Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(34 produtos)
- Cisteína Protease(96 produtos)
- DPP-4(20 produtos)
- Glutaminase(40 produtos)
- HIV Protease(449 produtos)
- PAI-1(25 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(53 produtos)
- Proteassoma(94 produtos)
- Protease serina(50 produtos)
- p97(14 produtos)
Exibir 3 mais subcategorias
Foram encontrados 1044 produtos de "Proteases/Proteassoma"
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Carbobenzoxyproline
CAS:<p>Carbobenzoxyproline (Carbobenzoxy-S-proline) is a prolidase inhibitor.</p>Fórmula:C13H15NO4Pureza:99.79%Cor e Forma:White To Light Yellow Crystal PowderPeso molecular:249.26PF-00835231
CAS:<p>PF-00835231 is a CoV-2 cysteine 3C-like protease (3CLpro) inhibitor, with IC50s of 0.27 nM and 4 nM for SARS CoV-2 and SARS CoV-1 3CLpro, respectively.PF-</p>Fórmula:C24H32N4O6Pureza:97.83%Cor e Forma:SolidPeso molecular:472.53CH 5450
CAS:<p>CH 5450 (Z-Ile-Glu-Pro-Phe-Ome) (Z-Ile-Glu-Pro-Phe-Ome) is a short peptide inhibitor of chymase in the human heart</p>Fórmula:C34H44N4O9Pureza:95.93%Cor e Forma:SolidPeso molecular:652.73Rusalatide acetate (497221-38-2 free base)
CAS:<p>Rusalatide acetate (TP508 amide acetate), a regenerated peptide, alleviates radiation-induced gastrointestinal injury by activating stem cells.</p>Fórmula:C99H151N29O37SPureza:>99.99%Cor e Forma:SolidPeso molecular:2371.5Hepln-13
CAS:<p>Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.</p>Fórmula:C17H13BrN2Pureza:97.67%Cor e Forma:SolidPeso molecular:325.2(Arg)9 TFA (143413-47-2 free base)
CAS:<p>(Arg)9 TFA (Peptide R9 TFA) is a cell-penetrating peptide. (Arg)9 TFA exhibits neuroprotective activity with an IC50 of 0.78 μM in the glutamic acid model.</p>Fórmula:C56H111F3N36O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:1537.714-Isopropylcatechol
CAS:<p>4-Isopropylcatechol is a potent depigmenting agent and is of use in the topical therapy of selected patients with hypermelanosis.</p>Fórmula:C9H12O2Pureza:97.93%Cor e Forma:SolidPeso molecular:152.19Azvudine
CAS:<p>Azvudine (FNC) is a powerful NRTI effective against HIV, HBV, HCV, and resistant strains.</p>Fórmula:C9H11FN6O4Pureza:99.76% - >99.99%Cor e Forma:SolidPeso molecular:286.22Z-YVAD-FMK
CAS:<p>AA-Z-YVAD-FMK is a Irreversible caspase-1 inhibitor,with anti-inflammatory and anti-tumor activities.</p>Fórmula:C31H39FN4O9Pureza:98.00%Cor e Forma:SolidPeso molecular:630.66Enfuvirtide acetate
CAS:<p>Enfuvirtide acetate salt is a linear synthetic peptide made of 36 amino acids. It has an acetylated N-terminus and a carboxamide C-terminus.</p>Fórmula:C206H305N51O66Pureza:99.34%Cor e Forma:SolidPeso molecular:4552Diprotin A
CAS:<p>Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.</p>Fórmula:C17H31N3O4Pureza:99.29%Cor e Forma:White PowderPeso molecular:341.45GI254023X
CAS:<p>GI254023X is a MMP9 and ADAM10 inhibitor with IC50 values of 2.5 and 5.3 nM.Cost-effective and quality-assured.</p>Fórmula:C21H33N3O4Pureza:98.21% - 98.56%Cor e Forma:SolidPeso molecular:391.5Paritaprevir free base
CAS:<p>Paritaprevir (ABT-450) is an oral HCV NS3/NS4A protease inhibitor with potential against genotype 1, disrupting viral replication.</p>Fórmula:C40H43N7O7SPureza:95% - 99.26%Cor e Forma:SolidPeso molecular:765.89Bictegravir
