Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,440 products)
- Cytoskeletal Signaling(1,527 products)
- DNA Damage/DNA Repair(2,968 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,005 products)
- Immunology and Inflammation(3,874 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,591 products)
- Neuroscience(10,382 products)
- Other Inhibitors(36,042 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,444 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66686 products of "Inhibitors"
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ERRγ Inverse Agonist 1
CAS:ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].Formula:C30H38Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:529.54Phenoprolamine Hydrochloride
CAS:Phenoprolamine HCl: α1 blocker with anti-hypertensive, brain, and heart protection; inhibits CYP2D/3A, crosses the blood-brain barrier.Formula:C21H30ClNO3Color and Shape:SolidMolecular weight:379.92(Iso)-FK-480
CAS:(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.Formula:C26H19FN4O2Purity:98.36% - 99.41%Color and Shape:SolidMolecular weight:438.45JTP-4819
CAS:JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.Formula:C19H25N3O4Color and Shape:SolidMolecular weight:359.42AZD8848
CAS:AZD8848 is a selective antedrug agonist of toll-like receptor 7 (TLR7). It is developed for the research of asthma and allergic rhinitis.Formula:C29H43N7O5Color and Shape:SolidMolecular weight:569.7Antibacterial agent 48
CAS:Antibacterial agent 48 is an antimicrobial agent that reduces the MIC of the antimicrobial agent Ceftazidime.Formula:C13H18N5NaO7SColor and Shape:SolidMolecular weight:411.36MMPX
CAS:calmodulin-sensitive cyclic GMP phosphodiesterase inhibitorFormula:C12H18N4O3Purity:98%Color and Shape:SolidMolecular weight:266.3Rha-PEG3-SMCC
CAS:Rha-PEG3-SMCC (Compound 13) serves as an ADC (antibody-drug conjugate) linkage agent with robust antitumor properties, utilizing the protein crosslinker SMCC,Formula:C24H38N2O10Color and Shape:SolidMolecular weight:514.57HDAC3 Inhibitor
CAS:HDAC3 inhibitor: allosteric, Ki=0.16 nM, favors HDAC3 over HDAC1/2, targets specific leukemia cells, EC50=36.37-151.7 nM.Formula:C20H23N3O2Color and Shape:SolidMolecular weight:337.42Dimethenamid
CAS:Dimethenamid is a chloroacetamide herbicide.Formula:C12H18ClNO2SColor and Shape:Yellow-Brown Viscous LiquidMolecular weight:275.807α,25-Dihydroxycholesterol
CAS:7α, 25-dihydroxycholesterol (7α,25-OHC) is a potent and selective agonist and endogenous ligand of the orphan GPCR receptor EBI2 (GPR183).Formula:C27H46O3Purity:98%Color and Shape:SolidMolecular weight:418.65JNJ-64264681
CAS:JNJ-64264681 is a potent, orally active, selective, and irreversible covalent inhibitor of Bruton's tyrosine kinase (BTK).Formula:C27H30N6O3SPurity:98%Color and Shape:SolidMolecular weight:518.63SYN20028567
CAS:SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].Formula:C20H29N3O3SColor and Shape:SolidMolecular weight:391.53Antibacterial agent 126
Antibacterial agent 126 combats biofilm, disrupts membranes, and boosts ROS/RNS to prevent drug resistance.Formula:C21H24NO6PColor and Shape:SolidMolecular weight:417.39J1075
CAS:<p>J1075 is an histone deacetylase 8 (HDAC8) inhibitor.</p>Formula:C9H6ClNO2SPurity:98%Color and Shape:SolidMolecular weight:227.67Razinodil
