Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,856 products)
- Apoptosis(6,375 products)
- Cell Cycle/Checkpoint(4,913 products)
- Chromatin/Epigenetics(2,633 products)
- Cytoskeletal Signaling(1,590 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,055 products)
- Immunology and Inflammation(3,957 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,162 products)
- Metabolism(10,157 products)
- Microbiology/Virology(7,674 products)
- Neuroscience(10,550 products)
- Other Inhibitors(35,861 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,438 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,992 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66511 products of "Inhibitors"
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Antibacterial agent 94
CAS:Compound 5b, an antibacterial, effectively targets MRSA and disrupts bacterial membranes and PG synthesis.Formula:C21H21FO4Color and Shape:SolidMolecular weight:356.39Niceritrol
CAS:Niceritrol (Cardiolipol) is a niacin ester that reduces cholesterol and triglycerides in total plasma and in the VLD and LD lipoprotein fractions.Formula:C29H24N4O8Purity:97.02%Color and Shape:SolidMolecular weight:556.52Ref: TM-T19861
1mg57.00€2mg80.00€5mg103.00€1mL*10mM (DMSO)142.00€10mg147.00€25mg255.00€50mg384.00€100mg567.00€KNI-272
CAS:Kynostatin-272 is a HIV protease inhibitor. KNI-272 blocked the maturation of viral particles.Formula:C33H41N5O6S2Color and Shape:SolidMolecular weight:667.84BACE1-IN-1
CAS:BACE1-IN-1 is a high brain penetrant BACE1 inhibitor (IC50s: 32 and 47 nM for human BACE1 and BACE2).Formula:C18H14F3N5O2Purity:98%Color and Shape:SolidMolecular weight:389.33Justicidin D
CAS:Justicidin D is a lignan that has antiviral activities.Formula:C21H14O7Purity:98%Color and Shape:SolidMolecular weight:378.33AR-13503
CAS:AR-13503, a Netarsudil metabolite, is a ROCK inhibitor, potentially treating glaucoma and lowering eye pressure.Formula:C19H19N3O2Color and Shape:SolidMolecular weight:321.37Cisd2 agonist 2
CAS:Cisd2 agonist 2 (compound 6), with an EC50 of 191 nM, is an orally active activator of Cisd2, a protein whose levels are associated with nonalcoholic fattyFormula:C14H14N2O4SColor and Shape:SolidMolecular weight:306.34GSK-2807 free base
CAS:GSK2807: potent, selective SMYD3 inhibitor (Ki=14 nM); targets SAM-binding site, potentially useful in cancer therapy.Formula:C19H32N8O5Color and Shape:SolidMolecular weight:452.51HDAC1/CDK7-IN-1
CAS:HDAC1/CDK7-IN-1 (compound 8e) serves as a dual inhibitor targeting both CDK7 and HDAC1, with IC50 values of 893 nM and 248 nM , respectively.Formula:C33H32ClN7O4Purity:98%Color and Shape:SolidMolecular weight:626.11BChE-IN-20
CAS:BChE-IN-20 (compound 7c) is a potent, selective inhibitor of BChE, demonstrating IC50 values of 105 nM for eqBChE and 2.3 nM for hBChE.Formula:C27H39N5O2Color and Shape:SolidMolecular weight:465.63KRAS degrader-1
CAS:KRAS degrader-1 (compound 1) is a potent agent that selectively targets KRAS proteins for destruction via the autophagy-lysosomal degradation pathway [1].Formula:C55H57Br2ClFIN8O7Color and Shape:SolidMolecular weight:1283.25LG 83-6-05
CAS:LG 83-6-05 is a novel kind of sodium channel blocking agent.Formula:C21H30ClNO3SColor and Shape:SolidMolecular weight:411.99YXG-158
CAS:YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1Formula:C30H36FN3OPurity:98%Color and Shape:SolidMolecular weight:473.62Sigma-1 receptor antagonist 3
CAS:Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM).Formula:C19H23ClFN3OPurity:99.95%Color and Shape:SolidMolecular weight:363.86ASP-8497