CAS:<p>Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).</p>Fórmula:C21H18F3N3O5Pureza:97.6% - 99.51%Cor e Forma:SolidPeso molecular:449.38ABT530
CAS:<p>ABT530 (Pibrentasvir) is an HCV NS5A inhibitor with EC50s ranging from 1.4-5.0 pM against HCV replicons containing NS5A from genotypes 1-6.</p>Fórmula:C57H65F5N10O8Pureza:99.15% - 99.93%Cor e Forma:SolidPeso molecular:1113.18TMC647055 Choline Hydroxide Salt
<p>TMC647055 is a potent HCV NS5B inhibitor with low toxicity and good pharmacokinetics, under clinical evaluation.</p>Fórmula:C37H53N5O8SPureza:99.44%Cor e Forma:SolidPeso molecular:727.91Brensocatib
CAS:<p>Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).</p>Fórmula:C23H24N4O4Pureza:97.55%Cor e Forma:SolidPeso molecular:420.46Apelin-17 (human, bovine) acetate
<p>Apelin-17 (human, bovine) acetate is an endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).</p>Fórmula:C98H160N34O22SPureza:99.36%Cor e Forma:SolidPeso molecular:2198.63Rilpivirine
CAS:<p>Rilpivirine (R278474) is a diarylpyrimidine derivative and reverse transcriptase inhibitor with antiviral activity against HIV-1 that is used in the treatment</p>Fórmula:C22H18N6Pureza:97.22% - 98.83%Cor e Forma:SolidPeso molecular:366.42CASP3 Activator 1541
CAS:<p>CASP3 Activator 1541 is an activator of the proenzyme forms of caspase-3, and induces cell death.</p>Fórmula:C24H17N3O4Pureza:98.84%Cor e Forma:SolidPeso molecular:411.41EIDD-1931
CAS:<p>EIDD-1931 (Beta-d-N4-hydroxycytidine) is a ribonucleoside analog with antiviral activity. It inhibits replication of SARS-CoV, MERS-CoV, and SARS-CoV-2.</p>Fórmula:C9H13N3O6Pureza:99.14% - 99.73%Cor e Forma:SolidPeso molecular:259.22GSK-690693
CAS:<p>GSK-690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also sensitive to the AGC kinase family: PKA, PrkX and PKC isozymes. Phase 1.</p>Fórmula:C21H27N7O3Pureza:98.07% - 99.77%Cor e Forma:SolidPeso molecular:425.483-O-Ethyl-L-ascorbic acid
CAS:3-O-Ethyl-L-ascorbic acid is a cosmetic tyrosinase inhibitor with whitening ability and is a stabilized vitamin C derivative.Fórmula:C8H12O6Pureza:97.35% - 99.99%Cor e Forma:White To Very Pale Yellow Crystalline Powder Solid PowderPeso molecular:204.18PSI-6130
CAS:<p>PSI-6130 (R 1656) is a potent and selective HCV NS5B polymerase inhibitor. PSI-6130 inhibits HCV replication with a mean IC50 of 0.6 μM.</p>Fórmula:C10H14FN3O4Pureza:98.63% - 99.79%Cor e Forma:SolidPeso molecular:259.23Asunaprevir
CAS:<p>Asunaprevir (BMS-650032) is an effective hepatitis C virus (HCV) NS3 protease inhibitor.</p>Fórmula:C35H46ClN5O9SPureza:99.34% - 99.8%Cor e Forma:SolidPeso molecular:748.29PTACH
CAS:<p>PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).</p>Fórmula:C20H26N2O2S2Pureza:87.44% - 99.74%Cor e Forma:SolidPeso molecular:390.56Daclatasvir
CAS:<p>Daclatasvir (EBP 883/BMS-790052) is a potent HCV NS5A inhibitor with EC50 9-50 pM across various genotypes. Phase 3.</p>Fórmula:C40H50N8O6Pureza:99.81%Cor e Forma:SolidPeso molecular:738.88CA-074 methyl ester
CAS:<p>CA-074 methyl ester (Cathepsin B Inhibitor IV) is a selective inhibitor of Cathepsin B (IC50=36.3 nM). neuroprotective effect. High-Quality, Low-Cost!</p>Fórmula:C19H31N3O6Pureza:97.26% - 99.58%Cor e Forma:SolidPeso molecular:397.47Peptide T acetate(106362-32-7 free base)
