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Neuroscience

Neuroscience

Neuroscience inhibitors are compounds designed to modulate the activity of specific proteins, enzymes, or receptors within the nervous system. These inhibitors are crucial for studying the molecular mechanisms underlying neural function, synaptic transmission, and neurodegenerative diseases. By targeting neurotransmitter receptors, ion channels, and signaling pathways, neuroscience inhibitors aid in the exploration of brain function and the development of therapeutic strategies for neurological disorders such as Alzheimer's, Parkinson's, and epilepsy. At CymitQuimica, we offer a comprehensive range of high-quality neuroscience inhibitors to support your research in neurobiology, neuropharmacology, and cognitive sciences.

Subcategories of "Neuroscience"

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Found 5389 products of "Neuroscience"

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  • CBP501

    CAS:
    <p>CBP501 peptide inhibits kinases like MAPKAP-K2/C-Tak1/CHK1, preventing Cdc25C function and blocking the entry into mitosis.</p>
    Formula:C86H122F5N29O17
    Color and Shape:Solid
    Molecular weight:1929.06
  • ST1936

    CAS:
    <p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>
    Formula:C13H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.74
  • GR-55562 dihydrobromide

    CAS:
    <p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>
    Formula:C23H26ClN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.93
  • Glutaminyl Cyclase Inhibitor 5


    <p>Glutaminyl Cyclase Inhibitor 5 is a potent, selective inhibitor of human glutaminyl cyclase (hQC), demonstrating an inhibition concentration half-max (IC 50) of</p>
    Formula:C22H30N6O
    Color and Shape:Solid
    Molecular weight:394.51
  • Safrazine

    CAS:
    <p>Safrazine is an irreversible, non-specific and orally active monoamine oxidase (MAO) inhibitor. Safrazine can be used in depression research[1].</p>
    Formula:C11H16N2O2
    Color and Shape:Solid
    Molecular weight:208.26
  • AChE/BChE-IN-5

    CAS:
    <p>AChE/BChE-IN-5 (BMC-16) crosses BBB; IC50: hAChE 266 nM, hBChE 10.6 nM. Dual AChE/BChE inhibitor.</p>
    Formula:C17H26N2O3
    Color and Shape:Solid
    Molecular weight:306.4
  • UCSF686

    CAS:
    <p>UCSF686, a UCSF678 analog, lacks 5-HT5A potency but keeps affinity for 5-HT1A, 5-HT2B, 5-HT7, and serves as a control.</p>
    Formula:C14H19N3O2S
    Color and Shape:Solid
    Molecular weight:293.38
  • WAY-361789

    CAS:
    <p>WAY-361789 is an agonist of alpha7 nicotinic acetylcholine receptor.</p>
    Formula:C22H31N5O3
    Color and Shape:Solid
    Molecular weight:413.51
  • AS19

    CAS:
    <p>AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).</p>
    Formula:C18H25N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.41
  • Etbicyphat

    CAS:
    <p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>
    Formula:C6H11O4P
    Color and Shape:Solid
    Molecular weight:178.12
  • Piperilate

    CAS:
    <p>Piperilate (Pipethanate), a hetrazepine PAF antagonist and anticholinergic used in asthma studies, counters organophosphate toxicity.</p>
    Formula:C21H25NO3
    Color and Shape:Solid
    Molecular weight:339.43
  • DMeOB

    CAS:
    DMeOB (3,3'-Dimethoxybenzaldazine) is a negative regulator with mGluR5 agonist activity and is used in the study of neurological disorders.
    Formula:C16H16N2O2
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:268.31
  • GW791343 trihydrochloride

    CAS:
    GW791343 trihydrochloride (GW791343 3HCl) is aHCl salt form of GW791343, which is a non-competitive allosteric modulator of human P2X7 receptor inhibitor with
    Formula:C20H24F2N4O·3HCl
    Purity:98%
    Color and Shape:Solid
    Molecular weight:483.81
  • JNJ-40068782

    CAS:
    <p>JNJ-40068782 is a potent, selective and systemically active positive allosteric modulator of the mGlu2 receptor.</p>
    Formula:C21H23N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.43
  • Distigmine Bromide

    CAS:
    <p>Distigmine Bromide is an acetylcholinesterase inhibitor. It is used for the treatment of underactive neurogenic bladder and myasthenia gravis.</p>
    Formula:C22H32BrN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:496.42
  • LY 2087101

    CAS:
    <p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>
    Formula:C15H11FN2OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.39
  • Pruvanserin hydrochloride

    CAS:
    <p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>
    Formula:C22H22ClFN4O
    Purity:99.6%
    Color and Shape:Solid
    Molecular weight:412.89
  • W-5 hydrochloride

    CAS:
    <p>W-5 hydrochloride (N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl) is a potent calmodulin antagonist.</p>
    Formula:C16H23ClN2O2S
    Purity:99.35%
    Color and Shape:Off-White Crystalline Solid
    Molecular weight:342.88
  • 5-Iodo-A-85380 dihydrochloride

