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EGFR
Daphnetin
CAS:486-35-1
Formula:
C9H6O4
Purity:
>90.0%(HPLC)
Color and Shape:
White to Light yellow to Light red powder to crystal
Molecular weight:
178.14
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin AG 1478
CAS:153436-53-4
Formula:
C16H14ClN3O2
Purity:
>98.0%(HPLC)
Color and Shape:
Light orange to Yellow to Green powder to crystal
Molecular weight:
315.76
Estimated delivery in United States, on Monday 31 Jan 2022
Butein
CAS:487-52-5
Formula:
C15H12O5
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
272.26
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin RG 14620
CAS:136831-49-7
Formula:
C14H8Cl2N2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
275.13
Estimated delivery in United States, on Monday 31 Jan 2022
Gefitinib
CAS:184475-35-2
Formula:
C22H24ClFN4O3
Purity:
>98.0%(HPLC)(T)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
446.91
Estimated delivery in United States, on Monday 31 Jan 2022
Genistein
CAS:446-72-0
Formula:
C15H10O5
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
270.24
Estimated delivery in United States, on Monday 31 Jan 2022
AEE 788
CAS:497839-62-0
Formula:
C27H32N6
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
440.60
Estimated delivery in United States, on Monday 31 Jan 2022
Dacomitinib
CAS:1110813-31-4
Formula:
C24H25ClFN5O2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
469.95
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin AG 494
CAS:133550-35-3
Formula:
C16H12N2O3
Purity:
>98.0%(HPLC)(N)
Color and Shape:
Light yellow to Amber to Dark green powder to crystal
Molecular weight:
280.28
Estimated delivery in United States, on Monday 31 Jan 2022
Mubritinib
CAS:366017-09-6
Formula:
C25H23F3N4O2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Gray to Brown powder to crystal
Molecular weight:
468.48
Estimated delivery in United States, on Monday 31 Jan 2022
Methyl 2,5-Dihydroxycinnamate
CAS:63177-57-1
Formula:
C10H10O4
Purity:
>96.0%(HPLC)
Color and Shape:
Very Pale Yellow - Yellow Solid
Molecular weight:
194.19
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin AG528
CAS:133550-49-9
Formula:
C18H14N2O3
Purity:
>97.0%(HPLC)
Color and Shape:
Light yellow to Amber to Dark green powder to crystal
Molecular weight:
306.32
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin AG 490
CAS:133550-30-8
Formula:
C17H14N2O3
Purity:
>98.0%(HPLC)(T)
Color and Shape:
Slightly Pale Yellow - Yellow Solid
Molecular weight:
294.31
Estimated delivery in United States, on Monday 31 Jan 2022
PD 153035 Hydrochloride
CAS:183322-45-4
Formula:
C16H14BrN3O2HCl
Purity:
>97.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
396.67
Estimated delivery in United States, on Monday 31 Jan 2022
BMS-599626
CAS:714971-09-2
Formula:
C27H27FN8O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
530.56
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin AG 835
CAS:133550-37-5
Formula:
C18H16N2O3
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Amber to Dark green powder to crystal
Molecular weight:
308.34
Estimated delivery in United States, on Monday 31 Jan 2022
Curcumin (Natural)
CAS:458-37-7
Formula:
C21H20O6
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
368.39
Estimated delivery in United States, on Monday 31 Jan 2022
WHI-P154
CAS:211555-04-3
Formula:
C16H14BrN3O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Yellow to Orange powder to crystal
Molecular weight:
376.21
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin A23
CAS:118409-57-7
Formula:
C10H6N2O2
Purity:
>98.0%(GC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
186.17
Estimated delivery in United States, on Monday 31 Jan 2022
Curcumin (Synthetic)
CAS:458-37-7
Formula:
C21H20O6
Purity:
>97.0%(T)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
