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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1045 products of "Proteases/Proteasome"

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  • N-CBZ-Phe-Arg-AMC

    CAS:
    <p>Z-FR-AMC substrate for serine proteases; cathepsins, kallikrein, plasmin. Substrate: 330/390 nm; Product: 342/441 nm.</p>
    Formula:C33H36N6O6
    Purity:98%
    Color and Shape:White To Off-White Powder
    Molecular weight:612.68
  • Zetomipzomib maleate

    CAS:
    <p>Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.</p>
    Formula:C34H46N4O12
    Color and Shape:Solid
    Molecular weight:702.758
  • CRA-2059

    CAS:
    <p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>
    Formula:C34H46N12O8
    Purity:97.68%
    Color and Shape:Solid
    Molecular weight:750.818
  • ADAM8-IN-1

    CAS:
    <p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>
    Formula:C44H44Br4N6O12S2
    Color and Shape:Solid
    Molecular weight:1232.6
  • MMP-3 Inhibitor

    CAS:
    <p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>
    Formula:C27H46N10O9S
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:686.78
  • (-)-Taxifolin

    CAS:
    <p>(-)-Taxifolin, less active enantiomer with anti-tyrosinase, collagenase inhibition (IC50 = 193.3 μM), antifibrotic, antioxidant properties.</p>
    Formula:C15H12O7
    Color and Shape:Solid
    Molecular weight:304.25
  • TP0597850

    CAS:
    <p>TP0597850, a selective MMP2 inhibitor with an IC50 value of 0.22 nM, demonstrates a prolonged dissociation half-life from MMP2 (t1/2 = 265 minutes) [1].</p>
    Formula:C41H57N9O13S
    Color and Shape:Solid
    Molecular weight:916.01
  • TAPI1 acetate


    <p>TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .</p>
    Formula:C28H41N5O7
    Purity:98.82% - 99.94%
    Color and Shape:Solid
    Molecular weight:559.65
  • Leptosin D

    CAS:
    <p>Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)</p>
    Formula:C25H24N4O3S2
    Color and Shape:Solid
    Molecular weight:492.61
  • HCVP-IN-1

    CAS:
    <p>HCVP-IN-1 (compound 1) is a hepatitis C viral polymerase (HCVP) inhibitor.</p>
    Formula:C30H34FN5O3
    Color and Shape:Solid
    Molecular weight:531.632
  • Cathepsin K inhibitor 7


    <p>Cathepsin K Inhibitor7 (compound 7) is an inhibitor of Cathepsin K, exhibiting a pKi value of 7.3. It is utilized in research on osteoporosis.</p>
    Color and Shape:Odour Solid
  • Sofosbuvir impurity A

    CAS:
    <p>Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.</p>
    Formula:C22H29FN3O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.45
  • Imitrodast

    CAS:
    <p>Imitrodast is a small molecule thromboxane A2 synthase (TXA2 synthase) inhibitor for the treatment of immune system disorders, respiratory disorders, and</p>
    Formula:C13H12N2O2S
    Purity:98.39%
    Color and Shape:Solid
    Molecular weight:260.31
  • Ellipyrone A


    <p>Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).</p>
    Formula:C25H34O8
    Color and Shape:Solid
    Molecular weight:462.53
  • Neutrophil elastase inhibitor 4


    <p>Neutrophil elastase inhibitor 4 (compound 4f) is a competitive inhibitor of human neutrophil elastase (HNE) with IC50 of 42.30 nM and Ki of 8.04 nM.</p>
    Formula:C20H21N3O5
    Color and Shape:Solid
    Molecular weight:383.4
  • HCV-IN-4

    CAS:
    <p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>
    Formula:C52H58FN9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:956.07
  • Chetoseminudin B

    CAS:
    <p>Chetoseminudin B exhibits inhibitory activity against mushroom tyrosinase, with an IC 50 value of 31.7 μM [1].</p>
    Formula:C17H21N3O3S2
    Color and Shape:Solid
    Molecular weight:379.5
  • Sofosbuvir impurity J