    CAS:
    α4β2 and α6β2 nicotinic acetylcholine receptors agonist
    Formula:C9H13Cl2IN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.02
  • BChE-IN-4

    CAS:
    <p>BChE-IN-4, a potent butyrylcholinesterase inhibitor, crosses blood-brain barrier, improves memory in mice; promising for Alzheimer's research.</p>
    Formula:C24H37N3O
    Color and Shape:Solid
    Molecular weight:383.57
  • Oxybutynin R-isomer HCl

    CAS:
    <p>Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.</p>
    Formula:C22H32ClNO3
    Color and Shape:Solid
    Molecular weight:393.95
  • Irindalone

    CAS:
    <p>IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.</p>
    Formula:C24H29FN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.51
  • LY456066

    CAS:
    <p>LY456066 is a mGluR1 receptor-selective, negative allosteric modulator.</p>
    Formula:C19H23N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.47
  • S16961

    CAS:
    <p>S16961 (S169611) is an agonist of nicotinic receptor.</p>
    Formula:C41H71NO6
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:674.01
  • (1R,2S)-VU0155041

    CAS:
    <p>(1R,2S)-VU0155041 is the cis regioisomer of VU0155041 and a partial agonist of mGluR4.</p>
    Formula:C14H15Cl2NO3
    Purity:98.85%
    Color and Shape:Solid
    Molecular weight:316.18
  • Ampreloxetine

    CAS:
    <p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>
    Formula:C18H18F3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.34
  • ATC0065 HCl

    CAS:
    <p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>
    Formula:C25H31BrCl2F3N5O
    Color and Shape:Solid
    Molecular weight:625.35
  • SSAO inhibitor-2

    CAS:
    <p>SSAO inhibitor-2 targets human SSAO (&lt;10 nM) and MAO-A (10-100 μM); useful in various diseases research.</p>
    Formula:C14H21FN4O2
    Color and Shape:Solid
    Molecular weight:296.34
  • Pirenzepine

    CAS:
    <p>Pirenzepine targets M1 mAChR, curbs acid secretion, eases spasms, and has anti-cancer properties.</p>
    Formula:C19H21N5O2
    Color and Shape:Solid
    Molecular weight:351.4
  • BuChE-IN-4

    CAS:
    <p>BuChE-IN-4 is a potent inhibitor of BuChE (IC50: 7.7 nM) and exhibits mild antioxidant capacity, non-toxicity, lipophilicity and neuroprotective effects.</p>
    Formula:C21H21BrFN3O4S
    Color and Shape:Solid
    Molecular weight:510.38
  • Z-Cyclopentyl-AP4

    CAS:
    Group III mGlu receptor agonist
    Formula:C6H12NO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.14
  • PNU-282987 S enantiomer hydrochloride

    CAS:
    <p>(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.</p>
    Formula:C14H18Cl2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:301.21
  • Indisetron Dihydrochloride

    CAS:
    <p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>
    Formula:C17H24ClN5O
    Color and Shape:Solid
    Molecular weight:349.86
  • MAO-IN-M30 dihydrochloride

    CAS:
    <p>MAO-IN-M30 dihydrochloride: potent, brain-specific MAO-A/B inhibitor, iron chelator with antioxidant effects, counters Parkinson's in mice.</p>
    Formula:C14H16Cl2N2O
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:299.2
  • VU0400195

    CAS:
    <p>VU0400195 is a oral effective, positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu(4)).</p>
    Formula:C21H16ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.82
  • Afacifenacin

    CAS:
    <p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>
    Formula:C27H26F3N3O2
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:481.51
  • Asoxime dichloride

    CAS:
    <p>Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.</p>
    Formula:C14H16Cl2N4O3
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:359.21
  • CGP 36216 hydrochloride

    CAS:
    <p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>
    Formula:C5H14NO2P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:151.14
  • RR-11a

    CAS:
    <p>RR-11a is a synthetic enzyme Legumain inhibitor.</p>
    Formula:C24H28N6O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:560.51
  • SIB 1508Y maleate

    CAS:
    <p>neuronal nicotinic ACh receptor agonist</p>
    Formula:C16H18N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.33
  • VU0418506

    CAS:
    <p>VU0418506 is a positive allosteric modulator (PAM) of the metabotropic glutamate receptor 4 (mGlu4).</p>
    Formula:C12H8ClFN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:262.67
  • TCS 1105

    CAS:
    <p>TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.</p>
    Formula:C17H13FN2O2
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:296.3
  • AP521

    CAS:
    <p>AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).</p>
    Formula:C20H19ClN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.89
  • Pipazethate

    CAS:
    <p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>
    Formula:C21H25N3O3S
    Color and Shape:Solid
    Molecular weight:399.51
  • EMD 56551

    CAS:
    <p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>
    Formula:C24H31N3O2
    Purity:95.64% - 99.39%
    Color and Shape:Solid
    Molecular weight:393.522
  • MAO-B-IN-11

    CAS:
    <p>MAO-B-IN-11 (Compound 8c) is a strong MAO-B blocker with a 1.3 μM IC50 and neuroprotective effects.</p>
    Formula:C22H32O3
    Color and Shape:Solid
    Molecular weight:344.49
  • SGS518 oxalate

