
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(34 products)
- Cysteine Protease(96 products)
- DPP-4(20 products)
- Glutaminase(40 products)
- HIV Protease(447 products)
- PAI-1(25 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(94 products)
- Serine Protease(50 products)
- p97(14 products)
Show 3 more subcategories
Found 1045 products of "Proteases/Proteasome"
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Galegenimab
CAS:<p>Galegenimab (FHTR 2163; RG 6147; RO 7171009) is an HTRA1 antibody fragment for AMD research.</p>Purity:95% - 95%Color and Shape:LiquidZampilimab
CAS:<p>Zampilimab (UCB-7858) is a humanised monoclonal antibody targeting TGM2, inhibits the cross-linking transamidase activity of TG2, renal fibrosis.</p>Purity:95%Color and Shape:LiquidHCV-IN-30
CAS:<p>HCV-IN-30 is an HCV NS5A replication complex inhibitor (IC50s: 901 and 102 nM for genotypes 1a and 1b replicons).</p>Formula:C36H44N6O4Purity:99.6%Color and Shape:SolidMolecular weight:624.77Carboxypeptidase G2 (CPG2) Inhibitor
CAS:<p>Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.</p>Formula:C13H15NO6SPurity:99.96%Color and Shape:SolidMolecular weight:313.33Cathepsin Inhibitor 1
CAS:<p>Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.</p>Formula:C20H24ClN5O2Purity:99.78%Color and Shape:SolidMolecular weight:401.89PK44 phosphate
CAS:<p>PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).</p>Formula:C17H19F5N7O5PColor and Shape:SolidMolecular weight:527.349DPP-4-IN-2
CAS:<p>DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.</p>Formula:C18H18N6OColor and Shape:SolidMolecular weight:334.38Alvelestat tosylate
CAS:<p>Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.</p>Formula:C32H30F3N5O7S2Purity:98%Color and Shape:SolidMolecular weight:717.73BAY8040
CAS:<p>BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.</p>Formula:C21H16F3N5O2Color and Shape:SolidMolecular weight:427.38HCV-IN-33
CAS:<p>HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.</p>Formula:C31H36ClN5Color and Shape:SolidMolecular weight:514.1AA10 TG2 inhibitor
CAS:<p>AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).</p>Formula:C32H36N4O5Color and Shape:SolidMolecular weight:556.65DPP-4-IN-1
CAS:<p>DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.</p>Formula:C19H19ClN6Color and Shape:SolidMolecular weight:366.85(Rac)-Tanomastat
CAS:<p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>Formula:C23H19ClO3SColor and Shape:SolidMolecular weight:410.91Thrombin Inhibitor 2
CAS:<p>Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.</p>Formula:C19H16ClF3N6O2Purity:98%Color and Shape:SolidMolecular weight:452.82PSI-7409 tetrasodium
CAS:<p>PSI-7409 tetrasodium, a sofosbuvir metabolite, inhibits GT 1b, 2a, 3a, 4a NS5B polymerases with IC50s of 1.6, 2.8, 0.7, 2.6 μM.</p>Formula:C10H16FN2Na4O14P3Purity:98%Color and Shape:SolidMolecular weight:592.117CAY10704
CAS:<p>CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.</p>Formula:C18H20Cl2N2Color and Shape:SolidMolecular weight:335.27ASPER-29
CAS:<p>ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.</p>Formula:C31H29BrN2O5SColor and Shape:SolidMolecular weight:621.54Evogliptin HCl
CAS:<p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>Formula:C19H27ClF3N3O3Color and Shape:SolidMolecular weight:437.88LY 806303
CAS:<p>LY 806303 is a highly selective thrombin inhibitor.</p>Formula:C16H14O5SPurity:98%Color and Shape:SolidMolecular weight:318.34Elasnin
CAS:<p>Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.</p>Formula:C24H40O4Color and Shape:SolidMolecular weight:392.57L 658758
CAS:<p>L 658758 is an inhibitor of serine proteinase.</p>Formula:C16H20N2O9SColor and Shape:SolidMolecular weight:416.4Glutaminase-IN-4
CAS:<p>Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).</p>Formula:C23H22N6O2S2Color and Shape:SolidMolecular weight:478.59Nucleoside-Analog-2