    CAS:
    <p>Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Formula:C22H30FN4O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:528.47
  • 6-Acetylnimbandiol

    CAS:
    <p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>
    Formula:C28H34O8
    Color and Shape:Solid
    Molecular weight:498.56
  • α 1(I) Collagen (614-639), human

    CAS:
    <p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>
    Formula:C134H189N37O39
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2942.16
  • PF 00356231

    CAS:
    <p>PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).</p>
    Formula:C25H20N2O3S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:428.5
  • Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2

    CAS:
    <p>Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic probe for MMP-1 and MMP-9 detection, releasing fluorescent Nma upon cleavage (Ex/Em: 340/440 nm).</p>
    Formula:C49H68N14O12S
    Color and Shape:Solid
    Molecular weight:1077.22
  • Bictegravir Sodium

    CAS:
    <p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>
    Formula:C21H17F3N3NaO5
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:471.36
  • HIV-1 inhibitor-6 

    CAS:
    <p>HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicing</p>
    Formula:C14H10N4O4S
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:330.32
  • JC-10

    CAS:
    <p>JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.</p>
    Formula:C25H29Cl2IN4
    Purity:95%
    Color and Shape:Solid
    Molecular weight:583.34
  • Enzyme-IN-1

    CAS:
    <p>Enzyme-IN-1(compound 1)为基于肽的N端亲核试剂(Ntn)水解酶抑制剂,特别针对20S蛋白酶体的糜胰蛋白酶样活性(CT-L)进行抑制,可能展现出抗炎特性。</p>
    Formula:C36H50N4O7
    Color and Shape:Solid
    Molecular weight:650.8
  • Cepeginterferon alfa-2b

    CAS:
    <p>Cepeginterferon alfa-2b: pegylated interferon with 20 kDa PEG for HCV, PV, ET research.</p>
    Color and Shape:Liquid
  • Cys-TAT(47-57) acetate(583836-55-9 Free base)


    <p>Cys-TAT(47-57) acetate is derived from the HIV-1 transactivating protein. Cys-TAT(47-57) acetate is an arginine rich peptide that can penetrate cells.</p>
    Formula:C69H128N34O16S
    Purity:95.1100%
    Color and Shape:Solid
    Molecular weight:1722.04
  • RJS308


    <p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>
    Formula:C63H75N13O11S
    Color and Shape:Solid
    Molecular weight:1222.42
  • Talabostat isomer mesylate


    <p>Talabostat isomer mesylate, a PT100/Val-boroPro variant, is a potent oral DPP-IV inhibitor (Ki: 0.18 nM).</p>
    Formula:C10H23BN2O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.18
  • PPACK II

    CAS:
    <p>PPACK II is an irreversible and specific glandular and plasma kallikreins inhibitor [1] .</p>
    Formula:C25H33ClN6O3
    Color and Shape:Solid
    Molecular weight:501.02
  • Rivulariapeptolides 1121


    <p>Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).</p>
    Formula:C56H83N9O15
    Color and Shape:Solid
    Molecular weight:1122.31
  • Fotagliptin

    CAS:
    <p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>
    Formula:C17H19FN6O
    Color and Shape:Solid
    Molecular weight:342.37
  • N-CBZ-Phe-Arg-AMC TFA


    <p>N-CBZ-Phe-Arg-AMC TFA (Z-FR-AMC TFA) is a fluorescent substrate for serine proteases. assess the activity of trypsin, plasmin, and cathepsin.</p>
    Formula:C35H37F3N6O8
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:726.7
  • CRA-2059 hydrochloride


    <p>CRA-2059 hydrochloride is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].</p>
    Color and Shape:Solid
  • 7-Methoxy obtusifolin

