
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(36 products)
- Cysteine Protease(110 products)
- DPP-4(24 products)
- Glutaminase(44 products)
- HIV Protease(498 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(91 products)
- Serine Protease(51 products)
- p97(15 products)
Show 3 more subcategories
Found 1014 products of "Proteases/Proteasome"
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Thrombin inhibitor 5
CAS:Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.Formula:C11H9FN4O3Purity:99.58%Color and Shape:SolidMolecular weight:264.21Ref: TM-T9845
2mg35.00€5mg56.00€10mg86.00€25mg154.00€50mg224.00€100mg320.00€200mg434.00€1mL*10mM (DMSO)55.00€Glutaminase-IN-3
CAS:Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.Formula:C19H19F3N6O2SPurity:98.51%Color and Shape:SolidMolecular weight:452.45Ubenimex Hydrochloride [for Biochemical Research]
CAS:Formula:C16H24N2O4·HClPurity:>97.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:344.84MMP-8 Inhibitor I
CAS:MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.Formula:C17H18N2O5SColor and Shape:SolidMolecular weight:362.4Sitagliptin fenilalanil
CAS:Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.Formula:C25H24F6N6O2Color and Shape:SolidMolecular weight:554.49PKSI-527
CAS:PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.Formula:C25H32ClN3O4Color and Shape:SolidMolecular weight:473.99Tilpisertib
CAS:Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).Formula:C33H33ClN8OColor and Shape:SolidMolecular weight:593.13Tomeglovir
CAS:Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).Formula:C23H27N3O4SPurity:98%Color and Shape:SolidMolecular weight:441.54BAY-677
CAS:BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.Formula:C20H15F3N4O2Color and Shape:SolidMolecular weight:400.35PD-166793
CAS:PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.Formula:C17H18BrNO4SPurity:99.86%Color and Shape:SolidMolecular weight:412.3Ref: TM-T20563
5mg42.00€10mg60.00€25mg112.00€50mg175.00€100mg261.00€200mg368.00€1mL*10mM (DMSO)46.00€H-Arg-4MβNA
CAS:H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.Formula:C17H23N5O2Purity:99.98%Color and Shape:SolidMolecular weight:329.4(Arg)9
CAS:(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).Formula:C54H110N36O10Color and Shape:SolidMolecular weight:1423.69Dabigatran ethyl ester
CAS:Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.Formula:C27H29N7O3Purity:99.98%Color and Shape:SolidMolecular weight:499.56DMP 777
CAS:DMP 777 is an orally active inhibitor of human leukocyte elastase.Formula:C31H40N4O6Color and Shape:SolidMolecular weight:564.675-Amino-8-hydroxyquinoline
CAS:5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.Formula:C9H8N2OPurity:99.69%Color and Shape:SolidMolecular weight:160.17ML-345
CAS:ML-345, Selective IDE inhibitor (IC50=188 nM) targeting Cys819, for type 2 diabetes and Alzheimer's research.Formula:C21H22FN3O5S2Purity:99.21%Color and Shape:SolidMolecular weight:479.55Ref: TM-T35802
1mgTo inquire2mg60.00€5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire1mL*10mM (DMSO)To inquireTeneligliptin D8
CAS:Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.Formula:C22H30N6OSPurity:98%Color and Shape:SolidMolecular weight:434.63Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]
CAS:Formula:C10H13N2Na3O8·xH2OPurity:>98.0%(T)Color and Shape:White to Almost white powder to crystalMolecular weight:358.19 (as Anhydrous)Urokinase
CAS:Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.
Color and Shape:SolidUbenimex
CAS:Formula:C16H24N2O4Purity:>98.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:308.38


