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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2277 products of "Membrane Transporter/Ion Channel"

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  • ATPase-IN-5

    CAS:
    <p>ATPase-IN-5 (Compound 11) is an antifungal Pma1p (H+ -ATPase) inhibitor (IC50 = 12.7 μM) that inhibits the growth of Candida albicans and Saccharomyces cerevisiae.</p>
    Formula:C10H10N4O3S
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:266.28
  • PDE1-IN-4


    <p>PDE1-IN-4: inhibits PDE1C/A/B with IC50s 10/145/354 nM, may help study idiopathic pulmonary fibrosis.</p>
    Formula:C33H33N3O4
    Color and Shape:Solid
    Molecular weight:535.63
  • P2X receptor-1


    <p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>
    Formula:C14H14ClN3O3S2
    Color and Shape:Solid
    Molecular weight:371.86
  • 5-O-Desmethyl donepezil

    CAS:
    <p>5-O-Desmethyl donepezil is a metabolite of Donepezil that acts as an inhibitor of hERG channels, with an IC50 of 1.5 μM.</p>
    Formula:C23H27NO3
    Color and Shape:Solid
    Molecular weight:365.465
  • ICA-105665

    CAS:
    <p>ICA-105665 is an orally active Kv7.2/7.3/7.5 channel opener, CNS-penetrant with antiseizure effects, and low hepatocyte cytotoxicity.</p>
    Formula:C19H15F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.34
  • GNE-616

    CAS:
    <p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>
    Formula:C24H23F4N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.53
  • (RS)-AMPA hydrobromide

    CAS:
    AMPAR agonist
    Formula:C7H11BrN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.08
  • KV1.3-IN-2

    CAS:
    <p>KV1.3-IN-2 (Compound I) selectively inhibits the kv1.3 potassium channel without affecting the hERG channel. It is applicable in research related to immune-associated diseases such as psoriasis, rheumatoid arthritis, and systemic lupus erythematosus.</p>
    Formula:C16H23ClN2O4
    Color and Shape:Solid
    Molecular weight:342.818
  • Opakalim

    CAS:
    <p>Opakalim is an activator of potassium channels (potassium channel) and exhibits anticonvulsant activity.</p>
    Formula:C18H22F2N4O
    Color and Shape:Solid
    Molecular weight:348.39
  • WS-898


    <p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>
    Formula:C33H25N7OS
    Color and Shape:Solid
    Molecular weight:567.66
  • Blixeprodil

    CAS:
    <p>Blixeprodil (GM-1020) is an orally active NMDA receptor antagonist with an affinity of Ki = 3.25 µM in rat cortical tissue. It inhibits NR1/2A-NMDAR-mediated currents in HEK293 cells with an IC50 of 1.192 µM. Blixeprodil demonstrates antidepressant effects in rat models and exhibits blood-brain barrier permeability.</p>
    Formula:C13H16FNO
    Color and Shape:Solid
    Molecular weight:221.271
  • IAA65

    CAS:
    <p>IAA65 is a potent inhibitor of T-type calcium channels, exhibiting an IC50 value of 18.9 μM, and holds potential for use in epilepsy research [1].</p>
    Formula:C16H13F6NO2
    Color and Shape:Solid
    Molecular weight:365.27
  • VU0463271 quarterhydrate


    <p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>
    Formula:C19H20N4O2S2
    Color and Shape:Solid
    Molecular weight:387
  • V-ATPase-IN-1

    CAS:
    <p>V-ATPase-IN-1 (Compound 3b-03) is an inhibitor of Vacuolar-type H+-ATPases (V-ATPase), exhibiting an inhibition constant (IC50) of 194.80 μM and effectively targeting the V-ATPase subunit A with a dissociation constant (Kd) of 0.803 μM. This compound demonstrates insecticidal activity against M. separata (LC50 = 2.64 mM), aiding in the development of chemical insecticides.</p>
    Formula:C21H20ClNO2
    Color and Shape:Solid
    Molecular weight:353.84
  • (S)-Albuterol

    CAS:
    <p>(S)-Albuterol functions as a muscarinic receptor and phospholipase C activator, enhancing the intracellular free calcium concentration in airway smooth muscle cells.</p>
    Formula:C13H21NO3
    Color and Shape:Solid
    Molecular weight:239.311
  • Lubeluzole dihydrochloride

