
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(38 products)
- Cysteine Protease(111 products)
- DPP-4(24 products)
- Glutaminase(44 products)
- HIV Protease(505 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(89 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 987 products of "Proteases/Proteasome"
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Rusalatide acetate (497221-38-2 free base)
CAS:Rusalatide acetate (TP508 amide acetate), a regenerated peptide, alleviates radiation-induced gastrointestinal injury by activating stem cells.Formula:C99H151N29O37SPurity:>99.99%Color and Shape:SolidMolecular weight:2371.5Ref: TM-TP1024
2mg40.00€5mg66.00€10mg95.00€25mg156.00€50mg225.00€100mg320.00€200mg434.00€1mL*10mM (DMSO)164.00€TAPI-1 trifluoroacetate (163847-77-6(free base))
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.Formula:C28H38F3N5O7Purity:98.06%Color and Shape:SolidMolecular weight:613.62SB-734117
CAS:SB-734117 inhibits productive replication of several HCMV strains.Formula:C14H16N6OPurity:99.72%Color and Shape:SolidMolecular weight:284.32Ref: TM-T9580
1mg115.00€5mg249.00€10mg369.00€25mg562.00€50mg787.00€100mg1,054.00€200mg1,406.00€1mL*10mM (DMSO)235.00€S 3304
CAS:S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.Formula:C24H20N2O4S2Purity:98.09%Color and Shape:SolidMolecular weight:464.56Ref: TM-T16966
1mg42.00€2mg60.00€5mg105.00€10mg170.00€25mg281.00€50mg395.00€100mg537.00€200mg725.00€1mL*10mM (DMSO)108.00€MDL-28170
CAS:MDL-28170 (Calpain Inhibitor III) is a Cysteine protease.Formula:C22H26N2O4Purity:95.06%Color and Shape:SolidMolecular weight:382.45Ref: TM-T2470
1mg34.00€2mg49.00€5mg71.00€10mg90.00€25mg128.00€50mg167.00€100mg284.00€1mL*10mM (DMSO)75.00€CH 5450
CAS:CH 5450 (Z-Ile-Glu-Pro-Phe-Ome) (Z-Ile-Glu-Pro-Phe-Ome) is a short peptide inhibitor of chymase in the human heartFormula:C34H44N4O9Purity:95.93%Color and Shape:SolidMolecular weight:652.73Ref: TM-TP1012
1mg50.00€5mg111.00€10mg177.00€25mg298.00€50mg424.00€100mg577.00€200mg778.00€1mL*10mM (DMSO)163.00€Grazoprevir
CAS:Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.Formula:C38H50N6O9SPurity:99.36% - >99.99%Color and Shape:SolidMolecular weight:766.9(R)-MG-132
CAS:(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.Formula:C26H41N3O5Purity:99.90%Color and Shape:SolidMolecular weight:475.62Ref: TM-T12628
2mg40.00€5mg60.00€10mg84.00€25mg127.00€50mg187.00€100mg283.00€200mg419.00€1mL*10mM (DMSO)74.00€Simeprevir
CAS:Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.Formula:C38H47N5O7S2Purity:99.45% - 99.92%Color and Shape:SolidMolecular weight:749.94Marimastat
CAS:Marimastat (BB2516) (BB-2516) is a potent, broad spectrum matrix metalloprotease (MMP) inhibitor.
