Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5598 produits trouvés pour "Apoptose"
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4-IBP
CAS :<p>4-IBP is a selective σ1 agonist with a high level of affinity for the σ1 receptor (Ki = 1.7 nM) and a moderate affinity for the σ2 receptor (Ki = 25.2 nM) .</p>Formule :C19H21IN2ODegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :420.29Lubiprostone
CAS :<p>Lubiprostone (RU-0211), an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.</p>Formule :C20H32F2O5Degré de pureté :97.31% - 98.54%Couleur et forme :White Odorless Crystals Or Crystalline PowderMasse moléculaire :390.46RH01687
CAS :<p>RH01687 is a potent β-cell protector , exhibits β-cell-protective activities against endoplasmic reticulum (ER) stress.</p>Formule :C12H9ClN6O2SDegré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :336.76Clodronic acid disodium salt
CAS :<p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>Formule :CH4Cl2O6P0·2NaDegré de pureté :>99.99% - ≥98%Couleur et forme :White SolidMasse moléculaire :288.86Sodium benzoate
CAS :<p>Sodium benzoate (Benzoic acid sodium salt) is a D-Amino Acid Oxidase Inhibitor.Sodium Benzoate is a Food Preservative.</p>Formule :C7H5NaO2Degré de pureté :99.72%Couleur et forme :White Solid CrystallineMasse moléculaire :144.10HX 531
CAS :<p>HX 531 is a RXR antagonist (IC50 of 18 nM).Cost-effective and quality-assured.</p>Formule :C29H29N3O4Degré de pureté :98.59% - 99.86%Couleur et forme :SolidMasse moléculaire :483.563-hydroxy-3-phenylpentanamide
CAS :<p>Chiral 3-hydroxy-3-phenylpentanamide: neuroprotective, may treat anxiety/depression/addiction, anticancer.</p>Formule :C11H15NO2Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :193.24Ceftiofur
CAS :<p>Ceftiofur is a semisynthetic antibiotic, with activity against various gram-positive/negative, anaerobic and aerobic bacteria encountered by domestic animals.</p>Formule :C19H17N5O7S3Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :523.56Dantrolene sodium hemiheptahydrate
CAS :<p>Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium</p>Formule :C14H9N4NaO5·5H2ODegré de pureté :99.72%Couleur et forme :Orange PowderMasse moléculaire :399.29GYY4137
CAS :<p>GYY4137 (GYY 4137 morpholine salt) is a novel water-soluble and slow releasing H2S donor with antihypertensive, anti-inflammatory and anticancer activity.</p>Formule :C11H16NO2PS2·C4H9NODegré de pureté :95.54% - 99.97%Couleur et forme :SolidMasse moléculaire :376.47DIM-C-pPhCO2Me
CAS :<p>DIM-C-pPhCO2Me is a nuclear receptor 4A1 (NR4A1) antagonist.</p>Formule :C25H20N2O2Degré de pureté :99.55% - 99.86%Couleur et forme :SolidMasse moléculaire :380.44Desciclovir
CAS :<p>Desciclovir (DCV), a prodrug of the antiherpetic agent acyclovir (ACV), is converted in humans to ACV, presumably by xanthine oxidase.</p>Formule :C8H11N5O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :209.212-HBA
CAS :<p>2-HBA, a synthetic analog of curcumin, is an indirect inducer of enzymes that catalyze detoxification reactions through the Keap1-Nrf2-ARE pathway.</p>Formule :C17H14O3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :266.293,4 Dichloroisocoumarin
CAS :<p>3,4 Dichloroisocoumarin is a granzyme, cathepsin G, and neutrolphil elastase inhibitor</p>Formule :C9H4Cl2O2Degré de pureté :97.94%Couleur et forme :SolidMasse moléculaire :215.03Thalidomide-NH-CH2-COOH TFA
CAS :<p>2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid (trifluoroacetic acid) is mainly used in compounds Synthesis.</p>Formule :C17H14F3N3O8Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :445.3036ILK-IN-2
CAS :<p>ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.</p>Formule :C30H30F3N5ODegré de pureté :99.30%Couleur et forme :SolidMasse moléculaire :533.59BMS202 hydrochloride (1675203-84-5(free base))
CAS :<p>BMS202 hydrochloride (1675203-84-5) is a potent PD-1/PD-L1 inhibitor (IC50: 18 nM) that promotes PD-L1 dimerization, blocking PD1 binding.</p>Formule :C25H30ClN3O3Degré de pureté :98.29% - 99.47%Couleur et forme :SolidMasse moléculaire :455.97Hexamethylene bisacetamide
CAS :<p>Hexamethylene bisacetamide inhibits BET Bromodomain Proteins.</p>Formule :C10H20N2O2Degré de pureté :99.94%Couleur et forme :White FlakesMasse moléculaire :200.28PDL-1 cpd 10
CAS :<p>PDL-1 cpd 10 is a novel small molecule PD-L1 inhititor.</p>Formule :C21H23N5O2Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :377.44Piperacetazine
CAS :<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57(E/Z)-Necrosulfonamide
CAS :<p>(E/Z)-Necrosulfonamide is a novel inhibitor of MLKL.</p>Formule :C18H15N5O6S2Degré de pureté :97.62% - 98%Couleur et forme :SolidMasse moléculaire :461.47OTS964 hydrochloride
CAS :<p>OTS964 hydrochloride (OTS964) is a potent and selective TOPK inhibitor with potential anticancer activity.</p>Formule :C23H24N2O2S·HClDegré de pureté :96.5% - 98.03%Couleur et forme :SolidMasse moléculaire :428.97Z-VAD-FMK
CAS :<p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>Formule :C21H28FN3O7Degré de pureté :98.24% - 99.79%Couleur et forme :SolidMasse moléculaire :453.46PD184161
CAS :<p>PD184161 is a novel, orally-active MEK inhibitor. PD184161 inhibited MEK activity (IC50 = 10-100 nM) in a time- and concentration-dependent manner[1].</p>Formule :C17H13BrClF2IN2O2Degré de pureté :99.40%Couleur et forme :SolidMasse moléculaire :557.56Nocodazole
CAS :<p>Nocodazole: synthetic microtubule polymerization blocker, also impedes Abl with low IC50; binds to beta-tubulin.</p>Formule :C14H11N3O3SDegré de pureté :98% - 99.91%Couleur et forme :Physical Description White Powder (Ntp 1992)Masse moléculaire :301.32Rhapontin
CAS :<p>Rhapontin may reduce liver fat and better blood sugar/lipids, showing potential for treating type 2 diabetes.</p>Formule :C21H24O9Degré de pureté :99% - 99.91%Couleur et forme :Light YellowMasse moléculaire :420.41Perillyl alcohol
