMP sodium
CAS:<p>8-Bromo-cGMP sodium: PKG activator, eases pain, dilates vessels, reduces Ca2+ currents & insulin release.</p>Formula:C10H10BrN5NaO7PPurity:99.45%Color and Shape:SolidMolecular weight:446.09WY-47766
CAS:<p>WY-47766, a proton pump inhibitor, is used potentially for the treatment of postmenopausal osteoporosis.</p>Formula:C14H13N3O2SPurity:97.63% - 99.83%Color and Shape:SolidMolecular weight:287.34FEMA-4809
CAS:<p>FEMA-4809 activates TRPM8, the ion channel for cold sensation, and is used as a cooling agent.</p>Formula:C17H17N3O2SPurity:99.9%Color and Shape:SolidMolecular weight:327.4TC-I 2014
CAS:<p>TC-I 2014 shows antiallodynic properties in pain models.</p>Formula:C23H19F6N3OPurity:99.07%Color and Shape:SolidMolecular weight:467.41Saripidem
CAS:<p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>Formula:C19H20ClN3OPurity:99.45%Color and Shape:SolidMolecular weight:341.83GNE-8324
CAS:<p>GNE-8324 is a GluN2A selective positive allosteric modulator that enhances NMDAR-mediated synaptic responses in inhibitory, but not excitatory, neurons.</p>Formula:C18H18FN3OSPurity:98.68% - 99.34%Color and Shape:SolidMolecular weight:343.42Temiverine hydrochloride
CAS:<p>Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.</p>Formula:C24H36ClNO3Purity:99.26% - 99.43%Color and Shape:SolidMolecular weight:422Nelonemdaz
CAS:<p>Nelonemdaz (Neu2000) is an NMDA receptor antagonist with antioxidant activity that can be used to study cerebral infarction reperfusion injury.</p>Formula:C15H8F7NO3Purity:99.52%Color and Shape:SolidMolecular weight:383.22Losigamone
CAS:<p>Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.</p>Formula:C12H11ClO4Purity:99.98%Color and Shape:SolidMolecular weight:254.67Suriclone
CAS:<p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>Formula:C20H20ClN5O3S2Purity:99.21% - 99.73%Color and Shape:SolidMolecular weight:477.99R 56865
CAS:<p>R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.</p>Formula:C23H28FN3OSPurity:99.52%Color and Shape:SolidMolecular weight:413.55MK-0448
CAS:<p>MK-0448 is a novel and selective blocker of the Kv1.5 (KCNA5) channel, a key channel involved in cardiac repolarization current I Kur.</p>Formula:C24H21FN4O2SPurity:99.25% - 99.79%Color and Shape:SolidMolecular weight:448.51DMP-543
CAS:<p>DMP-543 (XR-543) is a potassium channel (KV7 channel) blocker that enhances the release of neurotransmitters.</p>Formula:C26H18F2N2OPurity:99.89%Color and Shape:SolidMolecular weight:412.43KR-32568
CAS:<p>KR-32568 is a sodium/hydrogen exchanger 1 (NHE-1) inhibitor (IC50: 230 nM).</p>Formula:C13H12FN3O2Purity:99.91%Color and Shape:SolidMolecular weight:261.25PG01
CAS:<p>PG01 is a potent CFTR Cl-channel potentiator, effective against ΔF508 (Ka 0.3 μM), and also against E193K, G970R and G551D (CFTR mutants), with Kd values of 0.</p>Formula:C28H29N3O2Purity:99.87%Color and Shape:SolidMolecular weight:439.55AZD-1305
CAS:<p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>Formula:C22H31FN4O4Purity:99.31% - 99.86%Color and Shape:SolidMolecular weight:434.5NHE3-IN-1
CAS:<p>NHE3-IN-1 是钠/质子交换剂 3 (NHE-3) 的抑制剂。</p>Formula:C12H10ClN3SPurity:99.93%Color and Shape:SolidMolecular weight:263.75Nisoxetine hydrochloride
CAS:<p>Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor</p>Formula:C17H21NO2·HClPurity:99.21%Color and Shape:White SolidMolecular weight:307.82Golexanolone
CAS:<p>Golexanolone can be used to study neurological diseases.</p>Formula:C21H31NO2Purity:99.90% - 99.99%Color and Shape:SolidMolecular weight:329.48Ru-32514
CAS:<p>Ru-32514 is a benzodiazepine receptor agonist.</p>Formula:C18H17N3O2Purity:99.21%Color and Shape:SolidMolecular weight:307.35DFP00173
CAS:<p>DFP00173: Potent, selective AQP3 inhibitor; IC50 ~0.1-0.4 μM; less effective on AQP7, AQP9.</p>Formula:C11H7Cl2N3O3SPurity:99.53% - 99.53%Color and Shape:SolidMolecular weight:332.16UCL 2077
CAS:<p>UCL 2077 blocks KCNQ channels, related to epilepsy, and selective slow-afterhyperpolarization channels, with 500 nM IC50, sparing Ca2+ channels.</p>Formula:C25H22N2Purity:99.58%Color and Shape:SolidMolecular weight:350.46Riluzole hydrochloride
CAS:<p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>Formula:C8H6ClF3N2OSPurity:99.76%Color and Shape:SolidMolecular weight:270.66Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Formula:C24H35N3O8S2Purity:98.74%Color and Shape:SolidMolecular weight:557.68NNC 05-711