    CAS:
    <p>SGS518 oxalate is a 5-HT6 antagonist.</p>
    Formula:C23H24F2N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.51
  • LP44 hydrochloride

    CAS:
    <p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>
    Formula:C27H38ClN3OS
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:488.13
  • γ-Secretase modulator 12

    CAS:
    <p>γ-Secretase modulator 12 (Compound 1a) is a selective compound that effectively reduces amyloid-β42 (Aβ42) levels with an IC50 of 0.39 μM.</p>
    Formula:C25H23N3O2
    Color and Shape:Solid
    Molecular weight:397.47
  • WAY208466 dihydrochloride

    CAS:
    <p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>
    Formula:C17H20Cl2FN3O2S
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:420.33
  • NRA-0160

    CAS:
    <p>NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)</p>
    Formula:C24H23F2N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.52
  • (Rac)-SEP-363856

    CAS:
    <p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>
    Formula:C9H13NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:183.27
  • AY1511

    CAS:
    <p>AY1511 is a low cytotoxic inhibitor of amyloid β (Aβ) aggregation [1].</p>
    Formula:C17H14O6
    Color and Shape:Solid
    Molecular weight:314.29
  • AR-R 17779 hydrochloride

    CAS:
    <p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>
    Formula:C9H15ClN2O2
    Color and Shape:Solid
    Molecular weight:218.68
  • DFMTI

    CAS:
    <p>DFMTI can completely block the rmGlu1 L757V glutamate response.</p>
    Formula:C20H18F2N4O
    Color and Shape:Solid
    Molecular weight:368.38
  • GRN-529

    CAS:
    <p>GRN-529 is a selective negative allosteric modulator of the mGluR5 receptor.</p>
    Formula:C22H15F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.37
  • AChE/BChE-IN-2

    CAS:
    <p>AChE/BChE-IN-2 (Compound 13b) is a potent inhibitor of AChE/BChE with IC50 values of 0.96 ± 0.14 μM and 1.23 ± 0.23 μM for AChE and BChE, respectively.</p>
    Formula:C23H25N3O5
    Color and Shape:Solid
    Molecular weight:423.46
  • 2-Iodomelatonin

    CAS:
    <p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, &gt;5x selective over MT2, used to map melatonin sites in brain/tissues.</p>
    Formula:C13H15IN2O2
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:358.17
  • NNC052090

    CAS:
    <p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>
    Formula:C27H30N2O2
    Color and Shape:Solid
    Molecular weight:414.54
  • LY 302148

    CAS:
    <p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>
    Formula:C19H23FN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:326.41
  • MAO-B-IN-16

    CAS:
    <p>MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.</p>
    Formula:C18H19NO3
    Color and Shape:Solid
    Molecular weight:297.35
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Formula:C16H25ClN4O2
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:340.85
  • ML337

    CAS:
    ML337 is a negative allosteric modulator of mGlu3 with an IC50 of 593 nM.
    Formula:C21H20FNO3
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:353.39
  • VMY-2-95

    CAS:
    <p>VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.</p>
    Formula:C17H16N2O
    Color and Shape:Solid
    Molecular weight:264.32
  • AChE/BChE/BACE-1-IN-1

    CAS:
    <p>Compound 4k is an oral AChE, BChE, BACE-1 inhibitor with IC50s: 0.058, 0.082, 0.115 μM, crosses blood-brain barrier, and has neuroprotective effects.</p>
    Formula:C19H21F3N2O
    Color and Shape:Solid
    Molecular weight:350.38
  • BuChE-IN-1

    CAS:
    <p>BuChE-IN-1 is a potent BBB-permeable, low-toxic BuChE inhibitor with potential for AD research.</p>
    Formula:C23H23FN2O4S
    Color and Shape:Solid
    Molecular weight:442.5
  • Arecaidine propargyl ester tosylate

    CAS:
    <p>Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.</p>
    Formula:C17H21NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.42
  • MAP4

    CAS:
    <p>metabotropic glutamate receptor modulator</p>
    Formula:C5H12NO5P
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:197.13
  • mGlu4 receptor agonist 1

    CAS:
    <p>Compound 62, an mGlu4 agonist, has a 308 nM EC50 with anxiolytic and antipsychotic effects.</p>
    Formula:C21H15ClN4O2
    Color and Shape:Solid
    Molecular weight:390.82
  • S-14671

    CAS:
    <p>S-14671: 5-HT1A agonist (pKi 9.3), potent in vivo; 5-HT2A/2C antagonist (pKi 7.8).</p>
    Formula:C22H25N3O2S
    Color and Shape:Solid
    Molecular weight:395.52
  • GR 113808

    CAS:
    <p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>
    Formula:C19H27N3O4S
    Purity:98.16%
    Color and Shape:Solid
    Molecular weight:393.5
  • Foliglurax

    CAS:
    Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).
    Formula:C23H23N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.51
  • ACDPP hydrochloride

    CAS:
    <p>mGlu5 receptor antagonist</p>
    Formula:C12H13ClN6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.72
  • TIK-301