CAS :<p>Perillyl Alcohol, a monoterpene with antitumor properties, inhibits protein activation blocking cancer cell growth.</p>Formule :C10H16ODegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :152.23Euscaphic acid
CAS :<p>Euscaphic acid has anti-diabetic and anti-inflammatory effects, blocking IKK/MAPKs and NF-κB activation by disrupting TRAF6/IRAK1/TAK1 clustering.</p>Formule :C30H48O5Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :488.7Licochalcone B
CAS :<p>Licochalcone B inhibits human bladder cancer cells, reduces inflammation by NO, TNFalpha, and MCP-1, and a derivative protects against endotoxin shock.</p>Formule :C16H14O5Degré de pureté :99.33% - 99.93%Couleur et forme :SolidMasse moléculaire :286.28Avelumab
CAS :<p>Avelumab is a fully human IgG1 anti-PD-L1 monoclonal antibody. Avelumab shows potential antibody-dependent cell-mediated cytotoxicity.</p>Degré de pureté :95% - 97.17% (SDS-PAGE)Couleur et forme :LiquidMasse moléculaire :143.8 kDaEvofosfamide
CAS :<p>Evofosfamide (TH-302) is a hypoxia-activated prodrug that releases Br-IPM in tumors to cause DNA damage and potentially induce apoptosis.</p>Formule :C9H16Br2N5O4PDegré de pureté :98.74% - 99.75%Couleur et forme :SolidMasse moléculaire :449.04Buparlisib
CAS :<p>Buparlisib (BKM120) is an orally bioavailable specific oral inhibitor of the pan-class I PI3K (IC50s: 52/166/116/nM for p110α, p110β, and p110δ).</p>Formule :C18H21F3N6O2Degré de pureté :95.32% - 98.45%Couleur et forme :SolidMasse moléculaire :410.39NS-1619
CAS :<p>NS1619 have cardio-protective effects after ischemia-reperfusion injury.</p>Formule :C15H8F6N2O2Degré de pureté :97.66% - 98%Couleur et forme :SolidMasse moléculaire :362.23SSE15206
CAS :<p>SSE15206 is a microtubule polymerization inhibitor that overcomes multidrug resistance.</p>Formule :C19H21N3O3SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :371.45Amsilarotene
CAS :<p>Amsilarotene (TAC101) blocks RB phosphorylation, boosts 2 CDK inhibitors, halts cell cycle, and reduces thymidylate synthase and cyclin A levels.</p>Formule :C20H27NO3Si2Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :385.6Estramustine phosphate sodium
CAS :<p>Estramustine phosphate sodium (Ro 21-8837/001) is an antimicrotubule chemotherapy agent; arrests prostate cancer cells in the G2/M phase of the cell cycle.</p>Formule :C23H30Cl2NNa2O6PDegré de pureté :96.44% - 99.54%Couleur et forme :SolidMasse moléculaire :564.35Rigosertib sodium
CAS :<p>Rigosertib sodium (ON-01910), a non-ATP-competitive inhibitor of PLK1(IC50=9 nM), exhibits 30-fold higher specificity activity over Plk2 and no effect on Plk3.</p>Formule :C21H24NNaO8SDegré de pureté :98% - 99.37%Couleur et forme :SolidMasse moléculaire :473.47Tenovin-1
CAS :<p>Tenovin-1 inhibits protein-deacetylating activities of SirT1 and SirT2 and protects against MDM2-mediated p53 degradation, which involves ubiquitination.</p>Formule :C20H23N3O2SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :369.48SBI-0206965
CAS :<p>SBI-0206965 is a potent, selective and cell-permeable autophagy kinase ULK1 inhibitor with IC50 of 108 nM for ULK1 kinase activity and 711 nM for ULK2.</p>Formule :C21H21BrN4O5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :489.32D-Pantothenic acid hemicalcium salt
CAS :<p>D-Pantothenic acid hemicalcium salt (Calcium pantothenate), a kind of water soluble vitamin, can reduce the patulin content of the apple juice.</p>Formule :C9H17NO5CaDegré de pureté :98% - 99.89%Couleur et forme :White Crystalline PowderMasse moléculaire :239.28AZD1208
CAS :<p>AZD1208 is a novel, orally bioavailable, highly selective PIM kinase inhibitor with single nanomolar potency against all three PIM kinases.</p>Formule :C21H21N3O2SDegré de pureté :97.24% - 99.83%Couleur et forme :SolidMasse moléculaire :379.48Niraparib hydrochloride
CAS :<p>Niraparib hydrochloride (MK-4827) is a PARP inhibitor with potential cancer treatment effects, causing DNA damage and apoptosis.</p>Formule :C19H21ClN4ODegré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :356.85Bullatine A
CAS :<p>1.</p>Formule :C22H33NO2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :343.51Navitoclax
CAS :<p>View and buy Navitoclax from TargetMol.Navitoclax (ABT-263) is a potent, orally bioavailable Bcl-2 family protein inhibitor that avidly binds Bcl-2.Cited in 4 publications.</p>Formule :C47H55ClF3N5O6S3Degré de pureté :95.82% - >99.99%Couleur et forme :Pale Yellow SolidMasse moléculaire :974.61Dihydrokaempferol
CAS :<p>Dihydrokaempferol (Aromadendrin) is a natural product. It induces apoptosis and inhibits Bcl-2 and Bcl-xL expression, possesses anti-inflammatory activity.</p>Formule :C15H12O6Degré de pureté :97.79% - 99.96%Couleur et forme :SolidMasse moléculaire :288.25Prexasertib
CAS :<p>Prexasertib (LY2606368) is a selective checkpoint kinase 1 (CHK1) inhibitor (Ki 0.9 nM, IC50<1 nM). antitumor activity. High-Quality, Low-Cost!</p>Formule :C18H19N7O2Degré de pureté :97.3% - 98.23%Couleur et forme :SolidMasse moléculaire :365.39SC-236
CAS :<p>SC-236 (Sc 236) is an orally active and selective inhibitor of COX-2 (IC50 of 0.005 μM and 17.8 μM for COX-2 and COX-1, respectively).</p>Formule :C16H11ClF3N3O2SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :401.79SNS-032
CAS :<p>SNS-032 (BMS-387032) is a selective inhibitor of CDK2 and is 10- and 20-fold selective over CDK1/CDK4. SNS-032 is sensitive to CDK7/9, and no effect on CDK6.</p>Formule :C17H24N4O2S2Degré de pureté :98.27% - 99.91%Couleur et forme :SolidMasse moléculaire :380.53Quercetin
CAS :<p>Quercetin (Sophoretin) is a natural flavonoid and is an agonist of SIRT1.</p>Formule :C15H10O7Degré de pureté :96.29% - 98.05%Couleur et forme :Sensitive To Exposure To Air And Light Insoluble In Water Alcoholic Solutions Taste Very Bitter (Ntp 1992)Masse moléculaire :302.24SecinH3