CAS:<p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>Formula:C21H23ClN2O3Purity:99.92%Color and Shape:SolidMolecular weight:386.87TAK-653
CAS:<p>TAK-653 is a selective AMPA receptor PAM with minimal agonist activity, showing antidepressant-like effects and safety in rats.</p>Formula:C19H23N3O3SPurity:99.89%Color and Shape:SolidMolecular weight:373.47ELB-139
CAS:<p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>Formula:C14H16ClN3OPurity:>99.99%Color and Shape:SolidMolecular weight:277.75DSP-0565
CAS:<p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>Formula:C14H12FNOPurity:99.51% - 99.56%Color and Shape:SolidMolecular weight:229.25Progabide
CAS:<p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>Formula:C17H16ClFN2O2Purity:99.68%Color and Shape:SolidMolecular weight:334.77Cerebrocrast
CAS:<p>Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.</p>Formula:C26H35F2NO7Purity:99.71%Color and Shape:SolidMolecular weight:511.56Tiludronate disodium
CAS:Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.Formula:C7H7ClNa2O6P2SPurity:>99.99% - >99.99%Color and Shape:Fine White To Off-White Crystalline PowderMolecular weight:362.57Aptiganel
CAS:<p>Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.</p>Formula:C20H21N3Purity:98.13% - 98.90%Color and Shape:SolidMolecular weight:303.4Trombodipine
CAS:<p>Trombodipine (PCA-4230) is a platelet aggregation inhibitor with antithrombotic activity and protection against Listeria monocytogenes.</p>Formula:C21H24N2O7SPurity:98.73% - 99.14%Color and Shape:SolidMolecular weight:448.49Elpetrigine
CAS:<p>Elpetrigine (GW273293) is a potential sodium channel blocker with antiepileptic activity that can be used to study epilepsy.</p>Formula:C10H7Cl3N4Purity:99.04% - 99.43%Color and Shape:SolidMolecular weight:289.55Olvanil
CAS:<p>Olvanil (N-Vannilyloleoylamide) is a vanilloid receptor agonist with EC50 of 0.7nM.</p>Formula:C26H43NO3Purity:99.58%Color and Shape:SolidMolecular weight:417.62TASK-1-IN-1
CAS:<p>TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.</p>Formula:C22H20N2O2Purity:99.57%Color and Shape:SoildMolecular weight:344.41Nerisopam
CAS:<p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>Formula:C18H19N3O2Purity:97.07%Color and Shape:SolidMolecular weight:309.36DMT1 blocker 1
CAS:<p>DMT1 blocker 1 inhibits DMT1; IC50=0.64μM; may prevent intestinal iron absorption.</p>Formula:C16H14N4O2Purity:99.73%Color and Shape:SolidMolecular weight:294.31Muscimol HBr
CAS:<p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>Formula:C4H7BrN2O2Purity:98.13%Color and Shape:Off-White PowderMolecular weight:195.01Indecainide
CAS:<p>Indecainide (Ricainid) is an antiarrhythmic compound that is carcinogenic and may be used in studies secondary to coronary artery disease.</p>Formula:C20H24N2OPurity:98.01% - 98.96%Color and Shape:SolidMolecular weight:308.42Fengabine
CAS:<p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>Formula:C17H17Cl2NOPurity:99%Color and Shape:SolidMolecular weight:322.23ANO1-IN-1
CAS:<p>ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.</p>Formula:C18H28N2O2SPurity:99.66%Color and Shape:SolidMolecular weight:336.49Delucemine Hydrochloride
CAS:<p>Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.</p>Formula:C16H18ClF2NPurity:98.49% - 99.30%Color and Shape:SolidMolecular weight:297.77N106
CAS:<p>N106 is an activator of the SUMO-activating enzyme, E1 ligase, and triggers intrinsic sumoylation of SERCA2a. N106 can be used in studies about heart failure.</p>Formula:C17H14N4O3SPurity:99.69%Color and Shape:SolidMolecular weight:354.38SKF96067
CAS:<p>SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.</p>Formula:C21H22N2O2Purity:99.89%Color and Shape:SolidMolecular weight:334.41MSP3
CAS:<p>MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective effects.</p>Formula:C16H19NO3SPurity:99.89%Color and Shape:SolidMolecular weight:305.39Saviprazole
CAS:<p>Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer.</p>Formula:C15H10F7N3O2S2Purity:97.07% - 97.17%Color and Shape:SolidMolecular weight:461.38Rilmakalim