    CAS:
    <p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>
    Formula:C14H17ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.75
  • ADX71743

    CAS:
    <p>ADX71743 is a potent and selective negative allosteric modulator of metabotropic glutamate receptor 7.</p>
    Formula:C17H19NO2
    Color and Shape:Solid
    Molecular weight:269.34
  • FTEAA


    <p>FTEAA is a dual MAO-A and MAO-B inhibitor with IC50 of 0.52 μM and 1.02 μM, used in cardiovascular and neurological research.</p>
    Formula:C34H26F8N2O2
    Color and Shape:Solid
    Molecular weight:646.57
  • GABA-AT-IN-1

    CAS:
    <p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>
    Formula:C23H18N2O6
    Color and Shape:Solid
    Molecular weight:418.4
  • SB-221284

    CAS:
    5-HT2C/2B receptor antagonist
    Formula:C16H14F3N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.36
  • CCD-3693

    CAS:
    <p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>
    Formula:C21H31F3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:372.46
  • LY 125180

    CAS:
    LY 125180 is a serotonin antagonist.
    Formula:C18H24ClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:305.84
  • AChE/BChE/MAO-B-IN-2


    <p>AChE/BChE/MAO-B-IN-2 inhibits AChE (48.2 nM), BChE (83.9 nM), MAO-B (31.2 nM), has antioxidant activity, and aids Parkinson's research.</p>
    Formula:C25H31N3O3
    Color and Shape:Solid
    Molecular weight:421.53
  • (±)-Muscarine chloride

    CAS:
    <p>(±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].</p>
    Formula:C9H20ClNO2
    Color and Shape:Solid
    Molecular weight:209.71
  • RU 33965

    CAS:
    <p>RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.</p>
    Formula:C16H15N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:281.31
  • ML375

    CAS:
    <p>ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).</p>
    Formula:C23H15ClF2N2O2
    Color and Shape:Solid
    Molecular weight:424.83
  • MHP 133

    CAS:
    <p>MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).</p>
    Formula:C17H20ClN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.83
  • PRX933 hydrochloride

    CAS:
    <p>PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.</p>
    Formula:C16H22ClN5O2
    Purity:99.51% - 99.89%
    Color and Shape:Solid
    Molecular weight:351.84
  • Rapacuronium bromide

    CAS:
    Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.
    Formula:C37H61BrN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:677.8
  • 8-M-PDOT

    CAS:
    <p>8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.</p>
    Formula:C14H19NO2
    Purity:99.54% - 99.54%
    Color and Shape:Solid
    Molecular weight:233.31
  • KL8604166

    CAS:
    KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.
    Formula:C12H21N5O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:267.33
  • LY 334370 hydrochloride

    CAS:
    5-HT1F receptor agonist
    Formula:C21H23ClFN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:387.88
  • WAY 161503 hydrochloride

    CAS:
    <p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>
    Formula:C11H12Cl3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.59
  • FK960

    CAS:
    FK962 boosts somatostatin, enhances cognition, and raises synaptic density in rat hippocampus.
    Formula:C13H16FN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:265.28
  • 9-CP-Ade Mesylate

    CAS:
    <p>9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.</p>
    Formula:C11H17N5O3S
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:299.35
  • Deramciclane

    CAS:
    Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.
    Formula:C20H31NO
    Color and Shape:Solid
    Molecular weight:301.47
  • JI051

    CAS:
    JI051 has anti-tumor effects and can interact with PHB2 to inhibit the proliferation of HEK293 cells and pancreatic cancer cells.
    Formula:C22H24N2O3
    Purity:≥98% - ≥98.0%
    Color and Shape:Solid
    Molecular weight:364.44
  • Dimethyl-W84 (dibromide)

    CAS:
    <p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>
    Formula:C34H48Br2N4O4
    Color and Shape:Solid
    Molecular weight:736.59
  • Cimetropium Bromide

    CAS:
    <p>Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.</p>
    Formula:C21H28BrNO4
    Color and Shape:Solid
    Molecular weight:438.36
  • SC57666

    CAS:
    <p>SC57666 is a highly selective COX2 inhibitor (IC50 at 26 nM) that shows no activity against COX1.</p>
    Formula:C18H17FO2S
    Purity:98.83%
    Color and Shape:Solid
    Molecular weight:316.39
  • Pivalylbenzhydrazine

    CAS:
    <p>Pivhydrazine: strong MAO inhibitor, stunts rat cartilage growth, used in depression research.</p>
    Formula:C12H18N2O
    Color and Shape:Solid
    Molecular weight:206.28
  • Aβ42-IN-1 free base

    CAS:
    <p>Aβ42-IN-1 free base (compound 1v), an orally active γ-secretase modulator with high brain exposure, effectively lowers Aβ42 levels, exhibiting an IC 50 of 0.091</p>
    Formula:C29H26N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.54
  • VU 6008667

    CAS:
    VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).
    Formula:C24H17ClF2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.85
  • AChE-IN-9