CAS:<p>Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.</p>Formula:C9H11N5O6Purity:98%Color and Shape:SolidMolecular weight:285.21BI-L 45XX
CAS:<p>BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.</p>Formula:C10H9F3N2O2SColor and Shape:SolidMolecular weight:278.25Tyrphostin 47
CAS:<p>Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.</p>Formula:C10H8N2O2SColor and Shape:SolidMolecular weight:220.25Levovirin valinate HCl
CAS:<p>Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.</p>Formula:C13H22ClN5O6Purity:98%Color and Shape:SolidMolecular weight:379.8Ici 186756
CAS:<p>Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.</p>Formula:C33H49N5O9Purity:98%Color and Shape:SolidMolecular weight:659.77MMP2-IN-2
CAS:<p>MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.</p>Formula:C13H8N4O4Purity:98.09%Color and Shape:SolidMolecular weight:284.23SAP2-IN-1
CAS:<p>SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.</p>Formula:C34H29NO7Color and Shape:SolidMolecular weight:563.6Chymase-IN-2
CAS:<p>Chymase-IN-2 is a modulator of chymase.</p>Formula:C19H15ClF2NO3PSPurity:98%Color and Shape:SolidMolecular weight:441.82α-Glucosidase-IN-5
CAS:<p>α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.</p>Formula:C15H13NO3Color and Shape:SolidMolecular weight:255.27A-953227
CAS:<p>A-953227: Selective calpain inhibitor with improved cathepsin selectivity, strong microsomal stability, and cellular efficacy.</p>Formula:C25H20FN5O3Purity:98%Color and Shape:SolidMolecular weight:457.46Tyrosinase-IN-5
CAS:<p>Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.</p>Formula:C18H13N3O6Color and Shape:SolidMolecular weight:367.31Duazomycin
CAS:<p>Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.</p>Formula:C8H11N3O4Color and Shape:SolidMolecular weight:213.19BMS-363131
CAS:<p>BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.</p>Formula:C28H40N6O5Purity:97.99%Color and Shape:SolidMolecular weight:540.65Moxicoumone
CAS:<p>Moxicoumone is an anticoagulant agent.</p>Formula:C22H30N2O6Purity:98%Color and Shape:SolidMolecular weight:418.48BRD-8899
CAS:<p>BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].</p>Formula:C17H22N4O3SColor and Shape:SolidMolecular weight:362.45HCV-IN-36
CAS:<p>HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.</p>Formula:C30H36ClN5Color and Shape:SolidMolecular weight:502.09Tyrphostin A46
CAS:<p>Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.</p>Formula:C10H8N2O3Purity:98%Color and Shape:Off-White SolidMolecular weight:204.18GLS1 Inhibitor
CAS:<p>GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.</p>Formula:C19H21N7O2SColor and Shape:SolidMolecular weight:411.48MDK0734
CAS:<p>MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>Formula:C15H17N3O2Purity:98%Color and Shape:SolidMolecular weight:271.31NVP DPP 728 dihydrochloride
CAS:<p>NVP-DPP728 is a reversible DPP-IV inhibitor with a K i of 11 nM, enhancing insulin release by preventing GLP-1 degradation, used for diabetes research.</p>Formula:C15H18N6OColor and Shape:SolidMolecular weight:298.34Elastase-IN-1
CAS:<p>Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].</p>Formula:C17H12N4O3Color and Shape:SolidMolecular weight:320.3GLS1 Inhibitor-3
CAS:<p>GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.</p>Formula:C30H32N10O2SColor and Shape:SolidMolecular weight:596.71MMP-2/9-IN-1
CAS:<p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>Formula:C14H16IN7SColor and Shape:SolidMolecular weight:441.29AZD5248
CAS:<p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>Formula:C22H22N4O2Color and Shape:SolidMolecular weight:374.44FQ
CAS:<p>FQ is a novel reversible inhibitor of mixed-type tyrosinase.</p>Formula:C14H9FN2OColor and Shape:SolidMolecular weight:240.23VA4 TG2 inhibitor
CAS:<p>VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.</p>Formula:C33H41N5O6SColor and Shape:SolidMolecular weight:635.77Bz-D-Arg-pNA hydrochloride