    CAS:
    <p>Lubeluzole (dihydrochloride) acts as a neuroprotective agent by blocking neuronal voltage-gated sodium channels and also affects cardiac sodium channels, exhibiting both tonic and blocking effects. This compound is considered promising in the research of antiarrhythmic agents.</p>
    Formula:C22H27Cl2F2N3O2S
    Color and Shape:Solid
    Molecular weight:506.44
  • Kv7.2/Kv7.3 activator-1

    CAS:
    <p>Kv7.2/Kv7.3 Activator-1 (compound 517) serves as a powerful activator of the Kv7.2/Kv7.3 channels, exhibiting an EC50 value of less than 1 µM. It holds potential for use in neurological disease research.</p>
    Formula:C19H22F2N4O
    Color and Shape:Solid
    Molecular weight:360.40
  • PF-05661014

    CAS:
    <p>PF-05661014, a demethylated analogue of PF-06526290, selectively inhibits Nav1.3 and Nav1.7 currents by stabilizing the inactivated state through interaction with the D4 VSD. This compound is utilized in research focused on sodium channel modulation.</p>
    Formula:C17H16N4O3S2
    Color and Shape:Solid
    Molecular weight:388.46
  • CFTR corrector 16

    CAS:
    <p>CFTRcorrector 16 (Compound 39) is a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR), utilized in the research of cystic fibrosis disease.</p>
    Formula:C27H26ClN5O2S
    Color and Shape:Solid
    Molecular weight:520.05
  • SP100030 analogue 1

    CAS:
    SP100030 analogue 1 (compound 11) is a selective transcription activation (SITA) inhibitor within the SP100030 class, capable of inhibiting XPO1-dependent upregulation of IL2 in a Jurkat-based IL2-Luc reporter assay, with an EC50 of 137 nM.
    Formula:C13H5ClF7N3O
    Color and Shape:Solid
    Molecular weight:387.64
  • CFTR corrector 15

    CAS:
    <p>CFTR Corrector 15 (Compound 4172) serves as a corrector for cystic fibrosis transmembrane conductance regulator (CFTR). When used in combination with VX-809, it addresses the folding defects of F508del-CFTR. CFTR Corrector 15 is also applicable in the research of cystic fibrosis.</p>
    Formula:C24H22ClN5O2S
    Color and Shape:Solid
    Molecular weight:479.98
  • (2S,3S,11bR)-Dihydrotetrabenazine

    CAS:
    <p>(2S,3S,11bR)-Dihydrotetrabenazine ((2S,3S,11bR)-DHTBZ) is a highly selective inhibitor of vesicular monoamine transporter 2 (VMAT2) with a Ki value of 593 nM. It suppresses the vesicular transport of monoamine neurotransmitters, such as dopamine and serotonin, leading to reduced release into the synaptic cleft. This compound holds potential for research in Huntington's disease and other hyperkinetic movement disorders.</p>
    Formula:C19H29NO3
    Color and Shape:Solid
    Molecular weight:319.44
  • S 0960

    CAS:
    <p>S 0960 is a dimeric bile acid analogue, a specific inhibitor of the sodium-dependent bile salt transporter in the ileum, used in metabolic disease research.</p>
    Formula:C48H79NO8
    Purity:99.32% - >99.99%
    Color and Shape:Solid
    Molecular weight:798.14
  • PF-06462894

    CAS:
    PF-06462894: morpholinopyrimidone, mGlu5 antagonist (Ki=6nM), no immune activation in mouse model.
    Formula:C18H23N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.39
  • 2-PPA

    CAS:
    2-PPA serves as a selective TMEM175 inhibitor (IC 50 =32 μM), primarily influencing lysosomal activity. Through acute inhibition of TMEM175, 2-PPA enhances lysosomal macromolecular catabolism, which in turn boosts macrophage activity and other digestive processes. This compound holds significance in Parkinson's disease research.
    Formula:C11H10N2
    Color and Shape:Solid
    Molecular weight:170.21
  • Caramboxin

    CAS:
    <p>Caramboxin, a neurotoxin, can induce acute kidney injury.</p>
    Formula:C11H13NO6
    Color and Shape:Solid
    Molecular weight:255.22
  • Dehydroindapamide

    CAS:
    <p>Dehydroindapamide, an indole form of Indapamide, is utilized to quantify the turnover rate of Indapamide in CYP3A4, which is approximately 10 times higher than that of Indoline, with slightly enhanced affinity for CYP3A4.</p>
    Formula:C16H14ClN3O3S
    Color and Shape:Solid
    Molecular weight:363.82
  • Perfluoroheptanesulfonic acid