CAS:<p>Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.</p>Formula:C21H23NO5SPurity:99.8% - 99.9%Color and Shape:SolidMolecular weight:401.48Orphenadrine
CAS:<p>Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner,</p>Formula:C18H23NOPurity:98.91% - 99.11%Color and Shape:SolidMolecular weight:269.38L-Cysteine S-sulfate
CAS:<p>L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.</p>Formula:C3H7NO5S2Purity:99.90% - 99.92%Color and Shape:SolidMolecular weight:201.22Pyr3
CAS:<p>Pyr3 selectively blocks TRPC3 channels, reducing Ca2+ influx; it's effective at 700 nM.</p>Formula:C16H11Cl3F3N3O3Purity:98.04%Color and Shape:SolidMolecular weight:456.63Quinacainol
CAS:<p>Quinacainol (RP 54272) is a new antiarrhythmic compound with class I antiarrhythmic effects in rats.</p>Formula:C21H30N2OPurity:99.64%Color and Shape:SolidMolecular weight:326.48Leminoprazole
CAS:<p>Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.</p>Formula:C19H23N3OSPurity:99.08% - 99.56%Color and Shape:SolidMolecular weight:341.47Stepronin
CAS:<p>Stepronin (TTPG) shows expectorant activities and inhibits airway secretion.</p>Formula:C10H11NO4S2Purity:99.59%Color and Shape:White Or Off White CrystallineMolecular weight:273.33Lirequinil
CAS:<p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>Formula:C26H25ClN2O3Purity:98.54%Color and Shape:SolidMolecular weight:448.94ZTZ240
CAS:<p>ZTZ240 is a KCNQ2 channel activator used in the study of epilepsy.</p>Formula:C12H8ClFN2OPurity:99.89%Color and Shape:SolidMolecular weight:250.66YM758
CAS:<p>YM758 is an inhibitor of If current channel.</p>Formula:C26H32FN3O4Purity:99.65%Color and Shape:SolidMolecular weight:469.55Quinabactin
CAS:<p>Quinabactin (LC-66C6): ABA agonist, induces guard cell closure, reduces water loss, hinders germination, boosts drought resistance in Arabidopsis/soybean.</p>Formula:C20H24N2O3SPurity:99.63%Color and Shape:SolidMolecular weight:372.48NaV1.2/1.6 channel blocker-1
CAS:<p>NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.</p>Formula:C14H14N2OSPurity:99.54%Color and Shape:SolidMolecular weight:258.34Ralitoline
CAS:<p>Ralitoline (Ralitolinum) is an anticonvulsant with anticancer activity and sodium channel blocking activity.</p>Formula:C13H13ClN2O2SPurity:98.45%Color and Shape:SolidMolecular weight:296.77Mavatrep
CAS:<p>Mavatrep (JNJ-39439335) is a selective antagonist of TRPV1 with Ki of 6.5 nM and can be used for studies about inflammatory pain.</p>Formula:C25H21F3N2OPurity:98.51% - 99.31%Color and Shape:SolidMolecular weight:422.44Sarmazenil
CAS:<p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>Formula:C15H14ClN3O3Purity:99.46%Color and Shape:SolidMolecular weight:319.74Elismetrep
CAS:<p>Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.</p>Formula:C27H21F3N2O5SPurity:99.37% - 99.93%Color and Shape:SolidMolecular weight:542.53S 18986
CAS:<p>S 18986 is a selective, orally active, brain penetrant positive allosteric modulator of AMPA-type receptors, showcasing cognitive-enhancing properties in</p>Formula:C10H12N2O2SPurity:99.64%Color and Shape:SolidMolecular weight:224.28Divaplon
CAS:<p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>Formula:C17H17N3O2Purity:97.44% - 98.25%Color and Shape:SolidMolecular weight:295.34GW 542573X
CAS:<p>GW 542573X is a potent and selective small molecule Ca2+-activated K+ 2 (SK2) channel activator.GW 542573X induces a leftward shift in the Ca2+ response curve</p>Formula:C19H28N2O5Purity:99.91%Color and Shape:SolidMolecular weight:364.44CFTR corrector 8
CAS:<p>CFTR corrector 8: potent for cystic fibrosis research, modulates CFTR protein.</p>Formula:C29H27F2NO7Purity:99.57%Color and Shape:SolidMolecular weight:539.52VRT-532
CAS:<p>VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.</p>Formula:C16H14N2OPurity:99.88% - 99.93%Color and Shape:SolidMolecular weight:250.3VU 0240551
CAS:<p>VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.</p>Formula:C16H14N4OS2Purity:99.9%Color and Shape:SolidMolecular weight:342.44RWJ-51204
CAS:<p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>Formula:C21H19F2N3O3Purity:99.57% - 99.95%Color and Shape:SolidMolecular weight:399.39Bamocaftor
CAS:<p>Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF patients.</p>Formula:C28H32F3N5O4SPurity:99.71%Color and Shape:SolidMolecular weight:591.65IKs124