CAS:Razinodil is a vasodilator.Formula:C27H34N4O10Color and Shape:SolidMolecular weight:574.58ABCG2-IN-1
CAS:ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with an inhibitory concentration (IC50) of 0.13 μM.Formula:C26H36N4O4Purity:98%Color and Shape:SolidMolecular weight:468.59Chitin synthase inhibitor 4
CAS:Chitin synthase inhibitor 4: a CHS inhibitor with antimicrobial properties, potential fungicide.Formula:C20H15FN4OPurity:99.8%Color and Shape:SolidMolecular weight:346.36Ref: TM-T61147
2mg39.00€5mg62.00€10mg99.00€25mg195.00€50mg284.00€100mg393.00€200mg520.00€1mL*10mM (DMSO)67.00€KRAS4b-IN-D14
CAS:KRAS4b-IN-D14 inhibits oncogenic KRAS4b, shrinks tumors, and induces cancer cell apoptosis.Formula:C24H24ClN5O4Color and Shape:SolidMolecular weight:481.93CSF1R-IN-13
CAS:CSF1R-IN-13: potent cancer research CSF1R inhibitor impacting cell growth regulation.Formula:C21H20N4O3Color and Shape:SolidMolecular weight:376.41MMP-1-IN-1
MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .Formula:C14H17ClN2O3Color and Shape:SolidMolecular weight:296.757U-85 Hydrochloride
CAS:7U-85 Hydrochloride, a DNA-directed DNA polymerase inhibitor, is used potentially for the treatment of cancer.Formula:C22H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:384.96BrW
CAS:6BrW is an analog of tryptophan effector.Formula:C11H11BrN2O2Purity:98%Color and Shape:SolidMolecular weight:283.12Telomerase-IN-5
CAS:Telomerase-IN-5 is a potent inhibitor of telomerase with antiproliferative properties, and it induces apoptosis [1].Formula:C22H20N4OS2Purity:98%Color and Shape:SolidMolecular weight:420.55Detirelix acetate
CAS:Detirelix acetate is an LHRH AntagonistFormula:C82H113ClN18O17Color and Shape:SolidMolecular weight:1658.34TBK1/IKKε-IN-4
CAS:TBK1/IKKε-IN-4, a 6-aminopyrazolopyrimidine derivative, serves as a potent, selective inhibitor for TBK1 and IKKε, demonstrating IC50 values of 13 nM and 59 nMFormula:C28H35N7O4Color and Shape:SolidMolecular weight:533.62Dual AChE-MAO B-IN-2
CAS:Potent Dual AChE-MAO B-IN-2 inhibits AChE (0.12 μM) & MAO B (0.01 μM); promising for Alzheimer's research.Formula:C26H25NO4Color and Shape:SolidMolecular weight:415.48Mabuterol hydrochloride
CAS:Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.Formula:C13H19Cl2F3N2OColor and Shape:SolidMolecular weight:347.20APA-APA-MPO
CAS:APA-APA-MPO is a PCAF bromodomain/Tat-AcK50 association inhibitor.Formula:C12H25Cl2N5OPurity:98%Color and Shape:SolidMolecular weight:326.27N-Arachidonyldopamine
CAS:N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is also a potent and selective TRPV1Formula:C28H41NO3Purity:97.65%Color and Shape:SolidMolecular weight:439.63Keap1-Nrf2-IN-12
CAS:eap1-Nrf2-IN-12 is a potent inhibitor of Keap1-Nrf2 (IC50: 2.30 μM). eap1-Nrf2-IN-12 is metabolically stable in human liver microsomes.Formula:C26H28N2O10S2Color and Shape:SolidMolecular weight:592.64Relutrigine
CAS:Relutrigine (PRAX-562) is an oral persistent sodium channel inhibitor with anticonvulsant properties, IC50 of 141 nM/75 nM for ATX-II/SCN8A-N1768D.Formula:C15H11F6N5O2Color and Shape:SolidMolecular weight:407.27Ref: TM-T69652
1mgTo inquire5mgTo inquire10mg1,064.00€25mg1,586.00€50mg2,072.00€100mg2,660.00€1mL*10mM (DMSO)615.00€Hexestrol dibutyrate