    CAS:
    <p>Perfluoroheptanesulfonic acid (1-Perfluoroheptanesulfonic acid; Perfluoroheptanesulphonic acid) is a perfluoroalkyl substance (PFAS). This compound has been detected in landfill leachate and has been shown to induce deformities in zebrafish larvae (EC50=168.1 μM). Exposure to PFHpS in fetuses can lead to reduced birth weight.</p>
    Formula:C7HF15O3S
    Color and Shape:Solid
    Molecular weight:450.12
  • ZK 93426 hydrochloride

    CAS:
    <p>benzodiazepine receptor antagonist,competitive</p>
    Formula:C18H21ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.82
  • CAD204520

    CAS:
    <p>CAD204520 functions as an inhibitor of SERCA (IC50 = 0.34 μM), specifically targeting mutations in the wild-type NOTCH1 protein associated with T-cell acute lymphoblastic leukemia (T-ALL) and mantle cell lymphoma (MCL).</p>
    Formula:C23H32F3N3O2
    Color and Shape:Solid
    Molecular weight:439.51
  • AP-6

    CAS:
    AP-6, a selective TMEM175 inhibitor, enhances lysosomal macromolecular catabolism by acutely inhibiting TMEM175, thus speeding up macrophage and other digestive activities. This compound holds potential for use in Parkinson's disease research due to its role in modulating lysosomal function.
    Formula:C16H14N4
    Color and Shape:Solid
    Molecular weight:262.31
  • AN-988

    CAS:
    <p>AN-988 (compound 6) is a covalent CRM1 inhibitor.</p>
    Formula:C22H22N2O4S
    Color and Shape:Solid
    Molecular weight:410.49
  • Fletazepam

    CAS:
    <p>Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.</p>
    Formula:C17H13ClF4N2
    Color and Shape:Solid
    Molecular weight:356.74
  • SOAT-IN-1

    CAS:
    <p>SOAT-IN-1 (compound 40) is a potent and selective inhibitor targeting the sodium-dependent organic anion transporter (SOAT), exhibiting IC50 values of 1.6 µM for SOAT and 14.3 µM for NTCP.</p>
    Formula:C20H16ClN3O6S
    Color and Shape:Solid
    Molecular weight:461.88
  • LY 215490

    CAS:
    <p>LY 215490 is a selective AMPA receptor antagonist with neuroprotective properties in rat ischemia.</p>
    Formula:C13H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.34
  • Lorajmine

    CAS:
    <p>Lorajmine, a monochloroacetyl derivative of ajmaline, is a class Ia antiarrhythmic agent that is rapidly hydrolyzed to ajmaline by plasma and tissue esterases.</p>
    Formula:C22H27ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.91
  • PD-217014

    CAS:
    <p>PD-217014 is an α2δ ligand that exhibits visceral analgesic activity and can suppress visceral hypersensitivity. Its antihyperalgesic effects are dose-dependent.</p>
    Formula:C10H17NO2
    Color and Shape:Solid
    Molecular weight:183.25
  • SDZ 220-040

    CAS:
    <p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂,可诱导根系生长的部分无重力模式 。</p>
    Formula:C16H16Cl2NO6P
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:420.18
  • Suzetrigine

    CAS:
    <p>Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.</p>
    Formula:C21H20F5N3O4
    Purity:98.08% - 99.27%
    Color and Shape:Solid
    Molecular weight:473.39
  • Odevixibat

    CAS:
    <p>Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.</p>
    Formula:C37H48N4O8S2
    Purity:99.53% - 99.83%
    Color and Shape:Solid
    Molecular weight:740.93
  • (+)-Tetrabenazine

    CAS:
    <p>(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold</p>
    Formula:C19H27NO3
    Purity:98.31%
    Color and Shape:Solid
    Molecular weight:317.42
  • SYM2206

    CAS:
    <p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>
    Formula:C20H22N4O3
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:366.41
  • 5-Hydroxylansoprazole

    CAS:
    <p>5-Hydroxylansoprazole (AG1908) is the active metabolite of plasma Lansoprazole, inhibits the proton pump, and is used in the study of peptic ulcers.</p>
    Formula:C16H14F3N3O3S
    Purity:99.00%
    Color and Shape:Solid
    Molecular weight:385.36

    Ref: TM-T14051

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  • A-887826

    CAS:
    <p>A-887826 is a selective, orally bioavailable, and voltage-dependent Na(v1.8) channel blocker (IC50: 11 nM). It attenuates neuropathic tactile allodynia in vivo.</p>
    Formula:C26H29ClN4O3
    Color and Shape:Solid
    Molecular weight:480.99