CAS :<p>SecinH3 is selective cytohesin inhibitor.</p>Formule :C24H20N4O4SDegré de pureté :97.49% - 99.37%Couleur et forme :SolidMasse moléculaire :460.51EB-3D
CAS :<p>EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.</p>Formule :C30H36Br2N4O2Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :644.4Pogostone
CAS :<p>Pogostone: anti-bacterial/fungal, blocks T-cells, modulates cytokines, protects against gastric ulcers, boosts antioxidants/PGE2/NP-SH.</p>Formule :C12H16O4Degré de pureté :98.46% - 99.03%Couleur et forme :SolidMasse moléculaire :224.25NVP-CGM097
CAS :<p>NVP-CGM097 (CGM097) is an effective and specific MDM2 inhibitor (IC50: 1.7 nM for hMDM2).</p>Formule :C38H47ClN4O4Degré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :659.26NVP-TNKS656
CAS :<p>NVP-TNKS656 (TNKS656) is a highly potent, selective, and orally active TNKS2 inhibitor.</p>Formule :C27H34N4O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :494.58Linifanib
CAS :<p>Linifanib (AL-39324) (ABT-869) is a novel, potent ATP-competitive VEGFR/PDGFR inhibitor for KDR (IC50: 4 nM), CSF-1R (IC50: 3 nM), Flt-1/3 (IC50: 3/4 nM) and</p>Formule :C21H18FN5ODegré de pureté :98% - 98.24%Couleur et forme :SolidMasse moléculaire :375.4DC661
CAS :<p>DC661 is a palmitoyl-protein thioesterase 1 (PPT1) inhibitor that acts as an anti-lysosomal agent by inhibiting autophagy, demonstrating anti-cancer activity.</p>Formule :C31H39Cl2N5Degré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :552.58Cobimetinib
CAS :<p>Cobimetinib (GDC-0973) is a MEK1 inhibitor with selective and oral activity. Cobimetinib exhibits antitumor activity. Cost-effective and quality-assured.</p>Formule :C21H21F3IN3O2Degré de pureté :98% - 99.61%Couleur et forme :SolidMasse moléculaire :531.31GW 5074
CAS :<p>GW 5074 (Raf1 Kinase Inhibitor I)(IC50=9 nM) is an effective and specific c-Raf inhibitor.</p>Formule :C15H8Br2INO2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :520.94Tolcapone
CAS :<p>Tolcapone (Ro 40-7592) is a catechol-O-methyltransferase inhibitor used in the therapy of Parkinson disease as adjunctive therapy in combination with levodopa</p>Formule :C14H11NO5Degré de pureté :98.93% - 99.68%Couleur et forme :SolidMasse moléculaire :273.24Didymin
CAS :<p>Didymin, an antioxidant, may treat neuroblastoma and neurodegeneration by blocking N-Myc and boosting RKIP.</p>Formule :C28H34O14Degré de pureté :99.12% - 99.87%Couleur et forme :Faintly Beige PowderMasse moléculaire :594.56SCR7 pyrazine
CAS :<p>SCR7 pyrazine (SCR7) enhances CRISPR-Cas9-mediated homology-directed repair (HDR) efficiency in vitro up to 19-fold. Inhibits nonhomologous end-joining (NHEJ).</p>Formule :C18H12N4OSDegré de pureté :98.72% - 99.85%Couleur et forme :SolidMasse moléculaire :332.383,6-Dihydroxyflavone
CAS :<p>3,6-Dihydroxyflavone suppresses the epithelial-mesenchymal transition in breast cancer cells by inhibiting the Notch signaling pathway.</p>Formule :C15H10O4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :254.24PP1
CAS :<p>PP1 (AGL 1872), a specific and effective Src inhibitor, is with IC50 for Lck/Fyn is 5 nM/ 6 nM, respectively.</p>Formule :C16H19N5Degré de pureté :99% - 99.88%Couleur et forme :Off-White To Grey SolidMasse moléculaire :281.36Oroxin B
CAS :<p>Oroxin B (Hypocretin-2) has antioxidant activity.</p>Formule :C27H30O15Degré de pureté :98.22% - 99.81%Couleur et forme :SolidMasse moléculaire :594.52Nystatin
CAS :<p>Nystatin (Fungicidin) is a topical and oral antifungal agent with activity against many species of yeast and candida albicans, which is used largely to treat</p>Formule :C47H75NO17Degré de pureté :69.55% - 99.53%Couleur et forme :Yellow SuspensionMasse moléculaire :926.1Capmatinib
CAS :<p>Capmatinib (INCB28060) is an orally bioavailable inhibitor of the proto-oncogene c-Met (HGFR)with potential antineoplastic activity.</p>Formule :C23H17FN6ODegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :412.42CDDO-Im
CAS :<p>CDDO-Im (TP-235) is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).</p>Formule :C34H43N3O3Degré de pureté :98.3% - 99.61%Couleur et forme :SolidMasse moléculaire :541.72MK-4101
CAS :<p>MK-4101 inhibits Hedgehog pathway, causing apoptosis and reduced proliferation in cancer cells.</p>Formule :C24H24F5N5ODegré de pureté :98.2% - 99.13%Couleur et forme :SolidMasse moléculaire :493.47KEA1-97
CAS :<p>Kea1-97 is a selective disruptor of interaction between thioredoxin and caspase-3 (IC50 = 10 μ M).</p>Formule :C15H9Cl2FN4Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :335.16C188-9
CAS :<p>C188-9 (TTI-101) is a Stat3 inhibitor with an IC50 of 4-7 μM.</p>Formule :C27H21NO5SDegré de pureté :98.07% - >99.99%Couleur et forme :SolidMasse moléculaire :471.52NADPH tetrasodium salt
CAS :<p>NADPH tetrasodium salt is the reduced form of the electron acceptor nicotinamide adenine dinucleotide phosphate, which acts as an electron donor in a variety of</p>Formule :C21H26N7Na4O17P3Degré de pureté :97.15% - >99.99%Couleur et forme :SolidMasse moléculaire :833.35L-BUTHIONINE-(S,R)-SULFOXIMINE
CAS :<p>L-Buthionine-(S,R)-sulfoximine is a cell-permeable and irreversible inhibitor of γ-glutamylcysteine synthetase that induces oxidative stress by depleting GSH.</p>Formule :C8H18N2O3SDegré de pureté :97.07% - ≥98%Couleur et forme :White Fine PowderMasse moléculaire :222.31XL019
CAS :<p>XL019 is a potent and selective JAK2 inhibitor with IC50 of 2.2 nM, 100 fold selectivity over JAK1.</p>Formule :C25H28N6O2Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :444.53Vandetanib
CAS :<p>Vandetanib (ZD6474) is a potent inhibitor of VEGFR2 (IC50: 40 nM). It also inhibits VEGFR3 and EGFR.</p>Formule :C22H24BrFN4O2Degré de pureté :99.7% - >99.99%Couleur et forme :White SolidMasse moléculaire :475.35Domatinostat
