Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,849 products)
- Apoptosis(6,366 products)
- Cell Cycle/Checkpoint(4,907 products)
- Chromatin/Epigenetics(2,624 products)
- Cytoskeletal Signaling(1,585 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,759 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,051 products)
- Immunology and Inflammation(3,945 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,162 products)
- Metabolism(10,149 products)
- Microbiology/Virology(7,672 products)
- Neuroscience(10,549 products)
- Other Inhibitors(35,858 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,693 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,743 products)
Show 16 more subcategories
Found 66517 products of "Inhibitors"
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DGAT-1 inhibitor 2
CAS:DGAT-1 inhibitor 2: effective against obesity, targets enzyme in triglyceride synthesis for diabetes treatment.Formula:C24H28N4O3Purity:98.36%Color and Shape:SolidMolecular weight:420.5Ref: TM-T11016
1mg62.00€5mg133.00€1mL*10mM (DMSO)147.00€10mg205.00€25mg378.00€50mg580.00€100mg798.00€TAK-441
CAS:TAK-441: oral Hedgehog signal blocker, potent anticancer, IC50=4.4 nM, reduces Gli1 mRNA & tumor growth.Formula:C28H31F3N4O6Purity:99.82%Color and Shape:SolidMolecular weight:576.56SynuClean-D
CAS:SynuClean-D prevents α-synuclein clumps, breaks fibrils & protects neurons in Parkinson’s models.Formula:C13H5F3N4O5Purity:99.64% - 99.96%Color and Shape:SolidMolecular weight:354.2Ref: TM-T13048
1mg130.00€5mg268.00€1mL*10mM (DMSO)303.00€10mg439.00€25mg777.00€50mg1,108.00€100mg1,485.00€H-1152 dihydrochloride
CAS:H-1152 2HCl: ROCK inhibitor, IC50=12 nM, Ki=1.6 nM. Blocks PKA, PKC, PKG, Aurora A, CaMKII with higher IC50s.Formula:C16H23Cl2N3O2SPurity:99.85%Color and Shape:SolidMolecular weight:392.34Ref: TM-T35328
1mg60.00€5mg135.00€1mL*10mM (DMSO)147.00€10mg215.00€25mg415.00€50mg655.00€100mg888.00€IACS-52825
CAS:IACS-52825 is a DLK inhibitor that reverses para-mechanical aberrant pain in a CIPN mouse model and can be used to study neurological disorders.Formula:C16H13F7N4O2Purity:99.77%Color and Shape:SolidMolecular weight:426.29PARP-1-IN-4
CAS:PARP-1-IN-4 is a potent PARP-1 inhibitor with potential see anti-tumor activity, and inhibition of PARP-1 may be used in cancer development.Formula:C22H15Cl2N3O2Purity:99.82%Color and Shape:SolidMolecular weight:424.28PP5-IN-1
CAS:PP5-IN-1 is a serine/threonine protein phosphatase-5 (PP5) inhibitor with potential anticancer activity that induces apoptosis in cancer cells.Formula:C18H18N2O3SPurity:99.13%Color and Shape:SolidMolecular weight:342.41Salicyl-AMS
CAS:Salicyl-AMS is an inhibitor of mycobacterium auxin biosynthesis that inhibits the growth of mycobacterium in the presence of iron deficiency in vitro.Formula:C17H18N6O8SPurity:98.19%Color and Shape:SolidMolecular weight:466.43Lartesertib
CAS:Lartesertib (ATM Inhibitor-5) is an inhibitor of the serine/threonine protein kinase ATM with potential anticancer activity and can be used to study lung cancerFormula:C23H21FN6O3Purity:99.9%Color and Shape:SolidMolecular weight:448.45Ref: TM-T62684
1mg123.00€2mg177.00€5mg295.00€1mL*10mM (DMSO)326.00€10mg505.00€25mg982.00€50mg1,639.00€100mg2,538.00€UCL-TRO-1938
CAS:UCL-TRO-1938 is a subtype-selective PI3Kα allosteric activator with cardioprotective and neuroregenerative effects.Formula:C27H32N6OPurity:99.95%Color and Shape:SolidMolecular weight:456.58Ref: TM-T78092
5mg114.00€1mL*10mM (DMSO)114.00€10mg177.00€25mg371.00€50mg595.00€100mg954.00€200mg1,279.00€Holomycin
CAS:Holomycin, a dithiopyrrolidone antibiotic, promotes S2753 biofilm formation and has broad-spectrum antibacterial and antitumor properties.
