PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
Read more
Umbralisib
CAS:1532533-67-7
Umbralisib (TGR 1202) is a PI3Kδ inhibitor.
Formula:
C31H24F3N5O3
Purity:
99.56% - 99.56%
Color and Shape:
White Solid
Molecular weight:
571.55
Ref: TM-T4976
| 1mg | 48.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 449.00 € | ||
| 100mg | 658.00 € | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Friday 16 May 2025
AZD-8835
CAS:1620576-64-8
AZD-8835 is a mixed inhibitor of PI3Kα/δ (IC50: 6.2/5.7 nM), also with selectivity against PI3Kβ/γ …
Formula:
C22H31N9O3
Purity:
98.22% - 98.49%
Color and Shape:
Solid
Molecular weight:
469.54
Ref: TM-T6774
| 5mg | 50.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 170.00 € | ||
| 100mg | 301.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 16 May 2025
AS-604850
CAS:648449-76-7
AS-604850: ATP-competitive PI3Kγ inhibitor, IC50 250 nM, 18x >PI3Kα, 80x > PI3Kδ/β.
Formula:
C11H5F2NO4S
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
285.22
Ref: TM-T6394
| 10mg | 50.00 € | ||
| 25mg | 80.00 € | ||
| 50mg | 117.00 € | ||
| 100mg | 210.00 € | ||
| 200mg | 313.00 € | ||
| 1mL*10mM (DMSO) | 38.00 € |
Estimated delivery in United States, on Friday 16 May 2025
PIK-93
CAS:593960-11-3
PIK-93 is the first potent, synthetic PI4K inhibitor with IC50 of 19 nM; inhibits PI3Kα …
Formula:
C14H16ClN3O4S2
Purity:
97.72%
Color and Shape:
Solid
Molecular weight:
389.88
Ref: TM-T2616
| 1mg | 44.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 522.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 16 May 2025
CH5132799
CAS:1007207-67-1
CH5132799 has been used in trials studying the treatment of Solid Tumors.
Formula:
C15H19N7O3S
Purity:
98.81% - 99.87%
Color and Shape:
Solid
Molecular weight:
377.42
Ref: TM-T2619
| 1mg | 64.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 227.00 € | ||
| 25mg | 420.00 € | ||
| 50mg | 622.00 € | ||
| 100mg | 885.00 € | ||
| 500mg | 1,786.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Seletalisib
CAS:1362850-20-1
Seletalisib (UCB5857) (UCB5857) is a potent and specific PI3Kδ inhibitor (IC50: 12 nM).
Formula:
C23H14ClF3N6O
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
482.85
Ref: TM-TQ0044
| 1mg | 57.00 € | ||
| 2mg | 81.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 660.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Friday 16 May 2025
α-Linolenic acid
CAS:463-40-1
α-Linolenic Acid (ALA) is an essential fatty acid. α-Linolenic acid improves memory, inhibits thrombosis, and …
Formula:
C18H30O2
Purity:
98.19% - 99.81%
Color and Shape:
Physical Description Clear Colorless Liquid (Ntp 1992)
Molecular weight:
278.43
Ref: TM-T3P2904
| 50mg | To inquire | ||
| 100mg | 48.00 € | ||
| 500mg | 77.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 16 May 2025
GSK2636771
CAS:1372540-25-4
GSK2636771, an effective, specific, orally bioavailable, PI3Kβ inhibitor, has been used in cancer, lymphoma, solid …
Formula:
C22H22F3N3O3
Purity:
98.58% - ≥95%
Color and Shape:
Solid
Molecular weight:
433.42
Ref: TM-T2073
| 1mg | 43.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Vps34-IN-1
CAS:1383716-33-3
Vps34-IN-1: potent, selective Vps34 inhibitor, 25 nM IC50, spares class I/II PI3Ks.
