Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,657 products)
- Apoptosis(6,058 products)
- Cell Cycle/Checkpoint(4,657 products)
- Chromatin/Epigenetics(2,354 products)
- Cytoskeletal Signaling(1,460 products)
- DNA Damage/DNA Repair(2,908 products)
- Endocrinology/Hormones(3,601 products)
- Enzyme(3,655 products)
- GPCR/G-Protein(8,703 products)
- Immunology and Inflammation(3,737 products)
- Influenza Virus(298 products)
- JAK/STAT signaling(403 products)
- MAPK Signaling(1,227 products)
- Membrane Transporter/Ion Channel(2,922 products)
- Metabolism(9,881 products)
- Microbiology/Virology(7,303 products)
- Neuroscience(10,209 products)
- Other Inhibitors(36,770 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,669 products)
- Stem Cell and Derivatives(828 products)
- Tyrosine Kinase/Adaptors(2,042 products)
- Ubiquitination(1,681 products)
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Found 66609 products of "Inhibitors"
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CYP1B1-IN-2
<p>CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].</p>Formula:C20H11F3O2Color and Shape:SolidMolecular weight:340.3Metoquizine
CAS:Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.Formula:C22H27N5OPurity:98%Color and Shape:SolidMolecular weight:377.48VU6028418
<p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>Color and Shape:LiquidER272
CAS:<p>ER272 is a natural PKC activator, inducing hippocampal neurogenesis.</p>Formula:C24H34O6Color and Shape:SolidMolecular weight:418.52GW311616
CAS:GW-311616 is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).Formula:C19H31N3O4SColor and Shape:SolidMolecular weight:397.53CBR Agonist-1
CBR Agonist-1 targets CB1R and CB2R with Ki of 0.18 μM and 1.22 μM, useful for studying cannabinoid-related diseases.Formula:C27H27FN4OColor and Shape:SolidMolecular weight:442.53Ivaltinostat formic
Ivaltinostat (CG-200745) is an oral panHDAC inhibitor, inducing apoptosis and enhancing cancer drug sensitivity.Formula:C25H35N3O6Color and Shape:SolidMolecular weight:473.56EFdA-TP tetrasodium
CAS:EFdA-TP tetrasodium is a potent HIV-1 inhibitor that blocks DNA synthesis as an ICT or DCT.Formula:C12H11FN5Na4O12P3Purity:98%Color and Shape:SolidMolecular weight:621.12CGP 22979
CAS:CGP 22979 is a renal selective vasodilator prodrug.Formula:C16H24N4O4Color and Shape:SolidMolecular weight:336.39MDL-43291
CAS:<p>MDL-43291 is a leukotriene receptor antagonist.</p>Formula:C25H42O4SColor and Shape:SolidMolecular weight:438.66Trichostatin A S-isomer
CAS:<p>Trichostatin A S-isomer, a HDAC 1, 3, 4, 6, 10 inhibitor with IC50 ~20 nM, has wide-ranging epigenetic effects.</p>Formula:C17H22N2O3Purity:98%Color and Shape:SolidMolecular weight:302.37Cgs 25155
CAS:Cgs 25155 is an orally active inhibitor of NEP 24.11.Formula:C25H34N2O6SPurity:98%Color and Shape:SolidMolecular weight:490.61TSWV-IN-1
TSWV-IN-1 is an anti-TSWV drug with potential TSWV N.Formula:C26H31FO4S2Color and Shape:SolidMolecular weight:490.65TY 11223
CAS:TY 11223: stable homoisocarbacyclin analog, potently inhibits platelet aggregation with lasting effect and selective activity.Formula:C24H34O5Color and Shape:SolidMolecular weight:402.52EBOV-GP-IN-1
EBOV-GP-IN-1 (Compound 28) is a potent inhibitor of Ebola entry, acting on the Ebola virus envelope glycoprotein (EBOV-GP) (IC50: 0.05 μM).Formula:C25H40ClN3O2Color and Shape:SolidMolecular weight:450.06Nrf2 activator-2
Compound O15, an Osthole derivative, is a potent Nrf2 agonist with an EC50 of 2.9 μM; it inhibits Keap1-Nrf2 binding and Nrf2 ubiquitination.Formula:C20H17BrO3Color and Shape:SolidMolecular weight:385.25YM-355179
CAS:YM-355179 is a novel, selective antagonist of CC chemokine receptor 3 with oral activity.Formula:C33H34FN4O7Purity:98%Color and Shape:SolidMolecular weight:617.64PDHK-IN-3
PDHK-IN-3 (compound 7) is a potent inhibitor of pyruvate dehydrogenase kinase(PDHK) with IC50s of 0.21 and 1.54 μM for PDHK2 and PDHK4, respectively [1].Formula:C17H16N2O2Color and Shape:SolidMolecular weight:280.32Cryptopleurine
CAS:Cryptopleurine is an inhibitor of gene products associated with cell proliferation, survival, invasion and angiogenesis. It acts by targeting the NF-κB pathway.Formula:C24H27NO3Purity:98%Color and Shape:SolidMolecular weight:377.48C5aR-IN-3
CAS:C5aR-IN-3, a potent C5aR inhibitor, may treat autoimmune and inflammatory diseases.Formula:C36H40FN5O3Color and Shape:SolidMolecular weight:609.73TRPC4/5-IN-1
TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.Formula:C21H21N3OColor and Shape:SolidMolecular weight:331.41Ophiobolin C
