Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,754 products)
- Apoptosis(6,185 products)
- Cell Cycle/Checkpoint(4,805 products)
- Chromatin/Epigenetics(2,573 products)
- Cytoskeletal Signaling(1,502 products)
- DNA Damage/DNA Repair(2,893 products)
- Endocrinology/Hormones(3,702 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,963 products)
- Immunology and Inflammation(3,697 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,246 products)
- Membrane Transporter/Ion Channel(3,136 products)
- Metabolism(10,098 products)
- Microbiology/Virology(7,552 products)
- Neuroscience(10,304 products)
- Other Inhibitors(35,769 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,402 products)
- Proteases/Proteasome(1,670 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,923 products)
- Ubiquitination(1,715 products)
Show 16 more subcategories
Found 66573 products of "Inhibitors"
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GBR-13069 dimethanesulfonate
CAS:GBR-13069 dimethanesulfonate is a dopamine reuptake inhibitor.Formula:C30H38F2N2O7S2Color and Shape:SolidMolecular weight:640.76MAGL-IN-1
CAS:MAGL-IN-1 is a selective and potent monoacylglycerol lipase (MAGL) inhibitor with an IC50 of 80 nM.Formula:C22H24FNO3Purity:98%Color and Shape:SolidMolecular weight:369.43Sovleplenib
CAS:Sovleplenib (HMPL-523), oral SYK inhibitor, IC50 25 nM, targets tumors & ITP studies.Formula:C24H30N6O3SPurity:99.71%Color and Shape:SolidMolecular weight:482.6Ref: TM-T32088
1mg120.00€5mg289.00€10mg434.00€25mg737.00€50mg1,153.00€100mg1,791.00€200mg2,412.00€1mL*10mM (DMSO)308.00€Isoflupredone
CAS:Isoflupredone, a synthetic corticosteroid, inhibits inflammation and immune response in animals.Formula:C21H27FO5Purity:97.62% - 99.85%Color and Shape:SolidMolecular weight:378.43Ref: TM-T41303
1mg63.00€2mg90.00€5mg137.00€10mg235.00€25mg512.00€50mg740.00€100mg1,035.00€1mL*10mM (DMSO)150.00€LH 21
CAS:LH-21, a strong CB1 receptor antagonist, curbs eating and lessens weight gain in obese rats.Formula:C20H20Cl3N3Color and Shape:SolidMolecular weight:408.75Mps-BAY2b
CAS:Mps-BAY2b is a novel MPS1 inhibitor.Formula:C20H23N5OColor and Shape:SolidMolecular weight:349.43CAY10487
CAS:CAY10487 reduces aortic fatty streaks in high-cholesterol rabbits by 37.4% and inhibits LDL oxidation by 75% at 2μM, without altering lipids or ACAT activity.Formula:C13H15NO5Color and Shape:SolidMolecular weight:265.26FRAN-12
CAS:FRAN-12 is a histamine and 5-hydroxytryptamine antagonist with pressor properties.Formula:C19H21ClN4SColor and Shape:SolidMolecular weight:372.91Azalanstat mesylate
CAS:Azalanstat, an anti-obesity drug, inhibits cholesterol synthesis by targeting P450 enzyme lanosterol 14α-demethylase; reduces LDL more than HDL in hamsters.Formula:C23H28ClN3O5S2Color and Shape:SolidMolecular weight:526.063ACPT-I
CAS:Agonist for group III mGlu receptorsFormula:C8H11NO6Purity:98%Color and Shape:SolidMolecular weight:217.18SGK1 inhibitor
CAS:SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.Formula:C17H12Cl2N6O2SColor and Shape:SolidMolecular weight:435.29GSK1482160
CAS:GSK1482160 is a potent and selective P2X7 receptor allosteric modulator.Formula:C14H14ClF3N2O2Purity:98%Color and Shape:SolidMolecular weight:334.72Atuzaginstat
CAS:Atuzaginstat is a bacterial protease lysine gingipain inhibitor.Formula:C19H25F3N2O3Color and Shape:SolidMolecular weight:386.41BPN-15606
