
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(36 products)
- Cysteine Protease(111 products)
- DPP-4(24 products)
- Glutaminase(44 products)
- HIV Protease(501 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(89 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 993 products of "Proteases/Proteasome"
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Nostosin G
Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).Formula:C25H33N5O6Color and Shape:SolidMolecular weight:499.56Sofosbuvir impurity J
CAS:Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C22H30FN4O8PPurity:98%Color and Shape:SolidMolecular weight:528.47HIV-1 TAT (48-60) Acetate
Lilotomab (HH1) is a murine anti-CD37 antibody that can be used to synthesize anti-CD37 antibody-radionuclide couplings.Formula:C72H135N35O18Purity:99.93%Color and Shape:SoildMolecular weight:1779.07Dutogliptin tartrate
CAS:Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.Formula:C14H26BN3O9Purity:98%Color and Shape:SolidMolecular weight:391.18L-Methionine-DL-sulfoximine
CAS:MSO blocks glutamine synthetase, impacts astroglia, and is used in convulsant research.Formula:C5H12N2O3SPurity:99.56% - ≥98%Color and Shape:White Crystalline PowderMolecular weight:180.23Arabinosylhypoxanthine
CAS:Arabinosylhypoxanthine inhibits Ns5b polymerase in hepatitis C virus and can be used in biochemical experiments and organic synthesis.Formula:C10H12N4O5Purity:99.71%Color and Shape:SolidMolecular weight:268.23Diprotin A TFA
CAS:Diprotin A (TFA) is an inhibitor of dipeptidyl peptidase IV (DPP-IV).Formula:C19H32F3N3O6Color and Shape:SolidMolecular weight:455.47Urokinase
CAS:Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.Color and Shape:SolidUbenimex
CAS:Formula:C16H24N2O4Purity:>98.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:308.382'-β-C-Ethynyladenosine
CAS:2'-β-C-Ethynyladenosine is a nucleoside analog that potently inhibits hepatitis C virus (HCV) replication by targeting the viral NS5B polymerase.Formula:C12H13N5O4Color and Shape:SolidMolecular weight:291.26Retagliptin
CAS:Retagliptin is a DPP-4 inhibitor potentially used to treat Type 2 diabetes.Formula:C19H18F6N4O3Color and Shape:SolidMolecular weight:464.36Anguizole
CAS:Anguizole, a small molecule, effectively inhibits Hepatitis C Virus (HCV) replication by modifying the subcellular distribution of NS4B.Formula:C17H11ClF2N4O2SColor and Shape:SolidMolecular weight:408.81ML-345
CAS:ML-345, Selective IDE inhibitor (IC50=188 nM) targeting Cys819, for type 2 diabetes and Alzheimer's research.Formula:C21H22FN3O5S2Purity:99.21%Color and Shape:SolidMolecular weight:479.55Ref: TM-T35802
1mg39.00€5mg84.00€10mg120.00€25mg197.00€50mgTo inquire100mg434.00€1mL*10mM (DMSO)To inquireSaxagliptin hydrochloride
CAS:Saxagliptin: oral DPP-4 inhibitor, enhances incretins, manages type 2 diabetes by reducing glucose levels.Formula:C18H26ClN3O2Color and Shape:SolidMolecular weight:351.87Sivelestat Sodium Tetrahydrate
CAS:Formula:C20H21N2NaO7S·4H2OPurity:>95.0%(T)(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:528.50Tanaproget
CAS:Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.Formula:C16H15N3OSPurity:98%Color and Shape:SolidMolecular weight:297.38Alogliptin (13CD3)
CAS:Alogliptin (SYR-322) 13CD3 is the deuterium-labeled Alogliptin. Alogliptin is a selective inhibitor of DPP-4.Formula:C18H21N5O2Purity:98%Color and Shape:SolidMolecular weight:343.4(-)-Gallocatechin Gallate
CAS:Formula:C22H18O11Purity:>95.0%(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:458.38H-Pro-Lys-OH TFA
H-Pro-Lys-OH TFA is a dipeptide composed of proline and lysine, serving as a substrate for imino dipeptidase (prolinase). Additionally, it can be utilized in peptide synthesis.Formula:C13H22F3N3O5Color and Shape:SolidMolecular weight:357.33CTS-1027
CAS:CTS-1027 is a small molecule inhibitor of MMPs (IC50s: 0.3 nM, 0.5 nM for MMP2, MMP13). It has > 1,000 fold selectivity over MMP1.Formula:C19H20ClNO6SColor and Shape:SolidMolecular weight:425.88Pepstatin A
CAS:Formula:C34H63N5O9Purity:>90.0%(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:685.90LN5P45
LN5P45, an OTUB2 inhibitor (IC50: 2.3 μM), promotes monoubiquitination of OTUB2 at lysine 31 and is utilized in the study of tumor progression and metastasis [1Formula:C13H15ClN2O2Color and Shape:SolidMolecular weight:266.726-Chloro-7-deazapurine-2F-β-D-arabinofuranose
CAS:6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside.Formula:C11H11ClFN3O3Color and Shape:SolidMolecular weight:287.67Ref: TM-TNU0055
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireE-64d [for Biochemical Research]
CAS:Formula:C17H30N2O5Purity:>95.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:342.44Glutaminase-IN-3
CAS:Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.Formula:C19H19F3N6O2SPurity:98.51%Color and Shape:SolidMolecular weight:452.45PSI-6206 13C,d3
CAS:PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.