    CAS:
    <p>7-Methoxy obtusifolin (Compound 4) is a chemical compound that acts as a competitive inhibitor of the enzyme tyrosinase, displaying an inhibitory concentration</p>
    Formula:C17H14O6
    Color and Shape:Solid
    Molecular weight:314.29
  • Tyrosinase/elastase-IN-1


    <p>Tyrosinase/elastase-IN-1, a triterpenoid extracted from the leaves of Rubus fraxinifolius, exhibits inhibitory activities against both tyrosinase and elastase</p>
    Formula:C33H52O5
    Color and Shape:Solid
    Molecular weight:528.76
  • DPP8/9-IN-1


    <p>DPP8/9-IN-1 (Compound 16) is a selective covalent inhibitor of dipeptidyl peptidase 8 and 9 (DPP8/9), with IC50 values of 14 nM and 298 nM, respectively. It irreversibly binds to the active site serine (such as S730 in DPP9) through a phosphate ester warhead, blocking substrate binding and inhibiting DPP8/9-mediated protein processing. DPP8/9-IN-1 holds potential for research in cancer and inflammatory diseases.</p>
    Color and Shape:Odour Solid
  • Sofigatran

    CAS:
    <p>Sofigatran (MCC-977) is an oral anticoagulant targeting thrombin for cardiovascular research.</p>
    Formula:C24H44N4O4S
    Color and Shape:Solid
    Molecular weight:484.7
  • L 659286

    CAS:
    <p>L 659286 is one kind of cephalosporin derivative.</p>
    Formula:C17H21N5O7S2
    Color and Shape:Solid
    Molecular weight:471.51
  • Nitidanin


    <p>Nitidanin is a useful organic compound for research related to life sciences and the catalog number is T125599.</p>
    Formula:C21H24O8
    Color and Shape:Solid
    Molecular weight:404.415
  • Dutogliptin tartrate

    CAS:
    <p>Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>
    Formula:C14H26BN3O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.18
  • NS5A-IN-1


    <p>NS5A-IN-1 is a proagent of the HCV NS5A inhibitor Pibrentasvir (ABT-530).</p>
    Formula:C72H86F5N10O14P
    Color and Shape:Solid
    Molecular weight:1441.48
  • Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2

    CAS:
    <p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>
    Formula:C47H64N14O10
    Color and Shape:Solid
    Molecular weight:985.1
  • Sofosbuvir impurity M

    CAS:
    <p>Sofosbuvir impurity M is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Formula:C22H30N3O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.467
  • Cathepsin D and E FRET Substrate

    CAS:
    <p>Mca-GKPILFFRL-Dpa-r-amide, FRET substrate for cathepsin D and E. Also cleaved by napsin A.</p>
    Formula:C85H122N22O19
    Color and Shape:Solid
    Molecular weight:1756.046
  • FFAGLDD TFA


    <p>FFAGLDD TFA: MMP9 peptide for controlled DOX delivery to cytoplasm.</p>
    Formula:C39H50F3N7O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:897.85
  • L-Methionine-DL-sulfoximine

    CAS:
    <p>MSO blocks glutamine synthetase, impacts astroglia, and is used in convulsant research.</p>
    Formula:C5H12N2O3S
    Purity:99.56% - ≥98%
    Color and Shape:White Crystalline Powder
    Molecular weight:180.23
  • NS5A-IN-4

    CAS:
    <p>NS5A-IN-4 (Compound 1.12) is a hepatitis C inhibitor effective against multiple genotypes, with IC50 values ranging from 1.2 to 2296 pM.</p>
    Formula:C47H48N8O6
    Color and Shape:Solid
    Molecular weight:820.93
  • GCPII-IN-1

    CAS:
    <p>GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.</p>
    Formula:C12H21N3O7
    Color and Shape:Solid
    Molecular weight:319.314
  • AL-611