CAS:<p>IKs124 is a KCNE2/KCNQ1 potassium channel blocker, for hKCNE1 and hKCNE3, and can be used to study peptic ulcers.</p>Formula:C18H26N2O3SPurity:99.53%Color and Shape:SolidMolecular weight:350.48Cirsimaritin
CAS:<p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>Formula:C17H14O6Purity:99.9%Color and Shape:SolidMolecular weight:314.29UK 66914
CAS:<p>UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.</p>Formula:C18H24N4O3SPurity:99.75%Color and Shape:SolidMolecular weight:376.47ABT 102
CAS:<p>ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.</p>Formula:C21H24N4OPurity:98.38% - 99.86%Color and Shape:SolidMolecular weight:348.44Panadiplon
CAS:<p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>Formula:C18H17N5O2Purity:98.30% - 98.94%Color and Shape:SolidMolecular weight:335.36BTG 502
CAS:<p>BTG 502 is an alkylamide insecticide that binds to voltage-gated sodium channels, antagonising the activation of sodium channels by Batrachotoxin (BTX).</p>Formula:C21H24BrNOPurity:99.30%Color and Shape:SolidMolecular weight:386.33CGP 64213
CAS:<p>CGP 64213 is a GABAb receptor agonist.</p>Formula:C26H36IN2O7PPurity:98%Color and Shape:SolidMolecular weight:646.45A 425619
CAS:<p>A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonist</p>Formula:C18H14F3N3OPurity:99.75%Color and Shape:SolidMolecular weight:345.32Potassium Channel Activator 1
CAS:<p>Potassium Channel Activator 1 aids treatment of ADHD, schizophrenia, and mood disorders by targeting the dopaminergic system.</p>Formula:C19H23N3O3Purity:99.86%Color and Shape:SolidMolecular weight:341.4Coelenterazine h
CAS:<p>Coelenterazine H, a Ca2+ sensitive synthetic derivative, is a luminescent biomolecule used to measure Ca2+ changes.</p>Formula:C26H21N3O2Purity:99.49%Color and Shape:Yellow To Brownish PowderMolecular weight:407.46NS1219
CAS:<p>NS1219, an isomer of NS1209, is a selective AMPA antagonist for studying stroke, neuropathic pain, and epilepsy.</p>Formula:C24H28N4O7SColor and Shape:SolidMolecular weight:516.57GSK 2833503A
CAS:<p>GSK 2833503A: potent TRPC6/3 antagonist; IC50: 3-16/21-100 nM; >63x selective; inhibits cardiac hypertrophy signaling.</p>Formula:C18H21ClFN3OSColor and Shape:SolidMolecular weight:381.9Ebio1
CAS:<p>Ebio1, a selective activator of the voltage-gated potassium channel KCNQ2, enhances channel conductance by promoting the formation of an expanded gate at a saturation voltage of +50 mV, leading to increased channel activity [1].</p>Formula:C19H14FNOColor and Shape:SolidMolecular weight:291.32CS-526
CAS:<p>CS-526 is a reversible proton pump inhibitor targeting the K+ site on H+,K+-ATPase, reducing gastric acid secretion and preventing mucosal lesions.</p>Formula:C20H22FN3OColor and Shape:SolidMolecular weight:339.41COR659
CAS:<p>COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.</p>Formula:C16H16ClNO3SPurity:99.75%Color and Shape:SolidMolecular weight:337.82Nalanthalide
CAS:<p>Nalanthalide, serving as a voltage-gated potassium channel Kv1.3 blocker (IC50 = 3.9 µM) with potential immunosuppressive properties, is applicable in the research of inflammatory immune diseases including neuroinflammation [1] [2].</p>Formula:C30H44O5Color and Shape:SolidMolecular weight:484.67NPBA
CAS:<p>NPBA, a potassium K2P channel TASK-3 (KCNK9) agonist, concurrently functions as a blocker of the tandem pore domain weak inward rectifying K+ channel (TWIK2). This compound effectively inhibits NLRP3 inflammasome activation in macrophages [1].</p>Formula:C16H14F3N3O3Color and Shape:SolidMolecular weight:353.3Piprofurol
CAS:<p>Piprofurol is used as a Calcium channel blocker.</p>Formula:C26H33NO6Purity:98%Color and Shape:SolidMolecular weight:455.54Diproqualone
CAS:<p>Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].</p>Formula:C12H14N2O3Color and Shape:SolidMolecular weight:234.255A-1165442
CAS:<p>A-1165442 is a competitive TRPV1 antagonist. For human TRPV, the IC50 values is 9 nM.</p>Formula:C22H20ClF2N3O2Color and Shape:SolidMolecular weight:431.86Pristinamycin IA
CAS:<p>Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic.</p>Formula:C45H54N8O10Purity:97.44%Color and Shape:SolidMolecular weight:866.96PU-48