CAS :<p>Domatinostat (4SC202) is a selective class I HDAC inhibitor. Domatinostat also displays inhibitory activity against Lysine specific demethylase 1 (LSD1).</p>Formule :C23H21N5O3SDegré de pureté :99.57% - 99.74%Couleur et forme :SolidMasse moléculaire :447.51tubuloside B
CAS :<p>Tubuloside B from Cistanche salsa stems guards SH-SY5Y cells against TNFalpha-induced apoptosis.</p>Formule :C31H38O16Degré de pureté :97.59% - 99.72%Couleur et forme :SolidMasse moléculaire :666.62ABT-737
CAS :<p>ABT-737 is a BH3 mimetic and an inhibitor of Bcl-2, Bcl-xL, and Bcl-w. ABT-737 exhibits antitumor activity and anti-aging activity. Cost-effective and quality-assured.</p>Formule :C42H45ClN6O5S2Degré de pureté :98.15% - >99.99%Couleur et forme :SolidMasse moléculaire :813.43PF-4989216
CAS :<p>PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.</p>Formule :C18H13FN6OSDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :380.4C25-140
CAS :<p>C25-140 is a small-molecule inhibitor of TRAF6-Ubc13.</p>Formule :C26H31N7ODegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :457.57Ziyuglycoside II
CAS :<p>1.</p>Formule :C35H56O8Degré de pureté :99.52% - ≥95%Couleur et forme :SolidMasse moléculaire :604.81Diosgenin glucoside
CAS :<p>Diosgenin glucoside (Trillin) and other synthetic glycosides with similar activities may be of use in the management of hypercholesterolemia and atherosclerosis</p>Formule :C33H52O8Degré de pureté :97.17% - 99.44%Couleur et forme :SolidMasse moléculaire :576.76Tauroursodeoxycholate dihydrate
CAS :<p>Tauroursodeoxycholate (TUDCA ,Taurolite) dihydrate is a bile acid that reduces Caspase-3, Caspase-12, ERK, reducing endoplasmic reticulum stress mediated death.</p>Formule :C26H49NO8SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :535.73Isosilybin A
CAS :<p>Isosilybin A is a partial PPARγ agonist, it significantly induced ABCA1 protein expression, it inhibited both monophenolase (IC50=1.7-7.6μM) and diphenolase (</p>Formule :C25H22O10Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :482.44Pexidartinib
CAS :<p>Pexidartinib (PLX-3397) is a capsule formulation containing a small-molecule receptor tyrosine kinase (RTK) inhibitor of KIT, CSF1R and FLT3 with potential</p>Formule :C20H15ClF3N5Degré de pureté :98.34% - 99.45%Couleur et forme :SolidMasse moléculaire :417.81Linalool
CAS :<p>Linalool, in essential oils, offers antinociceptive, antimicrobial, and anti-inflammatory effects, protects the liver, and boosts plant defense.</p>Formule :C10H18ODegré de pureté :98.22%Couleur et forme :Colorless Liquid Drypowder Liquid Othersolid LiquidMasse moléculaire :154.25Nutlin-3b
CAS :<p>Nutlin-3b, a less potent (+)-enantiomer of Nutlin-3, inhibits p53/MDM2 at IC50: 13.6 μM, 150x weaker than Nutlin-3a.</p>Formule :C30H30Cl2N4O4Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :581.49SRS16-86
CAS :<p>SRS16-86 is a novel third-generation ferrostatin, is an inhibitor of ferroptosis.</p>Formule :C26H32N4O2Degré de pureté :97.73%Couleur et forme :SolidMasse moléculaire :432.56Rasagiline Mesylate
CAS :<p>Rasagiline Mesylate (AGN1135) is a novel MAO-B inhibitor, which can treat idiopathic Parkinson's disease.</p>Formule :C13H17NO3SDegré de pureté :99.33%Couleur et forme :White PowderMasse moléculaire :267.34dl-Maackiain
CAS :<p>1. dl-Maackiain (Demethylpterocarpin) induces apoptosis and growth suppression 2. MAK1 is the second functional gene cloned from Maackiain detoxification.</p>Formule :C16H12O5Degré de pureté :97.36% - 99.89%Couleur et forme :SolidMasse moléculaire :284.26G-749
CAS :<p>G-749, a new-type FLT3 inhibitor, exhibits effective and sustained inhibition of the FLT3 wild type and mutants.</p>Formule :C25H25BrN6O2Degré de pureté :98.32% - 99.60%Couleur et forme :SolidMasse moléculaire :521.41Aurintricarboxylic acid
CAS :<p>Aurintricarboxylic acid (NSC-4056) blocks nucleases and topoisomerases, stopping nucleic acid binding.</p>Formule :C22H14O9Degré de pureté :97.1%Couleur et forme :Deep Red Coarse Crystalline PowderMasse moléculaire :422.34PhiKan 083
CAS :<p>PhiKan 083 is a carbazole derivative</p>Formule :C16H18N2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :238.33Hirsutine
CAS :<p>Hirsutine induces apoptosis and is a potent Dengue virus inhibitor exhibiting low cytotoxicity.Hirsutine has anticancer, cardioprotective, anti-hypertensive and</p>Formule :C22H28N2O3Degré de pureté :99.36% - 99.98%Couleur et forme :SolidMasse moléculaire :368.47(Rac)-Antineoplaston A10
CAS :<p>Antineoplaston A10 is the first identified human antineoplaston, naturally occurring with anti-proliferative properties.</p>Formule :C13H14N2O3Degré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :246.26A-1210477
CAS :<p>A-1210477 is an effective and specific MCL-1 and Bcl-2 inhibitor (Ki/IC50: 0.454/26.2 nM).</p>Formule :C46H55N7O7SDegré de pureté :99.17% - 99.37%Couleur et forme :SolidMasse moléculaire :850.04Echinocystic acid
CAS :<p>EA, a natural triterpene, is found in herbs; it has anti-inflammatory and antioxidant properties.</p>Formule :C30H48O4Degré de pureté :98% - 99.57%Couleur et forme :SolidMasse moléculaire :472.7Pseudolaric Acid B
CAS :<p>Pseudolaric acid B, a natural diterpenoid compound, is isolated from Pseudolarix kaempferi.</p>Formule :C23H28O8Degré de pureté :98.91% - 99.84%Couleur et forme :SolidMasse moléculaire :432.46Loganin
CAS :<p>Loganin inhibits Cox-1, suppresses TNF-α, and has antioxidant and anti-melanogenic properties.</p>Formule :C17H26O10Degré de pureté :99.01% - >99.99%Couleur et forme :White PowderMasse moléculaire :390.38SHR0302
CAS :<p>SHR0302 (ARQ252) is a JAK inhibitor that binds JAK1 with stronger affinity than others (Selectivity for JAK1 is more than 10 times for JAK2, 77 times for JAK3,</p>Formule :C18H22N8O2SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :414.48NVP-HSP990
