
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(38 products)
- Cysteine Protease(111 products)
- DPP-4(27 products)
- Glutaminase(46 products)
- HIV Protease(506 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(55 products)
- Proteasome(86 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 984 products of "Proteases/Proteasome"
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Velpatasvir
CAS:Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.Formula:C49H54N8O8Purity:99.17% - 99.83%Color and Shape:SolidMolecular weight:883Ref: TM-T3334
5mg34.00€10mg49.00€1mL*10mM (DMSO)54.00€25mg79.00€50mg98.00€100mg152.00€200mg219.00€500mg358.00€Efegatran HCl
CAS:Efegatran (GYKI-14166, RGH-2958, LY294468) is a thrombin inhibitor in development by IVAX for thromboembolic disorders.Formula:C21H34Cl2N6O3Color and Shape:SolidMolecular weight:489.442Brensocatib
CAS:Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).Formula:C23H24N4O4Purity:97.55%Color and Shape:SolidMolecular weight:420.46STK16-IN-1
CAS:STK16-IN-1 is an inhibitor of STK16 kinase (IC50: 295 nM).Formula:C17H12FN3OPurity:99.52%Color and Shape:SolidMolecular weight:293.32-Benzylsuccinic acid
CAS:2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formula:C11H12O4Purity:99.01% - ≥95%Color and Shape:SolidMolecular weight:208.21Coblopasvir dihydrochloride
CAS:Coblopasvir dihydrochloride can be used to study chronic HCV infection and is a pan-genotypic nonstructural protein 5A (NS5A) inhibitor.Formula:C41H52Cl2N8O8Purity:99.33%Color and Shape:SolidMolecular weight:855.81Ref: TM-T25268L
1mg87.00€5mg187.00€1mL*10mM (DMSO)298.00€10mg305.00€25mg518.00€50mg742.00€100mg1,017.00€Grazoprevir
CAS:Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.Formula:C38H50N6O9SPurity:99.36% - >99.99%Color and Shape:SolidMolecular weight:766.9FT011
CAS:FT011, a direct anti-fibrotic agent,attenuates cardiac remodelling and dysfunction in experimental diabetic cardiomyopathy.Formula:C20H17NO5Purity:98.98%Color and Shape:SolidMolecular weight:351.35Tris(4-aminophenyl)methane
CAS:Tris(4-aminophenyl)methane (Leucopararosaniline), a triphenylmethane dye, is a weak HCV helicase inhibitor.Formula:C19H19N3Purity:95.73%Color and Shape:Beige Solid CrystallineMolecular weight:289.37Ilomastat
CAS:Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.Formula:C20H28N4O4Purity:97.04% - 99.51%Color and Shape:SolidMolecular weight:388.46Ref: TM-T2743
1mg46.00€2mg62.00€5mg89.00€1mL*10mM (DMSO)94.00€10mg145.00€25mg255.00€50mg429.00€100mg620.00€200mg880.00€TMC647055 Choline Hydroxide Salt
TMC647055 is a potent HCV NS5B inhibitor with low toxicity and good pharmacokinetics, under clinical evaluation.Formula:C37H53N5O8SPurity:99.44%Color and Shape:SolidMolecular weight:727.91Ref: TM-T21537L
1mg95.00€5mg200.00€1mL*10mM (DMSO)286.00€10mg289.00€25mg520.00€50mg742.00€100mg1,018.00€JNJ0966
CAS:JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).Formula:C16H16N4O2S2Purity:99.46% - 99.62%Color and Shape:SolidMolecular weight:360.45Ref: TM-T4783
2mg34.00€1mL*10mM (DMSO)35.00€5mg46.00€10mg64.00€25mg126.00€50mg219.00€100mg315.00€200mg434.00€UAMC00039 dihydrochloride
CAS:UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM.Formula:C16H26Cl3N3OPurity:>99.99%Color and Shape:SolidMolecular weight:382.76PythiDC
CAS:PythiDC is a selective collagen prolyl 4-hydroxylase inhibitor, neither causing general toxicity nor disrupting iron homeostasis.Formula:C10H6N2O4SPurity:98.13%Color and Shape:SolidMolecular weight:250.23Simeprevir
CAS:Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.Formula:C38H47N5O7S2Purity:99.45% - 99.92%Color and Shape:SolidMolecular weight:749.94Bz-RS-ISer(3-Ph)-Ome
CAS:Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.
Formula:C17H17NO4Purity:99.36% - 99.89%Color and Shape:White CrystalMolecular weight:299.32Glecaprevir
CAS:Glecaprevir (ABT-493) is an HCV NS3/4A protease inhibitor, (IC50s: 3.5-11.3 nM).Formula:C38H46F4N6O9SPurity:99.16% - 99.69%Color and Shape:SolidMolecular weight:838.87Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purity:98.75%Color and Shape:SolidMolecular weight:300.83VCH-916 free acid(1200133-34-1 free base)
CAS:VCH-916 is a novel nonnucleoside HCV NS5B polymerase inhibitor.Formula:C26H37NO4SPurity:98.45%Color and Shape:SolidMolecular weight:459.647-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
CAS:7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).Formula:C15H16N4Purity:99.22%Color and Shape:SolidMolecular weight:252.31