CAS:ASP8497 is a potent DPP-IV inhibitor enhancing GLP-1, used for type 2 diabetes and glucose intolerance.Formula:C18H27FN4O7SColor and Shape:SolidMolecular weight:462.49A-1293102
CAS:A-1293102 is a potent, selective inhibitor of BCL-XL, effective in inducing apoptosis in tumor cells reliant on BCL-XL [1].Formula:C42H40F3N7O7S5Color and Shape:SolidMolecular weight:972.13MNK inhibitor 9
CAS:MNK inhibitor 9 potently blocks MNK1/2 (IC50: 0.003 µM each), is cell-permeable, and useful for tumor research.Formula:C25H29N9OColor and Shape:SolidMolecular weight:471.56PDE4-IN-8
CAS:PDE4-IN-8 is a potent PDE4 inhibitor with IC50 0.93 nM for PDE4B2 and minor impact on IL13, IL4, IFNy (IC50: 4.04, 36.33, 2394 nM).Formula:C18H22BNO4Color and Shape:SolidMolecular weight:327.18PPAR agonist 1
CAS:PPAR agonist 1 is an agonist of PPAR α/γ, used for reducing blood glucose, lipid levels, reducing body weight, and lowering cholesterol.Formula:C20H25NO6SPurity:98%Color and Shape:SolidMolecular weight:407.48GLPG0259
CAS:GLPG-0259 is an inhibitor of mitogen-activated protein kinase-activated protein kinase 5 (MAPKAPK5).Formula:C24H28N8O2Color and Shape:SolidMolecular weight:460.53MoTPS1-IN-1
CAS:MoTPS1-IN-1 is a potent MoTPS1 inhibitor with antifungal anti-inflammatory activity that acts through interaction with Glu396 study ulcerative colitis.Formula:C23H27F3N2O4Purity:99.76%Color and Shape:SoildMolecular weight:452.47Fosfluridine tidoxil
CAS:Fosfluridine tidoxil, a thymidylate synthase inhibitor, is used potentially for the treatment of colorectal cancer, and breast cancer.Formula:C34H62FN2O10PSColor and Shape:SolidMolecular weight:740.9SKF 81297
CAS:SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].Formula:C16H16ClNO2Purity:98%Color and Shape:SolidMolecular weight:289.76AY 31906
CAS:AY 31906: High ceiling diuretic, boosts sodium/chloride excretion without affecting potassium, GFR, or renal flow in dogs.Formula:C15H24N6O3SColor and Shape:SolidMolecular weight:368.45Despropylene gatifloxacin
CAS:Despropylene gatifloxacin, a metabolite of AM-1155, exhibits potent antibacterial activity and has favorable pharmacokinetics [1].Formula:C16H18FN3O4Color and Shape:SolidMolecular weight:335.33Sialyllacto-N-tetraose b
CAS:Sialyllacto-N-tetraose b, a sialylated oligosaccharide, naturally occurs in mammalian milk [1].Formula:C37H62N2O29Color and Shape:SolidMolecular weight:998.88Val-Cit-PAB-MMAF
CAS:Val-Cit-PAB-MMAF is an agent-linker conjugate utilized for antibody-drug conjugates (ADCs), consisting of the peptide linker Val-Cit-PAB and the potent tubulinFormula:C58H92N10O13Color and Shape:SolidMolecular weight:1137.41FEN1-IN-5
CAS:FEN1-IN-5 (compound 12A) is a potent Flap endonuclease-1 (FEN1) inhibitor with an IC50 value of 12 nM, playing a role in DNA repair mechanisms [1].Formula:C21H17N3O4SPurity:98%Color and Shape:SolidMolecular weight:407.44A-849519
CAS:A-849519 is a reversible MetAP2 inhibitor with anti-angiogenic and anticancer properties, tested against prostate cancer and compared to TNP-470.Formula:C22H25FN2O4SColor and Shape:SolidMolecular weight:432.51LY-426965
CAS:LY-426965 is a selective, potent, orally bioavailable 5-HT1A antagonist.Formula:C28H38N2O2Color and Shape:SolidMolecular weight:434.61ERK1/2 inhibitor 9
CAS:ERK1/2 Inhibitor 9 (Probe 1), a covalent antagonist of ERK1/2, exhibits sub-micromolar efficacy in cellular assays (A375 GI50=0.47 μM) and facilitates theFormula:C31H32ClN7O3Purity:98%Color and Shape:SolidMolecular weight:586.08SIRT-IN-1
CAS:SIRT-IN-1 is a potent SIRT1/2/3 inhibitor(IC50s of 15, 10, 33 μM, respectively).