CAS:<p>Bz-D-Arg-pNA hydrochloride is a competitive trypsin inhibitor.</p>Formula:C19H23ClN6O4Color and Shape:SolidMolecular weight:434.88ADAMTS-5 Inhibitor
CAS:<p>ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.</p>Formula:C16H11ClF3N3OS3Purity:99.66%Color and Shape:SolidMolecular weight:449.92DPP-IV-IN-1
CAS:<p>DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).</p>Formula:C11H18FN3O2Purity:98%Color and Shape:SolidMolecular weight:243.28TNIK-IN-1
CAS:<p>TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).</p>Formula:C19H17N5O3SPurity:98%Color and Shape:SolidMolecular weight:395.43Kallikrein 5-IN-2
CAS:<p>Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.</p>Formula:C23H22N6OColor and Shape:SolidMolecular weight:398.46Diethyl pyimDC
CAS:<p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>Formula:C14H15N3O4Color and Shape:SolidMolecular weight:289.29Aldumastat
CAS:<p>Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.</p>Formula:C20H24F2N4O3Purity:99.87%Color and Shape:SolidMolecular weight:406.43ND-336
CAS:<p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>Formula:C16H18ClNO3S2Color and Shape:SolidMolecular weight:371.9Tyrosinase-IN-11
CAS:<p>Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.</p>Formula:C15H14O5Color and Shape:SolidMolecular weight:274.27MK-4882
CAS:<p>MK-4882 is an effective inhibitor of HCV NS5A.</p>Formula:C42H50N8O7Purity:98%Color and Shape:SolidMolecular weight:778.9YM-53601
CAS:<p>YM-53601 is an SQS inhibitor that inhibits adipogenic biosynthesis and lipid secretion in rodents.YM-53601 is a cholesterol-lowering agent that inhibits FDFT1.</p>Formula:C21H22ClFN2OPurity:99.65%Color and Shape:SolidMolecular weight:372.86Gosogliptin
CAS:<p>Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.</p>Formula:C17H24F2N6OPurity:99.74%Color and Shape:SolidMolecular weight:366.41(R)-ND-336
CAS:<p>(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.</p>Formula:C16H18ClNO3S2Color and Shape:SolidMolecular weight:371.89L-873724
CAS:<p>L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.</p>Formula:C23H26F3N3O3SPurity:98%Color and Shape:SolidMolecular weight:481.53JO146
CAS:<p>JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂,其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM,可应用于细菌感染的抑制。</p>Formula:C31H44N3O7PColor and Shape:SolidMolecular weight:601.67Sortin1
CAS:<p>Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.</p>Formula:C26H19NO6Purity:98%Color and Shape:SolidMolecular weight:441.43MDK7677
CAS:<p>MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>Formula:C12H10N4O3Color and Shape:SolidMolecular weight:258.23Furaprofen
CAS:<p>Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.</p>Formula:C17H14O3Purity:98.49% - 99.52%Color and Shape:SolidMolecular weight:266.29Immunoproteasome inhibitor 1
CAS:<p>Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.</p>Formula:C20H26N2O4Color and Shape:SolidMolecular weight:358.43GEMSA
CAS:<p>GEMSA is a potent inhibitor of enkephalin convertase ( K i =8.8 nM) with analgesic effect[1].</p>Formula:C7H13N3O4SColor and Shape:SolidMolecular weight:235.26Cysteine Protease inhibitor hydrochloride
CAS:<p>Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.</p>Formula:C18H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:338.79GSK2793660 HCl
CAS:<p>GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.</p>Formula:C22H32ClN3O3Color and Shape:SolidMolecular weight:421.96PMPA sodium
CAS:<p>PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.</p>Formula:C6H11Na4O7PPurity:98%Color and Shape:SolidMolecular weight:318.08Nucleoside-Analog-1
CAS:<p>Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.</p>Formula:C9H9N5O5Purity:98%Color and Shape:SolidMolecular weight:267.2AK 275
CAS:<p>AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.</p>Formula:C20H31N3O4Color and Shape:SolidMolecular weight:377.48AZD-9684
CAS:<p>AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.</p>Formula:C10H14N2O2SColor and Shape:SolidMolecular weight:226.3CAA0225
