Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,850 products)
- Apoptosis(6,367 products)
- Cell Cycle/Checkpoint(4,909 products)
- Chromatin/Epigenetics(2,631 products)
- Cytoskeletal Signaling(1,586 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,053 products)
- Immunology and Inflammation(3,946 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,156 products)
- Microbiology/Virology(7,671 products)
- Neuroscience(10,551 products)
- Other Inhibitors(35,855 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,989 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66515 products of "Inhibitors"
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Collagen proline hydroxylase inhibitor
CAS:Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.Formula:C18H18N4O4Purity:98%Color and Shape:SolidMolecular weight:354.36Oxamniquine
CAS:Oxamniquine is an effective compound for the treatment of schistosomiasis.Formula:C14H21N3O3Purity:98%Color and Shape:Pale Yellow Crystals From Isopropanol SolidMolecular weight:279.33M-0002
CAS:M-0002, a vasopressin V2 receptor antagonist, is used potentially for the treatment of ascites.Formula:C32H29Cl2N3O3Color and Shape:SolidMolecular weight:574.5ICMT-IN-41
CAS:ICMT-IN-41 (compound 20) serves as a potent inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), demonstrating an IC50 value of 0.069 μM [1].Formula:C23H31NOColor and Shape:SolidMolecular weight:337.5PSMA-Val-Cit-PAB-MMAE
CAS:PSMA-Val-Cit-PAB-MMAE is a novel PSMA-targeted small-molecule conjugate leveraging monomethyl auristatin E (MMAE) for prostate cancer chemotherapy.Formula:C114H165ClN20O26Color and Shape:SolidMolecular weight:2267.1β-Catenin modulator-1
CAS:β-Catenin modulator-1 (IIa-650) is a useful agent in cancer research for modulating β-Catenin [1].Formula:C21H28N2O4SColor and Shape:SolidMolecular weight:404.52Mdl 27013
CAS:Mdl 27013 is a derivative of methoxysuccinyl-alanyl-alanyl-prolyl-valine.Formula:C22H33F3N4O7Color and Shape:SolidMolecular weight:522.52Antitumor agent-29
CAS:Antitumor agent-29 is a hepatocyte-targeting prodrug with demonstrated efficacy and minimal toxicity in anticancer applications.Formula:C71H96N16O24S2Color and Shape:SolidMolecular weight:1621.75HBY-793
CAS:HBY-793 is an HIV-1 proteinase inhibitor.Formula:C64H82N4O10S2Color and Shape:SolidMolecular weight:1131.49L-783483
CAS:L-783483 is an agonist of PPAR.Formula:C22H21ClF3NO4SPurity:98%Color and Shape:SolidMolecular weight:487.92NK007
CAS:NK007 is a novel anti-SARS-CoV-2 agent with an EC 50 value of 30 nM.Formula:C28H33NO9Color and Shape:SolidMolecular weight:527.56OADS
CAS:OADS is an inhibitor of ClC-ec1 with low micromolar affinity. OADS has no specific effect on a CLC channel (ClC-1).Formula:C30H42N2O8S2Color and Shape:SolidMolecular weight:622.79NSC309401 dihydrochloride
CAS:NSC309401 is an E. coli dihydrofolate reductase inhibitor with an IC50 value of 189 nM and a dissociation constant (Kd) of 14.57 nM [1].Formula:C17H18Cl2N6Color and Shape:SolidMolecular weight:377.27Benzamide, N,N-bis(5-(p-aminophenoxy)pentyl)-
CAS:Benzamide, N,N-bis(5-(p-aminophenoxy)pentyl)- is a bioactive chemical.Formula:C29H37N3O3Color and Shape:SolidMolecular weight:475.62Docebenone
CAS:Docebenone is a selective and orally active inhibitor of 5-LO.Formula:C21H26O3Color and Shape:SolidMolecular weight:326.43WAY-639299
CAS:WAY-639299 is an investigational compound targeting amyloid disorders and synucleinopathies for research purposes.Formula:C19H19N3O2S2Color and Shape:SolidMolecular weight:385.5PI3Kγ inhibitor 2
