CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 985 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • CL 82198 hydrochloride

    CAS:
    CL 82198 hydrochloride selectively inhibits MMP-13, not MMP-1/9/TACE, and blocks HP75 invasion and neurotoxicity in zebrafish.
    Formula:C17H23ClN2O3
    Color and Shape:Solid
    Molecular weight:338.83

    Ref: TM-T41179

    10mg
    642.00€
  • Z-Leu-Tyr-Chloromethylketone

    CAS:
    Z-Leu-Tyr-Chloromethylketone is a calpain inhibitor [1].
    Formula:C24H29ClN2O5
    Color and Shape:Solid
    Molecular weight:460.95

    Ref: TM-T80103

    5mg
    To inquire
    50mg
    To inquire
  • Sofosbuvir impurity L


    Sofosbuvir impurity L is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.
    Formula:C22H29FN3O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:545.45

    Ref: TM-T12967

    25mg
    2,403.00€
    50mg
    2,952.00€
    100mg
    3,690.00€
  • KKI-5

    CAS:

    KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.

    Formula:C35H55N11O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:773.88

    Ref: TM-TP1792

    1mg
    64.00€
    5mg
    172.00€
    10mg
    299.00€
  • CRA-2059 TFA


    CRA-2059 is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].
    Color and Shape:Solid

    Ref: TM-T38052

    5mg
    1,295.00€
  • DPP8/9-IN-1


    DPP8/9-IN-1 (Compound 16) is a selective covalent inhibitor of dipeptidyl peptidase 8 and 9 (DPP8/9), with IC50 values of 14 nM and 298 nM, respectively. It irreversibly binds to the active site serine (such as S730 in DPP9) through a phosphate ester warhead, blocking substrate binding and inhibiting DPP8/9-mediated protein processing. DPP8/9-IN-1 holds potential for research in cancer and inflammatory diseases.
    Color and Shape:Odour Solid

    Ref: TM-T206718

    10mg
    To inquire
    50mg
    To inquire
  • NVP-DPP728 dihydrochloride

    CAS:
    NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.
    Formula:C15H20Cl2N6O
    Color and Shape:Solid
    Molecular weight:371.27

    Ref: TM-T39481

    25mg
    1,369.00€
  • Histatin 5

    CAS:
    Histatin 5, a human saliva peptide, blocks MMP-2 and MMP-9 at IC50s of 0.57/0.25 μM and kills fungi.
    Formula:C133H195N51O33
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3036.29

    Ref: TM-TP1741

    1mg
    163.00€
    5mg
    562.00€
    10mg
    892.00€
  • HCVP-IN-1

    CAS:
    HCVP-IN-1 (compound 1) is a hepatitis C viral polymerase (HCVP) inhibitor.
    Formula:C30H34FN5O3
    Color and Shape:Solid
    Molecular weight:531.632

    Ref: TM-T41002

    5mg
    873.00€
  • Leptosphaerodione

    CAS:
    Leptosphaerodione from Remotididymella sp.: a potent UPS inhibitor with 3.2 μM IC50 in HeLa cells; anti-tumor.
    Formula:C21H22O5
    Color and Shape:Solid
    Molecular weight:354.4

    Ref: TM-T75488

    5mg
    To inquire
    50mg
    To inquire
  • Sofosbuvir impurity J

    CAS:
    Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.
    Formula:C22H30FN4O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:528.47

    Ref: TM-T12965

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • PS 915

    CAS:
    PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.
    Formula:C27H36ClN7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:590.08

    Ref: TM-T24674

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • TR-107

    CAS:
    TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.
    Formula:C22H19ClN4O
    Color and Shape:Soild
    Molecular weight:390.87

    Ref: TM-T85310

    5mg
    49.00€
    10mg
    72.00€
    25mg
    130.00€
    50mg
    203.00€
    100mg
    320.00€
    500mg
    755.00€
  • OM-7D3-B3


    OM-7D3-B3 is a monoclonal antibody that targets human tight junction protein 1 (CLDN1) with a dissociation constant (Kd) of 4 nM. This antibody inhibits the role of CLDN1 in the cellular entry of the hepatitis C virus (HCV) and holds potential for research into HCV infection.
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-901

    1mg
    To inquire
    5mg
    To inquire
  • APC-6860

    CAS:
    APC-6860, a serine protease inhibitor, targets multiple enzymes; most potent against human urokinase (Ki: 0.1 µM). Used in cancer research.
    Formula:C9H7IN2S
    Color and Shape:Solid
    Molecular weight:302.13

    Ref: TM-T39029

    5mg
    873.00€
  • Anticancer agent 114


    Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.
    Formula:C28H33BF6N2O7
    Color and Shape:Solid
    Molecular weight:634.37

    Ref: TM-T74839

    5mg
    To inquire
    50mg
    To inquire
  • Elastatinal

    CAS:
    Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.
    Formula:C21H36N8O7
    Color and Shape:Yellowish Solid
    Molecular weight:512.56

    Ref: TM-T20130

    5mg
    304.00€
    10mg
    575.00€
    25mg
    1,251.00€
  • Tyrosinase/elastase-IN-1


    Tyrosinase/elastase-IN-1, a triterpenoid extracted from the leaves of Rubus fraxinifolius, exhibits inhibitory activities against both tyrosinase and elastase
    Formula:C33H52O5
    Color and Shape:Solid
    Molecular weight:528.76

    Ref: TM-T74243

    5mg
    To inquire
    50mg
    To inquire
  • LM11


    LM11 is a transglutaminase 2 (TG2) inhibitor that exhibits activity against glioblastoma cells by maintaining TG2 in a cytotoxic conformational state.

    Formula:C26H18Cl2N4O5
    Molecular weight:536.06543

    Ref: TM-T209326

    10mg
    To inquire
    50mg
    To inquire
  • Elastase (high purity)


    Elastase (high purity) is a serine protease that hydrolyzes proteins and peptides.
    Color and Shape:Odour Solid

    Ref: TM-TRP-00545

    10mg
    To inquire
    50mg
    To inquire