    Ref: TM-T10209

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  • (-)-Bicuculline methobromide

    CAS:
    <p>(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .</p>
    Formula:C21H20BrNO6
    Color and Shape:White
    Molecular weight:462.29

    Ref: TM-T12043

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  • Umbellulone

    CAS:
    <p>Umbellulone is a natural product isolated from Umbellularia californica, and stimulates the TRPA1 channel in a subset of peptidergic, nociceptive neurons, activating the trigeminovascular system via this mechanism.</p>
    Formula:C10H14O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:150.22

    Ref: TM-T13953

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  • Indapamide

    CAS:
    <p>Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.</p>
    Formula:C16H16ClN3O3S
    Purity:98.97% - 99.83%
    Color and Shape:Solid
    Molecular weight:365.83

    Ref: TM-T1498

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  • Filapixant

    CAS:
    <p>Filapixant, a purinoreceptor antagonist. This compound serves as the active reference substance for Eliapixant.</p>
    Formula:C24H26F3N5O3S
    Color and Shape:Solid
    Molecular weight:521.56

    Ref: TM-T39357

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  • 3-Methylglutaconic acid

    CAS:
    <p>3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].</p>
    Formula:C6H8O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:144.13

    Ref: TM-T78071

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  • Zastaprazan

    CAS:
    <p>Zastaprazan (JP-1366, compound 6) is a potassium-competitive acid blocker and proton pump inhibitor that suppresses gastric acid secretion, indicated for GERD.</p>
    Formula:C22H26N4O
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:362.48

    Ref: TM-T39583

    ne
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  • Verapamil EP Impurity C hydrochloride

    CAS:
    <p>NSC-609249 hydrochloride, an impurity of Verapamil, is a calcium channel blocker with potent orally active properties. It also functions as a first-generation P-glycoprotein (P-gp) inhibitor.</p>
    Formula:C12H20ClNO2
    Color and Shape:Solid
    Molecular weight:245.75

    Ref: TM-T40591

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  • (Rac)-Lanicemine

    CAS:
    <p>(Rac)-Lanicemine ((Rac)-AZD6765) is the racemate of Lanicemine. Lanicemine (AZD6765) is a low-trapping NMDA channel blocker with a Ki of 0.56-2.1 μM for the NMDA receptor and IC50 values of 4-7 μM and 6.4 μM in CHO and Xenopus oocyte cells, respectively. Lanicemine shows antidepressant effects [1].</p>
    Formula:C13H14N2
    Color and Shape:Solid
    Molecular weight:198.26

    Ref: TM-T60235

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  • 2-AEMP TFA

    CAS:
    <p>2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.</p>
    Formula:C3H10NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:139.091

    Ref: TM-T26380

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  • L-Cysteine S-sulfate sodium salt sesquihydrate

    CAS:
    <p>L-Cysteine S-sulfate sodium salt sesquihydrate is a useful organic compound for research related to life sciences. The catalog number is T64782 and the CAS number is 150465-29-5.</p>
    Formula:C9H25N3Na3O17S6
    Color and Shape:Solid
    Molecular weight:708.63

    Ref: TM-T64782

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  • Apcin A HCL

    CAS:
    <p>Apcin A HCL is an Apcin derivative. Apcin A HCL is an anaphase-promoting complex (APC) inhibitor. Apcin-A HCL interacts strongly with Cdc20, and inhibits the ubiquitination of Cdc20 substrates. Apcin-A HCL can be used to synthesize the PROTAC CP5V [1].</p>
    Formula:C10H15Cl4N5O2
    Purity:99.30%
    Color and Shape:Solid
    Molecular weight:379.07

    Ref: TM-T001

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  • Indoxacarb

    CAS:
    <p>Indoxacarb is an Oxadiazine insecticide.</p>
    Formula:C22H17ClF3N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.83

    Ref: TM-T20895

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  • GNE-9278

    CAS:
    <p>GNE-9278 is a highly selective NMDAR orthosteric modulator that targets the GluN1 transmembrane structural domain (TMD), enhancing peak current and agonist affinity in activated NMDAR.</p>
    Formula:C21H27N5O3S
    Color and Shape:Solid
    Molecular weight:429.54

    Ref: TM-T62376

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  • PF-06761281

    CAS:
    <p>PF-06761281 is a partially selective sodium-coupled citrate transporter protein (NaCT/SLC13A5) inhibitor, oral, reducing plasma glucose concentration.</p>
    Formula:C13H17NO6
    Color and Shape:Solid
    Molecular weight:283.28