<p>Peptide T acetate is an octapeptide from the V2 region of HIV-1 gp120.</p>Fórmula:C37H59N9O18Pureza:99.47%Cor e Forma:SolidPeso molecular:917.91Letermovir
CAS:<p>Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.</p>Fórmula:C29H28F4N4O4Pureza:99.85% - 99.87%Cor e Forma:SolidPeso molecular:572.55Bemnifosbuvir
CAS:<p>Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.</p>Fórmula:C24H33FN7O7PPureza:99.35% - 99.54%Cor e Forma:SolidPeso molecular:581.53LY 3000328
CAS:<p>LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.</p>Fórmula:C25H29FN4O5Pureza:97.83% - 99.54%Cor e Forma:SolidPeso molecular:484.524-Butylresorcinol
CAS:<p>4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.</p>Fórmula:C10H14O2Pureza:98.64% - ≥95%Cor e Forma:Light Beige Solid PowderPeso molecular:166.22Daclatasvir dihydrochloride
CAS:<p>Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.</p>Fórmula:C40H52Cl2N8O6Pureza:99.67%Cor e Forma:SolidPeso molecular:811.8Ixazomib citrate
CAS:<p>Ixazomib citrate (MLN9708), a prodrug of Ixazomib (MMLN-2238), is an oral 2nd-gen proteasome inhibitor with anti-cancer potential (IC50: 3.4 nM).</p>Fórmula:C20H23BCl2N2O9Pureza:98.37% - >99.99%Cor e Forma:SolidPeso molecular:517.12Paritaprevir
CAS:<p>Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂，对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂，IC50为 1.31 μM。</p>Fórmula:C40H43N7O7SPureza:99.72%Cor e Forma:SolidPeso molecular:765.88Avatrombopag
CAS:<p>Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiation</p>Fórmula:C29H34Cl2N6O3S2Pureza:99.01% - 99.63%Cor e Forma:SolidPeso molecular:649.65S 3304
CAS:<p>S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.</p>Fórmula:C24H20N2O4S2Pureza:98.09%Cor e Forma:SolidPeso molecular:464.56Velpatasvir
CAS:<p>Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.</p>Fórmula:C49H54N8O8Pureza:99.17% - 99.83%Cor e Forma:SolidPeso molecular:883Boc-Asp(OMe)-fluoromethyl ketone
CAS:<p>Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.</p>Fórmula:C11H18FNO5Pureza:≥98%Cor e Forma:SolidPeso molecular:263.26Obefazimod
CAS:<p>Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).</p>Fórmula:C16H10ClF3N2OPureza:99.86%Cor e Forma:SolidPeso molecular:338.71KKI-5 acetate(97145-43-2 free base)
<p>KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.</p>Fórmula:C37H59N11O11Pureza:99.44%Cor e Forma:SolidPeso molecular:833.95Tris(4-aminophenyl)methane
CAS:<p>Tris(4-aminophenyl)methane (Leucopararosaniline), a triphenylmethane dye, is a weak HCV helicase inhibitor.</p>Fórmula:C19H19N3Pureza:95.73%Cor e Forma:Beige Solid CrystallinePeso molecular:289.37JNJ0966
CAS:<p>JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).</p>Fórmula:C16H16N4O2S2Pureza:99.46% - 99.62%Cor e Forma:SolidPeso molecular:360.45Omarigliptin
CAS:<p>Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value of 1.6 nM. Cost-effective and quality-assured.</p>Fórmula:C17H20F2N4O3SPureza:99.68% - 99.77%Cor e Forma:SolidPeso molecular:398.43Thiamine disulfide
CAS:<p>Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.</p>Fórmula:C24H34N8O4S2Pureza:99.81%Cor e Forma:CoaPeso molecular:562.71Y-29794 Tosylate
