Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(101 products)
- Adiponectin receptor(5 products)
- CFTR(65 products)
- CGRP Receptor(54 products)
- Calcium Channel(541 products)
- Chloride channel(53 products)
- GABA Receptor(366 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(54 products)
- Potassium Channel(280 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(209 products)
- TRP/TRPV Channel(95 products)
Show 13 more subcategories
Found 2507 products of "Membrane Transporter/Ion Channel"
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ML418
CAS:ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.Formula:C19H24ClN3O3Purity:99.3%Color and Shape:SolidMolecular weight:377.87Z433927330
CAS:<p>Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).</p>Formula:C20H20N4O3Purity:99.78%Color and Shape:SolidMolecular weight:364.4Prilocaine hydrochloride
CAS:Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Formula:C13H21ClN2OPurity:99.97%Color and Shape:Needles White Or Off White Crystalline PowderMolecular weight:256.77IK1 inhibitor PA-6
CAS:IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouseFormula:C31H32N4O2Purity:98.9%Color and Shape:SolidMolecular weight:492.61Dooku1
CAS:Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.Formula:C13H9Cl2N3OSPurity:98.87% - 99.74%Color and Shape:SolidMolecular weight:326.2Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Formula:C20H16Cl2F3N3O3Purity:99.49%Color and Shape:SolidMolecular weight:474.26AZD 7009
CAS:AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.Formula:C23H34N4O5Purity:98.42% - 98.51%Color and Shape:SoildMolecular weight:446.54Tocainide hydrochloride
CAS:<p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>Formula:C11H17ClN2OPurity:97%Color and Shape:SolidMolecular weight:228.72Manidipine dihydrochloride
CAS:Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).Formula:C35H40Cl2N4O6Purity:99.76% - 99.86%Color and Shape:SolidMolecular weight:683.62Torsemide
CAS:<p>Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.</p>Formula:C16H20N4O3SPurity:99.81%Color and Shape:Crystalline SolidMolecular weight:348.42DSP-2230
CAS:<p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>Formula:C20H20F3N5O2Purity:97.14%Color and Shape:SolidMolecular weight:419.4Penicillin G sodium salt
CAS:<p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>Formula:C16H17N2NaO4SPurity:98.11%Color and Shape:White To Off-White Crystalline PowderMolecular weight:356.37Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formula:C10H12ClNO2Purity:98% - >99.99%Color and Shape:1992)Molecular weight:213.66NS13001
CAS:NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).Formula:C17H16ClN7Purity:99.55%Color and Shape:SolidMolecular weight:353.81Pramocaine hydrochloride
CAS:Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.Formula:C17H27NO3·HClPurity:99.15% - 99.61%Color and Shape:Crystals White Or Off White Crystalline PowderMolecular weight:329.86Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormula:C15H14FN3O3Purity:99.72% - 99.98%Color and Shape:Less Crystals Colourless CrystalsMolecular weight:303.294-Aminopyridine
CAS:4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.Formula:C5H6N2Purity:91.61%Color and Shape:SolidMolecular weight:94.11Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Formula:C11H15NO5Purity:99.96%Color and Shape:Crystals From Benzene SolidMolecular weight:241.24γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Formula:C4H9NO2Purity:99.95%Color and Shape:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderMolecular weight:103.12Clorsulon
CAS:Clorsulon (L631529) is utilized for the treatment of Fasciola hepatica infections in calves and sheep.Formula:C8H8Cl3N3O4S2Purity:99.66% - 99.87%Color and Shape:White To Off-White Crystalline PowderMolecular weight:380.66