CAS :<p>NVP-HSP990 (HSP990) is an effective and specific HSP90α/β inhibitor (IC50: 0.6 /0.8 nM).</p>Formule :C20H18FN5O2Degré de pureté :98.03% - 99.32%Couleur et forme :SolidMasse moléculaire :379.39Ethyl 3,4-dihydroxybenzoate
CAS :<p>Ethyl 3,4-dihydroxybenzoate (EDHB): a prolyl hydroxylase inhibitor attenuates acute hypobaric hypoxia mediated vascular leakage in brain.</p>Formule :C9H10O4Degré de pureté :99.88%Couleur et forme :White Crystal Or PowderMasse moléculaire :182.17PF-3758309 hydrochloride
CAS :<p>PF-3758309 hydrochloride (PF-03758309 hydrochloride) , is a PAK4 inhibitor, is also a n orally bioavailable small-molecule inhibitor of p21-activated kinase 4 (</p>Formule :C25H31ClN8OSDegré de pureté :98.83% - >99.99%Couleur et forme :SolidMasse moléculaire :527.08PP121
CAS :<p>PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from 2 to 60 nM.</p>Formule :C17H17N7Degré de pureté :98.45% - 99.67%Couleur et forme :SolidMasse moléculaire :319.36SZL P1-41
CAS :<p>SZL P1-41 inhibits Skp2, blocks complex formation, and halts ubiquitination, promoting cell senescence, reducing glycolysis, and exhibiting antitumor effects.</p>Formule :C24H24N2O3SDegré de pureté :99.60% - 99.87%Couleur et forme :SolidMasse moléculaire :420.52Garcinol
CAS :<p>Garcinol: inhibits HATs/PCAF (IC50=7/5 μM), anti-inflammatory, anti-cancer, anti-cholinesterase (AChE IC50=0.66 μM, BChE IC50=7.39 μM).</p>Formule :C38H50O6Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :602.8Panobinostat
CAS :<p>Panobinostat (NVP-LBH589) is a broad-spectrum HDAC inhibitor (IC50=5 nM) with oral activity and non-selectivity.</p>Formule :C21H23N3O2Degré de pureté :97.2% - 99.81%Couleur et forme :Yellow SolidMasse moléculaire :349.43Scopoletin
CAS :<p>Scopoletin (Esculetin 6-methyl ether) is a plant growth factor derived from the root of Scopolia carniolica, inhibits of acetylcholinesterase (AChE).</p>Formule :C10H8O4Degré de pureté :97.06% - 99.88%Couleur et forme :Yellow To Beige Crystalline PowderMasse moléculaire :192.17Cucurbitacin B
CAS :<p>Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells.</p>Formule :C32H46O8Degré de pureté :97.1% - 99.33%Couleur et forme :SolidMasse moléculaire :558.7Kinsenoside
CAS :<p>Kinsenoside ((+)-Kinsenoside) shows significant antihepatotoxic, and anti-inflammatory activities.</p>Formule :C10H16O8Degré de pureté :99.2% - >99.99%Couleur et forme :SolidMasse moléculaire :264.23NSC 23766 trihydrochloride
CAS :<p>NSC 23766 trihydrochloride (Rac1 Inhibitor) is an inhibitor of Rac GTPase targeting Rac activation by GEFs; no inhibitory for RhoA or Cdc42.</p>Formule :C24H35N7·3HClDegré de pureté :96.48% - 99.54%Couleur et forme :SolidMasse moléculaire :530.965-Geranoxy-7-methoxycoumarin
CAS :<p>5-Geranoxy-7-methoxycoumarin shows antifungal activity.</p>Formule :C20H24O4Degré de pureté :98.94% - 99.99%Couleur et forme :SolidMasse moléculaire :328.4INH1
CAS :<p>INH1 (IBT13131) is a cell-permeable Hec1 inhibitor that specifically disrupts the Hec1/Nek2 interaction.</p>Formule :C18H16N2OSDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :308.4FX1
CAS :<p>FX1 is an effective and selective BCL6 inhibitor (IC50: 35 μM).</p>Formule :C14H9ClN2O4S2Degré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :368.82ZM-447439
CAS :<p>ZM 447439 selectively inhibits Aurora A/B (IC50: 110/130 nM); 8x less effective on MEK1, Src, Lck; minimal impact on CDK1/2/4, Plk1, Chk1.</p>Formule :C29H31N5O4Degré de pureté :99.11% - 99.59%Couleur et forme :Pale Yellow SolidMasse moléculaire :513.59SP600125
CAS :<p>SP600125 (JNK Inhibitor II) is a JNK inhibitor that inhibits JNK1, JNK2, and JNK3 (IC50=40/40/90 nM) with oral potency, reversibility, and ATP-competitive</p>Formule :C14H8N2ODegré de pureté :97.63% - 99.82%Couleur et forme :SolidMasse moléculaire :220.23GSK-923295
CAS :<p>GSK923295 is a selective allosteric inhibitor of CENP-E kinesin motor ATPase(Ki=3.2 nM).</p>Formule :C32H38ClN5O4Degré de pureté :96.22% - 98.02%Couleur et forme :SolidMasse moléculaire :592.13Indinavir sulfate
CAS :<p>Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.</p>Formule :C36H49N5O8SDegré de pureté :99.75% - >99.99%Couleur et forme :White PowderMasse moléculaire :711.87KY-05009
CAS :<p>KY-05009 blocks TGF-β1 EMT in lung cancer cells, inhibits TNIK, Wnt genes, induces apoptosis, and is an ATP-competitive TNIK inhibitor (Ki = 100 nM).</p>Formule :C18H16N4O2SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :352.411A-116
CAS :<p>1A-116 is a specific Rac1 inhibitor.</p>Formule :C16H16F3N3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :307.31CP-724714
CAS :<p>CP-724714 (CP724714) is an effective and selective HER2/ErbB2 inhibitor (IC50: 10 nM), >640-fold selectivity against EGFR, Abl, InsR, PDGFR, IRG-1R, Src, VEGFR2</p>Formule :C27H27N5O3Degré de pureté :97.1% - 98.82%Couleur et forme :SolidMasse moléculaire :469.54ASP3026
CAS :<p>ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies,and Positive for Anaplastic Lymphoma Kinase.</p>Formule :C29H40N8O3SDegré de pureté :98.78% - 99.81%Couleur et forme :SolidMasse moléculaire :580.74CCT 137690
CAS :<p>CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).</p>Formule :C26H31BrN8ODegré de pureté :98.51% - 99.89%Couleur et forme :SolidMasse moléculaire :551.48COTI-2
CAS :<p>COTI-2, an orally available thiosemicarbazone, is an activator of mutant forms of the p53 protein with potential antineoplastic activity.</p>Formule :C19H22N6SDegré de pureté :99% - 99.55%Couleur et forme :SolidMasse moléculaire :366.48CI-1040
CAS :<p>CI-1040 (PD 184352) (PD184352) is an ATP non-competitive MEK1/2 inhibitor (IC50: 17 nM).</p>Formule :C17H14ClF2IN2O2Degré de pureté :99.64%Couleur et forme :Off-White To Pale Beige SolidMasse moléculaire :478.66Salidroside
