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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1045 products of "Proteases/Proteasome"

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  • Lenacapavir

    CAS:
    <p>Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.</p>
    Formula:C39H32ClF10N7O5S2
    Purity:99.61% - 99.87%
    Color and Shape:Solid
    Molecular weight:968.28
  • Etarotene

    CAS:
    <p>Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is a</p>
    Formula:C25H32O2S
    Purity:99.58% - 99.93%
    Color and Shape:Solid
    Molecular weight:396.59
  • BDCRB


    <p>BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.</p>
    Formula:C12H11BrCl2N2O4
    Purity:99.41% - 99.43%
    Color and Shape:Soild
    Molecular weight:398.04
  • BILB-1941

    CAS:
    <p>BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.</p>
    Formula:C34H34N4O4
    Purity:99.51% - 99.65%
    Color and Shape:Solid
    Molecular weight:562.66
  • 2'-C-Methyladenosine

    CAS:
    <p>2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.</p>
    Formula:C11H15N5O4
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:281.27
  • CPA inhibitor

    CAS:
    <p>CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.</p>
    Formula:C18H19NO4
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:313.35
  • Cathepsin X-IN-1

    CAS:
    <p>Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].</p>
    Formula:C15H13N3O3S
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:315.35
  • P32/98 hemifumarate

    CAS:
    <p>P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.</p>
    Formula:C22H40N4O6S2
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:520.71
  • Atevirdine

    CAS:
    <p>Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).</p>
    Formula:C21H25N5O2
    Purity:98.20%
    Color and Shape:Solid
    Molecular weight:379.46
  • DB04760

    CAS:
    <p>DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.</p>
    Formula:C22H20F2N4O2
    Purity:99.93% - 99.99%
    Color and Shape:Solid
    Molecular weight:410.42
  • JNJ-10311795

    CAS:
    <p>JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.</p>
    Formula:C40H35N2O6P
    Purity:97.43%
    Color and Shape:Solid
    Molecular weight:670.69
  • TG-2-IN-1

    CAS:
    <p>TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].</p>
    Formula:C8H13ClN2OS
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:220.72
  • CP-544439

    CAS:
    <p>CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.</p>
    Formula:C18H19FN2O6S
    Purity:95.02% - 98.66%
    Color and Shape:Solid
    Molecular weight:410.42
  • Setrobuvir

    CAS:
    <p>Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension with</p>
    Formula:C25H25FN4O6S2
    Purity:98.92% - >99.99%
    Color and Shape:Solid
    Molecular weight:560.62
  • Granotapide

    CAS:
    <p>Granotapide is a microsomal triglyceride transfer protein (MTP) inhibitor that treats and rather prevents atherosclerosis, coronary artery disease, metabolic</p>
    Formula:C39H37F3N2O8
    Purity:99.70% - 99.79%
    Color and Shape:Solid
    Molecular weight:718.71
  • PG-116800

    CAS:
    <p>PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.</p>
    Formula:C24H27N3O7S
    Purity:98.03% - 99.66%
    Color and Shape:Solid
    Molecular weight:501.55
  • Sovaprevir

    CAS:
    <p>Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.</p>
    Formula:C43H53N5O8S
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:799.97
  • Melagatran

    CAS:
    <p>Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.</p>
    Formula:C22H31N5O4
    Purity:98.29% - >99.99%
    Color and Shape:Solid
    Molecular weight:429.51
  • Opaviraline

    CAS:
    <p>Opaviraline (GW-420867X) is a potent reverse transcriptase inhibitor that inhibits Human immunodeficiency virus 1 and has the potential to treat HIV infection.</p>
    Formula:C14H17FN2O3
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:280.29
  • MMP2-IN-3

    CAS:
    <p>MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).</p>
    Formula:C23H21N3O
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:355.43
  • Uprifosbuvir

    CAS:
    <p>Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.</p>
    Formula:C22H29ClN3O9P
    Purity:99.73% - >99.99%
    Color and Shape:Solid
    Molecular weight:545.91
  • Sirpiglenastat

    CAS:
    <p>Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.</p>
    Formula:C22H27N5O5
    Purity:98.01% - 98.37%
    Color and Shape:Solid
    Molecular weight:441.48
  • Emivirine

