Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,855 products)
- Apoptosis(6,375 products)
- Cell Cycle/Checkpoint(4,911 products)
- Chromatin/Epigenetics(2,633 products)
- Cytoskeletal Signaling(1,588 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,054 products)
- Immunology and Inflammation(3,954 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,157 products)
- Microbiology/Virology(7,674 products)
- Neuroscience(10,550 products)
- Other Inhibitors(35,862 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,438 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,992 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66512 products of "Inhibitors"
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Ragaglitazar
CAS:Ragaglitazar(NNC-61-0029) is a potent dual activator of PPARγ and PPARα.Cost-effective and quality-assured.Formula:C25H25NO5Purity:97.46% - 98.56%Color and Shape:SolidMolecular weight:419.47LNA-Adenosine
CAS:LNA-Adenosine (LNA-A) is a nucleoside analogue that acts as a ligand for adenosine A3 receptors.Formula:C11H13N5O4Purity:99.15%Color and Shape:SolidMolecular weight:279.25JHU395
CAS:JHU395, an oral prodrug of glutamine antagonist DON, shows stable antitumor effects on MPNST in vitro and vivo.Formula:C22H29N3O7Purity:99.26% - 99.57%Color and Shape:SolidMolecular weight:447.48CCT129202
CAS:CCT129202 is an ATP-competitive pan-Aurora inhibitor for Aurora A, Aurora B and Aurora C with IC50 of 0.042 μM, 0.198 μM and 0.227 μM, respectively.Formula:C23H25ClN8OSPurity:98.14%Color and Shape:SolidMolecular weight:497.02p-Ethynylphenylalanine
CAS:p-Ethynylphenylalanine (4-Ethynyl-L-phenylalanine), a tryptophan hydroxylase (TPH) inhibitor, is competitive, effective, selective, and reversible, with a Ki ofFormula:C11H11NO2Purity:99.44%Color and Shape:SolidMolecular weight:189.21TZ3O
CAS:TZ3O is an anticholinergic compound with neuroprotective activity.TZ3O ameliorates memory impairment in Scopolamine-induced Alzheimer's type model in rats.Formula:C18H13NO4SPurity:99.84%Color and Shape:SolidMolecular weight:339.37Ertugliflozin L-pyroglutamic acid
CAS:Ertugliflozin is a potent oral hSGLT2 inhibitor (IC50: 0.877 nM) for type 2 diabetes treatment studies.Formula:C27H32ClNO10Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:566Ref: TM-T15244
5mg44.00€1mL*10mM (DMSO)50.00€10mg57.00€25mg85.00€50mg90.00€100mg133.00€200mg188.00€500mg323.00€NSC697923
CAS:NSC-697923 inhibits UBE2N, triggers p53-dependent and JNK-mediated apoptosis, blocks DNA damage and NF-κB signaling in neuroblastoma cells.Formula:C11H9NO5SPurity:97% - 99.84%Color and Shape:SolidMolecular weight:267.26Rislenemdaz
CAS:Rislenemdaz (CERC-301) (CERC-301) is an antagonist of the N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B).Formula:C19H23FN4O2Purity:98.50%Color and Shape:SolidMolecular weight:358.41Ref: TM-T12733
1mg62.00€5mg170.00€1mL*10mM (DMSO)187.00€10mg269.00€25mg447.00€50mg622.00€100mg837.00€200mg1,125.00€VH032
CAS:VH032 is a VHL/HIF-1α inhibitor and PROTAC precursor targeting VHL for ubiquitination.Formula:C24H32N4O4SPurity:99.72%Color and Shape:SolidMolecular weight:472.6CFTR corrector 4
CAS:Potent, oral CFTR corrector 4 targets cystic fibrosis, increasing cell surface CFTR levels.Formula:C29H27F2NO7Purity:99.32%Color and Shape:SolidMolecular weight:539.52Ref: TM-T10776