Formula:C15H29N3O5Purity:97.46% - 98.11%Color and Shape:SolidMolecular weight:331.41MUN57694
CAS:MUN57694 is an inhibitor of 26S proteasome.Formula:C23H25N3O4Purity:99%Color and Shape:SolidMolecular weight:407.46Ref: TM-T9090
2mg35.00€5mg52.00€10mg86.00€25mg145.00€50mg210.00€100mg296.00€200mg414.00€1mL*10mM (DMSO)64.00€Dabigatran
CAS:Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.Formula:C25H25N7O3Purity:97.44% - 98.7%Color and Shape:Tan SolidMolecular weight:471.51LY 3000328
CAS:LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.Formula:C25H29FN4O5Purity:97.83% - 99.54%Color and Shape:SolidMolecular weight:484.52Ref: TM-TQ0116
1mg90.00€2mg130.00€5mg198.00€10mg263.00€25mg462.00€50mg672.00€100mg945.00€1mL*10mM (DMSO)207.00€PF-00835231
CAS:PF-00835231 is a CoV-2 cysteine 3C-like protease (3CLpro) inhibitor, with IC50s of 0.27 nM and 4 nM for SARS CoV-2 and SARS CoV-1 3CLpro, respectively.PF-Formula:C24H32N4O6Purity:97.83%Color and Shape:SolidMolecular weight:472.53Ref: TM-T9458
1mg54.00€2mg77.00€5mg114.00€10mg177.00€25mg321.00€50mg482.00€100mg710.00€200mg982.00€1mL*10mM (DMSO)126.00€2-Benzylsuccinic acid
CAS:2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formula:C11H12O4Purity:99.01% - ≥95%Color and Shape:SolidMolecular weight:208.21CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)
CTTHWGFTLC, CYCLIC acetate is an inhibitor for matrix metalloproteinases (MMP)-2 and MMP-9.Formula:C54H75N13O16S2Purity:99.71%Color and Shape:SolidMolecular weight:1226.39Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purity:98.75%Color and Shape:SolidMolecular weight:300.83Ilomastat
CAS:Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.Formula:C20H28N4O4Purity:97.04% - 99.51%Color and Shape:SolidMolecular weight:388.46Ref: TM-T2743
1mg46.00€2mg62.00€5mg89.00€10mg145.00€25mg255.00€50mg429.00€100mg620.00€200mg880.00€1mL*10mM (DMSO)94.00€Elbasvir
CAS:Elbasvir (MK-8742) is an NS5A inhibitor developed for chronic HCV treatment.Formula:C49H55N9O7Purity:98.95% - 99.85%Color and Shape:SolidMolecular weight:882.02Ref: TM-T4544
1mg42.00€2mg52.00€5mg79.00€10mg113.00€25mg200.00€50mg334.00€100mg537.00€1mL*10mM (DMSO)111.00€Ledipasvir (acetone)
CAS:Ledipasvir (acetone) (GS-5885 acetone) is an HCV NS5A polymerase inhibitor, used for the treatment of hepatitis C virus infection.Formula:C52H60F2N8O7Purity:99.72%Color and Shape:SolidMolecular weight:947.08Ref: TM-T4203
1mg34.00€2mg46.00€5mg66.00€10mg88.00€25mg144.00€50mg222.00€100mg340.00€200mg504.00€1mL*10mM (DMSO)92.00€Carbobenzoxyproline
CAS:Carbobenzoxyproline (Carbobenzoxy-S-proline) is a prolidase inhibitor.Formula:C13H15NO4Purity:99.79%Color and Shape:White To Light Yellow Crystal PowderMolecular weight:249.26Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purity:>99.99%Color and Shape:SolidMolecular weight:362.3Teneligliptin
CAS:Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.Formula:C22H30N6OSPurity:99.73%Color and Shape:SolidMolecular weight:426.58KP-457
CAS:KP-457 is a ADAM17 and a TNFα converting enzyme TACE inhibitor that blocks the production of soluble TNF (sTNF).Formula:C21H24N2O7S2Purity:98.33%Color and Shape:SolidMolecular weight:480.56Ref: TM-T77778
1mg96.00€5mg205.00€10mg334.00€25mg620.00€50mg982.00€100mg1,333.00€1mL*10mM (DMSO)219.00€(R)-Trolox
CAS:(R)-Trolox is a selective tyrosinase inhibitor used in food, cosmetics, and pharmaceutical products.Formula:C14H18O4Purity:99.88%Color and Shape:SolidMolecular weight:250.29(1S,2R)-Alicapistat
CAS:(1S,2R)-Alicapistat inhibits calpains 1 and 2, shows promise for Alzheimer's, and has an IC50 of 395 nM.Formula:C25H27N3O4Purity:99.60%Color and Shape:SoildMolecular weight:433.5Ref: TM-T60150
1mg64.00€5mg142.00€10mg197.00€25mg299.00€50mg400.00€100mg537.00€1mL*10mM (DMSO)167.00€Ledipasvir
CAS:Ledipasvir (GS-5885) is a Hepatitis C Virus NS5A Inhibitor.Formula:C49H54F2N8O6Purity:99.96%Color and Shape:SolidMolecular weight:889Ref: TM-T6200
1mg35.00€2mg50.00€5mg74.00€10mg94.00€25mg150.00€50mg244.00€100mg421.00€500mg964.00€1mL*10mM (DMSO)94.00€Danoprevir
