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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1093 products of "Proteases/Proteasome"

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  • Fotagliptin benzoate

    CAS:
    Fotagliptin benzoate, a DPP-4 inhibitor (IC50=2.27 nM), is safe in rats/dogs, useful for Type 2 diabetes research.
    Formula:C24H25FN6O3
    Color and Shape:Solid
    Molecular weight:464.49

    Ref: TM-T73875

    5mg
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    50mg
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  • Rivulariapeptolides 1185


    Rivulariapeptolides 1185 inhibits serine proteases; IC50: chymotrypsin 13.17 nM, elastase 23.59 nM, proteinase K 55.26 nM.
    Formula:C61H87N9O15
    Color and Shape:Solid
    Molecular weight:1186.39

    Ref: TM-T75649

    5mg
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    50mg
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  • Recombinant Proteinase K


    Recombinant Proteinase K: serine protease, cleaves carboxy-terminus peptides, digests proteins, purifies nucleic acids.
    Color and Shape:Solid

    Ref: TM-T76202

    5mg
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    50mg
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  • Tilpisertib fosmecarbil TFA

    CAS:
    Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.
    Formula:C37H37ClF3N8O9P
    Color and Shape:Solid
    Molecular weight:861.16

    Ref: TM-T88817

    10mg
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    50mg
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  • STK33-IN-1

    CAS:
    STK33-IN-1 (compound 1) is a STK33 inhibitor, with an IC 50 of 7 nM.
    Formula:C24H27N7O2
    Color and Shape:Solid
    Molecular weight:445.527

    Ref: TM-T38835

    5mg
    922.00€
  • Relacatib

    CAS:
    Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.
    Formula:C27H32N4O6S
    Color and Shape:Solid
    Molecular weight:540.64

    Ref: TM-T40463

    5mg
    1,872.00€
  • HIV-1 Rev (34-50)

    CAS:
    HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) is a 17 amino acid peptide with anti-HIV-1 activity.
    Formula:C97H173N51O24
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:2437.74

    Ref: TM-TP1149

    1mg
    131.00€
    5mg
    198.00€
    10mg
    288.00€
    25mg
    452.00€
    50mg
    607.00€
    100mg
    785.00€
    200mg
    1,045.00€
  • Ichorcumab

    CAS:
    <p>Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.</p>
    Color and Shape:Liquid

    Ref: TM-T9901A-779

    1mg
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    5mg
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  • HCV-IN-7 hydrochloride

    CAS:
    HCV-IN-7 hydrochloride: Oral, potent HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.
    Formula:C40H50Cl2N8O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:841.85

    Ref: TM-T11548L

    25mg
    1,444.00€
  • RXP470

    CAS:
    RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).
    Formula:C35H35BrClN4O10P
    Color and Shape:Solid
    Molecular weight:818

    Ref: TM-T28633

    5mg
    4,884.00€
  • SFTI-1

    CAS:
    SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.
    Formula:C67H104N18O18S2
    Color and Shape:Solid
    Molecular weight:1513.78

    Ref: TM-TP2622

    10mg
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    50mg
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  • TP0628103 TFA

    CAS:
    TP0628103 (Compound 18) TFA is a selective MMP-7 inhibitor with an IC50 value of 0.17 nM, playing a significant role in cancer and fibrosis.
    Formula:C53H68ClF6N11O13S
    Color and Shape:Solid
    Molecular weight:1248.68

    Ref: TM-T210971

    10mg
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    50mg
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  • Paritaprevir dihydrate

    CAS:
    Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.
    Formula:C40H47N7O9S
    Color and Shape:Solid
    Molecular weight:801.91

    Ref: TM-T73898

    5mg
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    50mg
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  • PSI-353661

    CAS:
    PSI-353661 (GS-558093), inhibits HCV's NS5B polymerase; EC90: 8nM (wild-type), 11nM (S282T); active in human hepatocytes.
    Formula:C24H32FN6O8P
    Color and Shape:Solid
    Molecular weight:582.52

    Ref: TM-T74301

    5mg
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    50mg
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  • Hirudin (54-65) (TFA)


    Hirudin (54-65) TFA, a segment of the 65-amino-acid protein Hirudin, exhibits anticoagulant properties [1].
    Color and Shape:Odour Solid

    Ref: TM-T82197

    5mg
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    50mg
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  • Ellipyrone B


    Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50
    Formula:C25H38O7
    Color and Shape:Solid
    Molecular weight:450.57

    Ref: TM-T75493

    5mg
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    50mg
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  • DPP-4-IN-14


    <p>DPP-4-IN-14 (compound 30) is an inhibitor of DPP-4, with an IC50 value of 12.82 nM.</p>
    Formula:C33H27N7O3
    Color and Shape:Solid
    Molecular weight:569.613

    Ref: TM-T204855

    10mg
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    50mg
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  • Cepeginterferon alfa-2b

    CAS:
    Cepeginterferon alfa-2b: pegylated interferon with 20 kDa PEG for HCV, PV, ET research.
    Color and Shape:Liquid

    Ref: TM-T76943

    5mg
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    50mg
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  • Mca-(endo-1a-Dap(Dnp))-TNF-α (-5 to +6) amide (human)

    CAS:
    Mca-(endo-1a-Dap(Dnp))-TNF-Alpha (-5 to +6) amide (human) is a peptide utilized as a fluorescence resonance energy transfer (FRET) based substrate for
    Formula:C69H103N23O24
    Color and Shape:Solid
    Molecular weight:1638.7

    Ref: TM-T81838

    5mg
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    50mg
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  • NIM811

    CAS:
    NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.
    Formula:C62H111N11O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1202.635

    Ref: TM-T12226

    5mg
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