CAS:<p>PU-48 is a potent inhibitor of urea transporters A (UT-A) with an IC50 value of 0.32 μM, exhibiting a significant diuretic effect in mouse models without</p>Formula:C14H12N2O3SColor and Shape:SolidMolecular weight:288.32Ritivixibat
CAS:<p>Ritivixibat inhibits IBAT and modulates bile acids, used in research for cardiovascular, metabolic, GI, and liver diseases.</p>Formula:C26H36N2O5S2Color and Shape:SolidMolecular weight:520.7Antiarrhythmic agent-1
CAS:<p>Antiarrhythmic agent-1 (example I), functioning as an antiarrhythmic agent and an IKr potassium channel blocker (IC 50 <1 μM), effectively inhibits cardiac</p>Formula:C25H27N3O4SColor and Shape:SolidMolecular weight:465.568-Pcpt-cGMP
CAS:<p>8-Pcpt-cGMP acts as an agonist for cyclic nucleotide-gated (CNG) channels with an EC50 of 0.5 μM and exhibits good membrane permeability. This compound is utilized in research to explore the role of CNG channels in visual and olfactory signal transduction.</p>Formula:C16H15ClN5O7PSColor and Shape:SolidMolecular weight:487.81URAT1 inhibitor 8
CAS:<p>URAT1 Inhibitor 8 (example 247) serves as a highly potent inhibitor of URAT1, demonstrating an IC50 value of 0.001 μM.</p>Formula:C19H13ClFN3O4SColor and Shape:SolidMolecular weight:433.84NaV1.7 Blocker-801
CAS:<p>NaV1.7 Blocker-801 is a potent NaV1.7 blocker.</p>Formula:C20H15ClF2N6O3S2Color and Shape:SolidMolecular weight:524.95MCT1-IN-2
CAS:<p>SR13800 is a monocarboxylate transporter 1 (MCT1) inhibitor with cell-permeable.</p>Formula:C25H29N3O2SColor and Shape:SolidMolecular weight:435.58mGAT3/4-IN-2
CAS:<p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>Formula:C26H32ClN3OS2Color and Shape:SolidMolecular weight:502.13CP-409092
CAS:<p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>Formula:C17H19N3O2Purity:98%Color and Shape:SolidMolecular weight:297.35JT010
CAS:<p>JT010 is an effective agonist of TRPA1 (EC50 = 0.65 nM).</p>Formula:C16H19ClN2O3SPurity:99.75%Color and Shape:SolidMolecular weight:354.85GDC-6599
CAS:<p>GDC-6599 (Example 8) is an orally active inhibitor of the TRPA1 channel, potentially useful for researching TRPA1-mediated conditions, including pain [1].</p>Formula:C20H19ClN6O3Color and Shape:SolidMolecular weight:426.86TRPC5-IN-3
CAS:<p>TRPC5-IN-3 is a potent TRPC5 inhibitor (IC50= 10.75 nM).</p>Formula:C18H15ClF3N5OColor and Shape:SolidMolecular weight:409.79CP 154526
CAS:<p>CRF1 receptor antagonist</p>Formula:C23H33ClN4Purity:98%Color and Shape:SolidMolecular weight:400.99NMDA receptor modulator 6
CAS:<p>NMDA receptor regulator 6 (Compound 183) is an effective NMDA receptor regulator and has research value in neurological disorders.</p>Formula:C20H17FN2O4SColor and Shape:SolidMolecular weight:400.42MONIRO-1
CAS:<p>MONIRO-1 blocks T/N-type Ca²⁺ channels: hCav2.2 (IC50: 34μM), hCav3.1 (3.3μM), hCav3.2 (1.7μM), hCav3.3 (7.2μM).</p>Formula:C23H24ClFN4O3Color and Shape:SolidMolecular weight:458.92AMPA receptor modulator-2
CAS:<p>AMPA receptor modulator-2 is a modulator of AMPA receptor. The pIC50 value for TARPγ2 dependent AMPA receptor is 10.1.</p>Formula:C15H6F6N4OSPurity:99.8%Color and Shape:SolidMolecular weight:404.29TRPC3/6-IN-2
CAS:<p>TRPC3/6-IN-2 is a potent inhibitor of TRPC3 and TRPC6, exhibiting IC50 values of 16 nM for TRPC3 and 29.8 nM for TRPC6, respectively [1].</p>Formula:C18H23F2N5Color and Shape:SolidMolecular weight:347.41SN40 hydrochloride
CAS:<p>SN40 hydrochloride is a potent inhibitor of amino acid transport (AAT), exhibiting inhibitory constants (Kis) of 7.29 μM, 2.42 μM, 2.94 μM, 5.55 μM, 24.43 μM, and 5.55 μM for rat ASCT2, human ASCT2, EAAT1, EAAT2, EAAC1, and EAAT5, respectively. It is utilized in cancer research. [1]</p>Formula:C18H21ClN2O2Color and Shape:SolidMolecular weight:332.82KVI-020
CAS:<p>KVI-020: oral Kv1.5 blocker (IC50: 480nM), hERG inhibitor (IC50: 15100nM), potent antiarrhythmic for AF studies.</p>Formula:C20H25N3O5SColor and Shape:SolidMolecular weight:419.49L 663581
CAS:<p>L 663581 is the benzodiazepine receptor partial agonist.</p>Formula:C17H16ClN5O2Purity:98%Color and Shape:SolidMolecular weight:357.79Chromanol 293B
CAS:slow delayed rectifier K+ current (IKs) blockerFormula:C15H20N2O4SPurity:98%Color and Shape:SolidMolecular weight:324.4Xeniafaraunol A
CAS:<p>Xeniafaraunol A (compound 31) is a potent inhibitor of the transient receptor potential melastatin 7 (TRPM7) channel [1].</p>Formula:C20H28O2Color and Shape:SolidMolecular weight:300.44TROX-1