CAS:inhibitor of human CCR5 binding to HIV-1 gp120Formula:C25H38O3Purity:98%Color and Shape:SolidMolecular weight:386.57JAK3 covalent inhibitor-1
CAS:<p>JAK3 Covalent Inhibitor-1 is a compound characterized by its potent and selective inhibition of Janus kinase 3 (JAK3), possessing an IC50 of 11 nM and</p>Formula:C22H17FN6O2SPurity:98%Color and Shape:SolidMolecular weight:448.47AS1940477
CAS:<p>AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.</p>Formula:C24H22FN5O2Color and Shape:SolidMolecular weight:431.46TLR7/8 agonist 7
CAS:<p>TLR7/8 agonist 7 activates immune cells, useful in ISAC synthesis and immunity research.</p>Formula:C26H37N7O2Color and Shape:SolidMolecular weight:479.62Ganciclovir monophosphonate
CAS:Ganciclovir monophosphate treats CMV, inhibiting replication in human/animal strains (IC50: 0.01μM).Formula:C10H16N5O6PColor and Shape:SolidMolecular weight:333.24FNC-TP trisodium
<p>FNC-TP trisodium, active intracellular FNC form, inhibits NRTI, fights HIV, HBV, and HCV.</p>Formula:C9H11FN6Na3O13P3Color and Shape:SolidMolecular weight:592.11T-3764518
CAS:T-3764518 is a novel and potent inhibitor of stearoyl coenzyme A desaturase (SCD)(IC50 of 4.7 nM).Formula:C20H17F6N5O2Purity:98%Color and Shape:SolidMolecular weight:473.37ACT 178882
CAS:ACT 178882 is a new Renin inhibitor (IC50: 1.4 nM).Formula:C33H38Cl3N3O4Purity:98%Color and Shape:SolidMolecular weight:647.03PfPKG-IN-1
PfPKG-IN-1, an imidazole-based inhibitor, targets the Plasmodium falciparum cyclic guanosine monophosphate-dependent protein kinase (PfPKG).Formula:C24H22ClN7OSColor and Shape:SolidMolecular weight:492Antitumor agent-50
Antitumor agent-50 (compound 1a) is a thiazolidinone.Formula:C17H14FNO3SColor and Shape:SolidMolecular weight:331.36Samuraciclib hydrochloride hydrate
<p>Samuraciclib (CT7001) is a potent oral CDK7 inhibitor (IC50: 41 nM) with anti-breast cancer properties.</p>Formula:C22H35ClN6O3Color and Shape:SolidMolecular weight:521.7CDK9-IN-11
CAS:CDK9-IN-11 is a potent CDK9 inhibitor that is the ligand for the PROTAC CDK9 Degrader-1 [1].Formula:C20H25N3O4Purity:98%Color and Shape:SolidMolecular weight:371.43LY367385 hydrochloride
CAS:<p>LY367385 hydrochloride: selective mGluR1a antagonist, IC50 = 8.8 μM, neuroprotective, anticonvulsant, antiepileptic.</p>Formula:C10H12ClNO4Color and Shape:SolidMolecular weight:245.66Mcl-1 inhibitor 9
CAS:Mcl-1 Inhibitor 9 (Example 2) is a potent inhibitor of myeloid cell leukemia 1 (Mcl-1), demonstrating anti-tumor activity with an IC50 value of 0.21889 nM.Formula:C32H39ClN2O5SColor and Shape:SolidMolecular weight:599.18WM382
CAS:<p>WM382, a potent dual PMIX/X inhibitor, has IC50s of 1.4 nM/0.03 nM and effective against various malaria stages.</p>Formula:C29H36N4O4Color and Shape:SolidMolecular weight:504.62CS-0777
CAS:<p>CS-0777 is a potent, selective, and orally active S1P1 agonist (sphingosine 1-phosphate receptor modulator).</p>Formula:C21H31N2O5PColor and Shape:SolidMolecular weight:422.45HDAC-IN-37
HDAC-IN-37 inhibits HDACs 1, 3, 8, & 6, induces histone acetylation, halts G1 to S phase, and triggers early apoptosis.Formula:C23H24ClN7OColor and Shape:SolidMolecular weight:449.94Spliceostatin A
CAS:<p>Spliceostatin A is an anticancer agent and splicing inhibitor that induces apoptosis by inducing cell cycle arrest in the G1 and G2/M phases.</p>Formula:C28H43NO8Purity:94.66%Color and Shape:SolidMolecular weight:521.643NA 0346
CAS:NA 0346 is a derivative of SF 2370 that shows long lasting antihypertensive action as well as potent protein kinases inhibitory activity.Formula:C26H22N4O3Color and Shape:SolidMolecular weight:438.48Revamilast
CAS:Revamilast, also known as GRC4039, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritisFormula:C18H9Cl2F2N3O4Color and Shape:SolidMolecular weight:440.18PSB 36
CAS:A1 adenosine receptor antagonistFormula:C21H30N4O3Purity:98%Color and Shape:SolidMolecular weight:386.49SENP2-IN-1
CAS:SENP2-IN-1 selectively inhibits SENP2, SENP1, and SENP5 with low IC50 values; useful in cancer studies.Formula:C32H29N3O5S2Color and Shape:SolidMolecular weight:599.72SB 243213 dihydrochloride
CAS:SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8 forFormula:C22H21Cl2F3N4O2Purity:98%Color and Shape:SolidMolecular weight:501.33FGFR3-IN-4
CAS:FGFR3-IN-4 is a selective inhibitor targeting FGFR3, demonstrating an IC50 value of under 50 nM.Formula:C26H24ClN7OColor and Shape:SolidMolecular weight:485.97ETP-47037
CAS:ETP-47037: strong PI3Kα inhibitor (IC50: 0.99 nM), also targets PI3Kβ, δ, γ; may protect telomeres.Formula:C20H27N9O3SColor and Shape:SolidMolecular weight:473.55DAD dichloride
DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.Formula:C26H42Cl2N6OColor and Shape:SolidMolecular weight:525.56AY 17,605
CAS:AY 17,605 is an inhibitor of bovine heart and rat brain nucleoside-3',5'- monophosphate phosphodiesterase.Formula:C25H36O5Color and Shape:SolidMolecular weight:416.55CDK1-IN-4
CDK1-IN-4 inhibits CDK1 (IC50: 44.52 nM), CDK2/CDK5 less potently, impacts cell cycle, used in cancer studies.Formula:C26H24ClN5SColor and Shape:SolidMolecular weight:474.02P-gp modulator 2
P-gp modulator 2 (Compound 27) is a potent competitive and metabotropic P-glycoprotein (P-gp) modulator.Formula:C22H20BrN3O4Color and Shape:SolidMolecular weight:470.32Acetylpepstatin
CAS:<p>Acetylpepstatin is an inhibitor of HIV-1 protease, HIV-2 protease, aspartyl protease.</p>Formula:C33H61N5O11Purity:98%Color and Shape:SolidMolecular weight:703.875FP0429
CAS:FP0429 is an agonist of mGlu4.Formula:C10H12N2O7Purity:98%Color and Shape:SolidMolecular weight:272.21TAK-828F
CAS:<p>TAK-828F: potent, selective RORγt inverse agonist. Oral. IC50=1.9 nM; reporter gene IC50=6.1 nM.</p>Formula:C28H32FN3O5Purity:98%Color and Shape:SolidMolecular weight:509.57Thiolactomycin
CAS:Thiolactomycin is a novel reversible dual inhibitor of D-amino acid oxidase (DAO) and D-Aspartate oxidase (DDO).Formula:C11H14O2SPurity:98%Color and Shape:SolidMolecular weight:210.29CN-716 HCl
CAS:cn-716 is a novel Zika virus (ZIKV) NS2B-NS3pro protease inhibitor.Formula:C22H33BCl2N6O4Color and Shape:SolidMolecular weight:527.25Trk-IN-8
<p>Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).</p>Formula:C18H16F2N6O2Color and Shape:SolidMolecular weight:386.36Antitubercular agent-22
Antitubercular agent-22 combats Candida albicans (MIC: 2.34 μg/ml) and M. tuberculosis (MIC: 2 μg/ml).Formula:C24H28FN5O8Color and Shape:SolidMolecular weight:533.51BRD7929
CAS:BRD7929 is a multistage antimalarial inhibitor for single-dose treatment of malaria in mouse models.Formula:C33H38N4O2Color and Shape:SolidMolecular weight:522.68LPA5 antagonist 1
<p>LPA5 antagonist 1: selective, potent (IC50=32 nM), high brain permeability, studies inflammatory/neuropathic pain.</p>Formula:C28H26N2O4SColor and Shape:SolidMolecular weight:486.58Cimpuciclib tosylate
CAS:<p>Cimpuciclib tosylate, a selective CDK4 inhibitor (IC50: 0.49 nM), exhibits anti-tumor activity.</p>Formula:C37H43FN8O4SColor and Shape:SolidMolecular weight:714.85L-744832
CAS:<p>L-744832, also known as L-744,832, is a potent Farnesyltransferase inhibitor with potential anticancer activity.</p>Formula:C26H45N3O6S2Color and Shape:SolidMolecular weight:559.78KDOAM-25 citrate
CAS:KDOAM-25 citrate inhibits KDM5A/B/C/D (IC50: 71, 19, 69, 69 nM); boosts H3K4 methylation, hinders MM1S cell growth. [1]Formula:C21H33N5O9Purity:98%Color and Shape:SolidMolecular weight:499.51Mevidalen HBA
CAS:<p>Mevidalen (LY3154207), a potent D1 positive allosteric modulator, is in clinical trials for Lewy body dementia.</p>Formula:C31H35Cl2NO6Color and Shape:SolidMolecular weight:588.52β-N-Acetyl-D-hexosaminidase-IN-1
β-N-Acetyl-D-hexosaminidase-IN-1 is a newly discovered chemical compound that acts as an inhibitor for β-N-acetyl-D-hexosaminidase.Formula:C18H13F2NO2SColor and Shape:SolidMolecular weight:345.36Cap-dependent endonuclease-IN-14
CAS:Cap-dependent endonuclease-IN-14 hinders CEN and could treat influenza virus infections. (Patent CN113620948A, compound 1-c).Formula:C30H23FN2O6SColor and Shape:SolidMolecular weight:558.58XIAP degrader-1
<p>XIAP degrader-1 is a small primary amine molecule that promotes the degradation of X-linked apoptosis inhibitory protein (XIAP).</p>Formula:C34H45N5O4Color and Shape:SolidMolecular weight:587.75Antitumor agent-42
<p>Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.</p>Formula:C24H19BrN2O8SColor and Shape:SolidMolecular weight:575.39Antibacterial agent 66
Compound 6q, a trifluoromethylpyridine oxadiazole, targets Xanthomonas oryzae with EC50 of 7.2 μg/mL.Formula:C17H10ClF6N3O2SColor and Shape:SolidMolecular weight:469.79HIF-2α-IN-5
CAS:<p>HIF-2α-IN-5 is a potent HIF-2α inhibitor with an IC 50 of < 50 nM [1].</p>Formula:C15H12F4O3S2Color and Shape:SolidMolecular weight:380.38AP5 sodium
CAS:<p>AP5 sodium: potent oral GPR40 agonist, enhances ligands, may aid type II diabetes research.</p>Formula:C28H27FNNaO4Color and Shape:SolidMolecular weight:483.515LTD4 antagonist 1
CAS:LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM).Formula:C31H32F3N3O5SPurity:98%Color and Shape:SolidMolecular weight:615.66Tubulin polymerization-IN-4