    <p>AChE-IN-9: Tacrine-β-glucose glycoconjugate; IC50 0.4μM; reduced hepatotoxicity; Alzheimer's research.</p>
    Formula:C30H35N5O9
    Color and Shape:Solid
    Molecular weight:609.63
  • Neuroinflammatory-IN-2

    CAS:
    <p>Neuroinflammatory-IN-2: anti-neuroinflammatory, inhibits MAO-B (IC50: 10.30µM), 96.33% Aβ1-42 aggregation reduction, neuroprotective in PC-12 cells.</p>
    Formula:C25H27FN2O3
    Color and Shape:Solid
    Molecular weight:422.49
  • PAT-1251 Hydrochloride

    CAS:
    <p>PAT-1251 Hydrochloride: Potent, selective, oral LOXL2 inhibitor; IC50s - 0.71 μM (hLOXL2), 1.17 μM (hLOXL3).</p>
    Formula:C18H18ClF4N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.8
  • AChE/BChE-IN-8

    CAS:
    <p>AChE/BChE-IN-8 inhibits AChE (Ki=0.788 μM) &amp; BChE (Ki=2.364 μM), crosses the blood-brain barrier, and is low in cytotoxicity.</p>
    Formula:C26H32N2O2
    Color and Shape:Solid
    Molecular weight:404.54
  • SUN-C5174

    CAS:
    <p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>
    Formula:C22H29FN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:400.49
  • Piclozotan

    CAS:
    <p>Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)</p>
    Formula:C23H24ClN3O2
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:409.91
  • WAY 629 hydrochloride

    CAS:
    5-HT2C agonist
    Formula:C15H19ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:262.78
  • Tertatolol

    CAS:
    <p>Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.</p>
    Formula:C16H25NO2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.44
  • PCS1055 dihydrochloride

    CAS:
    <p>PCS1055 is a selective M4 antagonist (IC50: 18.1 nM, Ki: 6.5 nM) and potent AChE inhibitor with &gt;100-fold M1/M3/M5 selectivity.</p>
    Formula:C27H34Cl2N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:485.49
  • γ-Secretase modulator 11

    CAS:
    <p>5-{8-[(3,4'-Difluoro[1,1'-biphenyl]-4-yl)methoxy]-2-methylimidazo[1,2-a]pyridin-3-yl}-N-methylpyridine-2-carboxamide (1o) exhibited high in vitro potency and</p>
    Formula:C28H22F2N4O2
    Color and Shape:Solid
    Molecular weight:484.5
  • Alosetron ((Z)-2-butenedioate)

    CAS:
    <p>Alosetron (GR 68755) (Z)-2-butenedioate is a Serotonin 5HT3-receptor antagonist that is used in the treatment of irritable bowel syndrome.</p>
    Formula:C21H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.42
  • VU 0360223

    CAS:
    <p>VU 0360223 is a negative allosteric modulator of mGlu5.</p>
    Formula:C15H9FN2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:268.31
  • Oxetorone fumarate

    CAS:
    <p>Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.</p>
    Formula:C25H25NO6
    Purity:99.809%
    Color and Shape:Solid
    Molecular weight:435.48
  • Bibn 99

    CAS:
    <p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>
    Formula:C31H42ClN5O3
    Color and Shape:Solid
    Molecular weight:568.15
  • FR260010

    CAS:
    <p>FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.</p>
    Formula:C22H19N5
    Color and Shape:Solid
    Molecular weight:353.42
  • Pimprinine

    CAS:
    <p>Pimprinine: an alkaloid, inhibits MAO, and has anticonvulsant properties.</p>
    Formula:C12H10N2O
    Color and Shape:Solid
    Molecular weight:198.22
  • PD 118717

    CAS:
    PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.
    Formula:C20H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.41
  • p-MPPF dihydrochloride

    CAS:
    <p>p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.</p>
    Formula:C25H29Cl2FN4O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:507.43
  • β-CCB

    CAS:
    <p>benzodiazepine receptor ligand</p>
    Formula:C16H16N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:268.31
  • TC-2153

    CAS:
    <p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>
    Formula:C7H5ClF3NS5
    Color and Shape:Solid
    Molecular weight:355.89
  • Ro 64-5229

    CAS:
    <p>mGlu2 antagonist</p>
    Formula:C17H19Cl2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.26
  • Arecaidine but-2-ynyl ester tosylate

    CAS:
    mAChR M2 agonist
    Formula:C18H23NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:365.44
  • L-AP4 monohydrate

    CAS:
    <p>L-AP4 (L-APB) is a group III mGluR agonist with EC50s: 0.13μM (mGlu4), 0.29μM (mGlu8), 1.0μM (mGlu6), 249μM (mGlu7).</p>
    Formula:C4H12NO6P
    Color and Shape:Solid
    Molecular weight:201.115
  • RJR 2429 dihydrochloride

    CAS:
    <p>nAChR agonist that displays selectivity for α4β2</p>
    Formula:C12H18Cl2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:261.19
  • Milameline hydrochloride

    CAS:
    <p>Milameline hydrochloride is a Muscarinic receptor agonist.</p>
    Formula:C8H15ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:190.67
  • Cycrimine