1mg71.00€5mg166.00€1mL*10mM (DMSO)192.00€10mg250.00€25mg507.00€50mg713.00€100mg1,018.00€500mg2,035.00€RO5263397
CAS:RO5263397: TAAR1 agonist, orally active, studied as antidepressant, COX-2 inhibitor.Formula:C10H11FN2OPurity:98.58%Color and Shape:SolidMolecular weight:194.21Inolitazone
CAS:Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.Formula:C27H26N4O4SPurity:99.41% - 99.53%Color and Shape:SolidMolecular weight:502.58Ref: TM-T15581
500mgTo inquire1mg70.00€5mg149.00€1mL*10mM (DMSO)178.00€10mg230.00€25mg374.00€50mg532.00€100mg713.00€Rilapladib
CAS:Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activatingFormula:C40H38F5N3O3SPurity:99.92%Color and Shape:SolidMolecular weight:735.8Ref: TM-T16751
1mg87.00€5mg215.00€10mg349.00€1mL*10mM (DMSO)349.00€25mg537.00€50mg745.00€100mg1,108.00€200mg1,504.00€RH01386
CAS:RH01386, a small molecule, prevents ER stress in β cells, inhibits proapoptotic genes, and may treat type 2 diabetes by restoring insulin secretion.Formula:C18H15F3N4O3SPurity:99.16% - 99.67%Color and Shape:SolidMolecular weight:424.4Ref: TM-T13867
1mg66.00€2mg94.00€1mL*10mM (DMSO)128.00€5mg138.00€10mg197.00€25mg319.00€50mg429.00€100mg587.00€200mg795.00€(R)-Simurosertib
CAS:(R)-Simurosertib ((R)-TAK-931) is an inhibitor of the ATP-competitive cell division cycle 7 (CDC7) kinase.Formula:C17H19N5OSPurity:99.89%Color and Shape:SolidMolecular weight:341.43Nrf2-IN-3
CAS:Nrf2-IN-3 is an NRF2 inhibitor that selectively sensitizes xenografts of mouse mKEAP1 cancer cells to cisplatin.Formula:C22H26N4O4SPurity:98.07%Color and Shape:SolidMolecular weight:442.53Ref: TM-T78841
1mg58.00€5mg126.00€1mL*10mM (DMSO)138.00€10mg197.00€25mg371.00€50mg512.00€100mg707.00€200mg1,018.00€IACS-52825
CAS:IACS-52825 is a DLK inhibitor that reverses para-mechanical aberrant pain in a CIPN mouse model and can be used to study neurological disorders.Formula:C16H13F7N4O2Purity:99.77%Color and Shape:SolidMolecular weight:426.29(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Formula:C12H19NO3Purity:99.73%Color and Shape:SolidMolecular weight:225.28Aneratrigine hydrochloride
CAS:Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.Formula:C19H21Cl2F2N5O2S2Purity:98.37% - 99.16%Color and Shape:SolidMolecular weight:524.43Varespladib methyl
CAS:Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.Formula:C22H22N2O5Purity:99.42% - 99.97%Color and Shape:SolidMolecular weight:394.42Ref: TM-T17218
1mg93.00€2mg123.00€5mg200.00€1mL*10mM (DMSO)220.00€10mg319.00€25mg528.00€50mg730.00€100mg999.00€200mg1,333.00€KSQ-4279
CAS:KSQ-4279 (USP1-IN-1) is an inhibitor of USP1 and PARP.KSQ-4279 has anticancer activity and is used in the study of non-small cell lung cancer, osteosarcoma,Formula:C27H25F3N8OPurity:99.76% - 99.79%Color and Shape:SoildMolecular weight:534.54Zongertinib
CAS:Zongertinib is a human HER2-selective tyrosine kinase inhibitor, a novel TK that is highly selective for covalent binding to the HER2 tyrosine kinase domain (Formula:C29H29N9O2Purity:98.24%Color and Shape:SolidMolecular weight:535.6Ref: TM-T69534
1mg66.00€5mg145.00€1mL*10mM (DMSO)170.00€10mg222.00€25mg371.00€50mg522.00€100mg708.00€CDDO-3P-Im
CAS:CDDO-3P-Im is an orally active inhibitor of necroptosis with chemopreventive effects. CDDO-3P-Im can be used in studies about ischemia/reperfusion.Formula:C39H46N4O3Purity:97.72%Color and Shape:SolidMolecular weight:618.81Ref: TM-T13603