Formula:C7H6N2O2S2Purity:98.76%Color and Shape:SoildMolecular weight:214.26SAG 21k
CAS:SAG 21k is an orally bioactive and potent Hedgehog signaling activator that crosses the blood-brain barrier for the study of cartilage regeneration.Formula:C29H28ClF2N3O2SPurity:99.51%Color and Shape:SolidMolecular weight:556.07AZ PFKFB3 26
CAS:AZ PFKFB3 26 is an effective and selective PFKFB3 inhibitor with an IC50 of 23 nM. The IC50s for PFKFB1 and PFKFB2 are 2.06 and 0.384 μM, respectively.Formula:C24H26N4O2Purity:99.85%Color and Shape:SolidMolecular weight:402.49Fluspirilene
CAS:Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).Formula:C29H31F2N3OPurity:99.59%Color and Shape:SolidMolecular weight:475.57MB-07811
CAS:MB-07811 (VK-2809) is an orally active HepDirect prodrug of MB07344 with cholesterol and triglycerides lowering activity.Formula:C28H32ClO5PPurity:99.74% - 99.94%Color and Shape:SolidMolecular weight:514.98LNA-Adenosine
CAS:LNA-Adenosine (LNA-A) is a nucleoside analogue that acts as a ligand for adenosine A3 receptors.Formula:C11H13N5O4Purity:99.15%Color and Shape:SolidMolecular weight:279.25CXCR2-IN-1
CAS:CXCR2-IN-1 has a pIC50 of 9.3 and is a CXCR2 antagonist of the central nervous system penetration agent.Formula:C19H20Cl2FN3O4SPurity:99.89%Color and Shape:SolidMolecular weight:476.35C004019
CAS:C004019 is a small molecule PROTAC capable of targeting tau for selective protein degradation from the cell, while recruiting tau and E3 ligase (Vhl) for
Formula:C49H70N12O9S2Purity:99.89%Color and Shape:SoildMolecular weight:1035.29CCR3 antagonist 1
CAS:CCR3 antagonist 1 is a potent CCR3 antagonist, used for the research of inflammatory and immunologic diseases.Formula:C19H21Cl2N3O4S2Purity:98.28%Color and Shape:SolidMolecular weight:490.42Ref: TM-T10156
1mg96.00€5mg178.00€1mL*10mM (DMSO)212.00€10mg289.00€25mg462.00€50mg622.00€100mg837.00€Leritrelvir
CAS:Dermatan sulphate sodium (Chondroitin sulfate B sodium salt) is a linear sulfated polysaccharide, a glycosaminoglycan component of important proteoglycans.Formula:C31H44F3N5O6Purity:97.42%Color and Shape:SolidMolecular weight:639.71EGFR/ErbB-2 inhibitor-1
CAS:EGFR/ErbB-2 inhibitor-1 is a selective ErbB2/HER2 inhibitor that effectively blocks ErbB2 and HER2 signaling.Formula:C23H15ClFN3OS2Purity:98.93%Color and Shape:SolidMolecular weight:467.97ABR-238901
CAS:ABR-238901 is an oral, active S100A8/A9 blocker that inhibits the interaction of S100A8/A9 with its receptors RAGE(receptor for advanced glycation end productsFormula:C11H9BrClN3O4SPurity:98.71% - 99.04%Color and Shape:SolidMolecular weight:394.63Ref: TM-T39115
1mg116.00€5mg281.00€1mL*10mM (DMSO)310.00€10mg447.00€25mg710.00€50mg973.00€100mg1,333.00€Enerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Formula:C22H30N4O3Purity:99.7%Color and Shape:SoildMolecular weight:398.50Ref: TM-T67828
1mg49.00€2mg67.00€5mg102.00€1mL*10mM (DMSO)111.00€10mg166.00€25mg339.00€50mg439.00€100mg610.00€200mg827.00€PAOPA
CAS:dopamine D2 receptor modulatorFormula:C11H18N4O3Purity:>99.99%Color and Shape:SolidMolecular weight:254.29Aderamastat
CAS:Aderamastat (FP-025) is an orally active matrix metalloproteinase 12 (MMP-12) inhibitor indicated for the study of allergic asthma, COPD and pulmonary fibrosis.Formula:C21H18N2O4SPurity:99.35%Color and Shape:SolidMolecular weight:394.44BI-3231
CAS:BI-3231 is a hydroxysteroid 17ß-dehydrogenase 13 HSD17B13 inhibitor that inhibits hHSD17B13 .BI-3231 can be used to study cirrhosis.Formula:C16H14F2N4O3SPurity:98.2%Color and Shape:SolidMolecular weight:380.37Ref: TM-T73446
1mg69.00€5mg147.00€1mL*10mM (DMSO)164.00€10mg224.00€25mg358.00€50mg512.00€100mg707.00€200mg982.00€HS94
CAS:HS94 (DAPK3 inhibitor HS94) is a selective and potent DAPK3 inhibitor with a Ki value of 126 nM for Pim kinase inhibition and can be used to study hypertension.