CAS:Tubulin polymerization-IN-4: inhibits tubulin (IC50=4.6 μM), blocks G2/M phase, induces apoptosis, hinders cell cloning/migration, damages vasculature.Formula:C21H21ClN2O4Color and Shape:SolidMolecular weight:400.86BM635 hydrochloride (1493762-74-5 free base)
BM635 hydrochloride is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).Formula:C25H30ClFN2OPurity:98%Color and Shape:SolidMolecular weight:428.97Resolvin E4
CAS:RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45Dopamine D3 receptor ligand-1
Dopamine D 3 receptor ligand is a potent, selective, high-affinity dopamine D3 receptor ligand that is 89 times more selective for D3 (Ki: 8 nM) than D2 (Ki:Formula:C27H29N5OColor and Shape:SolidMolecular weight:439.55Homomoschatoline
CAS:Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.Formula:C19H15NO4Purity:98%Color and Shape:SolidMolecular weight:321.33AChE-IN-24
AChE-IN-24: Strong AChE blocker, crosses blood-brain barrier, IC50=0.053 μM, useful for AD research.Formula:C22H30N2O4S2Color and Shape:SolidMolecular weight:450.61TS010
TS010 is a highly potent inhibitor of GLO-I, with an IC50 value of 0.57 μM. It holds significant promise for advancements in cancer research [1].Formula:C16H12N4O4SColor and Shape:SolidMolecular weight:356.36KAG-308
CAS:KAG-308: selective EP4 agonist; Ki: 2.57 nM, EC50: 17 nM; suppresses colitis, promotes mucosal healing, inhibits TNF-α.Formula:C24H30F2N4O3Purity:98%Color and Shape:SolidMolecular weight:460.52KRAS G12D inhibitor 16
CAS:<p>KRAS G12D inhibitor 16 targets KRAS G12D with IC50 of 0.7 nM and mutant form at 0.35 μM, useful in various cancer studies.</p>Formula:C32H39IN6O3Color and Shape:SolidMolecular weight:682.59Anticancer agent 53
CAS:Anticancer agent 53 exhibits potent in vitro cytotoxicity, triggers apoptosis, halts S/G2/M cycle, and has antitumor effects without toxicity.Formula:C31H25FN4O6SColor and Shape:SolidMolecular weight:600.62(R)-ZG197
(R)-ZG197: Activates Sa ClpP (EC50=1.5μM) & Hs ClpP (EC50=31.4μM); selective for Sa ClpP.Formula:C28H35F3N4O3Color and Shape:SolidMolecular weight:532.6LJ-4517
LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.Formula:C19H21N5O3SColor and Shape:SolidMolecular weight:399.47GSK3527497 HCl
CAS:<p>GSK3527497: potent TRPV4 inhibitor, IC50=12 nM, targets heart/respiratory issues, for oral/IV use, low-dose effective.</p>Formula:C17H17Cl2FN4O4SColor and Shape:SolidMolecular weight:463.3054DYRKs-IN-1 hydrochloride
CAS:DYRKs-IN-1 HCl inhibits DYRK1A (5 nM IC50) & DYRK1B (8 nM IC50) with antitumor properties.Formula:C30H31Cl2N7O4Color and Shape:SolidMolecular weight:624.52CD33 splicing modulator 1
<p>Compound 1 modulates CD33, affects microglial cells, and may aid in neurodegenerative disease research.</p>Formula:C25H25FN6OColor and Shape:SolidMolecular weight:444.5CAII-IN-2
CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.Formula:C18H19BrN4SColor and Shape:SolidMolecular weight:403.34SS-RJW100
SS-RJW100 is an enantiomer of RJW100 targeting LRH-1, SF-1, enhances Tif2 interaction, and disrupts LRH-1 networks with lowered stability.Formula:C28H34OColor and Shape:SolidMolecular weight:386.57PPI-2458
CAS:PPI-2458, a fumagillin derivative, irreversibly blocks MetAP2, hindering abnormal cell growth and angiogenesis with improved toxicity.Formula:C22H36N2O6Color and Shape:SolidMolecular weight:424.53EGFR-IN-34
EGFR-IN-34 is a low-toxicity, acrylamide derivative antitumor agent that is a potent inhibitor of EGFR.Formula:C26H27ClN6O2Color and Shape:SolidMolecular weight:490.98GSK1820795A
CAS:<p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>Formula:C35H34N8Color and Shape:SolidMolecular weight:566.7Protectin D1
CAS:<p>Protectin D1 (Neuroprotectin D1) is a neuroprotectin produced by nerve cells and is a potential cardioprotective agent.</p>Formula:C22H32O4Purity:99.72% - 99.79%Color and Shape:SolidMolecular weight:360.49K203
K203 is a potent tabun-inhibited AChE reactivator and is an important antidote to organophosphorus poisoning.Formula:C16H18Br2N4O2Color and Shape:SolidMolecular weight:458.15A1-Phytoprostane-I
CAS:A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.Formula:C18H28O4Color and Shape:SolidMolecular weight:308.41CXCR7 antagonist-1 hydrochloride
CAS:CXCR7 antagonist-1 hydrochloride blocks SDF-1 and I-TAC from CXCR7; may prevent cancer and inflammation.Formula:C21H20ClFN6OColor and Shape:SolidMolecular weight:426.87MS8511
CAS:<p>MS8511: Selective, irreversible G9a/GLP inhibitor. IC50: 100 nM (G9a), 140 nM (GLP). Lowers H3K9me2, anti-proliferative. Useful in cancer/AD/PWS research.</p>Formula:C28H41N5O3Color and Shape:SolidMolecular weight:495.66FGFR4-IN-7