    Ref: TM-T60547

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  • Alfadolone acetate

    CAS:
    <p>Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.</p>
    Formula:C23H34O5
    Color and Shape:Solid
    Molecular weight:390.51

    Ref: TM-T26592

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  • (±)​-​Vasicine

    CAS:
    <p>(±)-Vasicine, the racemate of Vasicine, is isolated from Peganum harmala seeds and exhibits anti-ulcer activity.</p>
    Formula:C11H12N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:188.23

    Ref: TM-T12681

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  • CGP 44532

    CAS:
    <p>CGP 44532 a GABAB receptor agonist.</p>
    Formula:C4H12NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:153.12

    Ref: TM-T26991

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  • Gacyclidine

    CAS:
    <p>Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.</p>
    Formula:C16H25NS
    Purity:99.85% - 99.92%
    Color and Shape:Solid
    Molecular weight:263.44

    Ref: TM-T27397

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  • CMPDA

    CAS:
    <p>CMPDA is a positive allosteric modulator of AMPA receptors [EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor].</p>
    Formula:C16H28N2O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.53

    Ref: TM-TQ0114

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  • T16A(inh)-C01

    CAS:
    <p>T16A(inh)-C01 is the Ca(2+)-activated Cl(-) Channel, Ano1 class C inhibitor.</p>
    Formula:C18H16O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.32

    Ref: TM-T24846

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  • Fostedil

    CAS:
    <p>Fostedil enhances heart function, maintains blood flow during partial/total coronary occlusions, and lowers aortic pressure.</p>
    Formula:C18H20NO3PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.4

    Ref: TM-T27351

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  • Motugivatrep

    CAS:
    <p>Motugivatrep is a potent and selective TRPV1 antagonist that can be used to study TRPV1-related respiratory diseases.</p>
    Formula:C22H20F3NO3
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:403.39

    Ref: TM-T64312

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  • Tifenazoxide

    CAS:
    <p>Tifenazoxide is an effective and SUR1/Kir6.2 selective KATP channels opener. Tifenazoxide has an anti-diabetic effect, can inhibit glucose-stimulated insulin release in vitro and in vivo.</p>
    Formula:C9H10ClN3O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.78

    Ref: TM-T17094

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  • Pazinaclone

    CAS:
    <p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>
    Formula:C25H23ClN4O4
    Purity:97.79% - 99.07%
    Color and Shape:Solid
    Molecular weight:478.93

    Ref: TM-T28303

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  • Phenamil methanesulfonate

    CAS:
    <p>TRPP3 channel inhibitor</p>
    Formula:C13H16ClN7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.83

    Ref: TM-T23148

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Pipequaline

    CAS:
    <p>Pipequaline (PK-8165) is an anticonflict &amp; anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.</p>
    Formula:C22H24N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:316.44

    Ref: TM-T4655

    5mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • Xilmenolone

    CAS:
    <p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>
    Formula:C26H37N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:423.59

    Ref: TM-T78670

    5mg
    Discontinued
    25mg
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    50mg
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    100mg
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    Discontinued product
  • LFS-1107

    CAS:
    <p>LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering potential for cancer research applications [1].</p>
    Formula:C12H11N5OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:305.38

    Ref: TM-T81936

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • Belfosdil

    CAS:
    <p>Belfosdil is a blocker of antihypertensive calcium channel.</p>
    Formula:C27H50O7P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.63

    Ref: TM-T26764

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • CGP 56999A

    CAS:
    <p>CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.</p>
    Formula:C19H30NO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.42

    Ref: TM-T26993

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • HMR 1556

    CAS:
    <p>HMR 1556 is a chromanol derivative and is an IKs blocker (IC50s of 10.5 nM and 34 nM in canine and guinea pig left ventricular myocytes, respectively).</p>
    Formula:C17H24F3NO5S
    Color and Shape:Solid
    Molecular weight:411.44

    Ref: TM-T15487

    1mg
    Discontinued
    Discontinued product
  • VMAT2-IN-2 tosylate

    CAS:
    <p>VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].</p>
    Formula:C27H36F3NO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:559.64

    Ref: TM-T79061

    5mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Bumetanide sodium

    CAS:
    <p>Bumetanide sodium, a potent diuretic, blocks NKCC1 (IC50: 0.68 μM) and NKCC2 (IC50: 4.0 μM).</p>
    Formula:C17H19N2NaO5S
    Color and Shape:Solid
    Molecular weight:386.4

    Ref: TM-T61713

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product