368.39
Estimated delivery in United States, on Monday 31 Jan 2022
Tyrphostin RG 13022
CAS:136831-48-6
Formula:
C16H14N2O2
Purity:
>98.0%(GC)
Color and Shape:
White to Yellow to Green powder to crystal
Molecular weight:
266.30
Estimated delivery in United States, on Monday 31 Jan 2022
Pelitinib
CAS:257933-82-7
Formula:
C24H23ClFN5O2
Purity:
>97.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
467.93
Estimated delivery in United States, on Monday 31 Jan 2022
PD 158780
CAS:171179-06-9
Formula:
C14H12BrN5
Purity:
>97.0%(HPLC)
Color and Shape:
White to Yellow to Green powder to crystal
Molecular weight:
330.19
Estimated delivery in United States, on Monday 31 Jan 2022
EGFR-IN-1
CAS:1625677-63-5
EGFR-IN-1 displays strong antiproliferative activity against the H1975 cells and the first line mutant HCC827 …
Formula:
C28H30N6O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
514.58
Estimated delivery in United States, on Monday 7 Feb 2022
Mobocertinib
CAS:1847461-43-1
Mobocertinib is a potent inhibitor of epidermal growth factor receptor (EGFR) and an antineoplastic agent
Formula:
C32H39N7O4
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
585.71
Estimated delivery in United States, on Monday 7 Feb 2022
E-4031
CAS:113559-13-0
E-4031 is a methanesulfonanilide class III antiarrhythmic agent that prolongs cardiac action potential duration by …
Formula:
C21H29Cl2N3O3S
Molecular weight:
474.44
Estimated delivery in United States, on Monday 7 Feb 2022
Biochanin A
CAS:491-80-5
Biochanin A is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. …
Formula:
C16H12O5
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
284.26
Estimated delivery in United States, on Monday 7 Feb 2022
TX1-85-1
CAS:1603845-32-4
TX1-85-1 induces partial degradation of Her3 protein and attenuates Her3-dependent signaling. TX1-85-1 is an irreversible …
Formula:
C32H36N8O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
580.68
Estimated delivery in United States, on Monday 7 Feb 2022
Afatinib D6
CAS:1313874-96-2
Afatinib D6 (BIBW 2992 D6) is a deuterium-labeled Afatinib. Afatinib is an irreversible EGFR family …
Formula:
C24H19D6ClFN5O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
491.98
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR mutant-IN-1
EGFR mutant- in-1, A 5-methylpyrimidopyridone derivative are effective selective EGFRL858R/T790M/C797S mutant inhibitors with IC50 of …
Formula:
C34H39ClFN7O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
632.17
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR Inhibitor
CAS:879127-07-8
EGFR inhibitor is a cell permeable and selective inhibitor of EGFR kinase (IC50: 21 nM) …
Formula:
C21H18F3N5O
Purity:
99.15%
Color and Shape:
solid
Molecular weight:
413.4
Estimated delivery in United States, on Monday 7 Feb 2022
AST2818 mesylate
CAS:2130958-55-1
AST2818 mesylate,is an irreversible tyrosine kinase inhibitor that selectively inhibits EGFR mutations, especially T790M.
Formula:
C29H35F3N8O5S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
664.7
Estimated delivery in United States, on Monday 7 Feb 2022
lavendustin A
CAS:125697-92-9
lavendustin A is a potent, cell-permeable inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase.
Formula:
C21H19NO6
Purity:
98.17%
Color and Shape:
Off-White Solid
Molecular weight:
381.38
Estimated delivery in United States, on Monday 7 Feb 2022
Lifirafenib
CAS:1446090-79-4
Lifirafenib is a potent inhibitor of RAF family kinases and EGFR in biochemical assays with …
Formula:
C25H17F3N4O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
478.42
Estimated delivery in United States, on Monday 7 Feb 2022
BKI-1369
CAS:1951431-22-3
BKI-1369 is a bumped kinase inhibitor. BKI-1369 increases hERG-inhibitory activity (IC50:1.52 μM).