CAS:<p>CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.</p>Formula:C28H29N3O5Color and Shape:SolidMolecular weight:487.55ITX-4520
CAS:<p>ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.</p>Formula:C24H23F2N3OSColor and Shape:SolidMolecular weight:439.52WAY-151693
CAS:<p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>Formula:C21H22ClN3O5SColor and Shape:SolidMolecular weight:463.93L 722151
CAS:<p>L 722151 is an FXIIIa inhibitor.</p>Formula:C8H9ClN2O5S3Purity:98%Color and Shape:SolidMolecular weight:344.82Epostatin
CAS:<p>Epostatin is a new dipeptidyl peptidase II (DPP-II, EC 3.4.14.2) inhibitor.</p>Formula:C23H33N3O5Purity:98%Color and Shape:SolidMolecular weight:431.53Chymase-IN-1
CAS:<p>Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).</p>Formula:C20H15ClNO4PSPurity:99.17%Color and Shape:SolidMolecular weight:431.83AL-9
CAS:<p>AL-9 is a GT-1b and GT-2a replication inhibitor.</p>Formula:C23H22N4O3Purity:98%Color and Shape:SolidMolecular weight:402.45ADAMTS-5-IN-2
CAS:<p>ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.</p>Formula:C17H15N3OSColor and Shape:SolidMolecular weight:309.39GSK-2793660
CAS:<p>GSK-2793660, an oral, irreversible CTSC inhibitor, aids bronchiectasis research.</p>Formula:C20H27N3O3Purity:98%Color and Shape:SolidMolecular weight:357.45Safironil
CAS:<p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>Formula:C15H23N3O4Purity:99.83%Color and Shape:SolidMolecular weight:309.36RID-F
CAS:<p>RID-F is an inhibitor of the nonpeptidic proteasome.</p>Formula:C38H50N2O2Purity:98%Color and Shape:SolidMolecular weight:566.82SP-Chymostatin B
CAS:<p>SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.</p>Formula:C30H41N7O6Purity:98%Color and Shape:SolidMolecular weight:595.69TNK2-IN-1
CAS:<p>TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.</p>Formula:C23H24N6O2Color and Shape:SolidMolecular weight:416.48BC-05
CAS:<p>BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for</p>Formula:C21H29BN2O9Purity:98%Color and Shape:SolidMolecular weight:464.27A-933548
CAS:<p>A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.</p>Formula:C25H21N5O3Purity:98%Color and Shape:SolidMolecular weight:439.47Antiviral agent 30
CAS:<p>Antiviral Agent 30 (Example 118) is an active compound against HCV and RSV with an inhibitory concentration (IC 50) of greater than 25μM [1].</p>Formula:C21H32N2O3SColor and Shape:SolidMolecular weight:392.56K 579
CAS:<p>K 579 is a dipeptidyl peptidase IV inhibitor.</p>Formula:C17H24N6OPurity:98%Color and Shape:SolidMolecular weight:328.41Tyrosinase-IN-7
CAS:<p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>Formula:C15H10O5Purity:99%Color and Shape:SolidMolecular weight:270.24PTIQ
CAS:<p>MMP-3 expression inhibitor</p>Formula:C13H17NO3Purity:98%Color and Shape:SolidMolecular weight:235.28MDL 27399
CAS:<p>MDL 27399 suppresses human neutrophil cathepsin G.</p>Formula:C26H36N4O8Color and Shape:SolidMolecular weight:532.59AM 4299 B
CAS:<p>AM 4299 B is a novel inhibitor of a thiol protease.</p>Formula:C16H27N3O7Purity:98%Color and Shape:SolidMolecular weight:373.4BAY-678 racemate
CAS:<p>BAY-678 racemate: orally active, selective cell-permeable HNE inhibitor with IC50 of 20 nM.</p>Formula:C20H15F3N4O2Purity:98%Color and Shape:SolidMolecular weight:400.35HCV-IN-34
CAS:<p>HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.</p>Formula:C31H36ClN5Color and Shape:SolidMolecular weight:514.1ABT-770
CAS:<p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>Formula:C22H22F3N3O6Color and Shape:SolidMolecular weight:481.42Calpain Inhibitor XI
CAS:<p>Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.</p>Formula:C26H40N4O6Color and Shape:SolidMolecular weight:504.62Azo-Resveratrol
CAS:<p>Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.</p>Formula:C12H10N2O3Color and Shape:SolidMolecular weight:230.22WNK-IN-7