    CAS:
    Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.
    Formula:C19H29NO
    Color and Shape:Solid
    Molecular weight:287.44
  • Obidoxime dichloride

    CAS:
    <p>Obidoxime dichloride is an antidote for organophosphate poisoning that enhances the positive inotropic effect of phosphamidon on isolated working rat hearts.</p>
    Formula:C14H16Cl2N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.21
  • mAChr-in-1

    CAS:
    <p>mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).</p>
    Formula:C23H25IN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.36
  • LY 344864 hydrochloride

    CAS:
    <p>LY 344864 hydrochloride is a selective receptor agonist with an affinity of 6 nM (Ki) at the 5-HT1F receptor.</p>
    Formula:C21H23ClFN3O
    Color and Shape:Solid
    Molecular weight:387.88
  • MCI826

    CAS:
    <p>MCI826 is a potent and selective antagonist of P-glycoprotein (P-gp) and peptide leukotrienes (p-LTs), showing anti-asthmatic activity in a guinea pig model of</p>
    Formula:C22H28N2O3S
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:400.53
  • CP-601927

    CAS:
    <p>CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.</p>
    Formula:C12H12F3N
    Color and Shape:Solid
    Molecular weight:227.23
  • GS 39783

    CAS:
    <p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>
    Formula:C15H23N5O2S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:337.44
  • BChE-IN-15


    <p>BChE-IN-15 is a compound characterized as a pseudo-irreversible, covalent inhibitor of butyrylcholinesterase (BChE), demonstrating potent activity with an</p>
    Formula:C22H33N3O2
    Color and Shape:Solid
    Molecular weight:371.52
  • BHF-177

    CAS:
    <p>BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.</p>
    Formula:C19H20F3N3
    Color and Shape:Solid
    Molecular weight:347.38
  • (4E)-SUN9221

    CAS:
    (4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in
    Formula:C25H31FN4O3
    Purity:97.79%
    Color and Shape:Solid
    Molecular weight:454.54
  • VU0409106

    CAS:
    <p>VU0409106 is a potent, mGlu5-selective inhibitor.</p>
    Formula:C15H11FN4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:330.34
  • UoS 12258

    CAS:
    <p>UoS 12258 is a positive allosteric modulator of AMPA receptors, used for studying cognitive impairments.</p>
    Formula:C17H19FN2O2S
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:334.41
  • ZM 169369

    CAS:
    <p>ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.</p>
    Formula:C19H20N2S
    Color and Shape:Solid
    Molecular weight:308.44
  • Prucalopride hydrochloride

    CAS:
    <p>Prucalopride hydrochloride is a selective agonist of the 5-HT4.</p>
    Formula:C18H27Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.33
  • Rivanicline

    CAS:
    <p>Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with &gt;1,000x less affinity for α7 receptors.</p>
    Formula:C10H14N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:162.23
  • Tedatioxetine hydrobromide

    CAS:
    Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.
    Formula:C18H22BrNS
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:364.34
  • RR-11a analog

    CAS:
    <p>RR-11a (aza-peptide) inhibits asparaginyl endopeptidase: IC50 - 4.5 nM (T. Vaginalis, I. ricinus), 31 nM (S. mansoni).</p>
    Formula:C22H29N5O8
    Purity:98.80%
    Color and Shape:Solid
    Molecular weight:491.49
  • QF0301B

    CAS:
    QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
    Formula:C23H28N2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:364.48
  • Parapenzolate bromide

    CAS:
    <p>Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.</p>
    Formula:C21H26BrNO3
    Color and Shape:Solid
    Molecular weight:420.347
  • BisQ

    CAS:
    <p>BisQ is an agonist of photochromic. It used for the muscle-type nAChR.</p>
    Formula:C20H30IN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.392
  • CP 93129 dihydrochloride

    CAS:
    <p>5-HT1B agonist, potent and highly selective</p>
    Formula:C12H14ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:251.71
  • EMD 386088 hydrochloride

    CAS:
    <p>EMD 386088 hydrochloride is a 5-HT6 receptor agonist.</p>
    Formula:C14H16Cl2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.2
  • D-NMAPPD

    CAS:
    <p>Litifilimab (BIIB059) is a humanized antibody targeting BDCA2 and CLEC4C for the study of cutaneous lupus erythematosus.</p>
    Formula:C23H38N2O5
    Color and Shape:Solid
    Molecular weight:422.56
  • L-694,247

    CAS:
    <p>L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.</p>
    Formula:C20H21N5O3S
    Purity:98.36%
    Color and Shape:White Solid
    Molecular weight:411.48
  • Lidanserin

    CAS:
    <p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>
    Formula:C26H31FN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.53
  • CGS-12066 maleate salt

    CAS:
    <p>CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.</p>
    Formula:C21H21F3N4O4
    Color and Shape:Solid
    Molecular weight:450.41
  • TAK-070

    CAS:
    <p>TAK-070 is a non-competitive inhibitor of BACE1.</p>
    Formula:C27H31NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.54
  • Org37684

    CAS:
    <p>5-HT2 receptors agonist</p>
    Formula:C14H20ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:269.77
  • Ro 67-4853