Formula:C10H13FN2O5Purity:98%Color and Shape:SolidMolecular weight:264.23MMP-8 Inhibitor I
CAS:MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.Formula:C17H18N2O5SColor and Shape:SolidMolecular weight:362.4Sitagliptin fenilalanil
CAS:Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.Formula:C25H24F6N6O2Color and Shape:SolidMolecular weight:554.49Ubenimex Hydrochloride [for Biochemical Research]
CAS:Formula:C16H24N2O4·HClPurity:>97.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:344.84PKSI-527
CAS:PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.Formula:C25H32ClN3O4Color and Shape:SolidMolecular weight:473.99Tomeglovir
CAS:Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).Formula:C23H27N3O4SPurity:98%Color and Shape:SolidMolecular weight:441.54Tilpisertib
CAS:Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).Formula:C33H33ClN8OColor and Shape:SolidMolecular weight:593.13Dabigatran ethyl ester
CAS:Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.Formula:C27H29N7O3Purity:99.98%Color and Shape:SolidMolecular weight:499.56H-Arg-4MβNA
CAS:H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.Formula:C17H23N5O2Purity:99.98%Color and Shape:SolidMolecular weight:329.4(Arg)9
CAS:(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).Formula:C54H110N36O10Color and Shape:SolidMolecular weight:1423.69BAY-677
CAS:BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.Formula:C20H15F3N4O2Color and Shape:SolidMolecular weight:400.35PD-166793
CAS:PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.Formula:C17H18BrNO4SPurity:99.86%Color and Shape:SolidMolecular weight:412.3Ref: TM-T20563
5mg42.00€10mg60.00€25mg112.00€50mg175.00€100mg261.00€200mg368.00€1mL*10mM (DMSO)46.00€DMP 777
CAS:DMP 777 is an orally active inhibitor of human leukocyte elastase.Formula:C31H40N4O6Color and Shape:SolidMolecular weight:564.67Ilomastat
CAS:Formula:C20H28N4O4Purity:>95.0%(HPLC)(qNMR)Color and Shape:White to Light yellow powder to crystalMolecular weight:388.475-Amino-8-hydroxyquinoline
CAS:5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.Formula:C9H8N2OPurity:99.69%Color and Shape:SolidMolecular weight:160.17Teneligliptin D8
CAS:Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.Formula:C22H30N6OSPurity:98%Color and Shape:SolidMolecular weight:434.63Thrombin inhibitor 5
CAS:Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.Formula:C11H9FN4O3Purity:99.58%Color and Shape:SolidMolecular weight:264.21Ref: TM-T9845
2mg35.00€5mg56.00€10mg86.00€25mg154.00€50mg224.00€100mg320.00€200mg434.00€1mL*10mM (DMSO)55.00€Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]
CAS:Formula:C10H13N2Na3O8·xH2OPurity:>98.0%(T)Color and Shape:White to Almost white powder to crystalMolecular weight:358.19 (as Anhydrous)UAMC00039 dihydrochloride
CAS:UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM.Formula:C16H26Cl3N3OPurity:>99.99%Color and Shape:SolidMolecular weight:382.76GW280264X
CAS:GW280264X (Carbamic acid) is an inhibitor of ADAM17 .Formula:C28H41N5O6SPurity:99.51%Color and Shape:SolidMolecular weight:575.72Ref: TM-T8961
1mg156.00€5mg319.00€10mg477.00€25mg773.00€50mg1,063.00€100mg1,431.00€1mL*10mM (DMSO)404.00€Ledipasvir hydrochloride
CAS:Ledipasvir hydrochloride, a hepatitis C NS5A inhibitor, has EC50 of 34 pM (1a) and 4 pM (1b), also inhibits SARS-CoV 3CL pro (IC50 1.62 µM).Formula:C49H55ClF2N8O6Color and Shape:SolidMolecular weight:925.46Alloxan monohydrate
CAS:Alloxan Monohydrate is a glucose analog used to induce diabetes by destroying beta-cells.
Formula:C4H4N2O5Purity:99.01% - 99.42%Color and Shape:Off-White To Beige-Yellowish Crystalline PowderMolecular weight:160.09Clemizole
CAS:Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formula:C19H20ClN3Purity:98% - 99.65%Color and Shape:SolidMolecular weight:325.84Ref: TM-T1822
1mg44.00€5mg87.00€10mg106.00€25mg160.00€50mg270.00€100mg487.00€500mg1,026.00€1mL*10mM (DMSO)87.00€LY 3000328
CAS:LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.Formula:C25H29FN4O5Purity:97.83% - 99.54%Color and Shape:SolidMolecular weight:484.52Ref: TM-TQ0116
1mg90.00€2mg130.00€5mg198.00€10mg263.00€25mg462.00€50mg672.00€100mg945.00€1mL*10mM (DMSO)207.00€Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purity:98.75%Color and Shape:SolidMolecular weight:300.83