CAS:<p>TROX-1 is the activation state-dependent Cav2 channel antagonist.</p>Formula:C22H16ClFN6OPurity:98%Color and Shape:SolidMolecular weight:434.85(+)-Bicuculline methiodide
CAS:<p>(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.</p>Formula:C21H20INO6Purity:99.24%Color and Shape:SolidMolecular weight:509.29PF 04531083
CAS:<p>PF 04531083 is a selective blocker of the NaV1.8 channel. PF 04531083 can be used for neuropathic and inflammatory pain studies.</p>Formula:C17H16ClN5O2Purity:99.85%Color and Shape:SolidMolecular weight:357.79NMDA receptor modulator 4
CAS:<p>NMDA receptor modulator 4 (Compound 169) can be used for the research of neurological disorder that is a potent modulator of NMDA receptor [1].</p>Formula:C13H9F3N2O3SColor and Shape:SolidMolecular weight:330.28DNDS
CAS:<p>DNDS is a channel blocker of voltage-dependent cystic fibrosis transmembrane conductance regulator (CFTR).</p>Formula:C14H8N2Na2O10S2Purity:99.92%Color and Shape:Physical Description White Powder (Ntp 1992)Molecular weight:474.33GDC-0310
CAS:<p>GDC-0310 is a selective, orally available Nav1.7 inhibitor with an IC50 of 0.6 nM for human Nav1.7, suitable for pain research.</p>Formula:C25H29Cl2FN2O4SPurity:99.877%Color and Shape:SolidMolecular weight:543.48α,β-Methylene-ATP
CAS:<p>α,β-Methylene ATP，一种ATP的膦酸酯类似物，充当P2X3和P2X7受体的配体。该化合物对P2X1和P2X3表现出高选择性激动剂活性，而在P2X2, 4, 7受体上无活性。</p>Formula:C11H18N5O12P3Color and Shape:SolidMolecular weight:505.21Dasolampanel etibutil
CAS:<p>Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).</p>Formula:C23H32ClN5O3Color and Shape:SolidMolecular weight:461.98Kv3 modulator 2
CAS:<p>Kv3 modulator 2 is a potent Kv3 channels modulator.has analgesic activity and is used in the prophylaxis or treatment of related disorders.</p>Formula:C21H21N3O4Purity:98%Color and Shape:SolidMolecular weight:379.41UBP316
CAS:<p>GluR5-containing kainate receptor antagonist</p>Formula:C20H19N3O6SPurity:98%Color and Shape:SolidMolecular weight:429.45TPA 023
CAS:<p>TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).</p>Formula:C20H22FN7OPurity:99.75%Color and Shape:SolidMolecular weight:395.43GNE-0723
CAS:<p>GNE-0723 is a selective positive allosteric modulator of the NMDA receptor, GluN2A.blood-brain barrier (BBB) and Dravet syndrome and Alzheimer's disease (AD).</p>Formula:C16H8ClF6N5OSPurity:97.29% - 99.91%Color and Shape:SolidMolecular weight:467.78U 89843A
CAS:<p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>Formula:C16H23N5Purity:99.62%Color and Shape:SolidMolecular weight:285.39ADCI
CAS:<p>ADCI inhibits voltage-activated sodium and NMDA channels; boosts dopamine metabolism in prefrontal cortex and nucleus accumbens.</p>Formula:C16H14N2OPurity:98%Color and Shape:SolidMolecular weight:250.3PF-4778574
CAS:<p>PF-4778574 is a positive AMPA receptor allosteric modulation (EC50: 45 to 919 nM in different cells).</p>Formula:C19H22N2O3S2Purity:98%Color and Shape:SolidMolecular weight:390.52CFTR corrector 12
CAS:<p>CFTR corrector 12 is a CFTR corrector that rescues all mutant proteins except M760R ABCA3 and can be used to study cystic fibrosis.</p>Formula:C19H21ClN4O2S2Purity:99.47%Color and Shape:SolidMolecular weight:436.98TCS 46b
CAS:<p>TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.</p>Formula:C22H23N3OPurity:99.78% - 99.78%Color and Shape:SolidMolecular weight:345.4411-deoxy-PGF2a
CAS:<p>11-deoxy-PGF2a is a thromboxane A2 receptor agonist that partially alleviates crowding in Lpar3(−/−) female embryos and induces smooth muscle contraction</p>Formula:C20H34O4Color and Shape:SolidMolecular weight:338.48Zelquistinel
CAS:<p>Zelquistinel, an NMDA receptor agonist, aids research on depression, anxiety, and psychiatric disorders.</p>Formula:C15H25N3O5Color and Shape:SolidMolecular weight:327.38ZM 260384
CAS:<p>ZM 260384 is a potassium channel opener.</p>Formula:C15H11F4N3O4Color and Shape:SolidMolecular weight:373.26SLC13A5-IN-1
CAS:<p>SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5),completely blocks the uptake of 14C-citrate(IC50 : 0.022 μM in HepG2 cells).</p>Formula:C19H19Cl3N2O3SPurity:99.67%Color and Shape:SolidMolecular weight:461.79Nepaprazole