Formula:
C23H27N7O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
417.51
Estimated delivery in United States, on Monday 7 Feb 2022
Mutant EGFR inhibitor
CAS:1421373-62-7
Mutant EGFR inhibitor is a selective and potent Mutated EGFR inhibitor, inhibits L858R activating mutant, …
Formula:
C27H30ClN7O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
520.03
Estimated delivery in United States, on Monday 7 Feb 2022
Sigma-1 receptor antagonist 3
CAS:1639220-17-9
Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (1) receptor(Ki : …
Formula:
C19H23ClFN3O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
363.86
Estimated delivery in United States, on Monday 7 Feb 2022
Allitinib
CAS:897383-62-9
Allitinib (AST-1306) is an orally active and irreversible EGFR and ErbB2 inhibitor with IC50s of …
Formula:
C24H18ClFN4O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
448.88
Estimated delivery in United States, on Monday 7 Feb 2022
Dihydroberberine
CAS:483-15-8
Dihydroberberine has anti-atherosclerotic, anti-inflammatory, hypolipidemic and antitumor activities. It inhibits human ether-a-go-go-related gene (hERG) channels …
Formula:
C20H19NO4
Purity:
99.89%
Color and Shape:
solid
Molecular weight:
337.4
Estimated delivery in United States, on Monday 7 Feb 2022
PF 6274484
CAS:1035638-91-5
PF 6274484, a high affinity, irreversible covalent inhibitor of EGFR kinase with Ki of 0.14 …
Formula:
C18H14ClFN4O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
372.8
Estimated delivery in United States, on Monday 7 Feb 2022
AG-825
CAS:149092-50-2
AG-825(Tyrphostin AG-825) is a potential agent for overcoming Mn-induced neurotoxicity or AD development[5] and is …
Formula:
C19H15N3O3S2
Purity:
98.00%
Color and Shape:
Yellow Solid
Molecular weight:
397.47
Estimated delivery in United States, on Monday 7 Feb 2022
Nazartinib
CAS:1508250-71-2
Nazartinib (EGF816, NVS-816) is a covalent, irreversible, mutant-selective EGFR inhibitor that has nanomolar inhibitory potency …
Formula:
C26H31ClN6O2
Purity:
98.63%
Color and Shape:
Solid Powder
Molecular weight:
495.02
Estimated delivery in United States, on Monday 7 Feb 2022
Canertinib
CAS:267243-28-7
Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squamous cell carcinoma in …
Formula:
C24H25ClFN5O3
Purity:
100.00%
Color and Shape:
White Or Similar To White Crystalline Powder
Molecular weight:
485.94
Estimated delivery in United States, on Monday 7 Feb 2022
Naquotinib mesylate
CAS:1448237-05-5
Naquotinib mesylate is an orally available, mutant-selective and irreversible inhibitor of EGFR(iC50s of 8-33 nM …
Formula:
C31H46N8O6S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
658.81
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR-IN-2
CAS:1643497-70-4
EGFR-IN-2 is a non-covalent, mutation-selective and irreversible second-generation EGFR inhibitor.
Formula:
C26H33N9O3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
551.66
Estimated delivery in United States, on Monday 7 Feb 2022
Ginsenoside Rh2
CAS:78214-33-2
Ginsenoside Rh2, an extract of red Panax ginseng, is a potent anti-inflammatory and anticancer drug.