CAS:BPN-15606, an oral γ-secretase modulator, reduces Aβ42/Aβ40 with IC50 of 7/17 nM; promising PK/PD, lowers Aβ in rodent CNS.Formula:C23H23FN6OColor and Shape:SolidMolecular weight:418.47GW694481
CAS:GW694481 is a potent ApoA1 upregulator (EC170 = 500 nM).Formula:C21H18N4O2Color and Shape:SolidMolecular weight:358.39HIV-1 inhibitor-24
CAS:HIV-1 inhibitor-24 (S-12a) blocks HIV reverse transcription effectively (IC50: 9.5 nM), low toxicity, well-tolerated in mice, good heart safety.Formula:C26H19N5O2Color and Shape:SolidMolecular weight:433.46BDM14471
CAS:BDM14471 is a selective inhibitor of hydroxamate PfAM1.Formula:C17H15FN2O3Purity:98%Color and Shape:SolidMolecular weight:314.31Muscarine iodide
CAS:Muscarinic acetylcholine receptor agonistFormula:C9H20INO2Purity:98%Color and Shape:SolidMolecular weight:301.17A110
CAS:A110 is a potent and selective IMPDHs inhibitor. It binds to the NAD(+) cofactor site and forms a ternary complex with IMP.Formula:C19H15ClN4O2Purity:98%Color and Shape:SolidMolecular weight:366.8JNK-1-IN-1
CAS:JNK-1-IN-1 is an inhibitor specifically targeting JNK-1, also exhibiting inhibition of MKK7 with an IC50 value of 7.8μM.Formula:C24H22N6SColor and Shape:SolidMolecular weight:426.54DHP-218
CAS:DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) & 66 nmol/L (phenylephrine).Formula:C18H21N2O7PPurity:98%Color and Shape:SolidMolecular weight:408.34NSC 601980
CAS:NSC601980, an antitumor agent, inhibits COLO 205 and HT29 cell growth with Log GI50s of -6.6 and -6.9.Formula:C15H12N4Purity:98%Color and Shape:SolidMolecular weight:248.28PWZ-029
CAS:PWZ-029 is an inverse agonist selective for α₅ GABAA receptors with nootropic effects.Formula:C14H14ClN3O2Color and Shape:SolidMolecular weight:291.73Farnesyl pyrophosphate
CAS:Farnesyl pyrophosphate: 15-C isoprenoid, TRPM2 agonist, crucial for cholesterol, ubiquinones, protein farnesylation, and GGPP synthesis.Formula:C15H28O7P2Color and Shape:SolidMolecular weight:382.33Bucloxic acid
CAS:Bucloxic acid is an anti-inflammatory pyrazole derivative used in the treatment of chronic glomerular nephropathies.Formula:C16H19ClO3Purity:98%Color and Shape:SolidMolecular weight:294.77Ro 24-6392
CAS:Ro 24-6392, an ester co-drug of ciprofloxacin and desacetylcefotaxime, combats various aerobic bacteria.Formula:C31H31FN8O8S2Purity:98%Color and Shape:SolidMolecular weight:726.76Liothyronine HCl
CAS:Liothyronine is a T3 thyroid hormone normally synthesized and secreted by the thyroid gland in much smaller quantities than thyroxine.Formula:C15H13ClI3NO4Purity:98%Color and Shape:SolidMolecular weight:687.43Ketocaine
CAS:Ketocaine（Rec 7-0518） is a local anesthetic commonly used in animal experiments with potential antitumor activity for pain relief.Formula:C18H29NO2Purity:98.59%Color and Shape:SolidMolecular weight:291.43GNF-2-PEG-acid
GNF-2-PEG-acid is usually used as a fluorescent probe.Formula:C26H27F3N4O7Purity:98%Color and Shape:SolidMolecular weight:564.51GU-285
CAS:GU-285 is a potent non-selective adenosine receptor antagonist.Formula:C14H14N6OSColor and Shape:SolidMolecular weight:314.37LWG-301
LWG-301, a GLS1 allosteric inhibitor, IC50 7 nM, impedes glutamine metabolism and prompts apoptosis; shows antitumor effects.Formula:C28H38N8O3SColor and Shape:SolidMolecular weight:566.72Benzathine
CAS:Benzathine, a diamine, stabilizes and prolongs penicillin effects in medications like benzathine benzylpenicillin upon injection.Formula:C16H20N2Purity:98%Color and Shape:SolidMolecular weight:240.34Datelliptium chloride