CAS:<p>WNK-IN-7 is a potent and selective WNK1 kinase inhibitor.</p>Formula:C26H29N3OPurity:98%Color and Shape:SolidMolecular weight:399.53CA 074
CAS:<p>CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates</p>Formula:C18H29N3O6Purity:97.80%Color and Shape:SolidMolecular weight:383.44XMU-MP-2
CAS:<p>XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft</p>Formula:C32H33F3N8O2Purity:99.29%Color and Shape:SolidMolecular weight:618.65BR351 precursor
CAS:<p>BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Formula:C27H32N2O8S2Purity:98%Color and Shape:SolidMolecular weight:576.68RS-104966
CAS:<p>RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.</p>Formula:C19H21NO6SPurity:98%Color and Shape:SolidMolecular weight:391.44(3S,4S)-A2-32-01
<p>(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .</p>Formula:C19H27NO2Color and Shape:SolidMolecular weight:301.42Ono-3307 mesylate
CAS:<p>no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.</p>Formula:C15H18N4O7S2Purity:97.60% - 98.16%Color and Shape:SolidMolecular weight:430.462',5-Difluoro-2'-deoxycytidine
CAS:<p>2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.</p>Formula:C9H11F2N3O4Purity:98%Color and Shape:SolidMolecular weight:263.2MMP-1-IN-1
<p>MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .</p>Formula:C14H17ClN2O3Color and Shape:SolidMolecular weight:296.75Gü1303
CAS:<p>Gü1303 is a highly potent and reversible inhibitor of Cathepsin K (CatK), with a Ki value of 0.91 nM for mature CatK (mCatK).</p>Formula:C20H22N4O3Color and Shape:SolidMolecular weight:366.41HCV-IN-35
CAS:<p>HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.</p>Formula:C30H36ClN5Color and Shape:SolidMolecular weight:502.09Thrombin inhibitor 6
CAS:<p>Thrombin Inhibitor 6, with an IC 50 of 1 nM, acts as a potent anticoagulant by inhibiting thrombin.</p>Formula:C18H19ClN4O2SColor and Shape:SolidMolecular weight:390.89NAAA-IN-2
CAS:<p>NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.</p>Formula:C11H13N3O2SColor and Shape:SolidMolecular weight:251.3TAPI-0
CAS:<p>TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.</p>Formula:C24H32N4O5Color and Shape:SolidMolecular weight:456.53Tyrosinase-IN-10
CAS:<p>Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'</p>Formula:C16H12O4Color and Shape:SolidMolecular weight:268.26Calpain-2-IN-1
CAS:<p>Calpain-2-IN-1 is a selective calpain-2 inhibitor that prolongs ERK activation and thus enhances learning and memory.</p>Formula:C28H37N3O7Color and Shape:SolidMolecular weight:527.61LY 135305
CAS:<p>LY 135305 is a inhibition of spontaneous metastasis.</p>Formula:C19H20ClNPurity:98%Color and Shape:SolidMolecular weight:297.822-MPPA
CAS:<p>2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.</p>Formula:C8H14O4SPurity:99.81%Color and Shape:SolidMolecular weight:206.26Plasma kallikrein-IN-3
CAS:<p>Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.</p>Formula:C20H23N5O2Color and Shape:SolidMolecular weight:365.43Tec-IN-21
CAS:<p>Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).</p>Formula:C16H15ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:362.83RO-9187
CAS:<p>RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).</p>Formula:C9H12N6O5Purity:98%Color and Shape:SolidMolecular weight:284.23Flovagatran
CAS:<p>Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.</p>Formula:C27H36BN3O7Purity:99.56%Color and Shape:SolidMolecular weight:525.4HCV-IN-3
CAS:<p>HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).</p>Formula:C13H11F2NOPurity:98%Color and Shape:SolidMolecular weight:235.23Batimastat sodium salt
CAS:<p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>Formula:C23H31N3NaO4S2Purity:98%Color and Shape:SolidMolecular weight:500.63BrBzGCp2
CAS:<p>BrBzGCp2 (p BrBzGSH(Cp)2) is a GLO1 inhibitor with antitumor activities, relieving anxiety, and is useful in researching neurological disorders.</p>Formula:C27H38BrN3O6SPurity:98.68% - 98.68%Color and Shape:SolidMolecular weight:612.58ACH-806
