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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2507 products of "Membrane Transporter/Ion Channel"

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  • Flindokalner

    CAS:
    Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.
    Formula:C16H10ClF4NO2
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:359.7
  • Flumazenil

    CAS:
    Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous
    Formula:C15H14FN3O3
    Purity:99.72% - 99.98%
    Color and Shape:Less Crystals Colourless Crystals
    Molecular weight:303.29
  • NS5806

    CAS:
    NS5806 activates K+ currents, slows KV4.2/4.3 decay with KChIP2, and boosts KV4.3/KChIP2 peaks (EC50=5.3μM).
    Formula:C16H8Br2F6N6O
    Purity:97.95%
    Color and Shape:Solid
    Molecular weight:574.07
  • Eleclazine hydrochloride

    CAS:
    Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).
    Formula:C21H17ClF3N3O3
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:451.83
  • Cycloleucine

    CAS:
    Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.
    Formula:C6H11NO2
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:129.16
  • Dooku1

    CAS:
    Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.
    Formula:C13H9Cl2N3OS
    Purity:98.87% - 99.74%
    Color and Shape:Solid
    Molecular weight:326.2
  • Ciclopirox olamine

    CAS:
    Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.
    Formula:C14H24N2O3
    Purity:99.16% - >99.99%
    Color and Shape:White To Yellow Solid Solid Particulate/Powder
    Molecular weight:268.35
  • VU6036720


    <p>VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit</p>
    Formula:C20H22ClFN4O2S
    Purity:98.1%
    Color and Shape:Soild
    Molecular weight:436.93
  • Penicillin G sodium salt

    CAS:
    <p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>
    Formula:C16H17N2NaO4S
    Purity:98.11%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:356.37
  • Baclofen

    CAS:
    Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.
    Formula:C10H12ClNO2
    Purity:98% - >99.99%
    Color and Shape:1992)
    Molecular weight:213.66
  • AZD 7009

    CAS:
    AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.
    Formula:C23H34N4O5
    Purity:98.42% - 98.51%
    Color and Shape:Soild
    Molecular weight:446.54
  • Ethaverine hydrochloride

    CAS:
    Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.
    Formula:C24H30ClNO4
    Purity:99.66% - 99.90%
    Color and Shape:Solid
    Molecular weight:431.96
  • Prilocaine hydrochloride

    CAS:
    Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.
    Formula:C13H21ClN2O
    Purity:99.97%
    Color and Shape:Needles White Or Off White Crystalline Powder
    Molecular weight:256.77
  • Diphenidol hydrochloride

    CAS:
    Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.
    Formula:C21H28ClNO
    Purity:99.15% - 99.33%
    Color and Shape:Crystals Soluble In Methanol Water
    Molecular weight:345.91
  • Bupivacaine hydrochloride

    CAS:
    Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.
    Formula:C18H28N2O·HCl
    Purity:99.89% - 99.9%
    Color and Shape:Solid
    Molecular weight:324.89
  • CIQ

    CAS:
    CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.
    Formula:C26H26ClNO5
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:467.94
  • Bemegride

    CAS:
    Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.
    Formula:C8H13NO2
    Purity:99.89%
    Color and Shape:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)
    Molecular weight:155.19
  • IK1 inhibitor PA-6

    CAS:
    IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse
    Formula:C31H32N4O2
    Purity:98.9%
    Color and Shape:Solid
    Molecular weight:492.61
  • NBQX disodium

    CAS:
    NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and anticonvulsant activity.
    Formula:C12H6N4Na2O6S
    Purity:97.32% - 97.6%
    Color and Shape:Solid
    Molecular weight:380.2415
  • FG 7142

    CAS:
    <p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>
    Formula:C13H11N3O
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:225.25