CAS:PI3Kγ inhibitor 2 is an orally bioavailable inhibitor of PI3Kγ(Ki of 4 nM).Formula:C20H18F3N5O3Purity:98%Color and Shape:SolidMolecular weight:433.38(S)-FTY-720 Vinylphosphonate
CAS:(S)-FTY-720 Vinylphosphonate blocks sphingosine kinase 1 and aids its breakdown in various human cancer cells.Formula:C20H34NO4PColor and Shape:SolidMolecular weight:383.46MARK-IN-1
CAS:MARK-IN-1 is a potent microtubule affinity regulating kinase (MARK) inhibitor, (IC50<0.25 nM).Formula:C22H23F2N7OSPurity:98%Color and Shape:SolidMolecular weight:471.53CI-959 free acid
CAS:CI-959 Free Acid is an orally effective inhibitor of cell activation in vitro and in animal models and also has anti-allergic/anti-inflammatory properties.Formula:C14H15N5O3SColor and Shape:SolidMolecular weight:333.37AVG-233
CAS:AVG-233 is an RNA-dependent RNA polymerase (RdRp) inhibitor with antiviral activity for the study of respiratory syncytial virus infections.Formula:C26H22ClN5O3Purity:99%Color and Shape:SolidMolecular weight:487.94WAY-634964
CAS:WAY-634964 is an active molecule.Formula:C9H7N3O2Color and Shape:SolidMolecular weight:189.17ATAC21
CAS:ATAC21 is a linker-immune-stimulatory compound created by conjugating a noncleavable maleimide-PEG4 linker, which includes a succinimide group, with an immune-Formula:C38H50N12O21P2Color and Shape:SolidMolecular weight:1072.82CBP/p300-IN-17
CAS:CBP/p300-IN-17 (compound 7) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.18 μM) and LK2 H3K27 (IC50: 0.69 μM).Formula:C25H28N4O3Color and Shape:SolidMolecular weight:432.51MMP3 inhibitor 1
CAS:MMP3 inhibitor 1 is a potent and highly selective inhibitor of MMP-3 (IC50 of 1 nM).Formula:C23H31N3O6SPurity:98%Color and Shape:SolidMolecular weight:477.57FTI-2153
CAS:FTI-2153 inhibits farnesyltransferase with 1.4 nM IC50, >3000x more effective on H-Ras than Rap1A.Formula:C25H30N4O3SColor and Shape:SolidMolecular weight:466.67-(Dimethylamino)-4-methylcoumarin
CAS:7-(Dimethylamino)-4-methylcoumarin, a coumarin derivative, is utilized in the research of fluorescent brightener solutions [1].Formula:C12H13NO2Color and Shape:SolidMolecular weight:203.24Tirofiban HCl
CAS:Tirofiban HCl is an antagonist of platelet glycoprotein-IIb/IIIa receptor.
Formula:C22H37ClN2O5SPurity:98%Color and Shape:SolidMolecular weight:477.06PIM1-IN-4
CAS:PIM1-IN-4: strong PIM1 inhibitor, also blocks SGK-1, PKA, CaMK-1, GSK3β, MSK1; promising for cancer studies.Formula:C27H25BrCl2CuN6OPurity:98%Color and Shape:SolidMolecular weight:663.88AChE-IN-31
CAS:AChE-IN-31 (compound 1), a non-competitive acetylcholinesterase (AChE) inhibitor, exhibits potential for Alzheimer's disease research [1].Formula:C27H44Na2O9S2Color and Shape:SolidMolecular weight:622.74KRAS inhibitor-14
CAS:KRAS inhibitor-14 targets G12C (IC50: 0.249 μM) and inhibits p-ERK in cancer cells; promising for pancreatic, colorectal, lung cancers.Formula:C20H15Cl3FN3O2SColor and Shape:SolidMolecular weight:486.77TP-051
CAS:TP-051 is a FFAR1 agonist.Formula:C29H31FO6SPurity:99.45% - 99.96%Color and Shape:SolidMolecular weight:526.62JAK-IN-31
CAS:JAK-IN-31 (Example 75), a JAK inhibitor, demonstrates IC50 values of ≤0.01 µM for JAK1, ≤0.01 µM for JAK2, 0.01-0.1 µM for JAK3, and ≤0.01 µM for Tyk2,Formula:C21H19N7O2S2Purity:98%Color and Shape:SolidMolecular weight:465.557Ethanol-10NH2-11F-Camptothecin