Formula:
C36H62O8
Purity:
99.65%
Color and Shape:
White Powder
Molecular weight:
622.87
Estimated delivery in United States, on Monday 7 Feb 2022
PD158780
CAS:171179-06-9
PD 158780 reversibly inhibits auto and transphosphorylation of all four members of the ErbB receptor …
Formula:
C14H12BrN5
Purity:
99.16%
Color and Shape:
solid
Molecular weight:
330.19
Estimated delivery in United States, on Monday 7 Feb 2022
Lapatinib
CAS:231277-92-2
Lapatinib is a dual inhibitor of Lapatinib is a dual ErbB2/EGFR (IC50: 9.2/10.8 nM) inhibitor
Formula:
C29H26ClFN4O4S
Purity:
99.03%
Color and Shape:
Powder
Molecular weight:
581.06
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR-IN-11
EGFR-IN-11 significantly suppresses the EGFR phosphorylation, induce the apoptosis, and arrest cell cycle at G0/G1.EGFR-IN-11 …
Formula:
C29H35N9O2S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
573.71
Estimated delivery in United States, on Monday 7 Feb 2022
(Rac)-JBJ-04-125-02
CAS:2140807-05-0
JBJ-04-125-02 is effective as a single agent in both in vitro and in vivo models …
Formula:
C29H26FN5O3S
Purity:
95.85%
Molecular weight:
543.6
Estimated delivery in United States, on Monday 7 Feb 2022
Chrysophanic Acid
CAS:481-74-3
Chrysophanic acid is an EGFR/mTOR pathway inhibitor, which can be found in rhubarb, and sorrel.
Formula:
C15H10O4
Purity:
99.44%
Color and Shape:
Physical Description Golden Yellow Plates Or Brown Powder Melting Point 196°C
Molecular weight:
254.24
Estimated delivery in United States, on Monday 7 Feb 2022
AZD3759 hydrochloride
CAS:1626387-81-2
AZD3759 (hydrochloride) is an effective, orally active and central nervous system-penetrant EGFR inhibitor. At Km …
Formula:
C22H24Cl2FN5O3
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
496.36
Estimated delivery in United States, on Monday 7 Feb 2022
Desmethyl Erlotinib
CAS:183321-86-0
OSI-420 is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 nM).
Formula:
C21H21N3O4
Purity:
98.62%
Molecular weight:
379.41
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR-IN-9
CAS:1226549-39-8
EGFR-IN-9 has antitumor activity. EGFR-IN-9 is a potent EGFR kinase inhibitor with IC50s of 7 …
Formula:
C29H24N4O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
476.53
Estimated delivery in United States, on Monday 7 Feb 2022
Chalcone
CAS:94-41-7
Chalcone is an aromatic ketone that forms the central core for a variety of important …
Formula:
C15H12O
Purity:
97.89%
Color and Shape:
Solid
Molecular weight:
208.26
Estimated delivery in United States, on Monday 7 Feb 2022
ZD-4190
CAS:413599-62-9
ZD-4190 is a inhibitor of the vascular endothelial cell growth factor receptor 2 (VEGFR2) and …
Formula:
C19H16BrFN6O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
459.28
Estimated delivery in United States, on Monday 7 Feb 2022
Osimertinib
CAS:1421373-65-0
Osimertinib is a small molecule tyrosine kinase receptor inhibitor and antineoplastic agent that is used …
Formula:
C28H33N7O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
499.61
Estimated delivery in United States, on Monday 7 Feb 2022
O-Desmethyl gefitinib D8
O-Desmethyl gefitinib D8 is a deuterium labeled O-Desmethyl gefitinib that is an active metabolite of …
Formula:
C21H14D8ClFN4O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
440.93
Estimated delivery in United States, on Monday 7 Feb 2022
AG 99
CAS:122520-85-8
AG-99 is an inhibitor of EGFR kinase (IC50: 10 µM in the human epidermoid carcinoma …
Formula:
C10H8N2O3
Purity:
99.67%
Color and Shape:
solid
Molecular weight:
204.18
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR-IN-8
CAS:2407957-87-1
EGFR-IN-8 can be a promising candidate for further development to target EGFR TKI-resistant NSCLC. EGFR-IN-8 …
Formula:
C32H23ClF3N7O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
662.02
Estimated delivery in United States, on Monday 7 Feb 2022
Tyrphostin AG 112
CAS:144978-82-5
Tyrphostin AG 112 is an inhibitor of EGFR phosphorylation.