    CAS:
    <p>Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.</p>
    Formula:C17H22N2O3
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:302.37
  • Tyrosinase-IN-2

    CAS:
    <p>Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.</p>
    Formula:C8H8N4O2S
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:224.24
  • Isatoribine

    CAS:
    <p>Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.</p>
    Formula:C10H12N4O6S
    Purity:98.99% - 99.75%
    Color and Shape:Solid
    Molecular weight:316.29
  • AGPS-IN-2i

    CAS:
    <p>AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.</p>
    Formula:C18H17F2N3O2
    Purity:98.92%
    Color and Shape:Solid
    Molecular weight:345.34
  • HIV-1 integrase inhibitor 8

    CAS:
    <p>HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].</p>
    Formula:C21H24O2
    Purity:98.91%
    Color and Shape:Solid
    Molecular weight:308.41
  • TS-021

    CAS:
    <p>TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.</p>
    Formula:C17H24FN3O5S
    Purity:>99.99% - >99.99%
    Color and Shape:Solid
    Molecular weight:401.45
  • MMP-2/MMP-9 Inhibitor I

    CAS:
    <p>MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.</p>
    Formula:C21H19NO4S
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:381.44
  • KM-023

    CAS:
    <p>KM-023 is a new second-generation non-nucleoside reverse transcriptase inhibitor for the study of human immunodeficiency virus (HIV) type 1 infection.</p>
    Formula:C18H19N3O3
    Purity:99.47% - >99.99%
    Color and Shape:Solid
    Molecular weight:325.36
  • L 756423

    CAS:
    <p>L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.</p>
    Formula:C39H48N4O5
    Purity:99.34% - 99.88%
    Color and Shape:Solid
    Molecular weight:652.82
  • 20S Proteasome activator 1

    CAS:
    <p>20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.</p>
    Formula:C27H19ClF2N2OS
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:492.97
  • Gemigliptin

    CAS:
    <p>Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)</p>
    Formula:C18H19F8N5O2
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:489.36
  • MK-8325

    CAS:
    <p>MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailability</p>
    Formula:C43H54Cl2F2N8O6Si
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:915.93
  • Thrombin inhibitor 1

    CAS:
    <p>Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).</p>
    Formula:C22H20Cl2F2N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.32
  • GS-6620

    CAS:
    <p>GS-6620 is a HCV nonstructural protein 5B (NS5B) inhibitor.</p>
    Formula:C29H37N6O9P
    Color and Shape:Solid
    Molecular weight:644.61
  • SSR 69071

    CAS:
    <p>SSR69071: selective neutrophil elastase inhibitor, stronger for humans (Ki=0.0168 nM), may treat COPD, asthma, and reduce heart injury.</p>
    Formula:C27H32N4O7S
    Color and Shape:Solid
    Molecular weight:556.63
  • NS5A-IN-2

    CAS:
    <p>NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.</p>
    Formula:C46H45N7O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:807.89
  • XL-784

    CAS:
    <p>XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.</p>
    Formula:C42H42Cl2F4MgN6O16S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1122.15
  • Ravidasvir HCl

    CAS:
    <p>Ravidasvir, also known as PPI-668 and ASC16, is a second-generation, orally active, potent and selective HCV NS5A protein inhibitor.</p>
    Formula:C42H52Cl2N8O6
    Color and Shape:Solid
    Molecular weight:835.828
  • Inogatran

    CAS:
    <p>Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.</p>
    Formula:C21H38N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.56
  • Paltimatrectinib

    CAS:
    <p>Paltimatrectinib (PBI-200) is a tyrosine kinase inhibitor with anticancer activity, and is used in the study of bladder, breast, and colorectal cancers.</p>
    Formula:C20H15F5N6
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:434.37
  • ABP 25

    CAS:
    <p>ABP 25 is a highly potent and selective activity-based probe (ABP) for cathepsin K imaging.</p>
    Formula:C55H66ClN5O3
    Color and Shape:Solid
    Molecular weight:880.6
  • Beclabuvir HCl