CAS :<p>Salidroside is a bioactive phenolic glycoside compound isolated from Rhodiola rosea and is a prolyl endopeptidase inhibitor.Cost-effective and quality-assured.</p>Formule :C14H20O7Degré de pureté :97.81%Couleur et forme :Red-Brown Fine PowderMasse moléculaire :300.3Tomatine
CAS :<p>Tomatine (lycopersicin) is an antiproliferatve agent of breast adenocarcinoma cells.</p>Formule :C50H83NO21Degré de pureté :98.42% - 99.94%Couleur et forme :White To Light YellowMasse moléculaire :1034.19MG-101
CAS :<p>MG-101 (Calpain inhibitor I) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins.</p>Formule :C20H37N3O4Degré de pureté :98% - ≥98%Couleur et forme :SolidMasse moléculaire :383.53SJ-172550
CAS :<p>SJ-172550 is a small molecule inhibitor of MDMX (EC50: 5 μM).</p>Formule :C22H21ClN2O5Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :428.87Momelotinib
CAS :<p>Momelotinib (LM-1149), an oral JAK1/2 inhibitor with IC50s 11/18 nM, blocks ATP binding, disrupting JAK-STAT pathway and reducing tumor growth.</p>Formule :C23H22N6O2Degré de pureté :97.47% - 99.56%Couleur et forme :SolidMasse moléculaire :414.46Kahweol
CAS :<p>Kahweol has anticarcinogenic, anti-angiogenic,and anti-inflammatory activities, it can block the LPS-induced activation of NF-kappaB by preventing IkappaB</p>Formule :C20H26O3Degré de pureté :99.26% - 99.86%Couleur et forme :Off-White To Yellow SolidMasse moléculaire :314.42TC11
CAS :<p>TC11 (1H-Isoindole-1,3(2H)-dione, 5-amino-2-[2,6-bis(1-methylethyl)phenyl]-TC11) is a potent inhibitor of tumor cell proliferation and an inducer of apoptosis</p>Formule :C20H22N2O2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :322.4BC-1258
CAS :<p>BC-1258 is a unique small molecule F-box/LRR-repeat protein 2 (FBXL2) activator.</p>Formule :C22H22N4S2Degré de pureté :97.48% - 99.64%Couleur et forme :SolidMasse moléculaire :406.57GSK 872 hydrochloride
CAS :<p>GSK872 HCl（1346546-69-7 free base） (GSK2399872A) is an effective and specific RIP3 kinase inhibitor.</p>Formule :C19H18ClN3O2S2Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :419.94B-AP15
CAS :<p>B-AP15 (NSC-687852) selectively inhibits 26S proteasome enzymes Usp14 and UCHL5, blocking their activity.</p>Formule :C22H17N3O6Degré de pureté :91.43% - 98.77%Couleur et forme :SolidMasse moléculaire :419.39Niraparib
CAS :<p>Niraparib (MK-4827) inhibits PARP1/PARP2 (IC50: 3.8/2.1 nM), effective on BRCA mutant cancers, 330x less effective on PARP3, V-PARP, Tank1.</p>Formule :C19H20N4ODegré de pureté :98% - 99.91%Couleur et forme :SolidMasse moléculaire :320.39R406
CAS :<p>R406 (R-406 besylate) is an effective Syk inhibitor (IC50: 41 nM) and shows no effects on Lyn.</p>Formule :C22H23FN6O5·C6H6O3SDegré de pureté :97.67% - 98.82%Couleur et forme :SolidMasse moléculaire :628.63Mito-LND
CAS :<p>Mito-LND (Mito-Loidamine) is an orally active and mitochondria-targeted inhibitor of oxidative phosphorylation.</p>Formule :C43H45BrCl2N3OPDegré de pureté :97.25% - 98.34%Couleur et forme :SolidMasse moléculaire :801.62PR-619
CAS :<p>PR-619 (2,6-Diamino-3,5-dithiocyanopyridine) is a DUB inhibitor. PR-619 induces endoplasmic reticulum stress and activates autophagy. Cost-effective and quality-assured.</p>Formule :C7H5N5S2Degré de pureté :97.25% - >99.99%Couleur et forme :SolidMasse moléculaire :223.28Alisertib Sodium
CAS :<p>Alisertib Sodium (MLN 8237 Sodium)is a selective Aurora A inhibitor that causes G2/M phase arrest and chromosomal misalignment, leading to tumour cell apoptosis.</p>Formule :C27H19ClFN4NaO4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :540.91(R)-(-)-Gossypol acetic acid
CAS :<p>(R)-(-)-Gossypol acetic acid binds Bcl-2, Bcl-xL, Mcl-1 (Ki: 0.32, 0.48, 0.18 μM); no BIR3/BID inhibition. Phase 2.</p>Formule :C30H30O8·C2H4O2Degré de pureté :98.88% - 99.5%Couleur et forme :SolidMasse moléculaire :578.61Tiplaxtinin
CAS :<p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>Formule :C24H16F3NO4Degré de pureté :99.16% - 99.93%Couleur et forme :SolidMasse moléculaire :439.383-Dehydrotrametenolic acid
CAS :<p>3-Dehydrotrametenolic acid is a potential anticancer agent against H-ras transformed tumor and a promising candidate for a new type of insulin-sensitizing drug.</p>Formule :C30H46O3Degré de pureté :98.5% - 99.25%Couleur et forme :SolidMasse moléculaire :454.68K34C
CAS :<p>K34C is a selective inhibitor of Integrin α5β1, which inhibits cell survival and migration, promotes apoptosis, inhibits invasion.</p>Formule :C26H29N3O4Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :447.53Pilaralisib analogue
CAS :<p>Pilaralisib analogue (XL147 analogue) is a selective and reversible class I PI3K inhibitor for PI3Kα/δ/γ.</p>Formule :C21H16N6O2S2Degré de pureté :99.3% - 99.72%Couleur et forme :SolidMasse moléculaire :448.52Roquinimex
CAS :<p>Roquinimex (FCF89) (Linomide) is a quinoline derivative immunostimulant which increases NK cell activity and macrophage cytotoxicity; inhibits angiogenesis and</p>Formule :C18H16N2O3Degré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :308.33Toyocamycin
CAS :<p>Toyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage (</p>Formule :C12H13N5O4Degré de pureté :98.1% - 98.17%Couleur et forme :SolidMasse moléculaire :291.26Adalimumab
CAS :<p>Adalimumab (anti-TNF-alpha) is the first fully human recombinant IgG1 monoclonal antibody that specifically targets human TNF-alpha.</p>Degré de pureté :95% - 99.50%Couleur et forme :LiquidMasse moléculaire :145.4 kDatrans-Chalcone
CAS :<p>trans-Chalcone (Chalkone) is an aromatic ketone that forms the central core for a variety of important biological compounds, which are known collectively as</p>Formule :C15H12ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :208.26Solasodine
CAS :<p>Solasodine, a toxic alkaloid from Solanaceae, kills HeLa cervical cancer and U937 leukemia cells.</p>Formule :C27H43NO2Degré de pureté :99.64% - 99.94%Couleur et forme :SolidMasse moléculaire :413.64PTC-028