CAS:<p>Nepaprazole (TY-11345) is a potent proton pump inhibitor; IC50: 5.8µM at pH 6.0, 9.9µM at pH 7.4. Better inhibition in weak acid.</p>Formula:C18H19N3O2SPurity:98%Color and Shape:SolidMolecular weight:341.43PF-06456384
CAS:PF-06456384 is a highly potent and selective NaV1.7 inhibitor with IC50 value of 0.01 nM.Formula:C35H32F3N7O3S2Purity:98%Color and Shape:SolidMolecular weight:719.86,2'-Dihydroxyflavone
CAS:<p>6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.</p>Formula:C15H10O4Purity:99.44% - 99.67%Color and Shape:SolidMolecular weight:254.24URAT1 inhibitor 6
CAS:<p>URAT1 inhibitor 6 (Compound 1h), with an IC50 of 35 nM for hURAT1, demonstrates 200-fold and 8-fold greater potency compared to Lesinurad and Benzbromarone,</p>Formula:C9H7BrN3NaO2S2Color and Shape:SolidMolecular weight:356.2PF-05241328
CAS:<p>PF-05241328 is an effective and selective inhibitor of human Nav1.7 voltage-dependent sodium channels (IC50: 31 nM).</p>Formula:C19H21ClN4O4SPurity:98%Color and Shape:SolidMolecular weight:436.91XR9051
CAS:<p>XR9051, a synthetic derivative of a natural compound, potently reverses P-glycoprotein MDR (EC50 = 1.4 nM) by inhibiting cytotoxic binding.</p>Formula:C39H38N4O5Color and Shape:SolidMolecular weight:642.74NO-711ME
CAS:<p>NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.</p>Formula:C22H24N2O3Purity:99.54%Color and Shape:SolidMolecular weight:364.44L-822179
CAS:<p>L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.</p>Formula:C17H14N8O2Purity:98.5% - 99.61%Color and Shape:SolidMolecular weight:362.35(R)-3,4-DCPG
CAS:<p>AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors</p>Formula:C10H9NO6Purity:98%Color and Shape:SolidMolecular weight:239.18Clobutinol hydrochloride
CAS:<p>Clobutinol hydrochloride, an antitussive agent, influences heart rate and blood pressure, and is utilized in cough-related research [1] [2] [3].</p>Formula:C14H23Cl2NOPurity:98%Color and Shape:SolidMolecular weight:292.25AGN-201904Z
CAS:<p>AGN-201904Z is a slow-release, acid-resistant pro-PPI that turns into omeprazole, offering extended acid suppression.</p>Formula:C25H25N3NaO8S2Purity:98%Color and Shape:SolidMolecular weight:582.6GMA-839
CAS:<p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>Formula:C21H31F3O3Purity:98%Color and Shape:SolidMolecular weight:388.46VMAT2-IN-I HCl
CAS:<p>VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A.</p>Formula:C25H32ClF4NO4Purity:98%Color and Shape:SolidMolecular weight:521.97JM-1232
CAS:<p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>Formula:C24H27N3O2Color and Shape:SolidMolecular weight:389.49Mioflazine
CAS:<p>Mioflazine suppresses nucleoside uptake. Mioflazine is an orally active nucleoside transport inhibitor. It has the potential for sleep disorders treatment.</p>Formula:C29H30Cl2F2N4O2Purity:98%Color and Shape:SolidMolecular weight:575.48Afizagabar
CAS:<p>Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.</p>Formula:C19H12FN3O2SColor and Shape:SolidMolecular weight:365.38CGP-54626 free base
CAS:CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).Formula:C18H28Cl2NO3PPurity:98%Color and Shape:SolidMolecular weight:408.3AR-C141990
CAS:<p>AR-C141990 is a lactate transporters inhibitor.</p>Formula:C26H28N4O4SColor and Shape:SolidMolecular weight:492.59ROMK-IN-32
CAS:<p>ROMK-IN-32 is an inhibitor of the extra-renal medullary potassium channel (ROMK) (IC50: 35 nM) and also inhibits hERG (IC50: 22 μM).</p>Formula:C24H28N4O5Color and Shape:SolidMolecular weight:452.5M084 hydrochloride
CAS:<p>M084 hydrochloride, a TRPC4/5 channel blocker, exhibits IC50 values of 10.3 μM and 8.2 μM, respectively. This compound is noted for its antidepressant and anxiolytic effects [1] [2].</p>Formula:C11H16ClN3Color and Shape:SolidMolecular weight:225.72N-Linolenoylethanolamine
CAS:<p>N-Linolenoylethanolamine (18:3 NAE), an endocannabinoid, functions as a vanillin receptor (TRPV1) agonist [1].</p>Formula:C20H35NO2Color and Shape:SolidMolecular weight:321.5056-Iodoamiloride
CAS:<p>6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value of 88 nM.</p>Formula:C6H8IN7OPurity:98%Color and Shape:SolidMolecular weight:321.08D-erythro-Sphingosine hydrochloride
CAS:<p>D-erythro-Sphingosine HCl activates TRPM3 and dephosphorylates retinoblastoma protein.</p>Formula:C18H38ClNO2Color and Shape:SolidMolecular weight:335.95PPADS tetrasodium