    CAS:
    <p>Ro 67-4853 is a positive allosteric modulator of mGluR1, selectively enhancing the response to the agonist (S)-3,5-dihydroxy-phenylglycine (DHPG).</p>
    Formula:C19H19NO4
    Purity:98.57%
    Color and Shape:Solid
    Molecular weight:325.36
  • RX 801077

    CAS:
    <p>RX 801077 is a selective I2R agonist, Ki of 70.1 nM, with anti-inflammatory and neuroprotective properties for TBI research.</p>
    Formula:C11H10N2O
    Color and Shape:Solid
    Molecular weight:186.21
  • CGS 12066B dimaleate

    CAS:
    <p>5-HT1B full agonist</p>
    Formula:C25H25F3N4O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:566.48
  • BMS-911172

    CAS:
    <p>BMS-911172 is an adaptor associated kinase 1 (AAK1 kinase) inhibitor with an IC 50 of 35 nM.</p>
    Formula:C16H19F2N3O3
    Color and Shape:Solid
    Molecular weight:339.34
  • HexylHIBO

    CAS:
    <p>HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values of 140 and 110 μM, respectively.HexylHIBO decreases sEPSC in rats.</p>
    Formula:C12H20N2O4
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:256.3
  • Muscarine chloride

    CAS:
    <p>Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>
    Formula:C9H20ClNO2
    Color and Shape:Solid
    Molecular weight:209.71
  • AC-42

    CAS:
    <p>AC-42 is an allosteric agonist of M1 muscarinic receptor.</p>
    Formula:C20H31NO
    Color and Shape:Solid
    Molecular weight:301.47
  • NS 1209

    CAS:
    <p>NS 1209 (SPD 502) is a AMPA receptor antagonist.</p>
    Formula:C24H27N4NaO7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:538.55
  • AChE-IN-12

    CAS:
    <p>AChE-IN-12 inhibited rat/eel AChE, crossed BBB, prevented Aβ1-42 aggregation, and has potential for Alzheimer's research.</p>
    Formula:C33H41NO7
    Color and Shape:Solid
    Molecular weight:563.68
  • DPNB-ABT594


    <p>DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.</p>
    Formula:C31H46ClN3O11
    Color and Shape:Solid
    Molecular weight:672.16
  • Bisindolylmaleimide VII

    CAS:
    <p>Bisindolylmaleimide VII is a selective inhibitor of protein kinase C.</p>
    Formula:C27H27N5O2
    Color and Shape:Solid
    Molecular weight:453.54
  • Aβ Fibrillization modulator 1

    CAS:
    <p>Aβ Fibrillization Modulator 1 stabilizes amyloid-beta (Aβ) monomers, preventing their aggregation into fibrils.</p>
    Formula:C17H12N4O3SSe
    Color and Shape:Solid
    Molecular weight:431.33
  • S(-)-8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.</p>
    Formula:C16H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.29
  • VU6001966

    CAS:
    <p>VU6001966: potent, selective mGlu2 inhibitor (IC50=78 nM), negative modulator, with good CNS penetration.</p>
    Formula:C17H15FN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:326.33
  • VU6010572

    CAS:
    <p>VU6010572: potent, selective mGlu3 modulator, IC50 245 nM, high CNS penetration.</p>
    Formula:C20H18FNO3
    Color and Shape:Solid
    Molecular weight:339.36
  • Tebanicline tosylate

    CAS:
    <p>Tebanicline: synthetic, potent, non-opioid analgesic, less toxic than epibatidine; relieves neuropathic pain, acts on α3β4 and α4β2 nicotinic receptors.</p>
    Formula:C16H19ClN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.85
  • AFDX384

    CAS:
    <p>AFDX384 is potent M2/M4 selective antagonist.</p>
    Formula:C28H42N6O5S
    Color and Shape:Solid
    Molecular weight:574.74
  • Mimopezil

    CAS:
    <p>Mimopezil is an acetylcholinesterase (AChE) inhibitor.</p>
    Formula:C23H23ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.89
  • CP 135807

    CAS:
    <p>CP 135807 is a 5-HT1D receptor agonist.</p>
    Formula:C19H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.4
  • ZK93423

    CAS:
    <p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>
    Formula:C23H22N2O4
    Color and Shape:Solid
    Molecular weight:390.43
  • MAO-B-IN-14

    CAS:
    <p>MAO-B-IN-14 (Compound 9) is a potent and selective inhibitor of monoamine oxidase-B (MAO-B) with an IC 50 of 0.95 μM and a Ki of 0.55 μM for human MAO-B.</p>
    Formula:C17H14O3S
    Color and Shape:Solid
    Molecular weight:298.36
  • BuChE-IN-7


    <p>BuChE-IN-7: selective hBuChe &amp; eqBuChe inhibitor, IC50s 40/80 nM, boosts cognition &amp; memory, and penetrates blood-brain barrier.</p>
    Formula:C25H34N2O2
    Color and Shape:Solid
    Molecular weight:394.55
  • WAY 163909