CAS :<p>PTC-028 selectively suppresses cancer cells whereas normal cells remain unaffected.</p>Formule :C19H12F5N5Degré de pureté :97.61% - 98.12%Couleur et forme :SolidMasse moléculaire :405.32Divalproex Sodium
CAS :<p>Divalproex Sodium (Valproate semisodium) binds to and inhibits gamma-aminobutyric acid (GABA) transaminase and its anticonvulsant activity may be exerted by</p>Formule :C8H16O2·C8H15O2·NaDegré de pureté :99.87%Couleur et forme :A White Powder With A Characteristic OdorMasse moléculaire :310.41Tamibarotene
CAS :<p>Tamibarotene (Amnolake) is an orally active, synthetic retinoid, developed to overcome all-trans retinoic acid (ATRA) resistance, with potential antineoplastic</p>Formule :C22H25NO3Degré de pureté :98.55% - 99.73%Couleur et forme :Crystalline SolidMasse moléculaire :351.44PCI-34051
CAS :<p>PCI-34051 is an effective and selective HDAC8 inhibitor (IC50: 10 nM).</p>Formule :C17H16N2O3Degré de pureté :97.219% - 98.29%Couleur et forme :SolidMasse moléculaire :296.32(Rac)-Benpyrine
CAS :<p>(Rac)-Benpyrine is a potent and orally active inhibitor of TNF-α.</p>Formule :C16H16N6ODegré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :308.34Tyrphostin AG 879
CAS :<p>Tyrphostin AG 879 (AG 879) effectively inhibits HER2/ErbB2 (IC50: 1 μM), 100- and 500-fold higher selective to ErbB2 than EGFR and PDGFR.</p>Formule :C18H24N2OSDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :316.46RHPS4
CAS :<p>RHPS4 (RHPS 4 methosulfate) is a potent inhibitor of Telomerase at submicromolar.</p>Formule :C22H17F2N2·CH3O4SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :458.48Fidaxomicin
CAS :<p>Fidaxomicin (Tiacumicin B) is a semisynthetic macrolide antibiotic used to treat Clostridium difficile-associated diarrhea in adults.</p>Formule :C52H74Cl2O18Degré de pureté :99.76% - 99.82%Couleur et forme :SolidMasse moléculaire :1058.04L-Glutamic acid monosodium salt
CAS :<p>L-Glutamic acid monosodium salt (MSG) (Monosodium glutamate) is an activator of mGlu1 receptor.</p>Formule :C5H8NO4·NaDegré de pureté :99.93%Couleur et forme :White Solid CrystallineMasse moléculaire :169.11Kevetrin hydrochloride
CAS :<p>Kevetrin hydrochloride (4-Isothioureidobutyronitrile hydrochloride) is a small molecule and activator of the tumor suppressor protein p53, with potential</p>Formule :C5H10ClN3SDegré de pureté :99.32% - 99.93%Couleur et forme :SolidMasse moléculaire :179.67Parthenolide
CAS :<p>Parthenolide ((-)-Parthenolide) is a natural sesquiterpene lactone that is an NF-κB and HDAC1 inhibitor with anti-inflammatory effect. Cost-effective and quality-assured.</p>Formule :C15H20O3Degré de pureté :98.19% - 99.46%Couleur et forme :White To Pale Yellow Crystalline PowderMasse moléculaire :248.32PS210
CAS :<p>PS210 selectively activates PDK1 (Kd: 3 μM), doesn't affect PDK1 downstream kinases. Prodrug PS423 inhibits PDK1-mediated S6K phosphorylation.</p>Formule :C19H15F3O5Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :380.31Alofanib
CAS :<p>Alofanib (RPT835) selectively inhibits FGFR2 in KATO III cells with IC50 <10 nM; doesn’t affect FGFR1/3 or FGF2-FGFR2 binding.</p>Formule :C19H15N3O6SDegré de pureté :99.53% - 99.81%Couleur et forme :SolidMasse moléculaire :413.4ONO-4059 analog
CAS :<p>ONO-4059 analog (ONO-WG-307)ue is an analogue of ONO-4059, which is a highly potent and selective oral BTK inhibitor with IC50 of 23.9 nM. Phase 1.</p>Formule :C25H24N6O3Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :456.5Galgravin
CAS :<p>Galgravin combats inflammation, safeguards neurons, promotes neurite growth, and resists Abeta25-35 and MPP+ toxicity.</p>Formule :C22H28O5Degré de pureté :99.75% - 99.88%Couleur et forme :SolidMasse moléculaire :372.45SC-43
CAS :<p>SC-43 is a potent and orally active agonist of SHP-1 (PTPN6).</p>Formule :C21H13ClF3N3O2Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :431.8Sanguinarine
CAS :<p>Sanguinarine (Pseudochelerythrine) is a specific inhibitor of Rac1b with anti-microbial, anti-oxidant and anti-inflammatory properties.</p>Formule :C20H14NO4Degré de pureté :99.04% - 99.76%Couleur et forme :SolidMasse moléculaire :332.33Clovamide
CAS :<p>Trans-Clovamide (trans-Clovamide) is a naturally occurring caffeoyl conjugate identified in the antioxidant polyphenolic fraction of cocoa (T.</p>Formule :C18H17NO7Degré de pureté :97.12% - 97.68%Couleur et forme :SolidMasse moléculaire :359.33Salermide
CAS :<p>Salermide is an inhibitor of Sirt1 and Sirt2, causing strong cancer-specific apoptotic cell death.</p>Formule :C26H22N2O2Degré de pureté :97.09% - 99.55%Couleur et forme :SolidMasse moléculaire :394.47Piperlongumine
CAS :<p>Piperlongumine (Piplartine) is a natural alkaloid from Piper longum L.</p>Formule :C17H19NO5Degré de pureté :97.03% - 99.90%Couleur et forme :SolidMasse moléculaire :317.34Quercetin Dihydrate
CAS :<p>Quercetin Dihydrate (Sophoretin) is a flavonoid natural product that activates or inhibits the activity of many proteins. It activates SIRT1 and inhibits PI3K.</p>Formule :C15H10O7·2H2ODegré de pureté :97.77%Couleur et forme :Yellow SolidMasse moléculaire :338.27LY2409881 trihydrochloride
CAS :<p>LY2409881 trihydrochloride is a novel specific inhibitor of IKK2 (IC50: 30 nM); IC50 for IKK1 and other common kinases is at least one log higher.</p>Formule :C24H32Cl4N6OSDegré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :594.43ODQ
CAS :<p>ODQ is an effective and selective soluble guanylyl cyclase (sGC) inhibitor.</p>Formule :C9H5N3O2Degré de pureté :98.98%Couleur et forme :Off-White To Light Yellow PowderMasse moléculaire :187.15PS47
CAS :<p>PS-47(PS 47) is an inactive E-isomer of PS48. PS48 is an activator of PDK1.</p>Formule :C17H15ClO2Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :286.75Atractylenolide II