    CAS:
    <p>Beclabuvir (BMS-791325) is an HCV inhibitor targeting NS5B polymerase with sub-28 nM potency for genotypes 1, 3, 4, 5.</p>
    Formula:C36H46ClN5O5S
    Color and Shape:Solid
    Molecular weight:696.3
  • BAY-678

    CAS:
    <p>BAY-678: Oral selective human neutrophil elastase inhibitor; IC50: 20 nM; SGC-approved chemical probe.</p>
    Formula:C20H15F3N4O2
    Purity:97.89%
    Color and Shape:Solid
    Molecular weight:400.35
  • Proteasome-IN-5

    CAS:
    <p>Proteasome-IN-5, also known as compound 5, acts as a proteasome inhibitor [1].</p>
    Formula:C20H30BN5O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.29
  • Collagen proline hydroxylase inhibitor

    CAS:
    <p>Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.</p>
    Formula:C18H18N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:354.36
  • Ro 31-9790

    CAS:
    <p>Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).</p>
    Formula:C15H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.41
  • ONO 4817

    CAS:
    <p>ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.</p>
    Formula:C22H28N2O6
    Color and Shape:Solid
    Molecular weight:416.47
  • MMP-7-IN-3

    CAS:
    <p>MMP-7-IN-3 (compound 15) is a potent and selective MMP-7 inhibitor, inhibiting renal fibrosis in a unilateral ureteral obstruction mouse model.</p>
    Formula:C34H43ClF3N7O9S
    Purity:99.915%
    Color and Shape:Solid
    Molecular weight:818.26
  • KB-R7785

    CAS:
    <p>KB-R7785 is a novel ADAM12/MMP inhibitor improving heart function and insulin sensitivity by blocking HB-EGF and TNF-alpha.</p>
    Formula:C18H27N3O4
    Color and Shape:Solid
    Molecular weight:349.42
  • Cipemastat

    CAS:
    <p>Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).</p>
    Formula:C22H36N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.55
  • Azt-pmap

    CAS:
    <p>AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].</p>
    Formula:C20H25N6O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.42
  • XL-784 free base

    CAS:
    <p>XL-784 free base selectively inhibits MMPs with IC50: MMP-1 (1.9µM), MMP-2 (0.81nM), MMP-3 (120nM), MMP-8 (10.8nM), MMP-9 (18nM), MMP-13 (0.56nM).</p>
    Formula:C21H22ClF2N3O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:549.93
  • MDL 27324

    CAS:
    <p>MDL 27324 is an inhibitor of human neutrophil elastase.</p>
    Formula:C29H38F3N5O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:641.7
  • AA74-1

    CAS:
    <p>AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].</p>
    Formula:C16H28N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.42
  • Ro 32-7315

    CAS:
    <p>Ro 32-7315 is a selective inhibitor of ADAM17.</p>
    Formula:C22H35N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.6
  • MK-3281

    CAS:
    <p>MK-3281: Oral, potent HCV NS5B inhibitor with promising properties and efficacy in replication trials, suitable for clinical use.</p>
    Formula:C29H37N3O3
    Color and Shape:Solid
    Molecular weight:475.62
  • MDL 101146

    CAS:
    <p>MDL 101146 is an orally active neutrophil elastase inhibitor.</p>
    Formula:C29H37F5N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:632.62
  • JW 480

    CAS:
    <p>JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.</p>
    Formula:C22H23NO2
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:333.42
  • MMP-7-IN-2

    CAS:
    <p>MMP-7-IN-2 acts as a selective and potent MMP7 inhibitor and can be used to study inflammatory responses and vascular-related diseases.</p>
    Formula:C28H40ClF3N6O9S
    Purity:97.82%
    Color and Shape:Solid
    Molecular weight:729.17
  • Proteasome β2c/i-IN-1

    CAS:
    <p>Proteasome β2c/i-IN-1 (compound 37) serves as a selective inhibitor targeting the β2c and β2i subunits of the human proteasome [1].</p>
    Formula:C32H48N4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:600.75
  • ND-378

    CAS:
    <p>ND-378 is a potent and selective inhibitor of MMP-2 with no inhibition on MMP-9 and MMP-14.</p>
    Formula:C18H19NO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.48
  • AZD-7295