1mg92.00€5mg178.00€1mL*10mM (DMSO)250.00€10mg295.00€25mg502.00€50mg710.00€100mg1,009.00€200mg1,333.00€Calindol hydrochloride
CAS:Calindol (hydrochloride) is a positive allosteric modulator (PAM) of calcimimetic calcium-sensing receptor (CaSR) with an EC50 of 132 nM.Formula:C21H21ClN2Purity:99.47%Color and Shape:SolidMolecular weight:336.86Cdk1/2 Inhibitor III
CAS:Cdk1/2 Inhibitor III is a selective Cdk1/2 inhibitor with an IC50 value of 2.1 μM against CDK1/cyclin B.Formula:C15H13F2N7O2S2Purity:99.92%Color and Shape:SolidMolecular weight:425.44Ecopladib
CAS:Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) & 0.11 μM (rat blood).Formula:C39H33Cl3N2O5SPurity:95.15%Color and Shape:SolidMolecular weight:748.11Ref: TM-T11149
1mL*10mM (DMSO)To inquire1mg315.00€5mg630.00€10mg850.00€25mg1,234.00€50mg1,693.00€100mg2,305.00€AMG-0347
CAS:AMG-0347 inhibits TRPA1 ion channels in sensory neurons, blocking pain perception.Formula:C24H26F3N3O2Purity:99.93%Color and Shape:SolidMolecular weight:445.48Ref: TM-T29968
1mg215.00€5mg523.00€1mL*10mM (DMSO)537.00€10mg695.00€25mg1,054.00€50mg1,414.00€100mg1,900.00€200mg2,565.00€GI 181771
CAS:GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.Formula:C34H31N5O6Purity:95.02%Color and Shape:SolidMolecular weight:605.64Osemozotan HCl
CAS:Osemozotan is a 5-HT1A receptor agonist potentially for the treatment of generalized anxiety disorder.Formula:C19H22ClNO5Purity:98.87% - 99.63%Color and Shape:SolidMolecular weight:379.84Rheb inhibitor NR1
CAS:Rheb inhibitor NR1 is a Rheb inhibitor and selective mTORC1 inhibitor that promotes phosphorylation of S473pAKT.Formula:C25H19BrCl2N2O3SPurity:99.72%Color and Shape:SolidMolecular weight:578.3Ref: TM-T16741
1mL*10mM (DMSO)44.00€1mg87.00€5mg178.00€10mg295.00€25mg595.00€50mg895.00€100mg1,513.00€Maralixibat Chloride
CAS:Maralixibat Chloride (LUM001 chloride), an apical, sodium-dependent, bile acid transport inhibitor, prevents enterohepatic bile acid recirculation.Formula:C40H56ClN3O4SPurity:99.65% - 99.99%Color and Shape:SolidMolecular weight:710.41γ-Secretase-IN-1
CAS:γ-Secretase-IN-1 is a γ-secretase inhibitor that displays partial antiproliferative activity against T-47D cells.Formula:C27H24F2N4O3Purity:99.56%Color and Shape:SolidMolecular weight:490.5Ref: TM-T3521
1mg120.00€5mg385.00€1mL*10mM (DMSO)416.00€10mg618.00€25mg1,224.00€50mg1,648.00€100mg2,232.00€GW 833972A
CAS:GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.
Formula:C18H14Cl2F3N5OPurity:99.93%Color and Shape:SoildMolecular weight:444.24hRIO2 kinase ligand-1
CAS:hRIO2 kinase ligand-1 is a potent ligand for hRIO2 kinase (Kd: 520 nM).Formula:C17H14N2OPurity:99.89%Color and Shape:SolidMolecular weight:262.31PA452
CAS:PA452 is a selective antagonist of retinoic X receptor (RXR) and suppresses the effect of Retinoic acid on Th1/Th2 development.Formula:C26H37N3O3Purity:97.14%Color and Shape:SolidMolecular weight:439.59Ref: TM-T16425
1mg87.00€5mg236.00€1mL*10mM (DMSO)259.00€10mg380.00€25mg622.00€50mg888.00€100mg1,215.00€IMP-1710
CAS:IMP-1710 is a selective UCH-L1 inhibitor with an IC50 value of 38 nM in a fluorescence polarization assay.[1]Cost-effective and quality-assured.Formula:C23H19N5OPurity:99.3%Color and Shape:SolidMolecular weight:381.43AMPA receptor antagonist-3