    CAS:
    <p>AL-611 is an HCV NS5B polymerase inhibitor ( EC 50 = 5 nM).</p>
    Formula:C25H33F2N6O8P
    Color and Shape:Solid
    Molecular weight:614.544
  • Radalbuvir

    CAS:
    <p>Radalbuvir (GS-9669) is an investigational antiviral agent for the treatment of hepatitis C virus (HCV) infection as an NS5B inhibitor.</p>
    Formula:C30H41NO6S
    Color and Shape:Solid
    Molecular weight:543.71
  • Rivulariapeptolides 1155


    <p>Rivulariapeptolides 1155 inhibits chymotrypsin (41.84 nM), elastase (4.94 nM), and proteinase K (56.54 nM).</p>
    Formula:C59H81N9O15
    Color and Shape:Solid
    Molecular weight:1156.33
  • Recombinant Proteinase K


    <p>Recombinant Proteinase K: serine protease, cleaves carboxy-terminus peptides, digests proteins, purifies nucleic acids.</p>
    Color and Shape:Solid
  • GSK2336805

    CAS:
    <p>GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.</p>
    Formula:C42H52N8O8
    Color and Shape:Solid
    Molecular weight:796.91
  • Leptosphaerodione

    CAS:
    <p>Leptosphaerodione from Remotididymella sp.: a potent UPS inhibitor with 3.2 μM IC50 in HeLa cells; anti-tumor.</p>
    Formula:C21H22O5
    Color and Shape:Solid
    Molecular weight:354.4
  • Histargin

    CAS:
    <p>Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.</p>
    Formula:C14H25N7O4
    Color and Shape:Solid
    Molecular weight:355.39
  • Proteasome-IN-7


    <p>Proteasome-IN-7 (Compound 6f) is a macrolactam-based epoxyketone proteasome inhibitor with an IC50 value of 37.92 nM against the 20S proteasome ChT-L subunit. It exhibits potent antiproliferative effects on multiple myeloma, acute lymphoblastic leukemia, and non-small cell lung cancer.</p>
    Formula:C48H56N6O10S
    Color and Shape:Solid
    Molecular weight:909.06
  • Peptide 74

    CAS:
    <p>Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.</p>
    Formula:C62H107N23O20S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1558.79
  • α 1 Antichymotrypsin, Human Plasma

    CAS:
    <p>Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.</p>
    Color and Shape:Solid
  • APC-6860

    CAS:
    <p>APC-6860, a serine protease inhibitor, targets multiple enzymes; most potent against human urokinase (Ki: 0.1 µM). Used in cancer research.</p>
    Formula:C9H7IN2S
    Color and Shape:Solid
    Molecular weight:302.13
  • PSI-7409

    CAS:
    <p>PSI-7409 is the active 5'-triphosphate metabolite of Sofosbuvir (PSI-7977).</p>
    Formula:C10H16FN2O14P3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.16
  • AMG-222

    CAS:
    <p>AMG-222 (ALS-2-0426, ALS-20426) is a DPP-4 inhibitor and may be used in the treatment of type 2 diabetes.</p>
    Formula:C32H39N9O3
    Color and Shape:Solid
    Molecular weight:597.71
  • Ac-VDQQD-pNA

    CAS:
    <p>Ac-VDQQD-pNA serves as a substrate for Caspase 2, which cleaves it to yield the yellow compound pNA (p-nitroaniline).</p>
    Formula:C31H43N9O14
    Color and Shape:Solid
    Molecular weight:765.73
  • Sitagliptin fenilalanil hydrochloride

    CAS:
    <p>Sitagliptin phenylalanine hydrochloride, a dipeptidyl peptidase-4 (DPP-4) inhibitor [1], is a chemical compound utilized in medical applications.</p>
    Formula:C25H25ClF6N6O2
    Color and Shape:Solid
    Molecular weight:590.95
  • PS 915

    CAS:
    <p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>
    Formula:C27H36ClN7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:590.08
  • Fotagliptin benzoate