    CAS:
    <p>AZD-7295 (A-689) is an NS5A inhibitor that may be used to treat HCV infection.</p>
    Formula:C32H35F3N4O5S
    Color and Shape:Solid
    Molecular weight:644.7
  • PTC725

    CAS:
    <p>PTC725 is a selective HCV 1b replicons inhibitor. It has been shown to target the nonstructural protein 4B.</p>
    Formula:C23H18F4N6O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.49
  • EP1013

    CAS:
    <p>EP1013 is a broad-spectrum selective inhibitor of Caspase used in the study of type 1 diabetes.</p>
    Formula:C18H23FN2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.38
  • HIV-1 protease-IN-12

    CAS:
    <p>HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-</p>
    Formula:C25H35N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.63
  • GSK-2485852

    CAS:
    <p>GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.</p>
    Formula:C27H25BF2N2O6S
    Color and Shape:Solid
    Molecular weight:554.37
  • MMP13-IN-3

    CAS:
    <p>MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, &gt;1000x selective, for osteoarthritis treatment.</p>
    Formula:C24H22N4O5
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:446.46
  • TP0556351

    CAS:
    <p>TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.</p>
    Formula:C50H70N10O16
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1067.15
  • Apratastat

    CAS:
    <p>Apratastat is an orally active, potent, and reversible dual inhibitor of tumor necrosis factor-α converting enzyme (TACE) and matrix metalloproteinases (MMPs)</p>
    Formula:C17H22N2O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.5
  • MDL-101146, (R)-

    CAS:
    <p>MDL-101146, (R)- is an effective orally active inhibitor of human neutrophil elastase.</p>
    Formula:C29H37F5N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:632.62
  • LU-002i

    CAS:
    <p>LU-002i is a selective inhibitor targeting the human proteasome subunits β2c and β2i, demonstrating an inhibitory concentration (IC50) of 220 nM for β2i [1].</p>
    Formula:C35H52N4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:640.81
  • Phe-Pro-Ala-pNA

    CAS:
    <p>Phe-Pro-Ala-pNA is a chromogenic substrate utilized for assessing tripeptidyl peptidase activity.</p>
    Formula:C23H27N5O5
    Color and Shape:Solid
    Molecular weight:453.49
  • Flovagatran sodium

    CAS:
    <p>Flovagatran sodium, a thrombin inhibitor, is used potentially for the treatment of thrombosis.</p>
    Formula:C27H36BN3NaO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.4
  • Z-FG-NHO-BzOME

    CAS:
    <p>Z-FG-NHO-BzOME is a chemical compound functioning as a cysteine protease inhibitor, selectively targeting and inhibiting cathepsin B, cathepsin L, cathepsin S,</p>
    Formula:C27H27N3O7
    Color and Shape:Solid
    Molecular weight:505.52
  • HIV-1 protease-IN-7

    CAS:
    <p>HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].</p>
    Formula:C68H104N10O12S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1285.68
  • BAY-320

    CAS:
    <p>BAY-320 is a Bub1 inhibitor. With an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.</p>
    Formula:C26H26F2N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:492.52
  • Cyclotheonellazole A

    CAS:
    <p>Cyclotheonellazole A inhibits elastase (IC50=0.034nM) &amp; chymotrypsin (IC50=0.62nM), a natural macrocyclic peptide.</p>
    Formula:C44H54N9NaO14S2
    Color and Shape:Solid
    Molecular weight:1020.07
  • JTK-853

    CAS:
    <p>JTK-853: novel non-nucleoside HCV polymerase inhibitor with strong antiviral activity (EC50: 0.38 μM genotype 1a, 0.035 μM 1b).</p>
    Formula:C28H23F7N6O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:704.64
  • Z-PDLDA-NHOH

    CAS:
    <p>Z-PDLDA-NHOH is a potent, specific vertebrate collagenase inhibitor [1].</p>
    Formula:C22H32N4O6
    Color and Shape:Solid
    Molecular weight:448.51
  • HIV-1 protease-IN-9

    CAS:
    <p>HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and a</p>
    Formula:C37H41N7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:679.83
  • DCLK1-IN-2