CAS:Danoprevir (RG7227) is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).Formula:C35H46FN5O9SPurity:98% - 99.80%Color and Shape:SolidMolecular weight:731.83PSI
CAS:PSI is a proteasome inhibitor.Formula:C32H50N4O8Purity:97% - 98.33%Color and Shape:SolidMolecular weight:618.76Nelfinavir
CAS:Nelfinavir (AG1341), with Ki=2 nM, is an HIV treatment and broad-spectrum anticancer drug.Formula:C32H45N3O4SPurity:98.16% - 99.5%Color and Shape:White To Off-White Crystalline PowderMolecular weight:567.78Lanadelumab
CAS:Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.Purity:95% - 97.4% (SDS-PAGE); 99.2% (SEC-HPLC)Color and Shape:LiquidMolecular weight:145.70 kDaAnti-Matriptase Antibody
Anti-Matriptase Antibody is a human-derived antibody expressed in CHO cells, targeting Matriptase. It features a huIgG1 heavy chain and huκ light chain, with a predicted molecular weight (MW) of 150 kDa. The isotype control for Anti-Matriptase Antibody can be found in HumanIgG1kappa, Isotype Control.Color and Shape:Odour LiquidAnti-Human/Mouse denatured collagen type-I Antibody
Anti-Human/Mouse denatured collagen type-I Antibody (XL313) is an IgG1, κ inhibitor derived from mice, targeting denatured collagen type-I in both human and mouse.Color and Shape:Odour LiquidKZR-504
CAS:KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 nM, 4.274 μM for LMP2 and LMP7, respectively).Formula:C21H23N3O6Color and Shape:SolidMolecular weight:413.42Triton X-45(n=4)
CAS:Triton X-45: nonionic, low HLB surfactant, dispersible in water, high Krafft point, relevant for HCV research.Formula:C22H38O5Color and Shape:SolidMolecular weight:382.53MG-132
CAS:Formula:C26H41N3O5Purity:>95.0%(qNMR)Color and Shape:White to Light yellow powder to crystalMolecular weight:475.63HCV-IN-30
CAS:HCV-IN-30 is an HCV NS5A replication complex inhibitor (IC50s: 901 and 102 nM for genotypes 1a and 1b replicons).Formula:C36H44N6O4Purity:99.6%Color and Shape:SolidMolecular weight:624.77S 2160
CAS:S 2160 is a synthetic chromogenic substrate for thrombin.Formula:C33H40N8O6Color and Shape:SolidMolecular weight:644.72Cathepsin Inhibitor 1
CAS:Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.
Formula:C20H24ClN5O2Purity:99.78%Color and Shape:SolidMolecular weight:401.89Carboxypeptidase G2 (CPG2) Inhibitor
CAS:Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.Formula:C13H15NO6SPurity:99.96%Color and Shape:SolidMolecular weight:313.33Batimastat sodium salt
CAS:Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).Formula:C23H31N3NaO4S2Purity:98%Color and Shape:SolidMolecular weight:500.63Diprotin B
CAS:Diprotin B is a dipeptidyl peptidase IV inhibitor.Formula:C16H29N3O4Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:327.42Tyrosinase-IN-4
CAS:Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.Formula:C15H9ClO3Color and Shape:SolidMolecular weight:272.68Tanomastat
CAS:Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.Formula:C23H19ClO3SPurity:98%Color and Shape:SolidMolecular weight:410.91Gemigliptin Tartrate(911637-19-9 free base)
CAS:Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).Formula:C22H25F8N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:639.45BR351
CAS:BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).Formula:C20H25FN2O5SPurity:98%Color and Shape:SolidMolecular weight:424.49Adafosbuvir PM
CAS:Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.Formula:C10H13FN2O6Purity:98.39%Color and Shape:SolidMolecular weight:276.22OM-189
CAS:OM-189 is a selective inhibitor of synthetic thrombin.Formula:C24H36N6O3SPurity:98%Color and Shape:SolidMolecular weight:488.65Tyrosinase-IN-1
CAS:Tyrosinase-IN-1: potent inhibitor for skin-whitening & food preservation with uses in cosmetics & medicine.Formula:C10H9N3O2S2Color and Shape:SolidMolecular weight:267.33Gü1303
CAS:Gü1303 is a highly potent and reversible inhibitor of Cathepsin K (CatK), with a Ki value of 0.91 nM for mature CatK (mCatK).Formula:C20H22N4O3Color and Shape:SolidMolecular weight:366.41