    CAS:
    WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).
    Formula:C14H18N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:214.31
  • Flupyrimin

    CAS:
    <p>Flupyrimin is the insect nicotinic acetylcholine receptor (nAChR) antagonist [1].</p>
    Formula:C13H9ClF3N3O
    Color and Shape:Solid
    Molecular weight:315.68
  • GW-876167

    CAS:
    <p>GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.</p>
    Formula:C16H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.37
  • Lofepramine hydrochloride

    CAS:
    <p>Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.</p>
    Formula:C26H28Cl2N2O
    Purity:98%
    Color and Shape:Off-White Solid
    Molecular weight:455.42
  • VU0463841

    CAS:
    <p>VU0463841 is a mGlu5 negative allosteric modulators.</p>
    Formula:C13H8ClFN4O
    Color and Shape:Solid
    Molecular weight:290.68
  • VU 0360172 hydrochloride

    CAS:
    <p>positive allosteric modulator of mGlu5 receptors</p>
    Formula:C18H16ClFN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:330.78
  • KMS88009

    CAS:
    <p>KMS88009 is an amyloid-β aggregation inhibitor that acts by ameliorating neurodegenerative disorder.</p>
    Formula:C19H19NO2
    Color and Shape:Solid
    Molecular weight:293.36
  • VU0366248

    CAS:
    <p>VU0366248 is a mGlu5 negative allosteric modulator.</p>
    Formula:C14H7ClF2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.67
  • BGT1-IN-9

    CAS:
    <p>BGT1-IN-9 is an M1 muscarinic agonist.</p>
    Formula:C5H10ClN3O2
    Color and Shape:Solid
    Molecular weight:179.605
  • GABAA receptor agent 5

    CAS:
    <p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>
    Formula:C21H25N3O2S
    Color and Shape:Solid
    Molecular weight:383.51
  • (RS)-4-Carboxyphenylglycine

    CAS:
    <p>(RS)-4-Carboxyphenylglycine is a racemic mixture. (S)-4-Carboxyphenylglycine is a selective mGlu1α receptor antagonist.</p>
    Formula:C9H9NO4
    Purity:99.04% - >99.99%
    Color and Shape:Solid
    Molecular weight:195.17
  • PF-3246799

    CAS:
    <p>PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.</p>
    Formula:C15H17N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:239.32
  • Amitriptylinoxide

    CAS:
    <p>Amitriptylinoxide is an antidepressant.</p>
    Formula:C20H23NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:293.4
  • Ph-HTBA

    CAS:
    <p>Ph-HTBA: high-affinity CaMKIIα modulator, brain-penetrant, Kd 757 nM, used in ischemia/neurodegeneration research.</p>
    Formula:C19H18O3
    Color and Shape:Solid
    Molecular weight:294.34
  • BGC 20-761

    CAS:
    <p>BGC20-761: selective 5-HT6/Dopamine antagonist; enhances memory, potential antipsychotic. K i - 5-HT6: 20 nM, 5-HT2A: 69 nM, D2: 140 nM.</p>
    Formula:C19H22N2O
    Color and Shape:Solid
    Molecular weight:294.39
  • (S)-VQW-765


    <p>(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.</p>
    Formula:C19H22N2O
    Color and Shape:Solid
    Molecular weight:294.39
  • 2-PAT

    CAS:
    <p>2-PAT: reversible MAO-A inhib., IC50=0.721 µM; MAO-B inactivator, IC50=14.6 µM; potential in Parkinson's/depression study.</p>
    Formula:C13H15N
    Color and Shape:Solid
    Molecular weight:185.26
  • SGC-AAK1-1N

    CAS:
    <p>SGC-AAK1-1N is a potent and selective inhibitor of AAK1 (AP2 associated kinase 1) with an IC 50 of 1.8 μM [1].</p>
    Formula:C20H22N4O3S
    Color and Shape:Solid
    Molecular weight:398.48
  • Way 100289

    CAS:
    <p>Way 100289 is a selective 5-HT3 receptor antagonist.</p>
    Formula:C20H27N3O3
    Color and Shape:Solid
    Molecular weight:357.45
  • S 32212 hydrochloride

    CAS:
    <p>S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .</p>
    Formula:C25H29ClN4O2
    Purity:97.11% - 99.57%
    Color and Shape:Solid
    Molecular weight:452.98
  • 3,3'-Difluorobenzaldazine

    CAS:
    <p>allosteric potentiator of mGlu5</p>
    Formula:C14H10F2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.24
  • CIA-1 hcl(452087-38-6 Free base)

    CAS:
    <p>CIA-1 inhibits the nuclear receptor COUP-TFII, with IC50s ranging from 1.2 μM to 7.6 μM in prostate cancer cell lines.CIA-1 inhibits the growth of a variety of</p>
    Formula:C17H20ClN3O2S
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:365.88
  • Ifoxetine sulfate

    CAS:
    <p>Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.</p>
    Formula:C13H19NO2H2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:270.34
  • CGP 46381

    CAS:
    <p>CGP 46381 is a GABAB receptor antagonist.</p>
    Formula:C10H22NO2P
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:219.26