Formula:
C21H24ClN7O
Purity:
97.04%
Color and Shape:
Solid
Molecular weight:
425.91
Ref: TM-T7015
| 1mg | 46.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 219.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 505.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Friday 16 May 2025
SAR405
CAS:1523406-39-4
SAR-405 inhibits PIK3C3/Vps34 (IC50: 1.2 nM, Kd: 1.5 nM), blocks autophagy, and enhances MTOR inhibitor …
Formula:
C19H21ClF3N5O2
Purity:
99.42% - 99.79%
Color and Shape:
Solid
Molecular weight:
443.85
Ref: TM-T12831L
| 1mg | 149.00 € | ||
| 2mg | 217.00 € | ||
| 5mg | 368.00 € | ||
| 10mg | 580.00 € | ||
| 25mg | 882.00 € | ||
| 50mg | 1,596.00 € | ||
| 1mL*10mM (DMSO) | 444.00 € |
Estimated delivery in United States, on Friday 16 May 2025
PIK-90
CAS:677338-12-4
PIK-90, a DNA-PK and PI3K inhibitor, suppresses p110α( IC50=11 nM), p110γ(IC50=18 nM) and DNA-PK(IC50=13 nM) …
Formula:
C18H17N5O3
Purity:
98.25% - ≥95%
Color and Shape:
Solid
Molecular weight:
351.36
Ref: TM-T2461
| 5mg | 47.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 144.00 € |
Estimated delivery in United States, on Friday 16 May 2025
A66
CAS:1166227-08-2
A66 is a specific and effective p110α inhibitor(IC50=32 nM).
Formula:
C17H23N5O2S2
Purity:
99.51% - ≥95%
Color and Shape:
Solid
Molecular weight:
393.53
Ref: TM-T2418
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 246.00 € | ||
| 100mg | 364.00 € | ||
| 200mg | 512.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Linperlisib
CAS:1702816-75-8
Linperlisib (PI3Kδ-IN-2) is a potent and selective inhibitor of PI3Kδ
Formula:
C28H37FN6O5S
Purity:
99.01%
Color and Shape:
Solid
Molecular weight:
588.69
Ref: TM-T6330
| 1mg | 35.00 € | ||
| 2mg | 48.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 311.00 € | ||
| 100mg | 487.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Friday 16 May 2025
VPS34 inhibitor 1 (Compound 19, PIK-III analogue)
CAS:1383716-46-8
VPS34 inhibitor 1 (Compound 19, PIK-III analogue) (PIK-III analogue) is a potent and selective inhibitor …
Formula:
C21H25N7O
Purity:
98.60%
Color and Shape:
Solid
Molecular weight:
391.47
Ref: TM-T7944
| 1mg | 66.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 227.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 567.00 € | ||
| 100mg | 753.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Friday 16 May 2025
CAY10505
CAS:1218777-13-9
CAY10505, a form of dehydroxyl of AS-252424, is a PI3Kγ inhibitor (IC50: 33 nM).
Formula:
C14H8FNO3S
Purity:
99.74% - 99.79%
Color and Shape:
Solid
Molecular weight:
289.28
Ref: TM-T6433
| 10mg | 35.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 153.00 € | ||
| 200mg | 216.00 € | ||
| 500mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 40.00 € |
Estimated delivery in United States, on Friday 16 May 2025
GDC-0326
CAS:1282514-88-8
GDC-0326 is a potent and selective inhibitor of α-Isoform of Phosphoinositide 3-Kinase (PI3Kalpha inhibitor).
Formula:
C19H22N6O3
Purity:
100% - 99.35%
Color and Shape:
Solid
Molecular weight:
382.42
Ref: TM-T3985
| 1mg | 35.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 592.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Friday 16 May 2025
AZD8186
CAS:1627494-13-6
AZD8186 is an effective and specific PI3Kβ/δ inhibitor (IC50: 4/12 nM).
Formula:
C24H25F2N3O4
Purity:
99.89% - 99.91%
Color and Shape:
Solid
Molecular weight:
457.47
Ref: TM-T6773
| 2mg | 46.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 505.00 € | ||
| 500mg | 1,121.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Selective PI3Kδ Inhibitor 1
CAS:2088525-31-7
Selective PI3Kδ Inhibitor 1 is a PI3Kδ Inhibitor( IC50 = 0.9 nM).
Formula:
C23H20FN7O
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
429.45
Ref: TM-T5831
| 1mg | 58.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 373.00 € | ||
| 50mg | 509.00 € | ||
| 100mg | 695.00 € | ||
| 200mg | 937.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Pilaralisib analogue
CAS:956958-53-5
Pilaralisib analogue (XL147 analogue) is a selective and reversible class I PI3K inhibitor for PI3Kα/δ/γ.
Formula:
C21H16N6O2S2
Purity:
99.30% - 99.72%
Color and Shape:
Solid
Molecular weight:
448.52
Ref: TM-T2377
| 2mg | 38.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 139.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | 374.00 € | ||
| 200mg | 485.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 16 May 2025
AZD 6482
CAS:1173900-33-8
AZD 6482 (KIN-193) is a potent and selective inhibitor of p110β and PI3Kβ with IC50 …
Formula:
C22H24N4O4
Purity:
99.79% - 99.95%
Color and Shape:
Solid
Molecular weight:
408.45
Ref: TM-T6087
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Friday 16 May 2025
