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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 980 products of "Proteases/Proteasome"

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  • PF-00356231 hydrochloride

    CAS:
    PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.
    Formula:C25H21ClN2O3S
    Purity:98.39%
    Color and Shape:Solid
    Molecular weight:464.96

    Ref: TM-T12414

    500mg
    To inquire
    1mg
    67.00€
    5mg
    177.00€
    10mg
    284.00€
    25mg
    464.00€
    50mg
    642.00€
    100mg
    853.00€
  • Tyrosinase-IN-5

    CAS:
    Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.
    Formula:C18H13N3O6
    Color and Shape:Solid
    Molecular weight:367.31

    Ref: TM-T61425

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BRD-8899

    CAS:
    BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].
    Formula:C17H22N4O3S
    Color and Shape:Solid
    Molecular weight:362.45

    Ref: TM-T61361

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GS-9256

    CAS:
    GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].
    Formula:C46H56ClF2N6O8PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:957.46

    Ref: TM-T71653

    25mg
    14,013.00€
    50mg
    19,926.00€
    100mg
    28,288.00€
  • Z-LLF-CHO

    CAS:
    Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.
    Formula:C29H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:509.64

    Ref: TM-T78640

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BC-23

    CAS:
    BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.
    Formula:C21H14ClN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.87

    Ref: TM-T26754

    1mg
    99.00€
    5mg
    187.00€
    10mg
    303.00€
    25mg
    547.00€
    50mg
    817.00€
    100mg
    1,225.00€
  • Gemigliptin Tartrate(911637-19-9 free base)

    CAS:
    Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).
    Formula:C22H25F8N5O8
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:639.45

    Ref: TM-T7369L

    2mg
    38.00€
    5mg
    57.00€
    1mL*10mM (DMSO)
    90.00€
    10mg
    93.00€
    25mg
    148.00€
    50mg
    245.00€
  • HCV-IN-36

    CAS:
    HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.
    Formula:C30H36ClN5
    Color and Shape:Solid
    Molecular weight:502.09

    Ref: TM-T63407

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • NNGH

    CAS:
    NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.
    Formula:C13H20N2O5S
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:316.37

    Ref: TM-T21735

    1mg
    71.00€
    5mg
    105.00€
    10mg
    178.00€
    25mg
    313.00€
    50mg
    464.00€
    100mg
    660.00€
  • PK44 phosphate

    CAS:
    PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).
    Formula:C17H19F5N7O5P
    Color and Shape:Solid
    Molecular weight:527.349

    Ref: TM-T63698

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • AGLME

    CAS:
    AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.
    Formula:C11H21N3O4
    Color and Shape:Solid
    Molecular weight:259.3

    Ref: TM-T25007

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GLS1 Inhibitor-3

    CAS:
    GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.
    Formula:C30H32N10O2S
    Color and Shape:Solid
    Molecular weight:596.71

    Ref: TM-T64211

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ZM223 hydrochloride (2031177-48-5 free base)


    ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.
    Formula:C23H18ClF3N4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:538.99

    Ref: TM-T13412L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tanomastat

    CAS:
    Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.
    Formula:C23H19ClO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.91

    Ref: TM-T16986

    500µg
    92.00€
    1mg
    159.00€
    5mg
    487.00€
    10mg
    892.00€
  • MMP13-IN-4

    CAS:
    MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].
    Formula:C21H17BrN4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:485.29

    Ref: TM-T78774

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BI-L 45XX

    CAS:
    BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.
    Formula:C10H9F3N2O2S
    Color and Shape:Solid
    Molecular weight:278.25

    Ref: TM-T26813

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tyrphostin 47

    CAS:
    Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.
    Formula:C10H8N2O2S
    Color and Shape:Solid
    Molecular weight:220.25

    Ref: TM-T24908

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Levovirin valinate HCl

    CAS:
    Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.
    Formula:C13H22ClN5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.8

    Ref: TM-T25702L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ici 186756

    CAS:
    Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.
    Formula:C33H49N5O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.77

    Ref: TM-T25518

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Chymase-IN-2

    CAS:
    Chymase-IN-2 is a modulator of chymase.
    Formula:C19H15ClF2NO3PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.82

    Ref: TM-T12450

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€