    CAS:
    <p>Fotagliptin benzoate, a DPP-4 inhibitor (IC50=2.27 nM), is safe in rats/dogs, useful for Type 2 diabetes research.</p>
    Formula:C24H25FN6O3
    Color and Shape:Solid
    Molecular weight:464.49
  • HCV-IN-41

    CAS:
    <p>HCV-IN-41: potent HCV inhibitor; EC50 - 0.006762 nM (1b), 5.183 nM (2a), 1.365 nM (3a), 142.2 nM (4a); hinders RNA replication.</p>
    Formula:C48H56N6O8
    Color and Shape:Solid
    Molecular weight:844.99
  • Befovacimab

    CAS:
    <p>Befovacimab, a human IgG2 antibody, targets TFPI for hemophilia A/B research.</p>
    Color and Shape:Liquid
  • Berotralstat

    CAS:
    <p>Berotralstat (BCX7353) is an oral, low-toxicity, specific kallikrein inhibitor for hereditary angioedema research, blocking bradykinin release.</p>
    Formula:C30H26F4N6O
    Color and Shape:Solid
    Molecular weight:562.56
  • Tyrosinase-IN-34


    <p>Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.</p>
    Formula:C19H14BrClN4O
    Color and Shape:Solid
    Molecular weight:429.7
  • Histatin 5 (TFA)(115966-68-2,free)


    <p>Histatin 5 (TFA)(115966-68-2,free) (Histatin 5 (TFA)) inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μM</p>
    Formula:C135H196F3N51O35
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3150.32
  • NVP-DPP728 dihydrochloride

    CAS:
    <p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>
    Formula:C15H20Cl2N6O
    Color and Shape:Solid
    Molecular weight:371.27
  • Stevia Powder


    <p>Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.</p>
    Color and Shape:Odour Solid
  • CP-346086 dihydrate

    CAS:
    <p>CP-346086 dihydrate is a strong oral MTP inhibitor with 2.0 nM IC50, reducing cholesterol and triglycerides in vivo.</p>
    Formula:C26H26F3N5O3
    Color and Shape:Solid
    Molecular weight:513.521
  • Ecallantide TFA


    <p>Ecallantide (DX-88) TFA, a specific recombinant plasma kallikrein inhibitor, directly inhibits bradykinin production and is indicated for the prevention of</p>
    Color and Shape:Odour Solid
  • Pseudostellarin G

    CAS:
    <p>Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.</p>
    Formula:C42H56N8O9
    Color and Shape:Solid
    Molecular weight:816.94
  • MK-6169

    CAS:
    <p>MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.</p>
    Formula:C54H62FN9O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1016.2
  • KKI-5

    CAS:
    <p>KKI 5: Serine protease inhibitor, blocks kallikrein &amp; plasmin, potential for cancer therapy &amp; angioedema treatment.</p>
    Formula:C35H55N11O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:773.88
  • Dutogliptin

    CAS:
    <p>Dutogliptin (PHX-1149 free base) is an oral, effective and selective dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>
    Formula:C10H20BN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:241.10
  • CL 82198 hydrochloride

    CAS:
    <p>CL 82198 hydrochloride selectively inhibits MMP-13, not MMP-1/9/TACE, and blocks HP75 invasion and neurotoxicity in zebrafish.</p>
    Formula:C17H23ClN2O3
    Color and Shape:Solid
    Molecular weight:338.83
  • Acetyl-Calpastatin(184-210)(human)

    CAS:
    <p>Calpain inhibitor, Ki 0.2 nM for calpain I/II, doesn't affect papain/trypsin/cat L. Raises Aβ42, Aβ40 secretion &amp; Aβ42/Aβ40 ratio.</p>
    Formula:C142H230N36O44S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3177.65
  • Anticancer agent 114


    <p>Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.</p>
    Formula:C28H33BF6N2O7
    Color and Shape:Solid
    Molecular weight:634.37
  • AP-C2