CAS:<p>ACH-806 is an NS4A antagonist. It can inhibit Hepatitis C Virus (HCV) replication with an EC50 of 14 nM.</p>Formula:C19H20F3N3O2SPurity:98%Color and Shape:SolidMolecular weight:411.44Sheng Gelieting
CAS:<p>CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.</p>Formula:C17H16F6N4OColor and Shape:SolidMolecular weight:406.33HCV-IN-37
CAS:<p>HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.</p>Formula:C31H35F2N5Color and Shape:SolidMolecular weight:515.64Tyrosinase-IN-1
CAS:<p>Tyrosinase-IN-1: potent inhibitor for skin-whitening & food preservation with uses in cosmetics & medicine.</p>Formula:C10H9N3O2S2Color and Shape:SolidMolecular weight:267.33Calpain Inhibitor XII
CAS:<p>Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.</p>Formula:C26H34N4O5Color and Shape:SolidMolecular weight:482.57Diprotin B
CAS:<p>Diprotin B is a dipeptidyl peptidase IV inhibitor.</p>Formula:C16H29N3O4Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:327.42ZM223 hydrochloride (2031177-48-5 free base)
<p>ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.</p>Formula:C23H18ClF3N4O2S2Purity:98%Color and Shape:SolidMolecular weight:538.99MK-2048
CAS:<p>MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.</p>Formula:C21H21ClFN5O4Purity:98%Color and Shape:SolidMolecular weight:461.87Navuridine
CAS:<p>Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.</p>Formula:C9H11N5O4Purity:99.83%Color and Shape:SolidMolecular weight:253.22KIN1400
CAS:<p>KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.</p>Formula:C24H17F2N3O2SPurity:98%Color and Shape:SolidMolecular weight:449.47Cathepsin L/S-IN-1
<p>Cathepsin L/S-IN-1 inhibits Cathepsin L & S (IC50: 4.10 & 1.79 μM) and reduces metastasis in pancreatic cancer cells.</p>Formula:C29H33BrN4O4SColor and Shape:SolidMolecular weight:613.57OM-189
CAS:<p>OM-189 is a selective inhibitor of synthetic thrombin.</p>Formula:C24H36N6O3SPurity:98%Color and Shape:SolidMolecular weight:488.65NNGH
CAS:<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Formula:C13H20N2O5SPurity:98.41%Color and Shape:SolidMolecular weight:316.37Cofrogliptin
CAS:<p>Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).</p>Formula:C18H19F5N4O3SColor and Shape:SolidMolecular weight:466.43Ro 09-1679
CAS:<p>Ro 09-1679 is a thrombin inhibitor.</p>Formula:C22H39N9O6Purity:98%Color and Shape:SolidMolecular weight:525.6Gü2602
CAS:<p>Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for mature</p>Formula:C16H22N4O3Color and Shape:SolidMolecular weight:318.37Adafosbuvir PM
CAS:<p>Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.</p>Formula:C10H13FN2O6Purity:97.08%Color and Shape:SolidMolecular weight:276.22BC-23
CAS:<p>BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.</p>Formula:C21H14ClN3O4SPurity:98%Color and Shape:SolidMolecular weight:439.87CP-471474
CAS:<p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>Formula:C16H17FN2O5SPurity:98%Color and Shape:SolidMolecular weight:368.38PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Formula:C25H21ClN2O3SPurity:98.39%Color and Shape:SolidMolecular weight:464.96Tyrosinase-IN-3
CAS:<p>Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.</p>Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.41AGLME
CAS:<p>AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.</p>Formula:C11H21N3O4Color and Shape:SolidMolecular weight:259.3p-Aminobenzamidine dihydrochloride
CAS:<p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>Formula:C7H11Cl2N3Purity:99.00% - 99.56%Color and Shape:SolidMolecular weight:208.088FK-448 Free base
CAS:<p>FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.</p>Formula:C25H30N2O3Purity:98%Color and Shape:SolidMolecular weight:406.52N-Phenylthiourea
CAS:<p>N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.</p>Formula:C7H8N2SPurity:99.71%Color and Shape:SolidMolecular weight:152.22BR351