Formula:
C13H8N4O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
236.23
Estimated delivery in United States, on Monday 7 Feb 2022
Poziotinib hydrochloride
CAS:1429757-68-5
Poziotinib hydrochloride irreversibly inhibits EGFR (HER1 or ErbB1), including EGFR mutants, HER2, and HER4, thereby …
Formula:
C23H22Cl3FN4O3
Purity:
99.69%
Molecular weight:
527.8
Estimated delivery in United States, on Monday 7 Feb 2022
PF-06459988
CAS:1428774-45-1
PF-06459988 is an irreversible T790M-Containing EGFR Mutants inhibitor.
Formula:
C19H22ClN7O3
Color and Shape:
Solid
Molecular weight:
431.88
Estimated delivery in United States, on Monday 7 Feb 2022
Lapatinib ditosylate monohydrate
CAS:388082-78-8
Lapatinib is a tyrosine kinase receptor inhibitor used in the therapy of advanced breast cancer …
Formula:
C29H26ClFN4O4S·2(C7H8O3S)·H2O
Purity:
99.00%
Color and Shape:
Colourless To Light-Yellow Crystal
Molecular weight:
943.47
Estimated delivery in United States, on Monday 7 Feb 2022
HS-10296 hydrochloride
CAS:2134096-03-8
HS-10296 hydrochloride is a small molecule inhibitor of EGFR-activating mutations and T790M-resistant mutation with limited …
Formula:
C30H36ClN7O2
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
562.1
Estimated delivery in United States, on Monday 7 Feb 2022
Astragaloside VI
CAS:84687-45-6
Astragaloside VI could improve wound healing by activating the EGFR/ERK signaling pathway.
Formula:
C47H78O19
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
947.11
Estimated delivery in United States, on Monday 7 Feb 2022
JCN037
CAS:2305154-31-6
JCN037 is potent, non-covalent and brain-penetrant inhibitor of EGFR(EGFR, p-wtEGFR and pEGFRv with IC50 of …
Formula:
C16H11BrFN3O2
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
376.18
Estimated delivery in United States, on Monday 7 Feb 2022
Erlotinib hydrochloride
CAS:183319-69-9
Erlotinib is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment of …
Formula:
C22H23N3O4·HCl
Purity:
99.52%
Color and Shape:
White Or Off-White Powder
Molecular weight:
429.9
Estimated delivery in United States, on Monday 7 Feb 2022
Sapitinib
CAS:848942-61-0
AZD8931, a reversible, ATP competitive inhibitor of EGFR(IC50=4 nM), ErbB2(IC50=3 nM) and ErbB3(IC50=4 nM), is …
Formula:
C23H25ClFN5O3
Purity:
99.83%
Color and Shape:
solid
Molecular weight:
473.93
Estimated delivery in United States, on Monday 7 Feb 2022
Osimertinib dimesylate
CAS:2070014-82-1
Osimertinib dimesylate is an irreversible and mutant selective EGFR inhibitor (IC50s: 12 and 1 nM …
Formula:
C30H41N7O8S2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
691.82
Estimated delivery in United States, on Monday 7 Feb 2022
BI-4020
BI-4020 is a fourth-generation, non-covalent, and orally active inhibitor of EGFR tyrosine kinase.
Formula:
C30H38N8O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
542.68
Estimated delivery in United States, on Monday 7 Feb 2022
Mutated EGFR-IN-2
CAS:2050906-97-1
Mutated EGFR-IN-2 is an inhibitor of mutant-selective EGFR.
Formula:
C29H35FN8O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
562.64
Estimated delivery in United States, on Monday 7 Feb 2022
AG-1557 hydrochloride (189290-58-2(free base))
AG-1557 is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: 8.194).