Formula:C19H27N5O2SPurity:99.29%Color and Shape:SolidMolecular weight:389.52JNJ-37822681 dihydrochloride
CAS:JNJ-37822681 dihydrochloride 是特异性的、有中枢活性的，可快速解离的多巴胺 D2受体拮抗剂，与多巴胺 D2L 受体结合的亲和力适中 (Ki=158 nM)。JNJ-37822681 dihydrochloride 在精神分裂症和躁郁症领域有研究价值。Formula:C17H19Cl2F5N4Purity:99.78%Color and Shape:SolidMolecular weight:445.26N-Methyl Palbociclib
CAS:N-Methyl Palbociclib is an impurity of the orally active selective CDK4 and CDK6 inhibitor Palbociclib (PD 0332991).Formula:C25H31N7O2Purity:98%Color and Shape:SolidMolecular weight:461.56Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurity:99.73%Color and Shape:SolidMolecular weight:555.65CIL62
CAS:CIL62 is a caspase-3/7-independent inducer of cell death. The mechanism of action of CIL62 is Necrostatin-1 dependent cell death [1].Formula:C23H26O5Purity:97.07%Color and Shape:SolidMolecular weight:382.45Ref: TM-T8468
1mg38.00€5mg86.00€1mL*10mM (DMSO)94.00€10mg116.00€25mg222.00€50mg371.00€100mg504.00€200mg675.00€Vatinoxan hydrochloride
CAS:Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.Formula:C20H27ClN4O4SPurity:98%Color and Shape:SolidMolecular weight:454.97N-Acetylanonaine
CAS:N-Acetylanonaine may be used as a substrate for the identification, differentiation, and characterization of aminoacylase(s)/amidohydrolase(s).Formula:C19H17NO3Color and Shape:SolidMolecular weight:307.34MK-7725
CAS:Mk-7725 is an effective selective bombesin receptor subtype 3 agonist for the treatment of obesity.Formula:C25H19F6N5O5SColor and Shape:SolidMolecular weight:615.5RET-IN-5
CAS:RET-IN-5 is a potent inhibitor of RET (IC50: 4.57 nM).Formula:C29H26FN9OColor and Shape:SolidMolecular weight:535.57Pralatrexate, (S)-
CAS:Pralatrexate is a DHFR inhibitor with antineoplastic properties, targeting cells via RFC-1 and blocking folate synthesis.Formula:C23H23N7O5Color and Shape:SolidMolecular weight:477.47Dezapelisib
CAS:Dezapelisib, an oral delta PI3K inhibitor, blocks PIP3 production and PI3K/AKT pathway, hindering tumor cell growth and survival.Formula:C20H16FN7OSColor and Shape:SolidMolecular weight:421.45uPSEM 817 tartrate
CAS:Potent α7L-GlyR & PSAM4-5-HT3 agonist (EC50: 0.3/0.5 nM). Reduces cortical neuron activity; induces contralateral rotation in mice (LED 0.1 mg/kg).Formula:C20H25N3O7Color and Shape:SolidMolecular weight:419.434Vepafestinib
CAS:Vepafestinib is a RET inhibitor with potential antineoplastic activity[1].Formula:C26H30N6O3Purity:98.56%Color and Shape:SolidMolecular weight:474.55RXFP1 receptor agonist-8
CAS:Example 2 (RXFP1 receptor agonist-8) is a potent RXFP1 receptor agonist that suppresses cAMP production in HEK293 cells expressing human RXFP1, exhibiting anFormula:C40H36F5N3O7Color and Shape:SolidMolecular weight:765.72Deacetylanisomycin
CAS:Deacetylanisomycin is a potent growth regulator in plants Anisomycin and protein synthesis inhibitor. It is an inactive derivative of Anisomycin.Formula:C12H17NO3Purity:98%Color and Shape:SolidMolecular weight:223.27ROCK2-IN-2
CAS:ROCK2-IN-2 is a selective inhibitor of ROCK2 (IC50 of <1 μM).Formula:C18H12N6OSPurity:99.65%Color and Shape:SolidMolecular weight:360.39Ref: TM-T12747
1mg50.00€5mg111.00€1mL*10mM (DMSO)136.00€10mg177.00€25mg304.00€50mg447.00€100mg692.00€200mg888.00€Lin281632
CAS:Lin281632 is an inhibitor of RNA binding protein Lin28 and bromodomain. Lin281632 promotes mESC differentiation.Formula:C15H15N5OPurity:99.84%Color and Shape:SolidMolecular weight:281.31Ref: TM-T27835
1mg34.00€5mg71.00€1mL*10mM (DMSO)79.00€10mg101.00€25mg212.00€50mg340.00€100mg535.00€500mg1,144.00€Cholesterol 24-hydroxylase-IN-2
CAS:Cholesterol 24-hydroxylase-IN-2 is a potent inhibitor of cholesterol 24-hydroxylase (CH24H or CYP46A1), exhibiting an IC50 value of 5.4 nM, and has potentialFormula:C20H23FN4OColor and Shape:SolidMolecular weight:354.422-MT-63
CAS:2-MT 63: Novel, selective TIE-2 kinase inhibitor with >30-fold specificity over other angiogenesis-related kinases like KDR, PDGFR, EPHB4.Formula:C29H30F4N8O2Color and Shape:SolidMolecular weight:598.59
