
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(34 products)
- Cysteine Protease(96 products)
- DPP-4(20 products)
- Glutaminase(40 products)
- HIV Protease(449 products)
- PAI-1(25 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(53 products)
- Proteasome(94 products)
- Serine Protease(50 products)
- p97(14 products)
Show 3 more subcategories
Found 1044 products of "Proteases/Proteasome"
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Azo-Resveratrol
CAS:<p>Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.</p>Formula:C12H10N2O3Color and Shape:SolidMolecular weight:230.22AM 4299 B
CAS:<p>AM 4299 B is a novel inhibitor of a thiol protease.</p>Formula:C16H27N3O7Purity:98%Color and Shape:SolidMolecular weight:373.4HCV-IN-34
CAS:<p>HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.</p>Formula:C31H36ClN5Color and Shape:SolidMolecular weight:514.1MDL 27399
CAS:<p>MDL 27399 suppresses human neutrophil cathepsin G.</p>Formula:C26H36N4O8Color and Shape:SolidMolecular weight:532.59Tyrosinase-IN-7
CAS:<p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>Formula:C15H10O5Purity:99%Color and Shape:SolidMolecular weight:270.24CAA0225
CAS:<p>CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.</p>Formula:C28H29N3O5Color and Shape:SolidMolecular weight:487.55BC-05
CAS:<p>BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for</p>Formula:C21H29BN2O9Purity:98%Color and Shape:SolidMolecular weight:464.27RID-F
CAS:<p>RID-F is an inhibitor of the nonpeptidic proteasome.</p>Formula:C38H50N2O2Purity:98%Color and Shape:SolidMolecular weight:566.82AL-9
CAS:<p>AL-9 is a GT-1b and GT-2a replication inhibitor.</p>Formula:C23H22N4O3Purity:98%Color and Shape:SolidMolecular weight:402.45Immunoproteasome inhibitor 1
CAS:<p>Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.</p>Formula:C20H26N2O4Color and Shape:SolidMolecular weight:358.43PMPA sodium
CAS:<p>PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.</p>Formula:C6H11Na4O7PPurity:98%Color and Shape:SolidMolecular weight:318.08JO146
CAS:<p>JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂,其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM,可应用于细菌感染的抑制。</p>Formula:C31H44N3O7PColor and Shape:SolidMolecular weight:601.67L-873724
CAS:<p>L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.</p>Formula:C23H26F3N3O3SPurity:98%Color and Shape:SolidMolecular weight:481.53(R)-ND-336
CAS:<p>(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.</p>Formula:C16H18ClNO3S2Color and Shape:SolidMolecular weight:371.89Tyrosinase-IN-11
CAS:<p>Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.</p>Formula:C15H14O5Color and Shape:SolidMolecular weight:274.27Kallikrein 5-IN-2
CAS:<p>Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.</p>Formula:C23H22N6OColor and Shape:SolidMolecular weight:398.46VA4 TG2 inhibitor
CAS:<p>VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.</p>Formula:C33H41N5O6SColor and Shape:SolidMolecular weight:635.77AZD5248
CAS:<p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>Formula:C22H22N4O2Color and Shape:SolidMolecular weight:374.44MMP-2/9-IN-1
CAS:<p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>Formula:C14H16IN7SColor and Shape:SolidMolecular weight:441.29GLS1 Inhibitor-3
CAS:<p>GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.</p>Formula:C30H32N10O2SColor and Shape:SolidMolecular weight:596.71