Formula:
C16H15ClIN3O2
Purity:
98.95%
Color and Shape:
solid
Molecular weight:
443.66
Estimated delivery in United States, on Monday 7 Feb 2022
RG 13022
CAS:136831-48-6
RG13022 is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF receptor (IC50: …
Formula:
C16H14N2O2
Purity:
99.42%
Color and Shape:
solid
Molecular weight:
266.29
Estimated delivery in United States, on Monday 7 Feb 2022
Lapatinib Ditosylate
CAS:388082-77-7
Lapatinib is an effective EGFR and ErbB2 inhibitor (IC50: 10.8/9.2 nM for EGFR/ErbB2).
Formula:
C29H26ClFN4O4S·2C7H8O3S
Purity:
98.42%
Color and Shape:
Yellow Solid
Molecular weight:
925.46
Estimated delivery in United States, on Monday 7 Feb 2022
O-Desmethyl gefitinib
CAS:847949-49-9
O-Desmethyl gefitinib inhibits EGFR (IC50: 36 nM in subcellular assays). In human plasma, O-Desmethyl gefitinib …
Formula:
C21H22ClFN4O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
432.88
Estimated delivery in United States, on Monday 7 Feb 2022
Lazertinib
CAS:1903008-80-9
Lazertinib is an effective, highly mutant-selective and irreversible EGFR-TKI with IC50 values of 1.7 nM, …
Formula:
C30H34N8O3
Purity:
98.70%
Color and Shape:
Solid
Molecular weight:
554.64
Estimated delivery in United States, on Monday 7 Feb 2022
Nuvenzepine
CAS:96487-37-5
Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.
Formula:
C19H20N4O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
336.39
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR/ErbB2 Inhibitor
CAS:179248-61-4
EGFR/ErbB2 Inhibitor is a cell-permeable inhibitor of EGFR and c-ErbB2 (IC50s = 20 and 79 …
Formula:
C23H21N3O3
Molecular weight:
387.43
Estimated delivery in United States, on Monday 7 Feb 2022
Tyrphostin AG 528
CAS:133550-49-9
Tyrphostin AG 528 is an inhibitor of EGFR (IC50: 4.9 μM) and ErbB2 (IC50: 2.1 …
Formula:
C18H14N2O3
Purity:
99.74%
Color and Shape:
solid
Molecular weight:
306.32
Estimated delivery in United States, on Monday 7 Feb 2022
Epertinib
CAS:908305-13-5
Epertinib is a reversible and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 (IC50s: …
Formula:
C30H27ClFN5O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
560.02
Estimated delivery in United States, on Monday 7 Feb 2022
Ligustroside
CAS:35897-92-8
Ligustroside shows little antioxidant, and anti-inflammatory properties, it shows a significant inhibition effect on prostaglandin …
Formula:
C25H32O12
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
524.5
Estimated delivery in United States, on Monday 7 Feb 2022
WZ3146
CAS:1214265-56-1
WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and EGFR(E746_A750) with IC50 of 2 nM …
Formula:
C24H25ClN6O2
Purity:
98.95%
Color and Shape:
solid
Molecular weight:
464.95
Estimated delivery in United States, on Monday 7 Feb 2022
Afatinib free base
CAS:850140-72-6
Afatinib is an irreversible inhibitor of EGFR family (EGFR-wt, EGFR-L858R, EGFR-L858R/T790M and HER2 with IC50s …
Formula:
C24H25ClFN5O3
Purity:
99.90%
Color and Shape:
Off-White Solid
Molecular weight:
485.94
Estimated delivery in United States, on Monday 7 Feb 2022
CHMFL-EGFR-202
CAS:2089381-40-6
CHMFL-EGFR-202 is a potent, irreversible inhibitor of EGFR mutant kinase (IC50s: 5.3 nM and 8.3 …
Formula:
C25H24ClN7O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
489.96
Estimated delivery in United States, on Monday 7 Feb 2022
DBPR112
CAS:1226549-49-0
DBPR112 has an IC50 of 15 nM and 48 nM for EGFRWT and EGFRL858R / …
Formula:
C32H31N5O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
533.62
Estimated delivery in United States, on Monday 7 Feb 2022
EGFR-IN-1 hydrochloride
CAS:2227455-78-7
EGFR-IN-1 hydrochloride displays strong antiproliferative activity against the H1975 cells and the first line mutant …
Formula:
C28H31ClN6O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
551.04
Estimated delivery in United States, on Monday 7 Feb 2022
ICA-105574
CAS:316146-57-3
ICA-105574 is an activator of hERG that binds to the channel to remove inactivation, thus …
Formula:
C19H14N2O4
Purity:
99.77%
Molecular weight:
334.33
Estimated delivery in United States, on Monday 7 Feb 2022
PD153035
CAS:153436-54-5
PD153035 hydrochloride is an effective and selective inhibitor of EGFR (Ki/IC50: 5.2/29 pM, in cell-free …
Formula:
C16H14BrN3O2
Purity:
99.29%
Color and Shape:
solid
Molecular weight:
360.21
Estimated delivery in United States, on Monday 7 Feb 2022
AG1557
CAS:189290-58-2
AG-1557 is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: 8.194).