<p>FGFR4-IN-7 is a covalent, reversible FGFR4 inhibitor (IC50: 0.42 μM) that blocks the FGFR4 signaling pathway, thereby inducing apoptosis.</p>Formula:C26H25Cl2N5O3Color and Shape:SolidMolecular weight:526.41Asukamycin
CAS:<p>Asukamycin, from S. nodosus asukaensis, is a polyketide antibiotic inhibiting tumor cells by activating caspases 8 and 3.</p>Formula:C31H34N2O7Color and Shape:SolidMolecular weight:546.61FGFR-IN-5
CAS:FGFR-IN-5 is a potent inhibitor of FGFR. FGFR-IN-5 has potential for research in cancer diseases.Formula:C25H22N6O3Color and Shape:SolidMolecular weight:454.48RO5101576
CAS:RO5101576 is a potent antagonist of LTB4 receptor.Formula:C36H38O8SPurity:98%Color and Shape:SolidMolecular weight:630.75Antitumor agent-72
CAS:Antitumor agent-72 (compound 6w) is a potent anticancer agent that exhibits its anticancer activity by inducing apoptosis via caspase-3 activation and PARPFormula:C25H20ClNO6Color and Shape:SolidMolecular weight:465.88L-97-1
CAS:L-97-1 is an antagonist of the adenosine A1 receptor.Formula:C29H38N6O3Purity:98%Color and Shape:SolidMolecular weight:518.65PF-06273340
CAS:<p>PF-06273340 是一种口服具有活力的、具有选择性的外周限制性Trk 泛抑制剂。</p>Formula:C23H22ClN7O3Purity:98% - 98.00%Color and Shape:SolidMolecular weight:479.92PTP1B-IN-17
PTP1B-IN-17, a benzimidazole derivative, inhibits PTP1B (Ki: 30.2 μM) and may help study type 2 diabetes.Formula:C26H19N3O4SColor and Shape:SolidMolecular weight:469.51HBV-IN-18
HBV-IN-18 (Compound 3) is an HBV capsid assembly modulator (CpAM) (EC50: 2790 nM).Formula:C17H15F6N5O2Color and Shape:SolidMolecular weight:435.32LIT-001 free base
CAS:<p>LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.</p>Formula:C28H33N7O2SPurity:98%Color and Shape:SolidMolecular weight:531.67hCAII-IN-4
CAS:hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.Formula:C31H23NO9Color and Shape:SolidMolecular weight:553.52Nevirapine dimer
CAS:Nevirapine dimer is a non-nucleoside reverse transcriptase inhibitor (NNRTI).Formula:C30H26N8O2Color and Shape:SolidMolecular weight:530.58Glutamate-5-kinase-IN-1
Glutamate-5-kinase-IN-1 is a potent G5K inhibitor with a 4.1 μM MIC, showing promise in anti-TB research.Formula:C20H18N2OColor and Shape:SolidMolecular weight:302.37VEGFR-2-IN-5 hydrochloride
VEGFR-2-IN-5 hydrochloride is an effective VEGFR2 inhibitor.Formula:C19H25ClN8Color and Shape:SolidMolecular weight:400.91RET-IN-11
RET-IN-11 selectively inhibits RET (IC50: 6.20 nM), promotes apoptosis, and hinders cell proliferation and migration.Formula:C27H30FN9OColor and Shape:SolidMolecular weight:515.59Diacylglycerol acyltransferase inhibitor-1
CAS:<p>Diacylglycerol Acyltransferase Inhibitor-1, a diacylglycerol acyltransferase (DGAT1) inhibitor, effectively suppresses the activity of DGAT1.</p>Formula:C21H23N5O2Purity:98%Color and Shape:SolidMolecular weight:377.44Taprostene
CAS:<p>Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.</p>Formula:C24H30O5Color and Shape:SolidMolecular weight:398.49SAR-114137
CAS:<p>SAR-114137 is a histone sphingomyelin kinase inhibitor used in the study of molluscum arteriosum and peripheral neuropathic pain.</p>Formula:C25H34N4O7SPurity:99.09% - 99.91%Color and Shape:SolidMolecular weight:534.63L-697639
CAS:L-697639 inhibits of HIV-1 reverse transcriptase and HIV-1 replication.Formula:C18H21N3O2Color and Shape:SolidMolecular weight:311.38GSK8814
CAS:GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan).Formula:C28H35F2N5O3Purity:98%Color and Shape:SolidMolecular weight:527.61CBR Agonist-2
<p>CBR Agonist-2: CB1 receptor agonist, EC50 - 960 nM, Ki - 970 nM, useful for hCB1R-related disease research.</p>Formula:C27H27FN4OColor and Shape:SolidMolecular weight:442.53JH295 hydrate
<p>JH295 hydrate: potent, irreversible Nek2 inhibitor (IC50 = 770 nM), selective, doesn't target Cdk1, Aurora B or Plk1.</p>Formula:C18H18N4O3Color and Shape:SolidMolecular weight:338.36Butaprost
CAS:<p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>Formula:C24H40O5Purity:98%Color and Shape:SolidMolecular weight:408.57FLT3-IN-13
<p>FLT3-IN-13 inhibits topoisomerase II/FLT3 in leukemia with IC50 of 2.26 μM, causes G2/M arrest, and promotes apoptosis.</p>Formula:C20H14N4O2Color and Shape:SolidMolecular weight:342.35Carbacyclin
CAS:Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.Formula:C21H34O4Purity:98%Color and Shape:SolidMolecular weight:350.49Mu opioid receptor antagonist 5
Compound NAP: MOR antagonist, crosses blood-brain barrier, EC50: 1.14 nM, Ki: 0.37 nM, useful for OUD research.Formula:C26H29N3O4Color and Shape:SolidMolecular weight:447.53RWJ-56110