CAS:<p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Formula:C20H25FN2O5SPurity:98%Color and Shape:SolidMolecular weight:424.49BMS-986094
CAS:<p>INX 08189 is an RNA-directed RNA polymerase (NS5B) inhibitor.</p>Formula:C30H39N6O9PColor and Shape:SolidMolecular weight:658.64(S)-BI-1001
CAS:<p>(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).</p>Formula:C19H15BrClNO3Purity:98%Color and Shape:SolidMolecular weight:420.68JPM-OEt
CAS:<p>JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.</p>Formula:C20H28N2O6Purity:98%Color and Shape:SolidMolecular weight:392.45LB-30057
CAS:<p>LB-30057 is used as an oral thrombin inhibitor.</p>Formula:C26H31N5O3SPurity:98%Color and Shape:SolidMolecular weight:493.62Grazoprevir sodium salt
CAS:<p>Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.</p>Formula:C38H50N6NaO9SPurity:98%Color and Shape:SolidMolecular weight:789.9Anticancer agent 82
CAS:<p>Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.</p>Formula:C19H18Cl2N4OColor and Shape:SolidMolecular weight:389.28U 27391
CAS:<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Formula:C23H36N4O5Purity:98%Color and Shape:SolidMolecular weight:448.56Tyrosinase-IN-4
CAS:<p>Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.</p>Formula:C15H9ClO3Color and Shape:SolidMolecular weight:272.68Gemigliptin Tartrate(911637-19-9 free base)
CAS:<p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>Formula:C22H25F8N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:639.45Cysteine protease inhibitor-2
CAS:<p>Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.</p>Formula:C13H5N5OPurity:98%Color and Shape:SolidMolecular weight:247.21ZD8321
CAS:<p>ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).</p>Formula:C18H28F3N3O5Purity:98%Color and Shape:SolidMolecular weight:423.43Proteasome-IN-1
CAS:<p>Proteasome-IN-1 is an inhibitor of proteasome.</p>Formula:C42H35N5O3Purity:98%Color and Shape:SolidMolecular weight:657.76Tanomastat
CAS:<p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>Formula:C23H19ClO3SPurity:98%Color and Shape:SolidMolecular weight:410.91MDL-101146, (S)-
CAS:<p>MDL-101146, (S)- is an effective orally active inhibitor of human neutrophil elastase.</p>Formula:C29H37F5N4O6Purity:98%Color and Shape:SolidMolecular weight:632.62IMB-26
CAS:<p>IMB-26 is an HCV inhibitor (EC50: 2.1 μM) and has shown potent anti-HCV effects.</p>Formula:C20H23BrN2O6Color and Shape:SolidMolecular weight:467.31Tyrosinase-IN-6
CAS:<p>Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.</p>Formula:C24H31N3O2Color and Shape:SolidMolecular weight:393.52ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Formula:C24H32F3N3O5Purity:95% - 99.53%Color and Shape:SolidMolecular weight:499.52SLK/STK10-IN-1
CAS:<p>SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.</p>Formula:C17H13ClN2O3Purity:99.34%Color and Shape:SolidMolecular weight:328.75Prodipine hydrochloride
CAS:<p>Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).</p>Formula:C20H26ClNPurity:98%Color and Shape:SolidMolecular weight:315.88DTS
CAS:<p>DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.</p>Formula:C14H14S3Purity:98%Color and Shape:SolidMolecular weight:278.46TAPI-1
CAS:<p>TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.</p>Formula:C26H37N5O5Purity:≥95%Color and Shape:SolidMolecular weight:499.6ZYZ-488
CAS:<p>ZYZ-488 is an Apoptosis protease activating factor-1 (Apaf-1) inhibitor, which suppresses the activation of procaspase-9 and procaspase-3.</p>Formula:C20H29N3O11Purity:99.04%Color and Shape:SolidMolecular weight:487.46Desethyl KBT-3022
CAS:<p>Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.</p>Formula:C23H20N2O4SPurity:98%Color and Shape:SolidMolecular weight:420.48ND-322 HCl
CAS:<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Formula:C15H16ClNO3S2Purity:99.49%Color and Shape:SolidMolecular weight:357.88Cyclophilin inhibitor 3
CAS:<p>Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.</p>Formula:C34H38N4O6Color and Shape:SolidMolecular weight:598.69STOCK2S-26016