CAS:Datelliptium chloride is a DNA-intercalating agent derived from ellipticine. Datelliptium chloride shows anti-tumor activities.Formula:C23H28ClN3OPurity:98%Color and Shape:SolidMolecular weight:397.94NS004
CAS:NS004 is a large-conductance K+ channel opener, it inhibits mitochondrial function in glioma cells.Formula:C14H8ClF3N2O2Purity:98%Color and Shape:SolidMolecular weight:328.67Bradanicline HCl
CAS:Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.Formula:C22H24ClN3O2Color and Shape:SolidMolecular weight:397.9Oxydipentonium chloride
CAS:Oxydipentonium chloride is a cholinesterase inhibitor that was studied as a muscle relaxant.Formula:C16H38Cl2N2OColor and Shape:SolidMolecular weight:345.39WK-298
CAS:WK-298 is an effective MDM2/MDMX-p53 interaction inhibitor.Formula:C35H38Cl2N6OPurity:98%Color and Shape:SolidMolecular weight:629.62(R,1R)-Tenofovir amibufenamide
CAS:(R,1R)-Tenofovir amibufenamide ((R,1R)-HS-10234) can be used as a Tenofovir prodrug, which can be taken orally and has antiviral activity.Formula:C22H31N6O5PPurity:98.79% - 99.02%Color and Shape:SolidMolecular weight:490.49Ref: TM-T63290
1mg58.00€5mg133.00€10mg190.00€25mg328.00€50mg442.00€100mg598.00€200mg792.00€1mL*10mM (DMSO)145.00€SUN-C5174
CAS:"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."Formula:C22H29FN4O2Purity:98%Color and Shape:SolidMolecular weight:400.49MRS2395
CAS:MRS2395, a dipivaloyl P2Y12 receptor blocker, inhibits ADP-induced platelet activation with a Ki of 3.6 μM and boosts TRAP-6-triggered dense granule release.Formula:C20H30ClN5O4Color and Shape:SolidMolecular weight:439.94AT2R antagonist 1
CAS:AT2R antagonist 1: potent, selective ligand, Ki 29 nM, inhibits CYP enzymes, stable in liver microsomes.Formula:C23H30N4O4S2Color and Shape:SolidMolecular weight:490.64FPL-64170XX
CAS:FPL-64170XX is a selective inhibitor of the enzyme 5-lipoxygenase.Formula:C19H19N3O2Color and Shape:SolidMolecular weight:321.374-(β-aminoethyl)thiazole
CAS:4-(Beta-aminoethyl)thiazole is a histamine analog which can induce cross-tolerance to histamine.Formula:C5H8N2SColor and Shape:SolidMolecular weight:128.2BLM-IN-1
CAS:BLM-IN-1: BLM inhibitor, KD 1.81 μM, IC50 0.95 μM; causes DNA damage, apoptosis, stops cancer cell growth.Formula:C28H35FN4OColor and Shape:SolidMolecular weight:462.6S 11566
CAS:S 11566 is a selective dopamine D3 receptor antagonist.Formula:C18H27NOColor and Shape:SolidMolecular weight:273.41MDL-105212A HCl
CAS:MDL-105212A HCl is a nonpeptide NK-1 and NK-2 receptor antagonist.Formula:C34H40Cl3N3O5Color and Shape:SolidMolecular weight:677.06Anticancer agent 58
Anticancer agent 58 targets A549/T24 cell lines; IC50: 0.6/0.7 μM. It triggers apoptosis, ups Ca2+/ROS, and lowers mitochondrial potential.Formula:C39H55NO5Color and Shape:SolidMolecular weight:617.86Cetamolol (free base)
CAS:Cetamolol (free base) is a beta adrenergic antagonist, more specifically a β₁-adrenergic blocker.Formula:C16H26N2O4Color and Shape:SolidMolecular weight:310.39LY-393615
CAS:LY-393615 is a neuronal calcium channel blocker.Formula:C21H26ClF2NOColor and Shape:SolidMolecular weight:381.89Metallo-β-lactamase-IN-6
CAS:Metallo-β-lactamase-IN-6 is a highly effective inhibitor of VIM-Type metallo-β-lactamase, demonstrating IC 50 values of 0.56 μM, 29.50 μM, and 5.78 μM for VIM-2Formula:C10H9N3O2Color and Shape:SolidMolecular weight:203.2