CAS:protease-activated receptor-1 (PAR1) antagonistFormula:C41H43Cl2F2N7O3Purity:98%Color and Shape:SolidMolecular weight:790.73Cav 3.2 inhibitor 3
Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.Formula:C32H37N3O2Color and Shape:SolidMolecular weight:495.66NR1H4 activator 1
CAS:NR1H4 activator 1 is a potent and selective agonist of Famesoid X Receptor (FXR).Formula:C34H53NO7SPurity:98%Color and Shape:SolidMolecular weight:619.85CCR7 Ligand 1
CAS:CCR7-Cmp2105 is a thiadiazole-dioxide allosteric antagonist for CCR7 with a Kd of 3 nM and IC50 of 7.3 μM against arrestin binding.Formula:C22H29N5O5SColor and Shape:SolidMolecular weight:475.56TRK-IN-19
<p>TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) & TRKAG595R (5.3 nM), promising for cancer research.</p>Formula:C22H26FN5O2Color and Shape:SolidMolecular weight:411.47JAK1/TYK2-IN-3
JAK1/TYK2-IN-3, orally active, selectively inhibits TYK2 (IC50: 6 nM), JAK1 (37 nM), JAK2 (140 nM), JAK3 (362 nM), and has anti-inflammatory effects.Color and Shape:SolidNumidargistat
CAS:CB-1158 is a potent and orally bioavailable inhibitor of arginase (IC50s: 86 and 296 nM for recombinant human arginase 1 and 2).Formula:C11H22BN3O5Purity:98%Color and Shape:SolidMolecular weight:287.12P300 bromodomain-IN-1
P300 bromodomain-IN-1 blocks c-Myc, induces G1/G0 arrest, apoptosis. Potent EP300 inhibitor (IC50: 49 nM).Formula:C29H31ClN4O4Color and Shape:SolidMolecular weight:535.03Human enteropeptidase-IN-2
<p>Human enteropeptidase-IN-2 is a potent inhibitor of enteropeptidase (enteropeptidase) and can be used in anti-obesity studies.</p>Formula:C20H19F3N4O7Color and Shape:SolidMolecular weight:484.38KNI 10033
CAS:<p>KNI 10033 is a potent inhibitor of HIV protease</p>Formula:C40H45N5O7S2Color and Shape:SolidMolecular weight:771.95JH-XVII-10
JH-XVII-10: potent, oral DYRK1A/B inhibitor (IC50: 3/5 nM), shows antitumor activity in HNSCC.Formula:C21H16F4N8OColor and Shape:SolidMolecular weight:472.4PRN694
CAS:PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.Formula:C28H35F2N5O2SPurity:98%Color and Shape:SolidMolecular weight:543.67Atiratecan
CAS:Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.Formula:C31H34N6O6Purity:98%Color and Shape:SolidMolecular weight:586.64MraY-IN-3
MraY-IN-3 (12a) is a potent inhibitor of the bacterial translocase MraY (IC50: 140 μM). 46 μg/ml).Formula:C35H45N3O5Color and Shape:SolidMolecular weight:587.75BTK-IN-16
CAS:BTK-IN-16 is a potential inhibitor of wild-type BTK and C481S mutants.BTK-IN-16 can be used to study various autoimmune diseases and cancers caused by BTK.Formula:C15H14N4O2Purity:99.04%Color and Shape:SoildMolecular weight:282.3Dot1L-IN-1
CAS:The Ki value of DOT1L-in-1 is 2pm.It is a highly effective, selective and novel Dot1L inhibitor.Formula:C32H36ClN9O2SPurity:98%Color and Shape:SolidMolecular weight:646.21MAO-B-IN-7
MAO-B-IN-7 inhibits MAO-B/AChE, crossing the blood-brain barrier; IC50: 41/87 nM (h/eel AChE), 0.3 μM (MAO-B). Reduces oxidative stress and neuroinflammation.Formula:C25H31NO4Color and Shape:SolidMolecular weight:409.52KF26777
CAS:KF26777 is a potent and selective antagonist of adenosine A3 receptor.Formula:C16H16BrN5OPurity:98%Color and Shape:SolidMolecular weight:374.23Nrf2/HO-1 activator 2
Compound 13m, a difluoro derivative, activates Nrf2/HO-1, showing neuroprotective and antioxidant effects, useful in PD research.Formula:C20H16F2O5Color and Shape:SolidMolecular weight:374.33ACT-777991
CAS:ACT-777991: oral CXCR3 blocker, stable in microsomes/hepatocytes, inhibits T-cell migration to CXCL11.Formula:C20H20F6N8O2SColor and Shape:SolidMolecular weight:550.48PDHK-IN-4
PDHK-IN-4 inhibits PDHK2 (IC50: 0.0051 μM) & PDHK4 (IC50: 0.0122 μM), with potential for cancer research.Formula:C24H25N5O3Color and Shape:SolidMolecular weight:431.49Heme Oxygenase-2-IN-1
Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).Formula:C19H17N3O2Color and Shape:SolidMolecular weight:319.36E 5090
CAS:E5090 is a novel orally active inhibitor of IL-1 generation. It also has anti-inflammatory properties.Formula:C19H20O5Purity:98%Color and Shape:SolidMolecular weight:328.36Isoleucyl tRNA synthetase-IN-2
CAS:Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).Formula:C22H33N5O8SColor and Shape:SolidMolecular weight:527.59RXR antagonist 1
RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.Formula:C28H33F3N2O3Color and Shape:SolidMolecular weight:502.57Pelecopan
CAS:<p>Pelecopan (BCX9930), an oral complement factor D inhibitor, prevents hemolysis in PNH (IC50=14.3 nM).</p>Formula:C23H19FN2O4Color and Shape:SolidMolecular weight:406.41SHR0687