CAS:<p>Y-29794 Tosylate (Y-29794) is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.</p>Fórmula:C30H42N2O4S3Pureza:99.86%Cor e Forma:SolidPeso molecular:590.86GK921
CAS:<p>GK921 is a transglutaminase 2 (TGase) inhibitor.</p>Fórmula:C21H20N4OPureza:97.44% - 99.49%Cor e Forma:SolidPeso molecular:344.41HIV-1 Inhibitor 18A
CAS:<p>HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.</p>Fórmula:C14H11N5O2SPureza:99.79%Cor e Forma:SolidPeso molecular:313.33CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)
<p>CTTHWGFTLC, CYCLIC acetate is an inhibitor for matrix metalloproteinases (MMP)-2 and MMP-9.</p>Fórmula:C54H75N13O16S2Pureza:99.71%Cor e Forma:SolidPeso molecular:1226.39Dabigatran
CAS:<p>Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.</p>Fórmula:C25H25N7O3Pureza:97.44% - 98.7%Cor e Forma:Tan SolidPeso molecular:471.51CeMMEC13
CAS:<p>CeMMEC13 is an isoquinolinone that selectively inhibits the second bromodomain of TAF1 (IC50 = 2.1 μM).</p>Fórmula:C19H16N2O4Pureza:98.52%Cor e Forma:SolidPeso molecular:336.34Doravirine
CAS:<p>Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.</p>Fórmula:C17H11ClF3N5O3Pureza:99.65% - 99.79%Cor e Forma:SolidPeso molecular:425.75L-Albizziin
CAS:<p>L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.</p>Fórmula:C4H9N3O3Pureza:99.98%Cor e Forma:White PowderPeso molecular:147.13Anagliptin
CAS:<p>Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.</p>Fórmula:C19H25N7O2Pureza:97.59% - 99.98%Cor e Forma:SolidPeso molecular:383.45P-113 acetate
<p>P-113 acetate: AMP from histatin 5, treats gingivitis and HIV-related oral candidiasis safely and effectively.</p>Fórmula:C73H114N28O15Pureza:97.4%Cor e Forma:SolidPeso molecular:1623.86Samatasvir
CAS:<p>Samatasvir (ATOLIHZIXHZSBA-BTSKBWHGSA-N) is a pan-genotypic inhibitor of the HCV non-structural protein 5A.</p>Fórmula:C47H48N8O6S2Pureza:98.03%Cor e Forma:SolidPeso molecular:885.06Glutaminase C-IN-1
CAS:<p>Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.</p>Fórmula:C27H27BrN2OPureza:99.68% - >99.99%Cor e Forma:SolidPeso molecular:475.422,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:<p>2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urine</p>Fórmula:C13H16O3Pureza:99.53% - 99.81%Cor e Forma:SolidPeso molecular:220.26Ixazomib
CAS:<p>Ixazomib (MLN2238) is a boron-based peptide proteasome inhibitor targeting β5 site (IC50: 3.4 nM), also affecting β1 and β2 sites.</p>Fórmula:C14H19BCl2N2O4Pureza:98% - 98.92%Cor e Forma:SolidPeso molecular:361.03Batimastat
CAS:<p>Batimastat (BB94) (BB-94) is an effective, broad-spectrum matrix metalloprotease (MMP) inhibitor.</p>Fórmula:C23H31N3O4S2Pureza:98.15% - 99.5%Cor e Forma:SolidPeso molecular:477.64Elvitegravir
CAS:<p>Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.</p>Fórmula:C23H23ClFNO5Pureza:98.43% - 99.57%Cor e Forma:SolidPeso molecular:447.88Telaprevir
CAS:<p>Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).</p>Fórmula:C36H53N7O6Pureza:96.9% - 98.89%Cor e Forma:SolidPeso molecular:679.854-Chloro-2-(trifluoroacetyl)aniline hydrochloride