Formula:
C16H14IN3O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
407.21
Estimated delivery in United States, on Monday 7 Feb 2022
AZD3759
CAS:1626387-80-1
AZD3759 is an orally active, effective and central nervous system-penetrant EGFR inhibitor. The IC50 values …
Formula:
C22H23ClFN5O3
Purity:
99.36%
Color and Shape:
White To Off-White Solid
Molecular weight:
459.9
Estimated delivery in United States, on Monday 7 Feb 2022
BMS-690514
CAS:859853-30-8
BMS-690514 is a potent and orally active inhibitor of EGFR and VEGFR. It has IC50s …
Formula:
C19H24N6O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
368.43
Estimated delivery in United States, on Monday 7 Feb 2022
Endoxifen Z-isomer
CAS:112093-28-4
Endoxifen (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity …
Formula:
C25H27NO2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
373.49
Estimated delivery in United States, on Monday 7 Feb 2022
HKI-357
CAS:848133-17-5
HKI-357 is an irreversible dual inhibitor of EGFR and ERBB2 (IC50s: 34 nM and 33 …
Formula:
C31H29ClFN5O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
574.05
Estimated delivery in United States, on Monday 7 Feb 2022
BGB-102
CAS:807640-87-5
BGB-102 is a potent multi-kinase inhibitor against HER2, EGFR, and HER4 (IC50s: 18 nM, 9.6 …
Formula:
C22H25BrN4O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
457.36
Estimated delivery in United States, on Monday 7 Feb 2022
Theliatinib
CAS:1353644-70-8
Theliatinib, a potent and highly selective EGFR inhibitor, with anti-tumor activity. Ki of 0.05 nM …
Formula:
C25H26N6O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
442.5
Estimated delivery in United States, on Monday 7 Feb 2022
Avitinib maleate
CAS:1557268-88-8
Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor.
Formula:
C30H30FN7O6
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
603.61
Estimated delivery in United States, on Monday 7 Feb 2022
Tyrphostin A1
CAS:2826-26-8
Tyrphostin A1 is an inhibitor of EGFR tyrosine kinase .
Formula:
C11H8N2O
Purity:
99.13%
Color and Shape:
solid
Molecular weight:
184.19
Estimated delivery in United States, on Monday 7 Feb 2022
Erlotinib
CAS:183321-74-6
Erlotinib is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment of …
Formula:
C22H23N3O4
Purity:
99.98%
Color and Shape:
White To Off-White Powder
Molecular weight:
393.44
Estimated delivery in United States, on Monday 7 Feb 2022
JH-XI-10-02
CAS:2209085-22-1
JH-XI-10-02 causes proteasomal degradation, does not affect CDK8 mRNA levels. JH-XI-10-02 shows no effect on …
Formula:
C53H69N5O9
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
920.14
Estimated delivery in United States, on Monday 7 Feb 2022