    CAS:
    <p>DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cell</p>
    Formula:C26H32N8O3S
    Color and Shape:Solid
    Molecular weight:536.65
  • Berotralstat HCl

    CAS:
    <p>Berotralstat HCl is a selective plasma kallikrein inhibitor, reducing pain and swelling in HAE by blocking bradykinin release.</p>
    Formula:C30H28Cl2F4N6O
    Color and Shape:Solid
    Molecular weight:635.4886
  • Z-DEVD-CMK

    CAS:
    <p>Z-DEVD-CMK irreversibly inhibits various cathepsins in vitro [1].</p>
    Formula:C27H35ClN4O12
    Color and Shape:Solid
    Molecular weight:643.04
  • I-XW-053

    CAS:
    <p>I-XW-053 is an inhibitor of capsid targeted HIV-1 replication using the hybrid structure based method to block the interface between CA N-terminal domains (NTD-</p>
    Formula:C22H16N2O2
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:340.37
  • O-Benzoylhydroxylamine

    CAS:
    <p>O-Benzoyl hydroxylamine exhibits properties as a dipeptidyl peptidase-IV (DPP-IV) inhibitor and demonstrates antidiabetic effects[1].</p>
    Formula:C7H7NO2
    Color and Shape:Solid
    Molecular weight:137.14
  • Kallikrein-IN-2

    CAS:
    <p>Kallikrein-IN-2 (compound 1) is an inhibitor of the kinin-releasing enzyme Kallikrein.</p>
    Formula:C28H25F3N4O4
    Color and Shape:Solid
    Molecular weight:538.52
  • Neurodegenerative Disorder-Targeting Compound 1

    CAS:
    <p>Neurodegenerative Disorder-Targeting Compound 1 is an inhibitor of calpain [1].</p>
    Formula:C28H28N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:484.55
  • NCI-B16

    CAS:
    <p>NCI-B16 is a small-molecule RNA binder that inhibits HCV (hepatitis C virus) replication [1].</p>
    Formula:C27H26N8O4
    Color and Shape:Solid
    Molecular weight:526.55
  • KCC009

    CAS:
    <p>KCC009 is a potent and selective Transglutaminase 2 Inhibitor.</p>
    Formula:C21H22BrN3O5
    Color and Shape:Solid
    Molecular weight:476.32
  • SQ 32056

    CAS:
    <p>SQ 32056 is a cathepsin E inhibitor.</p>
    Formula:C37H56N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:636.86
  • BMS-189664 HCl

    CAS:
    <p>BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.</p>
    Formula:C22H35ClN6O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.07
  • Ecallantide

    CAS:
    <p>Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.</p>
    Formula:C305H448N88O91S8
    Color and Shape:Solid
    Molecular weight:7059.88
  • Proteasome-IN-4


    <p>Proteasome-IN-4, a potent non-covalent inhibitor (IC50=8.39nM), halts cancer cell growth, useful for oncology studies.</p>
    Formula:C44H58N6O5
    Color and Shape:Solid
    Molecular weight:750.97
  • MMP-145

    CAS:
    <p>MMP-145 is used as a protease inhibitor.</p>
    Formula:C20H20N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.45
  • HIV-1 protease-IN-8

    CAS:
    <p>HIV-1 protease-IN-8 (compound 34b) is a potent inhibitor of the HIV-1 protease enzyme, exhibiting an IC50 of 0.32 nM.</p>
    Formula:C25H35N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.63
  • Human enteropeptidase-IN-1

    CAS:
    <p>Enteropeptidase-IN-1: orally active, potent inhibitor, low systemic exposure, for anti-obesity research.</p>
    Formula:C20H18N4O7
    Color and Shape:Solid
    Molecular weight:426.38
  • MeOSuc-AAPV-CMK

    CAS:
    <p>MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediated</p>
    Formula:C22H35ClN4O7
    Color and Shape:Solid
    Molecular weight:502.99
  • NK3201

    CAS:
    <p>NK3201, a specific chymase inhibitor, suppresses bleomycin-induced pulmonary fibrosis in hamsters.</p>
    Formula:C31H29N5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:567.59