CAS:<p>SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.</p>Formula:C39H60N8O5Color and Shape:SolidMolecular weight:720.94RSK4-IN-1
CAS:RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.Formula:C19H20F2N4O3Color and Shape:SolidMolecular weight:390.38FAAH/MAGL-IN-2
CAS:<p>FAAH/MAGL-IN-2: potent, reversible, oral FAAH & MAGL inhibitor, IC50: 11/36 nM, may research neuropathic pain, no locomotion issue.</p>Formula:C15H13Cl2N3O3SColor and Shape:SolidMolecular weight:386.25PF-06815345 hydrochloride
CAS:<p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>Formula:C27H30Cl2FN9O4Color and Shape:SolidMolecular weight:634.49CCR4 antagonist 2
CAS:CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits TregFormula:C26H28Cl2N6OPurity:98%Color and Shape:SolidMolecular weight:511.45Nrf2 activator-6
CAS:Nrf2 activator-6, a tetrahydroisoquinoline, inhibits Kelch-Nrf2 at 5 nM IC50 (WO2021214470A1).Formula:C31H37ClFN5O5Color and Shape:SolidMolecular weight:614.11ND-654
CAS:ND-654 is an acetyl CoA carboxylase inhibitor.Formula:C29H33N3O8SColor and Shape:SolidMolecular weight:583.65PF 03709270
CAS:PF 03709270 is an oral prodrug of sulopenem with broad-spectrum antibacterial effects on gram-positive and gram-negative bacteria.Formula:C19H27NO7S3Purity:98%Color and Shape:SolidMolecular weight:477.61HER2-IN-11
HER2-IN-11 is a psoralen derivative that induces apoptosis. HER2-IN-11 shows light-activated cytotoxicity and also exhibits anti-breast cancer activity [1].Formula:C17H11NO6Color and Shape:SolidMolecular weight:325.27U 75875
CAS:U 75875 is a protease inhibitor.Formula:C45H61N7O7Color and Shape:SolidMolecular weight:812.01T01-1
CAS:<p>T01-1, a derivative of camptothecin, is an anticancer agent demonstrating significant anti-proliferative activity.</p>Formula:C26H29N3O6SColor and Shape:SolidMolecular weight:511.59MtTMPK-IN-5
<p>MtTMPK-IN-5 inhibits Mtb TMPK with IC50 of 34 μM and fights tuberculosis with MIC of 12.5 μM, aiding TB research.</p>Formula:C21H23N5O2Color and Shape:SolidMolecular weight:377.44SSR 146977
CAS:<p>NK3 receptor antagonist</p>Formula:C35H42Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:621.64Prohibitin ligand 1
Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.Formula:C20H22N2OColor and Shape:SolidMolecular weight:306.4AChE-IN-22
<p>AChE-IN-22 (10q) selectively inhibits AChE (IC50: 0.88 μM), less on BuChE (IC50: 10 μM), targets CAS and PAS, useful in Alzheimer's research.</p>Formula:C21H20N4O5SColor and Shape:SolidMolecular weight:440.47(S)-MALT1-IN-5
CAS:<p>(S)-MALT1-IN-5: Potent MALT1 protease inhibitor, may help in abnormal T/B-cell signalling and MALT1-linked diseases.</p>Formula:C17H17ClF2N6O3Color and Shape:SolidMolecular weight:426.80Thiomuscimol hydrobromide
CAS:Thiomuscimol hydrobromide is an agonist of GABAA receptor.Formula:C4H6N2OSPurity:98%Color and Shape:SolidMolecular weight:130.17AZ13824374
AZ13824374: potent, selective ATAD2 inhibitor; anti-proliferative in breast cancer; pIC50: FRET 8.2, NanoBRET 6.2.Formula:C30H39FN8O2Color and Shape:SolidMolecular weight:562.68L 731735
CAS:L 731735 is a farnesyltransferase inhibitor.Formula:C19H40N4O4SPurity:98%Color and Shape:SolidMolecular weight:420.61AChE-IN-10
<p>AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.</p>Formula:C23H27F2NO4SColor and Shape:SolidMolecular weight:451.53Elacestrant S enantiomer dihydrochloride
Elacestrant (RAD1901) dihydrochloride, an oral ERR degrader, has IC50 of 48 nM (ERα) and 870 nM (ERβ). Its S enantiomer has low activity.Formula:C30H40Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:531.56XN methyl pyrazole
<p>XN methyl pyrazole exhibits beneficial effects on diet-induced obesity and enhances energy expenditure in mice fed with a high-fat diet [1].</p>Formula:C22H24N2O4Color and Shape:SolidMolecular weight:380.44Purine phosphoribosyltransferase-IN-1
Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.Formula:C11H15N5Na4O10P2Color and Shape:SolidMolecular weight:531.17JNJ-1250132
CAS:JNJ-1250132 is a steroidal progesterone receptor modulator that inhibits binding of the receptor to DNA in vitro.Formula:C33H41NO4Color and Shape:SolidMolecular weight:515.68COX-2-IN-10
COX-2-IN-10 is a potent COX-2 inhibitor, reducing IL-6, TNF-α, IL-1β, PGE2 (IC50=2.54 μM), and iNOS expression.Formula:C31H32FN5O2SColor and Shape:SolidMolecular weight:557.68Antiallergic agent-1
Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.Formula:C27H19F6N5OColor and Shape:SolidMolecular weight:543.46NDM-1 inhibitor-3