CAS:<p>WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.</p>Formula:C20H19N3O2Color and Shape:SolidMolecular weight:333.38MMP13-IN-4
CAS:<p>MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].</p>Formula:C21H17BrN4O5Purity:98%Color and Shape:SolidMolecular weight:485.29Efegatran sulfate
CAS:<p>Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.</p>Formula:C21H34N6O7SPurity:≥98% - ≥98%Color and Shape:SolidMolecular weight:514.6Desirudin
CAS:<p>Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.</p>Color and Shape:SolidZ-LLF-CHO
CAS:<p>Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.</p>Formula:C29H39N3O5Purity:98%Color and Shape:SolidMolecular weight:509.64SJA6017
CAS:<p>SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.</p>Formula:C17H25FN2O4SPurity:98%Color and Shape:SolidMolecular weight:372.45AA9 TG2 inhibitor
CAS:<p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>Formula:C32H36N4O5Color and Shape:SolidMolecular weight:556.65GS-9256
CAS:<p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>Formula:C46H56ClF2N6O8PSPurity:98%Color and Shape:SolidMolecular weight:957.46Cysteine Protease inhibitor
CAS:<p>Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease</p>Formula:C18H14N4OPurity:98%Color and Shape:SolidMolecular weight:302.33SQ 32602
CAS:<p>SQ 32602 is a cathepsin E inhibitor.</p>Formula:C32H52N3O7PColor and Shape:SolidMolecular weight:621.74Tyrosinase-IN-8
<p>Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity while</p>Formula:C16H12O4Color and Shape:SolidMolecular weight:268.26Alicapistat
CAS:<p>Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).</p>Formula:C25H27N3O4Purity:98%Color and Shape:SolidMolecular weight:433.5VEL-0230
CAS:<p>VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.</p>Formula:C14H24NNaO5Color and Shape:SolidMolecular weight:309.33JNJ-10329670
CAS:<p>JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.</p>Formula:C30H34ClF3N6O3SColor and Shape:SolidMolecular weight:651.14BMS-488043
CAS:<p>BMS-488043 is a novel and unique oral small molecule HIV fusion inhibitor that inhibits the attachment of Human Immunodeficiency Virus type 1 (HIV-1) to CD4(+)</p>Formula:C22H22N4O5Purity:99.95%Color and Shape:SolidMolecular weight:422.43BAY-43-9695
CAS:<p>BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.</p>Formula:C22H25N3O4SPurity:99.50% - 99.65%Color and Shape:SolidMolecular weight:427.52BMS-929075
CAS:<p>BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokinetic</p>Formula:C31H24F2N4O3Purity:98.44% - 99.94%Color and Shape:SolidMolecular weight:538.54NP-313
CAS:<p>NP-313 (NSC-4264) is a potent antithrombotic that blocks platelet aggregation via thromboxane A2 synthesis inhibition and targets SOCC-mediated Ca2+ efflux.</p>Formula:C12H8ClNO3Purity:98.97%Color and Shape:SolidMolecular weight:249.65TY-51469
CAS:<p>TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).</p>Formula:C20H15FN2O6S4Purity:99.65%Color and Shape:SolidMolecular weight:526.6CZL55
CAS:<p>CZL55 is a potent caspase-1 inhibitor with an IC50 value of 0.024 μM.CZL55 has low cytotoxicity and can be used in the study of febrile seizures (FS).</p>Formula:C20H22N2O6Purity:98.19%Color and Shape:SolidMolecular weight:386.4(2RS)-FPMPA
CAS:<p>(2RS)-FPMPA(FPMPA) has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).</p>Formula:C9H13FN5O4PPurity:99.9% - >99.99%Color and Shape:SolidMolecular weight:305.2GSK-364735
CAS:<p>GSK-364735 is an HIV-1 IN inhibitor.</p>Formula:C19H18FN3O4Purity:97.73%Color and Shape:SolidMolecular weight:371.36TG2-IN-3h
CAS:<p>TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitor</p>Formula:C21H26N4O4SPurity:99.34% - 99.76%Color and Shape:SolidMolecular weight:430.52UPGL00004
CAS:<p>UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.</p>Formula:C25H26N8O2S2Purity:97.93%Color and Shape:SolidMolecular weight:534.66