CAS:Hexestrol dibutyrate: Synthetic ER activator, microtubule blocker, possible carcinogen, causes mitotic arrest, aneuploidy, and DNA adducts.Formula:C26H34O4Color and Shape:SolidMolecular weight:410.55CDK9-IN-14
CAS:CDK9-IN-14: Potent CDK9 inhibitor, IC50=6.92 nM, effective on MV-4-11 cells and in vivo tumors, low toxicity, minimal side effects.Formula:C21H23F2N3O4Color and Shape:SolidMolecular weight:419.42Clathrin-IN-2
CAS:Clathrin-IN-2: CME inhibitor, IC50 - 2.3μM; also blocks dyn I GTPase, IC50 - 7.7μM.Formula:C17H18Br2N2OColor and Shape:SolidMolecular weight:426.15Vapendavir
CAS:Vapendavir binds enterovirus capsids; effective against EV71 with EC50 of 0.5-1.4 μM.Formula:C21H26N4O3Purity:98%Color and Shape:SolidMolecular weight:382.46Teroxalene hydrochloride
CAS:Teroxalene Hydrochloride is disubstituted piperazine used to treat animals with Schistosoma mansoni.Formula:C28H42Cl2N2OColor and Shape:SolidMolecular weight:493.55Iodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Formula:C15H20BrIN4SPurity:98%Color and Shape:SolidMolecular weight:495.22KRN2
CAS:KRN2, an NFAT5 inhibitor with a 100 nM IC50, may treat Chronic Arthritis.Formula:C27H23ClFNO4Purity:98%Color and Shape:SolidMolecular weight:479.93CP-53631
CAS:CP-53631 is a selective serotonin reuptake inhibitor (SSRI)Formula:C17H19BrClNColor and Shape:SolidMolecular weight:352.7Edivoxetine
CAS:Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.Formula:C18H26FNO4Color and Shape:SolidMolecular weight:339.4YPC-22026
CAS:YPC-22026 has potential anticancer activity, inducing tumor regression in a mouse xenograft model while inhibiting ZNF143-regulated genes.Formula:C16H8F3N3O2Purity:99.78% - 99.98%Color and Shape:SolidMolecular weight:331.25Iprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Formula:C19H28N2Purity:99.54%Color and Shape:SolidMolecular weight:284.44Ref: TM-T37015
2mg37.00€5mg52.00€10mg80.00€25mg154.00€50mg266.00€100mg455.00€200mg652.00€1mL*10mM (DMSO)84.00€Aminopeptidase-IN-1
CAS:Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.Formula:C18H16N2O6Purity:98.34%Color and Shape:SolidMolecular weight:356.33MBM-17S
CAS:MBM-17S, a potent NIMA-related kinase 2 (Nek2) inhibitor with an IC50 of 3 nM, effectively inhibits cancer cell proliferation by inducing cell cycle arrest andFormula:C36H40N6O10Purity:98%Color and Shape:SolidMolecular weight:716.74OX01914
CAS:OX01914 is a soluble modulator to increase utrophin in DMD studies, EC50 20.5 μM.Formula:C17H14N4OColor and Shape:SolidMolecular weight:290.32N-(3-Oxooctanoyl)-DL-homoserine lactone
CAS:N-(3-Oxooctanoyl)-DL-homoserine lactone with stereochemistry-dependent growth regulatory activity for roots .Formula:C12H19NO4Purity:98%Color and Shape:SolidMolecular weight:241.28hCAIX-IN-8
CAS:hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.Formula:C19H16N4O6Color and Shape:SolidMolecular weight:396.35TRK-IN-23
CAS:TRK-IN-23 (compound 24b) is a potent, orally active inhibitor of TRK with IC50s of 0.5 nM for TRKA, 9 nM for TRKC, 14 nM for TRKA G595R, 4.4 nM for TRKA F589L,Formula:C20H17FN4O2Purity:98%Color and Shape:SolidMolecular weight:364.37PDE5-IN-5
CAS:PDE5-IN-5 is a selective inhibitor of phosphodiesterase 5 (PDE5) (IC50: 2.0 nM).Formula:C23H20BrN3O4Color and Shape:SolidMolecular weight:482.33