CAS :<p>Atractylenolide II inhibits STAT3, activates p38, deactivates ERK/Akt, and induces p53-dependent cytotoxicity against melanoma.</p>Formule :C15H20O2Degré de pureté :99.89% - 99.93%Couleur et forme :SolidMasse moléculaire :232.32D4476
CAS :<p>D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).</p>Formule :C23H18N4O3Degré de pureté :99.7% - 99.96%Couleur et forme :SolidMasse moléculaire :398.41Capsazepine
CAS :<p>Capsazepine, a TRPV1 antagonist (IC50: 562 nM), blocks capsaicin-induced heat pain.</p>Formule :C19H21ClN2O2SDegré de pureté :98% - 99.78%Couleur et forme :White To Off-White PowderMasse moléculaire :376.9Pectolinarin
CAS :<p>Pectolinarin is a Cirsium isolate with anti-inflammatory activity.</p>Formule :C29H34O15Degré de pureté :98% - 99.79%Couleur et forme :SolidMasse moléculaire :622.57SC144
CAS :<p>SC144 is an orally active small-molecule gp130 inhibitor.</p>Formule :C16H11FN6ODegré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :322.3Dapivirine
CAS :<p>Dapivirine (R147681) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.</p>Formule :C20H19N5Degré de pureté :98% - 99.77%Couleur et forme :SolidMasse moléculaire :329.4Bafetinib
CAS :<p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>Formule :C30H31F3N8ODegré de pureté :94.16% - 99.68%Couleur et forme :SolidMasse moléculaire :576.62PHT-427
CAS :<p>PHT-427 (CS-0223) is a dual Akt (Ki: 2.7 μM) and PDPK1 (Ki: 5.2 μM) inhibitor (high-affinity binding for the PH domains of Akt and PDPK1).</p>Formule :C20H31N3O2S2Degré de pureté :97.54% - >99.99%Couleur et forme :SolidMasse moléculaire :409.61KPT-251
CAS :<p>KPT-251 is a selective nuclear export inhibitor.</p>Formule :C14H7F6N5ODegré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :375.23Menin-MLL inhibitor MI-2
CAS :<p>Menin-MLL inhibitor MI-2 (MI2) is a potent menin-MLL interaction inhibitor with IC50 of 446 nM.</p>Formule :C18H25N5S2Degré de pureté :97.46%Couleur et forme :SolidMasse moléculaire :375.55Baohuoside I
CAS :<p>Baohuoside I (Icariside-II) is a component of Epimedium koreanum, exhibits anti-inflammatory activity and anti-osteoporosis activities.</p>Formule :C27H30O10Degré de pureté :97.64% - 98.14%Couleur et forme :SolidMasse moléculaire :514.52R547
CAS :<p>R547 (Ro 4584820) is a potent ATP-competitive inhibitor of CDK1/2/4 with Ki of 2 nM/3 nM/1 nM.</p>Formule :C18H21F2N5O4SDegré de pureté :90% - 99.64%Couleur et forme :SolidMasse moléculaire :441.45DCH36_06
CAS :<p>DCH36_06 ((5E)-1-(3-chloro-4-methylphenyl)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-ylidene]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione) as a bona fide is a potent</p>Formule :C18H13ClN2O3SDegré de pureté :97.78%Couleur et forme :SolidMasse moléculaire :372.83Arctigenin
CAS :<p>(-)-Arctigenin ((-)-Arctigenin) is found in burdock.</p>Formule :C21H24O6Degré de pureté :98% - 99.51%Couleur et forme :SolidMasse moléculaire :372.41Ethoxysanguinarine
CAS :<p>Ethoxysanguinarine inhibits HuAChE and HuBuChE with IC50s of 0.83 and 4.20 μM, respectively.</p>Formule :C22H19NO5Degré de pureté :99.24% - 99.48%Couleur et forme :SolidMasse moléculaire :377.39Tofacitinib
CAS :<p>Tofacitinib (Tasocitinib) is an orally Janus kinase inhibitor. Tofacitinib is used for the treatment of rheumatoid arthritis. Cost effective and quality assured.</p>Formule :C16H20N6ODegré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :312.37Furanodienone
CAS :<p>1.</p>Formule :C15H18O2Degré de pureté :98% - 99.91%Couleur et forme :SolidMasse moléculaire :230.3Avadomide
CAS :<p>Avadomide (CC 122) is an orally available pleiotropic pathway modulator with potential antineoplastic activity.</p>Formule :C14H14N4O3Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :286.29PHA-793887
CAS :<p>PHA-793887 has been used in trials studying the treatment of Advanced/Metastatic Solid Tumors.</p>Formule :C19H31N5O2Degré de pureté :98.02% - >99.99%Couleur et forme :SolidMasse moléculaire :361.48Sincalide
CAS :<p>Sincalide (CCK-8) is an injectable drug used to diagnose gallbladder and pancreas disorders; it's a cholecystokinin fragment.</p>Formule :C49H62N10O16S3Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :1143.27Hematoporphyrin dihydrochloride
CAS :<p>Hematoporphyrin dihydrochloride (Hematoporphyrin IX dihydrochloride) is a substrate for affinity chromatography of heme-binding proteins.</p>Formule :C34H40Cl2N4O6Degré de pureté :90.11%Couleur et forme :SolidMasse moléculaire :671.61PluriSIn 1
CAS :<p>PluriSIn 1 (NSC 14613) blocks SCD1, key in oleic acid creation, showing lipid metabolism's role in hPSCs.</p>Formule :C12H11N3ODegré de pureté :99.19% - 99.63%Couleur et forme :SolidMasse moléculaire :213.24BTSA1
CAS :<p>BTSA1: High-affinity BAX activator inducing conformational changes for apoptosis.</p>Formule :C21H14N6OS2Degré de pureté :99.60% - 99.71%Couleur et forme :SolidMasse moléculaire :430.51Cambinol
CAS :<p>Cambinol is a SIRT1/2 inhibitor (IC50: 56/59 μM), non-competitive with NAD, weak on SIRT5, and prompts apoptosis in lymphoma cells.</p>Formule :C21H16N2O2SDegré de pureté :98.02% - 99.83%Couleur et forme :SolidMasse moléculaire :360.43Cinobufagin
CAS :<p>Cinobufagin (Cinobufagine) is a selective Na+/K+-ATPase inhibitor. The activity of Cinobufagin is same as ouabain.</p>Formule :C26H34O6Degré de pureté :97.77% - 99.97%Couleur et forme :SolidMasse moléculaire :442.54Euphorbia Factor L2
CAS :<p>Euphorbia Factor L2 alleviates lipopolysaccharide-induced acute lung injury and inflammation through inhibits NF-κB activation.</p>Formule :C38H42O9Degré de pureté :99.53% - 99.96%Couleur et forme :SolidMasse moléculaire :642.73Omaveloxolone
CAS :<p>Omaveloxolone (RTA-408) (RTA-408) is a synthetic triterpenoid that activates the cytoprotective transcription factor Nrf2 and inhibits NF-κB signaling. Phase 2.</p>Formule :C33H44F2N2O3Degré de pureté :98.7% - 99.92%Couleur et forme :SolidMasse moléculaire :554.71