CAS:7Ethanol-10NH2-11F-Camptothecin, an antibody drug conjugate (ADC), demonstrates inhibitory effects on tumor growth and is utilized in cancer research [1].Formula:C21H18FN3O5Color and Shape:SolidMolecular weight:411.38NS1219
CAS:NS1219, an isomer of NS1209, is a selective AMPA antagonist for studying stroke, neuropathic pain, and epilepsy.Formula:C24H28N4O7SColor and Shape:SolidMolecular weight:516.57OSMI-1
CAS:OSMI-1: cell-permeable OGT inhibitor, blocks O-GlcNAcylation (IC50: 2.7 μM), no effect on other cell glycans.Formula:C28H25N3O6S2Purity:96.79% - 99.39%Color and Shape:SolidMolecular weight:563.64R-130823
CAS:R-130823 inhibits MAP kinase p38alpha (IC50=22 nM) and blocks cytokine release, reducing rat arthritis swelling and pain better than methotrexate.Formula:C28H26FN3Color and Shape:SolidMolecular weight:423.52Carbonic anhydrase inhibitor 12
CAS:CA Inhibitor 12 strongly blocks CA II (K_i 1.72 nM), also inhibits CA I (271 nM), shows anticancer effects.Formula:C27H22BrN5O5S2Purity:98%Color and Shape:SolidMolecular weight:640.53Orexin receptor antagonist 4
CAS:Orexin antagonist 4: potent, selective for OX2R (IC50=4.27 nM); less for OX1R (IC50=295 nM).Formula:C22H24FN5O2Color and Shape:SolidMolecular weight:409.46IIIM-290
CAS:IIIM-290 is an oral CDK inhibitor (IC50s: 90 and 94 nM for CDK2/A and CDK9/T1).Formula:C23H21Cl2NO5Purity:98%Color and Shape:SolidMolecular weight:462.32KF21213
CAS:KF21213 shows a high affinity for the adenosine A2A receptors (Ki=3.0 nM). KF21213 is a highly selective ligand for mapping CNS adenosine A2A receptors.Formula:C19H22N4O3Purity:98%Color and Shape:SolidMolecular weight:354.4Y18501
CAS:Y18501, an oxysterol-binding protein (OSBPI) inhibitor structurally akin to Oxathiapiprolin, demonstrates potent inhibition against Phytophthora spp.Formula:C27H26F2N6O2SColor and Shape:SolidMolecular weight:536.6Tyk2-IN-9
CAS:Tyk2-IN-9: selective Tyk-2 inhibitor, IC50 of 0.076 nM (TYK2-JH2), 1.8 nM (JAK1-JH2), for inflammation/autoimmune research.Formula:C20H17N9Purity:98%Color and Shape:SolidMolecular weight:383.41BACE1-IN-13
CAS:BACE1-IN-13 (Compound 36), an orally active inhibitor of BACE1, exhibits high potency with an IC50 of 2.9 nM and demonstrates greater efficacy in hAβ42 cells (Formula:C20H17FN8O2Purity:98%Color and Shape:SolidMolecular weight:420.4BRD4 Inhibitor-28
CAS:BRD4 Inhibitor-28 (Compound 18), an orally active molecule, selectively inhibits the bromodomains of BRD4 (BRD4-BD1 and BRD4-BD2) with IC50 values of 15 and 55Formula:C23H21N3O3Purity:98%Color and Shape:SolidMolecular weight:387.43Anticancer agent 101
CAS:Anticancer Agent 101, a tetracaine derivative, exhibits anti-cancer activity [1].Formula:C19H20F3N3OColor and Shape:SolidMolecular weight:363.38AGN 192836
CAS:AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).Formula:C12H13N3O2Color and Shape:SolidMolecular weight:231.25CPUY201112
CAS:CPUY201112, a novel inhibitor of heat shock protein Hsp90, induces p53-mediated apoptosis in MCF-7 cells.Formula:C19H23N3O4Color and Shape:SolidMolecular weight:357.46-Methoxypurine arabinoside
CAS:6-Methoxypurine arabinoside (Ara-m), a potent inhibitor of the varicella-zoster virus (VZV), exhibits 50% inhibitory concentrations (IC50) between 0.5 and 3Formula:C11H14N4O5Color and Shape:SolidMolecular weight:282.25YM-08
CAS:YM-08 (Compound 7a), a brain-penetrant SIRT2 inhibitor, exhibits an IC50 of 19.9 μM. Additionally, it acts as an inhibitor of Hsp70 [1].Formula:C19H17N3OS2Purity:98%Color and Shape:SolidMolecular weight:367.49