CAS:<p>PPADS tetrasodiuma is a P2X receptor antagonist and an inhibitor of the inverse mode of Na/Ca²⁺ exchange in guinea pig airway smooth muscle.</p>Formula:C14H10N3Na4O12PS2Purity:95% - ≥95%Color and Shape:SolidMolecular weight:599.3α,β-Methylene ATP trisodium
CAS:<p>α,β-Methylene ATP trisodium is a ligand of P2X3 and P2X7 receptor.</p>Formula:C11H15N5Na3O12P3Purity:99.66%Color and Shape:SolidMolecular weight:571.15Crobenetine hydrochloride
CAS:<p>Crobenetine hydrochloride, a sodium channel antagonist, is used potentially for the treatment of stroke.</p>Formula:C25H34ClNO2Color and Shape:SolidMolecular weight:416OADS
CAS:<p>OADS is an inhibitor of ClC-ec1 with low micromolar affinity. OADS has no specific effect on a CLC channel (ClC-1).</p>Formula:C30H42N2O8S2Color and Shape:SolidMolecular weight:622.79Oct4 inducer-2
CAS:<p>Oct4 Inducer-2, an OCT4 inducer, sustains hiPSC formation by enhancing endogenous OCT4 expression and has applications in anti-aging research [1].</p>Formula:C14H16N2O2SColor and Shape:SolidMolecular weight:276.35ARN 11391
CAS:<p>ARN 11391 enhances the function of the IP3-gated calcium channel ITPR1 (Inositol 1,4,5-trisphosphate (IP3) receptor type 1), boosting intracellular calcium ion</p>Formula:C22H29N3O3Color and Shape:SolidMolecular weight:383.49CFTR corrector 6
CAS:<p>CFTR corrector 6, a potent CFTR potentiator, aids cystic fibrosis research and related disorders.</p>Formula:C22H13F4N9Color and Shape:SolidMolecular weight:479.39MK-2295
CAS:<p>MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.</p>Formula:C27H31FN6O2Purity:98.83% - 99.44%Color and Shape:SolidMolecular weight:490.57(Rac)-AMG8379
CAS:<p>(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.</p>Formula:C25H16ClF2N3O5SPurity:99.6%Color and Shape:SolidMolecular weight:543.93Lingdolinurad
CAS:<p>Lingdolinurad is a uric acid transporter protein inhibitor targeting hURAT1 for the study of hyperuricemia or gout.</p>Formula:C17H12BrN3O2Purity:96.26%Color and Shape:SolidMolecular weight:370.2XR9051 Hydrochloride
CAS:<p>XR9051 Hydrochloride, a potent modulator of P-glycoprotein-mediated multidrug resistance (MDR), inhibits the binding of cytotoxics to P-glycoprotein.</p>Formula:C39H39ClN4O5Color and Shape:SolidMolecular weight:679.21(R)-Vanzacaftor
CAS:<p>(R)-Vanzacaftor ((R)-VX-121) is a cystic fibrosis transmembrane conductance regulator (CFTR) modulator [1].</p>Formula:C32H39N7O4SColor and Shape:SolidMolecular weight:617.76VU6007477
CAS:<p>VU6007477: M1 PAM, EC50=230 nM, min. agonist activity, penetrates CNS, no seizure AEs.</p>Formula:C24H26N6O2Color and Shape:SolidMolecular weight:430.5JYL-1511
CAS:<p>JYL-1511 is the TRPV1 channel partial agonist.</p>Formula:C21H29N3O3S2Purity:98%Color and Shape:SolidMolecular weight:435.6Naltiazem
CAS:<p>Naltiazem, a calcium channel antagonist, is used potentially for the treatment of arrhythmias, hypertension and myocardial infarction.</p>Formula:C26H28N2O4SPurity:98%Color and Shape:SolidMolecular weight:464.58BMT-108908
CAS:<p>BMT-108908 is a Negative Allosteric Modulator. It is selective for the NR2B Subtype of The NMDA Receptor Impair Cognition in Multiple Domains.</p>Formula:C22H25FN2O2Color and Shape:SolidMolecular weight:368.44TRPC5 modulator-1
CAS:<p>TRPC5 modulator-1 (Compound 9) is a TRPC5 modulator (IC50<1 nM) that can be used to study neuropsychiatric disorders.</p>Formula:C23H27FN2O4Color and Shape:SolidMolecular weight:414.47DPO-1
CAS:<p>DPO-1 可以高效抑制电压门控钾离子通道Kv1.5，也可以阻断超快速延迟整流钾电流。它能够预防房性心律失常。</p>Formula:C22H29OPPurity:99.78%Color and Shape:SolidMolecular weight:340.44CGP 55845 hydrochloride
CAS:<p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>Formula:C18H23Cl3NO3PColor and Shape:SolidMolecular weight:438.71γ-Kainylglutamic acid
CAS:<p>gamma-Kainylglutamic acid is a selective amino acid-induced neuroexcitation antagonist.</p>Formula:C15H22N2O7Purity:98%Color and Shape:SolidMolecular weight:342.34CRF1 receptor antagonist-1
CAS:<p>CRF1 Receptor Antagonist-1 (Compound 2), a CRF1 receptor antagonist, is utilized in research pertaining to congenital adrenal hyperplasia (CAH) [1].</p>Formula:C27H28ClFN2O2SPurity:98%Color and Shape:SolidMolecular weight:499.04