CAS:AMPA receptor antagonist-3 is an AMPA receptor antagonist.Formula:C20H19N5O2SPurity:99.79%Color and Shape:SolidMolecular weight:393.46Ref: TM-T61813
1mg185.00€5mg425.00€1mL*10mM (DMSO)455.00€10mg625.00€25mg938.00€50mg1,311.00€100mg1,795.00€LB42708
CAS:LB42708 is an orally active farnesyltransferase (FTase) inhibitor (IC50: 0.8/1.2/2.0 nM toward H/N/K-ras).Formula:C30H27BrN4O2Purity:99.36%Color and Shape:SolidMolecular weight:555.47TAK-020
CAS:TAK-020 is a potent covalent inhibitor of Btk with potential antitumor activity for the study of rheumatoid arthritis and immune-related diseases.Formula:C18H17N5O3Purity:98.66%Color and Shape:SolidMolecular weight:351.36Ref: TM-T9529
1mg138.00€5mg334.00€1mL*10mM (DMSO)358.00€10mg597.00€25mg1,234.00€50mg1,908.00€100mg2,952.00€OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purity:99.79%Color and Shape:SolidMolecular weight:421.58Ref: TM-T13804
1mg177.00€5mg432.00€1mL*10mM (DMSO)537.00€10mg587.00€25mg892.00€50mg1,198.00€100mg1,575.00€200mg2,133.00€Kras4B G12D-IN-1
CAS:Kras4B G12D-IN-1 is an inhibitor of Kras4B G12D with anticancer activity.Kras4B G12D-IN-1 inhibits Kras protein expression.Formula:C16H21ClN2O4SPurity:99.75%Color and Shape:SolidMolecular weight:372.87Ref: TM-T78170
2mg93.00€5mg144.00€1mL*10mM (DMSO)161.00€10mg230.00€25mg467.00€50mg745.00€100mg1,134.00€500mg2,277.00€GSK3186899
CAS:GSK3186899 is an inhibitor of Cdc2-related kinase 12 with an EC50 of 1.4 μM for L. donovani.Formula:C19H28F3N7O3SPurity:98.35% - 99.61%Color and Shape:SolidMolecular weight:491.53ZNL 02-096
CAS:ZNL 02-096 (Pomalidomide-C3-adavosertib) is a rapid and selective degrader of Wee1 (IC50=3.58 nM).ZNL 02-096 selectively degrades Wee1 at submolarFormula:C42H45N11O6Purity:98.2% - 99.84%Color and Shape:SolidMolecular weight:799.88Piflufolastat
CAS:Piflufolastat (DCFPYL) is a PET imaging agent for prostate cancer PSMA.Formula:C18H23FN4O8Purity:99.95%Color and Shape:SolidMolecular weight:442.4Ref: TM-T31224
1mg54.00€5mg114.00€1mL*10mM (DMSO)138.00€10mg178.00€25mg409.00€50mg708.00€100mg1,224.00€Nothofagin
CAS:Nothofagin: Antioxidant, anti-inflammatory, prevents clotting, inhibits leukocyte activity, may treat vascular inflammation.Formula:C21H24O10Purity:98.51%Color and Shape:SolidMolecular weight:436.41Ref: TM-TN1996
1mg264.00€5mg587.00€1mL*10mM (DMSO)665.00€10mg800.00€25mg1,198.00€50mg1,575.00€100mg2,142.00€Terbufibrol
CAS:Terbufibrol reduces the levels of serum total cholesterol in normal and hypercholesterolemic male rats.Formula:C20H24O5Purity:98.345%Color and Shape:SolidMolecular weight:344.4Ref: TM-T13919
1mg82.00€5mg178.00€1mL*10mM (DMSO)197.00€10mg285.00€25mg494.00€50mg665.00€100mg900.00€200mg1,215.00€MK-0674
CAS:MK-0674 is a cathepsin K inhibitor (IC50: 0.4 nM) that inhibits Cat B, Cat F, Cat L, and Cat S for metabolism-related diseases.Formula:C26H27F6N3O2Purity:97.3% - 99.91%Color and Shape:SolidMolecular weight:527.5Fluspirilene
CAS:Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).Formula:C29H31F2N3OPurity:99.59%Color and Shape:SolidMolecular weight:475.57SMN-C3
CAS:SMN-C3 (MV8T2MCK57) is an orally active modulator of SMN2 splicing, and has the potential to treat spinal muscular atrophy (SMA).Formula:C24H28N6OPurity:99.01% - 99.05%Color and Shape:SolidMolecular weight:416.52