<p>NDM-1 inhibitor-3 is a New Delhi Metallo-β-lactamase-1 (NDM-1) inhibitor (Ki : 4 μM) widely found in nature and is associated with antibiotic resistance.</p>Formula:C16H12O4Purity:98.66%Color and Shape:SolidMolecular weight:268.26DENV-IN-6
CAS:<p>DENV-IN-6, a potent anti-DENV (I-IV) and HIV-1 IIIB inhibitor with EC50 ranging 6.8-17.5 μM for DENV and EC50 0.0181 μM for HIV-1.</p>Formula:C23H26ClFN4OSColor and Shape:SolidMolecular weight:461Unoprostone
CAS:Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.Formula:C22H38O5Purity:98%Color and Shape:SolidMolecular weight:382.53MDL-27210
CAS:<p>MDL-27210 is the ethyl ester prodrug of a potent angiotensin-converting enzyme inhibitor, MDL-27088.</p>Formula:C27H32N2O5Color and Shape:SolidMolecular weight:464.55GC 14
CAS:GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 200 nM and 35 nM for hTRα and hTRβ, respectively.Formula:C26H27NO6Purity:98%Color and Shape:SolidMolecular weight:449.5Ataprost
CAS:Ataprost (ONO 41483), an oral Carboprostacyclin analogue, is 2.6x more potent in inhibiting ADP-induced platelet aggregation and can relieve coronary spasm.Formula:C21H32O4Color and Shape:SolidMolecular weight:348.48LSD1-IN-21
<p>LSD1-IN-21: potent LSD1 inhibitor, crosses blood-brain barrier, IC50 of 0.956 μM; lowers TNF-α, anti-cancer, anti-inflammatory.</p>Formula:C24H25N5O2SColor and Shape:SolidMolecular weight:447.55BI-1388
CAS:BI-1388 is a potent HCV NS3 protease inhibitor; halts replication across genotypes, including D168V/R155K mutants.Formula:C41H53N7O9SColor and Shape:SolidMolecular weight:819.97Nrf2/HO-1 activator 1
CAS:Compound 24: Potent Nrf2/HO-1 activator with neuroprotective, antioxidant properties; useful in PD research.Formula:C21H18O5Color and Shape:SolidMolecular weight:350.36XR8-89
CAS:XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.Formula:C29H36N4O2SColor and Shape:SolidMolecular weight:504.69S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Formula:C12H13N4O6PPurity:98%Color and Shape:SolidMolecular weight:340.23Antibacterial agent 118
Antibacterial agent 118, potent against various mycobacteria, has MIC values ranging from 10.2 to 163.0 μM. Useful in TB research.Formula:C19H21N5O2SColor and Shape:SolidMolecular weight:383.47BRD50837
CAS:BRD50837 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Formula:C26H32ClN3O6SPurity:98%Color and Shape:SolidMolecular weight:550.07TAK-637
CAS:<p>TAK-637 is a tachykinin 1 (NK1) receptor antagonist.</p>Formula:C30H25F6N3O2Purity:98%Color and Shape:SolidMolecular weight:573.53DNA-PK-IN-6
CAS:DNA-PK-IN-6 inhibits DNA-PKcs, disrupting tumor DNA repair and triggering apoptosis; enhances radiotherapy and targets various tumors (WO2021197159A1).Formula:C19H21N7OColor and Shape:SolidMolecular weight:363.42Alpibectir
CAS:<p>Alpibectir has antibacterial activity [1].</p>Formula:C12H14F6N2O2Color and Shape:SolidMolecular weight:332.24VEGFR-2-IN-12
VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.Formula:C22H24N6O3SColor and Shape:SolidMolecular weight:452.53Anticancer agent 30
<p>Anticancer agent 30 (6f-Z), a 3-arylidene-2-oxindole, selectively inhibits CDK2, showing potent anticancer potential.</p>Formula:C22H15ClFNOColor and Shape:SolidMolecular weight:363.81Pibrozelesin
CAS:Pibrozelesin, a water-soluble duocarmycin B2 derivative, binds AT-rich DNA, blocking replication and inducing cell death.Formula:C32H36BrN5O8Color and Shape:SolidMolecular weight:698.56Hoe 892
CAS:<p>Hoe 892 is a stable thia-thimo-analogue of prostacyclin and acts as a platelet aggregation inhibitor.</p>Formula:C20H33NO4SColor and Shape:SolidMolecular weight:383.55QTX125 TFA
QTX125 TFA: Potent, selective HDAC6 inhibitor with antitumor effects.Formula:C25H20F3N3O7Color and Shape:SolidMolecular weight:531.44ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Formula:C29H33ClF2N6O9Purity:98%Color and Shape:SolidMolecular weight:683.06Elacestrant S enantiomer
<p>Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.</p>Formula:C30H38N2O2Purity:98%Color and Shape:SolidMolecular weight:458.63MK-2748
CAS:MK-2748 is an inhibitor of NS3 protease, hepatitis C virus.Formula:C42H56N6O10SColor and Shape:SolidMolecular weight:836.99Macropa-NCS
CAS:Macropa-NCS is a macropa bifunctional analog with antitumor activity and can be used to study prostate cancer.Formula:C27H35N5O8SPurity:98%Color and Shape:SolidMolecular weight:589.66c-Met/HDAC-IN-2
CAS:Potent dual c-Met/HDAC inhibitor, IC50: HDAC1 5.4 nM, c-Met 18.49 nM; anti-cancer, induces apoptosis, G2/M arrest in HCT-116.Formula:C34H33N5O7Color and Shape:SolidMolecular weight:623.66