    CAS:
    <p>AP-C2 is a potent small molecule guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) inhibitor with a pIC50 of 5.2 for cGKII.</p>
    Formula:C18H16N4S
    Purity:99.87%
    Color and Shape:Soild
    Molecular weight:320.41
  • C-telopeptide

    CAS:
    <p>C-telopeptide from type I collagen is released during bone resorption; it correlates with bone mineral density.</p>
    Formula:C34H56N14O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:868.9
  • Tyrosinase-IN-32


    <p>Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.</p>
    Formula:C15H19NO3
    Color and Shape:Solid
    Molecular weight:261.32
  • EP 171

    CAS:
    <p>EP 171 is a potent agonist of TP-receptors.</p>
    Formula:C23H29FO5
    Color and Shape:Solid
    Molecular weight:404.47
  • Elastatinal

    CAS:
    <p>Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.</p>
    Formula:C21H36N8O7
    Color and Shape:Yellowish Solid
    Molecular weight:512.56
  • Ac-DEMEEC-OH

    CAS:
    <p>Ac-DEMEEC-OH is a competitive inhibitor of the HCV NS3 protease with a Ki of 0.6 µM.</p>
    Formula:C29H44N6O16S2
    Color and Shape:Solid
    Molecular weight:796.82
  • HIV-1 TAT (48-60) Acetate


    <p>Lilotomab (HH1) is a murine anti-CD37 antibody that can be used to synthesize anti-CD37 antibody-radionuclide couplings.</p>
    Formula:C72H135N35O18
    Purity:99.93%
    Color and Shape:Soild
    Molecular weight:1779.07
  • STK33-IN-1

    CAS:
    <p>STK33-IN-1 (compound 1) is a STK33 inhibitor, with an IC 50 of 7 nM.</p>
    Formula:C24H27N7O2
    Color and Shape:Solid
    Molecular weight:445.527
  • GSK2818713

    CAS:
    <p>GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.</p>
    Formula:C46H56N8O8
    Color and Shape:Solid
    Molecular weight:849.002
  • FiVe1

    CAS:
    <p>FiVe1 is a vimentin-binding compound that disrupts mitosis in cancer cells, causing cell death, with an IC50 of 234 nM in FOXC2-HMLER.</p>
    Formula:C18H16Cl2N4
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:359.25
  • BMS-767778

    CAS:
    <p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>
    Formula:C19H20Cl2N4O2
    Color and Shape:Solid
    Molecular weight:407.29
  • Linagliptin Methyldimer

    CAS:
    <p>Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.</p>
    Formula:C50H56N16O4
    Purity:97.23%
    Color and Shape:Solid
    Molecular weight:945.08
  • RXP470

    CAS:
    <p>RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).</p>
    Formula:C35H35BrClN4O10P
    Color and Shape:Solid
    Molecular weight:818
  • Plasma kallikrein-IN-1

    CAS:
    <p>Plasma kallikrein-IN-1 is a PKK inhibitor with an IC 50 value of 0.5 nM.</p>
    Formula:C23H25F2N7O
    Color and Shape:Solid
    Molecular weight:453.498
  • Paritaprevir dihydrate

    CAS:
    <p>Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.</p>
    Formula:C40H47N7O9S
    Color and Shape:Solid
    Molecular weight:801.91
  • CTTHWGFTLC, CYCLIC

    CAS:
    <p>CTT Gelatinase Inhibitor peptide blocks MMP-2/9, hindering cancer by stopping tumor growth.</p>
    Formula:C52H71N13O14S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1166.33
  • midesteine

    CAS:
    <p>Midesteine (MR-889) is a small molecule neutrophil elastase inhibitor used in the treatment of bronchitis, asthma and chronic lung disease.</p>
    Formula:C12H13NO3S3
    Purity:99.52% - 99.98%
    Color and Shape:Solid
    Molecular weight:315.43