CAS:<p>4-Chloro-2-(trifluoroacetyl)aniline hydrochloride is an inhibitor of HIV-1 RT (HIV reverse transcriptase) .</p>Fórmula:C8H6Cl2F3NOPureza:97.15%Cor e Forma:SolidPeso molecular:260.04Ceritinib
CAS:<p>Ceritinib (LDK378) is an ALK inhibitor with selective, ATP-competitive, and oral activity. Ceritinib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C28H36ClN5O3SPureza:98.52% - 99.77%Cor e Forma:SolidPeso molecular:558.14CGS 27023A
CAS:<p>CGS 27023A is a non-peptidic, potent, and orally active stromelysin inhibitor.</p>Fórmula:C18H24ClN3O5SPureza:99.08%Cor e Forma:SolidPeso molecular:429.92Picolamine
CAS:<p>Picolamine acts as a potential inhibitor of DPP-4.</p>Fórmula:C6H8N2Pureza:98.3%Cor e Forma:Light Yellow LiquidPeso molecular:108.14SB-3CT
CAS:<p>SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM).</p>Fórmula:C15H14O3S2Pureza:98% - 99.38%Cor e Forma:SolidPeso molecular:306.4S-methyl-KE-298
CAS:S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) productionFórmula:C13H16O3SPureza:97.33%Cor e Forma:SolidPeso molecular:252.33Tenofovir alafenamide hemifumarate
CAS:<p>Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.</p>Fórmula:C21H29N6O5PC4H4O4Pureza:99.33% - 99.96%Cor e Forma:SolidPeso molecular:534.51Trelagliptin succinate
CAS:<p>Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (</p>Fórmula:C22H26FN5O6Pureza:99.27% - 99.92%Cor e Forma:SolidPeso molecular:475.47Ilomastat
CAS:<p>Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.</p>Fórmula:C20H28N4O4Pureza:97.04% - 99.51%Cor e Forma:SolidPeso molecular:388.462-Benzylsuccinic acid
CAS:<p>2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.</p>Fórmula:C11H12O4Pureza:99.01% - ≥95%Cor e Forma:SolidPeso molecular:208.21(R)-MG-132
CAS:<p>(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.</p>Fórmula:C26H41N3O5Pureza:98.45%Cor e Forma:SolidPeso molecular:475.62NBD-557
CAS:<p>NBD-557 is a potentially HIV-1 inhibitor.</p>Fórmula:C17H24BrN3O2Pureza:99.52%Cor e Forma:SolidPeso molecular:382.3Sofosbuvir
CAS:<p>Sofosbuvir (GS 7977) is a uridine monophosphate analog inhibitor of hepatitis C virus (HCV) polymerase NS5B that is used as an antiviral agent in the treatment</p>Fórmula:C22H29FN3O9PPureza:99.77% - 99.82%Cor e Forma:SolidPeso molecular:529.45Vesnarinone
CAS:<p>Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, but</p>Fórmula:C22H25N3O4Pureza:96.69% - 98.13%Cor e Forma:SolidPeso molecular:395.45Lersivirine
CAS:<p>Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.</p>Fórmula:C17H18N4O2Pureza:98.01%Cor e Forma:SolidPeso molecular:310.35Boceprevir
CAS:<p>Boceprevir (SCH 503034), an oral HCV NS3 protease inhibitor, has a Ki of 14 nM and EC90 of 350 nM.</p>Fórmula:C27H45N5O5Pureza:95% - 99.16%Cor e Forma:SolidPeso molecular:519.68Trovirdine
CAS:<p>Trovirdine (LY300046) is a thiourea non-nucleoside reverse transcriptase inhibitor.</p>Fórmula:C13H13BrN4SPureza:98.12% - 98.50%Cor e Forma:SolidPeso molecular:337.24HCV-IN-31
CAS:<p>HCV-IN-31 is a HCV inhibitor with an EC50/EC95 of 15.7 μM.</p>Fórmula:C12H17FN6O3Pureza:99.83%Cor e Forma:SolidPeso molecular:312.3VCH-916
CAS:<p>VCH-916 is a new nonnucleoside inhibitor of HCV NS5B polymerase.</p>Fórmula:C26H36KNO4SPureza:98%Cor e Forma:SolidPeso molecular:497.732-PMPA
