CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 977 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • TAPI-1

    CAS:
    TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.
    Formula:C26H37N5O5
    Purity:≥95%
    Color and Shape:Solid
    Molecular weight:499.6

    Ref: TM-T6009

    1mg
    177.00€
  • GS-9256

    CAS:
    GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].
    Formula:C46H56ClF2N6O8PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:957.46

    Ref: TM-T71653

    25mg
    14,013.00€
    50mg
    19,926.00€
    100mg
    28,288.00€
  • Z-LLF-CHO

    CAS:
    Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.
    Formula:C29H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:509.64

    Ref: TM-T78640

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MMP13-IN-4

    CAS:
    MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].
    Formula:C21H17BrN4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:485.29

    Ref: TM-T78774

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ND-322 HCl

    CAS:
    ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.
    Formula:C15H16ClNO3S2
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:357.88

    Ref: TM-T28145

    1mg
    152.00€
    5mg
    334.00€
    1mL*10mM (DMSO)
    349.00€
    10mg
    492.00€
    25mg
    780.00€
    50mg
    1,044.00€
    100mg
    1,414.00€
  • PF-00356231 hydrochloride

    CAS:
    PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.
    Formula:C25H21ClN2O3S
    Purity:98.39%
    Color and Shape:Solid
    Molecular weight:464.96

    Ref: TM-T12414

    500mg
    To inquire
    1mg
    67.00€
    5mg
    177.00€
    10mg
    284.00€
    25mg
    464.00€
    50mg
    642.00€
    100mg
    853.00€
  • NNGH

    CAS:
    NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.
    Formula:C13H20N2O5S
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:316.37

    Ref: TM-T21735

    1mg
    71.00€
    5mg
    105.00€
    10mg
    178.00€
    25mg
    313.00€
    50mg
    464.00€
    100mg
    660.00€
  • ZM223 hydrochloride (2031177-48-5 free base)


    ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.
    Formula:C23H18ClF3N4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:538.99

    Ref: TM-T13412L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Flovagatran

    CAS:
    Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.
    Formula:C27H36BN3O7
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:525.4

    Ref: TM-T31806

    1mg
    685.00€
    5mg
    1,431.00€
    10mg
    1,783.00€
    50mg
    2,322.00€
  • RO-9187

    CAS:
    RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).
    Formula:C9H12N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:284.23

    Ref: TM-T16774

    2mg
    105.00€
    1mL*10mM (DMSO)
    197.00€
    5mg
    212.00€
    50mg
    648.00€
    100mg
    898.00€
  • 2-MPPA

    CAS:
    2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.
    Formula:C8H14O4S
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:206.26

    Ref: TM-T22497

    1mg
    50.00€
    5mg
    99.00€
    1mL*10mM (DMSO)
    109.00€
    10mg
    160.00€
    25mg
    358.00€
    50mg
    620.00€
    100mg
    1,108.00€
    200mg
    1,504.00€
  • Cofrogliptin

    CAS:
    Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).
    Formula:C18H19F5N4O3S
    Purity:99.25%
    Color and Shape:Solid
    Molecular weight:466.43

    Ref: TM-T62985

    25mg
    To inquire
    1mg
    73.00€
    5mg
    160.00€
    1mL*10mM (DMSO)
    164.00€
    10mg
    250.00€
    50mg
    803.00€
  • Gosogliptin

    CAS:
    Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.
    Formula:C17H24F2N6O
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:366.41

    Ref: TM-T11450

    1mg
    123.00€
    5mg
    295.00€
    10mg
    477.00€
    25mg
    982.00€
    50mg
    1,603.00€
    100mg
    2,142.00€
  • Efegatran sulfate

    CAS:
    Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.
    Formula:C21H34N6O7S
    Purity:≥98% - ≥98%
    Color and Shape:Solid
    Molecular weight:514.6

    Ref: TM-T25364L

    1mg
    290.00€
    5mg
    648.00€
    10mg
    858.00€
    25mg
    1,288.00€
  • ZD-0892

    CAS:
    ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).
    Formula:C24H32F3N3O5
    Purity:95% - 99.53%
    Color and Shape:Solid
    Molecular weight:499.52

    Ref: TM-T13389

    1mg
    73.00€
    5mg
    164.00€
    10mg
    261.00€
    25mg
    485.00€
    50mg
    665.00€
  • Calpain Inhibitor XII

    CAS:

    Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.

    Formula:C26H34N4O5
    Color and Shape:Solid
    Molecular weight:482.57

    Ref: TM-T21949

    1mg
    139.00€
    5mg
    512.00€
    10mg
    753.00€
    25mg
    1,064.00€
    50mg
    1,444.00€
  • MMP2-IN-2

    CAS:
    MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.
    Formula:C13H8N4O4
    Purity:98.09%
    Color and Shape:Solid
    Molecular weight:284.23

    Ref: TM-T60551

    1mg
    38.00€
    5mg
    80.00€
    10mg
    114.00€
    25mg
    215.00€
    50mg
    340.00€
    100mg
    557.00€
    500mg
    1,153.00€
  • TG2-IN-3h

    CAS:
    TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitor
    Formula:C21H26N4O4S
    Purity:99.34% - 99.76%
    Color and Shape:Solid
    Molecular weight:430.52

    Ref: TM-T70413

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
  • Gemigliptin

    CAS:
    Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)
    Formula:C18H19F8N5O2
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:489.36

    Ref: TM-T7369

    2mg
    38.00€
    5mg
    57.00€
    1mL*10mM (DMSO)
    84.00€
    10mg
    93.00€
    25mg
    148.00€
    50mg
    245.00€
    100mg
    385.00€
    500mg
    873.00€
  • Etarotene

    CAS:
    Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is a
    Formula:C25H32O2S
    Purity:99.58% - 99.98%
    Color and Shape:Solid
    Molecular weight:396.59

    Ref: TM-T25393

    1mg
    144.00€
    5mg
    346.00€
    10mg
    494.00€
    25mg
    740.00€