Formula:C15H15N5O2SPurity:95.04%Color and Shape:SolidMolecular weight:329.38Giredestrant tartrate
CAS:Giredestrant tartrate: a new oral, selective non-steroidal ER antagonist, inhibits ER-mediated gene activation and degrades ER protein, treating tumors.Formula:C31H37F5N4O7Purity:97.01%Color and Shape:SolidMolecular weight:672.64ML400
CAS:ML400 (CID73050863) is an allosteric inhibitor of LMPTP with an EC50 of 1μM. ML400 displays good cell-based activity and rodent pharmacokinetics.Formula:C24H29N3OPurity:99.95%Color and Shape:SolidMolecular weight:375.51Ref: TM-T25824
1mg92.00€5mg172.00€1mL*10mM (DMSO)222.00€10mg281.00€25mg447.00€50mg618.00€100mg853.00€500mg1,701.00€TP-10
CAS:TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.Formula:C26H19F3N4OPurity:99.21%Color and Shape:SolidMolecular weight:460.45Ref: TM-T13189
1mg87.00€2mg114.00€5mg177.00€1mL*10mM (DMSO)178.00€10mg264.00€25mg460.00€50mg668.00€100mg945.00€500mg1,783.00€Aneratrigine hydrochloride
CAS:Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.Formula:C19H21Cl2F2N5O2S2Purity:98.37% - 99.16%Color and Shape:SolidMolecular weight:524.43NEP-IN-1
CAS:NEP-IN-1 is an inhibitor of neutral endopeptidase (NEP, IC50 = 2 nM) and can be used in studies about female sexual arousal disorders.Formula:C21H30ClNO4Purity:99.69%Color and Shape:SolidMolecular weight:395.92HIF-2α agonist 2
CAS:HIF-2α agonist 2 is an HIF-2α agonist with an EC50 value of 1.68 μM for HIF-2α.Formula:C13H8Br2N2O2SPurity:98.87%Color and Shape:SoildMolecular weight:416.09OGT 2115
CAS:OGT 2115 blocks heparanase (IC50=0.4µM), cleaving heparan sulfate; antiangiogenic (IC50=1µM).Formula:C24H16BrFN2O4Purity:97.27%Color and Shape:SolidMolecular weight:495.3PDDC inhibitor
CAS:PDDC inhibitor (Phenyl (R)-(1-(3-(3,4-dimethoxyphenyl)-2,6-dimethylimidazo[1,2-b]pyridazin-8-yl)pyrrolidin-3-yl)carbamate) is an nSMase2 inhibitor.Formula:C27H29N5O4Purity:96.09% - 99.39%Color and Shape:SolidMolecular weight:487.55DuP-697
CAS:DuP-697 is an irreversible, specific COX-2 inhibitor with IC50 values of 10 nM and 800 nM for human COX-2 and COX-1.Cost-effective and quality-assured.Formula:C17H12BrFO2S2Purity:99.92%Color and Shape:SolidMolecular weight:411.31Ref: TM-T15181
1mg50.00€5mg99.00€1mL*10mM (DMSO)117.00€10mg145.00€25mg235.00€50mg350.00€100mg515.00€200mg732.00€Piflufolastat
CAS:Piflufolastat (DCFPYL) is a PET imaging agent for prostate cancer PSMA.Formula:C18H23FN4O8Purity:99.95%Color and Shape:SolidMolecular weight:442.4Ref: TM-T31224
1mg54.00€5mg114.00€1mL*10mM (DMSO)138.00€10mg178.00€25mg409.00€50mg708.00€100mg1,224.00€Zidesamtinib
CAS:Zidesamtinib (NVL-520) is a ROS1 fusion and resistance mutation inhibitor that inhibits ROS1 and can be used to study non-small cell lung cancer.Formula:C22H22FN7OPurity:99.74%Color and Shape:SolidMolecular weight:419.455Ref: TM-T72953
1mg71.00€5mg152.00€1mL*10mM (DMSO)167.00€10mg236.00€25mg480.00€50mg767.00€100mg1,224.00€200mg1,648.00€CE-224535
CAS:CE-224535 (PF-04905428) is a selective antagonist of P2X7 receptor. CE-224535 can be used in disease-modifying antirheumatic studies.Formula:C22H29ClN4O6Purity:99.68%Color and Shape:SolidMolecular weight:480.94Ref: TM-T14920