CAS:<p>2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).</p>Fórmula:C6H11O7PPureza:97.4% - 99.5%Cor e Forma:SolidPeso molecular:226.12Bz-RS-ISer(3-Ph)-Ome
CAS:<p>Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.</p>Fórmula:C17H17NO4Pureza:99.36% - 99.89%Cor e Forma:White CrystalPeso molecular:299.32Ledipasvir (acetone)
CAS:<p>Ledipasvir (acetone) (GS-5885 acetone) is an HCV NS5A polymerase inhibitor, used for the treatment of hepatitis C virus infection.</p>Fórmula:C52H60F2N8O7Pureza:99.72%Cor e Forma:SolidPeso molecular:947.08Methylchloroisothiazolinone/Methylisothiazolinone Mixture
CAS:<p>Methylchloroisothiazolinone/Methylisothiazolinone Mixture (Kathon 886MW),a preservative, activates MMPs in human bronchial epithelial cells.</p>Fórmula:C8H9ClN2O2S2Cor e Forma:SolidPeso molecular:264.75KP-457
CAS:<p>KP-457 is a ADAM17 and a TNFα converting enzyme TACE inhibitor that blocks the production of soluble TNF (sTNF).</p>Fórmula:C21H24N2O7S2Pureza:98.33%Cor e Forma:SolidPeso molecular:480.56Sitagliptin phosphate monohydrate
CAS:<p>Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.</p>Fórmula:C16H15F6N5O·H3PO4·H2OPureza:99.85% - 99.98%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:523.33(1S,2R)-Alicapistat
CAS:<p>(1S,2R)-Alicapistat inhibits calpains 1 and 2, shows promise for Alzheimer's, and has an IC50 of 395 nM.</p>Fórmula:C25H27N3O4Pureza:99.60%Cor e Forma:SoildPeso molecular:433.5Ledipasvir
CAS:<p>Ledipasvir (GS-5885) is a Hepatitis C Virus NS5A Inhibitor.</p>Fórmula:C49H54F2N8O6Pureza:99.96%Cor e Forma:SolidPeso molecular:889Rilpivirine HCl
CAS:<p>Rilpivirine HCl (Rilpivirine hydrochloride) is an NNRTI inhibitor with antiviral activity that inhibits the HIV virus.</p>Fórmula:C22H19ClN6Pureza:99.48%Cor e Forma:SolidPeso molecular:402.88(R)-Trolox
CAS:<p>(R)-Trolox is a selective tyrosinase inhibitor used in food, cosmetics, and pharmaceutical products.</p>Fórmula:C14H18O4Pureza:99.88%Cor e Forma:SolidPeso molecular:250.29Teneligliptin
CAS:<p>Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.</p>Fórmula:C22H30N6OSPureza:99.73%Cor e Forma:SolidPeso molecular:426.58Nelfinavir
CAS:<p>Nelfinavir (AG1341), with Ki=2 nM, is an HIV treatment and broad-spectrum anticancer drug.</p>Fórmula:C32H45N3O4SPureza:98.16% - 99.5%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:567.78Danoprevir
CAS:<p>Danoprevir (RG7227) is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).</p>Fórmula:C35H46FN5O9SPureza:98% - 99.35%Cor e Forma:SolidPeso molecular:731.83PSI
CAS:<p>PSI is a proteasome inhibitor.</p>Fórmula:C32H50N4O8Pureza:97% - 98.33%Cor e Forma:SolidPeso molecular:618.76Lanadelumab
CAS:<p>Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.</p>Pureza:95% - 95%Cor e Forma:LiquidGalegenimab
CAS:<p>Galegenimab (FHTR 2163; RG 6147; RO 7171009) is an HTRA1 antibody fragment for AMD research.</p>Pureza:95% - 95%Cor e Forma:LiquidKZR-504
CAS:KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 nM, 4.274 μM for LMP2 and LMP7, respectively).Fórmula:C21H23N3O6Cor e Forma:SolidPeso molecular:413.42Triton X-45(n=4)
CAS:<p>Triton X-45: nonionic, low HLB surfactant, dispersible in water, high Krafft point, relevant for HCV research.</p>Fórmula:C22H38O5Cor e Forma:SolidPeso molecular:382.53
