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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1014 products of "Proteases/Proteasome"

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  • Thrombin inhibitor 5

    CAS:
    Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.
    Formula:C11H9FN4O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:264.21

    Ref: TM-T9845

    2mg
    35.00€
    5mg
    56.00€
    10mg
    86.00€
    25mg
    154.00€
    50mg
    224.00€
    100mg
    320.00€
    200mg
    434.00€
    1mL*10mM (DMSO)
    55.00€
  • Glutaminase-IN-3

    CAS:
    Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
    Formula:C19H19F3N6O2S
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:452.45

    Ref: TM-T37385

    5mg
    59.00€
    10mg
    84.00€
    25mg
    119.00€
    50mg
    170.00€
    100mg
    251.00€
    1mL*10mM (DMSO)
    73.00€
  • Ubenimex Hydrochloride [for Biochemical Research]

    CAS:
    Formula:C16H24N2O4·HCl
    Purity:>97.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:344.84

    Ref: 3B-B4000

    25mg
    196.00€
  • MMP-8 Inhibitor I

    CAS:
    MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.
    Formula:C17H18N2O5S
    Color and Shape:Solid
    Molecular weight:362.4

    Ref: TM-T69666

    1mg
    642.00€
  • Sitagliptin fenilalanil

    CAS:
    Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.
    Formula:C25H24F6N6O2
    Color and Shape:Solid
    Molecular weight:554.49

    Ref: TM-T63915

    2mg
    60.00€
  • PKSI-527

    CAS:
    PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.
    Formula:C25H32ClN3O4
    Color and Shape:Solid
    Molecular weight:473.99

    Ref: TM-T35579

    2mg
    81.00€
  • Tilpisertib

    CAS:
    Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).
    Formula:C33H33ClN8O
    Color and Shape:Solid
    Molecular weight:593.13

    Ref: TM-T39466

    5mg
    873.00€
  • Tomeglovir

    CAS:
    Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).
    Formula:C23H27N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.54

    Ref: TM-TQ0030

    2mg
    54.00€
  • BAY-677

    CAS:
    BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.
    Formula:C20H15F3N4O2
    Color and Shape:Solid
    Molecular weight:400.35

    Ref: TM-T10473L

    2mg
    85.00€
  • PD-166793

    CAS:
    PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.
    Formula:C17H18BrNO4S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:412.3

    Ref: TM-T20563

    5mg
    42.00€
    10mg
    60.00€
    25mg
    112.00€
    50mg
    175.00€
    100mg
    261.00€
    200mg
    368.00€
    1mL*10mM (DMSO)
    46.00€
  • H-Arg-4MβNA

    CAS:
    H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.
    Formula:C17H23N5O2
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:329.4

    Ref: TM-T19347

    5mg
    33.00€
  • (Arg)9

    CAS:
    (Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).
    Formula:C54H110N36O10
    Color and Shape:Solid
    Molecular weight:1423.69

    Ref: TM-T13976

    100mg
    To inquire
    500mg
    To inquire
  • Dabigatran ethyl ester

    CAS:
    Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.
    Formula:C27H29N7O3
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:499.56

    Ref: TM-T15046

    2mg
    38.00€
    5mg
    51.00€
    10mg
    94.00€
    25mg
    155.00€
    50mg
    261.00€
    100mg
    410.00€
  • DMP 777

    CAS:
    DMP 777 is an orally active inhibitor of human leukocyte elastase.
    Formula:C31H40N4O6
    Color and Shape:Solid
    Molecular weight:564.67

    Ref: TM-T15144

    2mg
    88.00€
    5mg
    152.00€
    1mL*10mM (DMSO)
    205.00€
  • 5-Amino-8-hydroxyquinoline

    CAS:
    5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.
    Formula:C9H8N2O
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:160.17

    Ref: TM-T60234

    25mg
    35.00€
    50mg
    47.00€
    100mg
    59.00€
    500mg
    119.00€
    1mL*10mM (DMSO)
    47.00€
  • ML-345

    CAS:
    ML-345, Selective IDE inhibitor (IC50=188 nM) targeting Cys819, for type 2 diabetes and Alzheimer's research.
    Formula:C21H22FN3O5S2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:479.55

    Ref: TM-T35802

    1mg
    To inquire
    2mg
    60.00€
    5mg
    To inquire
    10mg
    To inquire
    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
    1mL*10mM (DMSO)
    To inquire
  • Teneligliptin D8

    CAS:
    Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.
    Formula:C22H30N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.63

    Ref: TM-T13121

    1mg
    595.00€
    5mg
    1,431.00€
    10mg
    1,963.00€
    25mg
    2,907.00€
  • Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]

    CAS:
    Formula:C10H13N2Na3O8·xH2O
    Purity:>98.0%(T)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:358.19 (as Anhydrous)

    Ref: 3B-T2599

    5g
    22.00€
    25g
    41.00€
  • Urokinase

    CAS:

    Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.

    Color and Shape:Solid

    Ref: TM-T73701

    1mg
    170.00€
    5mg
    425.00€
    10mg
    596.00€
    25mg
    951.00€
  • Ubenimex

    CAS:
    Formula:C16H24N2O4
    Purity:>98.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:308.38

    Ref: 3B-U0111

    1g
    416.00€
    250mg
    136.00€