1mg110.00€1mL*10mM (DMSO)222.00€5mg268.00€10mg378.00€25mg612.00€50mg858.00€100mg1,153.00€200mg1,558.00€γ-Secretase-IN-1
CAS:γ-Secretase-IN-1 is a γ-secretase inhibitor that displays partial antiproliferative activity against T-47D cells.Formula:C27H24F2N4O3Purity:99.56%Color and Shape:SolidMolecular weight:490.5Ref: TM-T3521
1mg120.00€5mg385.00€1mL*10mM (DMSO)416.00€10mg618.00€25mg1,224.00€50mg1,648.00€100mg2,232.00€INT-777
CAS:INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM.Formula:C27H46O5Purity:99.78%Color and Shape:SolidMolecular weight:450.65Ref: TM-T11662L
1mg130.00€5mg313.00€1mL*10mM (DMSO)343.00€10mg447.00€25mg715.00€50mg999.00€100mg1,395.00€Phos-tag Acrylamide AAL-107
CAS:Phos-tag Acrylamide AAL-107 is a polyacrylamide-conjugated phosphate-binding tag,visualizing phosphorylated proteins. High-Quality, Low-Cost!Formula:C33H38N8O3Purity:99.86% - >99.99%Color and Shape:SoildMolecular weight:594.71A7132
CAS:A7132 is an antibacterial agent and possesses broad and potent antibacterial activity.Formula:C19H16F2N4O3Purity:96.64%Color and Shape:SolidMolecular weight:386.35Inolitazone
CAS:Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.Formula:C27H26N4O4SPurity:99.41% - 99.53%Color and Shape:SolidMolecular weight:502.58Ref: TM-T15581
500mgTo inquire1mg70.00€5mg149.00€1mL*10mM (DMSO)178.00€10mg230.00€25mg374.00€50mg532.00€100mg713.00€AVP-13358
CAS:AVP-13358: a CD23/IgE inhibitor for treating immune, infection, and ENT disorders.Formula:C30H29N5O2Purity:98.45%Color and Shape:SolidMolecular weight:491.58MK-2461
CAS:MK-2461 is a novel inhibitor that targets multiple proteins and competitively binds to ATP sites, specifically inhibiting the activated c-Met protein with anFormula:C24H25N5O5SPurity:95.41% - 99.67%Color and Shape:SolidMolecular weight:495.55Ref: TM-T6094
1mg50.00€5mg114.00€1mL*10mM (DMSO)127.00€10mg177.00€25mg344.00€50mg523.00€100mg798.00€200mg1,071.00€CFI-402257
CAS:CFI-402257 is a selective inhibitor of Mps1/TTK kinase (Mps1 Ki = 0.09 nM; EC50 = 6.5 nM)and can be used in studies about hepatocellular carcinoma diseases.Formula:C28H30N6O3Purity:96.66% - 99.51%Color and Shape:SolidMolecular weight:498.58FHT-1015
CAS:FHT-1205 is a potent inhibitor (IC50 ≤ 10 nM) of SMARCA4/SMARCA2 ATPase (BRG1 and BRM).Formula:C25H25N5O4S3Purity:98.57%Color and Shape:SolidMolecular weight:555.69Ref: TM-T63925
1mg54.00€5mg114.00€1mL*10mM (DMSO)138.00€10mg178.00€25mg356.00€50mg580.00€100mg888.00€Rheb inhibitor NR1
CAS:Rheb inhibitor NR1 is a Rheb inhibitor and selective mTORC1 inhibitor that promotes phosphorylation of S473pAKT.Formula:C25H19BrCl2N2O3SPurity:99.72%Color and Shape:SolidMolecular weight:578.3Ref: TM-T16741
1mL*10mM (DMSO)44.00€1mg87.00€5mg178.00€10mg295.00€25mg595.00€50mg895.00€100mg1,513.00€Dalzanemdor
CAS:Dalzanemdor (SAGE-718) is an NMDA receptor-positive modulator of metabolism that can be used to study Huntington's chorea, Alzheimer's disease, and cognitiveFormula:C27H43F3O2Purity:98.2% - >99.99%Color and Shape:SolidMolecular weight:456.62
