
Cell Cycle/Checkpoint
Cell cycle/checkpoint inhibitors are compounds that disrupt the normal progression of the cell cycle, particularly at key regulatory checkpoints. These inhibitors are crucial for studying cell division, understanding cancer cell proliferation, and developing anti-cancer therapies. By targeting specific phases of the cell cycle, these inhibitors can induce cell cycle arrest, leading to apoptosis or senescence in rapidly dividing cells. At CymitQuimica, we offer a diverse range of high-quality cell cycle/checkpoint inhibitors to support your research in cancer biology, cell biology, and drug development.
Subcategories of "Cell Cycle/Checkpoint"
- Aurora Kinase(115 products)
- CDK(547 products)
- Cell Cycle Arrest(5 products)
- Chk(48 products)
- DYRK(46 products)
- Dynamin(27 products)
- Ferroptosis(227 products)
- HSP(180 products)
- Integrin(275 products)
- Kinesin(87 products)
- LIM Kinase(21 products)
- Microtubule Associated(273 products)
- PKC(127 products)
- PLK(25 products)
- ROCK(61 products)
- Rho(6 products)
- Wee1(14 products)
- c-Myc(77 products)
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Found 3920 products of "Cell Cycle/Checkpoint"
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4-Deoxy-xylo-uridine
CAS:Nucleoside Derivatives - Xylo-nucleosides; 4-Deoxy pyrimidine nucleosidesFormula:C9H12N2O5Color and Shape:SolidMolecular weight:228.2Ref: TM-TNU1366
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2'-Deoxy-2'-fluoro-3',5'-bis-O-TBDMS-uridine
CAS:Nucleoside Derivatives –Fluoro-modified nucleosides;Formula:C21H39FN2O5Si2Color and Shape:SolidMolecular weight:474.71Ref: TM-TNU1512
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire4-Chloro-5-iodo-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine
CAS:4-Chloro-5-iodo-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine is a Nucleoside Derivative - Halo-nucleoside, 7-Deaza-purine nucleoside.Formula:C11H11ClIN3O3Color and Shape:SolidMolecular weight:395.58Ref: TM-TNU1025
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireN4-Desmethyl-N5-Methyl wyosine
CAS:N4-Desmethyl-N5-Methyl wyosine is a Nucleoside Derivative - Bi-/Tri-cyclic nucleoside; naturally modified ribo-nucleoside.Formula:C14H17N5O5Color and Shape:SolidMolecular weight:335.32Ref: TM-TNU0179
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire1-[6-(Diethoxyphosphinyl)-2-O-(2-methoxyethyl)-β-D-ribo-hexofuranosyl]uracil
Nucleoside Derivatives - Phosphorus-containing nucleosides; 2’-Modified nucleosides; 5’-Modified nucleosidesColor and Shape:SoildRef: TM-TNU1286
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire1,2'-O-Dimethyl guanosine
CAS:1,2'-O-Dimethyl guanosine is a Nucleoside Derivative - 3'-Modified nucleoside, N-Methylated/ alkylated nucleoside.Formula:C12H17N5O5Color and Shape:SolidMolecular weight:311.29Ref: TM-TNU0572
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireIsocytidine
CAS:Nucleosides - isocytidine derivativeFormula:C9H13N3O5Color and Shape:SolidMolecular weight:243.22Ref: TM-TNU0049
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2',3',5'-Tri-O-benzoyl-5-methoxyuridine
CAS:2',3',5'-Tri-O-benzoyl-5-methoxyuridine is a 5-Modified Pyrimidine Nucleoside.Formula:C31H26N2O10Color and Shape:SolidMolecular weight:586.55Ref: TM-TNU0806
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2-Methoxy-9-(β-D-ribofuranosyl)purine
CAS:Nucleoside Derivatives - 6-De-aminopurine nucleosides, 2-Modified purine nucleosidesFormula:C11H14N4O5Color and Shape:SolidMolecular weight:282.25Ref: TM-TNU1109
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2'-Deoxy-2'-fluoro-N1-methyl inosine
CAS:Nucleoside Derivatives - 2’-Modified nucleosides, Fluoro-modified nucleosides, N-Methylated /alkylated nucleosidesFormula:C11H13FN4O4Color and Shape:SolidMolecular weight:284.24Ref: TM-TNU0548
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2'-Chloro-2'-deoxyuridine
CAS:2'-Chloro-2'-deoxyuridine is a Halo-nucleoside.Formula:C9H11ClN2O5Color and Shape:SolidMolecular weight:262.65Ref: TM-TNU0073
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2'-Deoxy-N6,N6-dimethyladenosine
CAS:2'-Deoxy-N6,N6-dimethyladenosine is a Nucleoside Derivative - 6-Modified purine nucleoside.Formula:C12H17N5O3Color and Shape:SolidMolecular weight:279.3Ref: TM-TNU1369
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire1-(b-D-Xylofuranosyl)-5-methylcytosine
CAS:Nucleoside Derivatives –5-Modified pyrimidine nucleosides;Xylo-nucleosidesFormula:C10H15N3O5Color and Shape:SolidMolecular weight:257.24Ref: TM-TNU0521
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire3'-O-Methyl-5-methyluridine
CAS:3'-O-Methyl-5-methyluridine is a Nucleoside Derivative - 3'-Modified nucleoside.Formula:C11H16N2O6Color and Shape:SolidMolecular weight:272.25Ref: TM-TNU1393
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire1-Amino-7-cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl)guanine
CAS:Nucleoside Derivatives - Xylo-nucleosides; 8-Modified purine nucleosides; Amino nucleosides; N-Methylated alkylated nucleosidesFormula:C14H20N6O6Color and Shape:SolidMolecular weight:368.35Ref: TM-TNU0387
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire6-Chloro-9-(2,3,5-tri-O-benzoyl-2-C-methyl-β-D-ribofuranosyl)-9H-purine
CAS:6-Chloro-9-(2,3,5-tri-O-benzoyl-2-C-methyl-β-D-ribofuranosyl)-9H-purine is a 2'-C-Methyl nucleoside; Halo-nucleoside.Formula:C32H25ClN4O7Color and Shape:SolidMolecular weight:613.02Ref: TM-TNU0772
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire1-(b-D-Xylofuranosyl)-5-trifluoromethyluracil
1-(b-D-Xylofuranosyl)-5-trifluoromethyluracil is a Nucleoside Derivative - Xylo-nucleoside, Fluoro-modified nucleoside, 5-Modified pyrimidine nucleoside.Color and Shape:SoildRef: TM-TNU1483
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2-Cyanoadenosine
CAS:Nucleoside Derivatives - 2’-Modified purine nucleosidesFormula:C11H12N6O4Color and Shape:SolidMolecular weight:292.25Ref: TM-TNU0296
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire5-Iodoarabinouridine
CAS:5-Iodoarabinouridine is a Halo-nucleoside; Arabino-nucleoside.Formula:C9H11IN2O6Color and Shape:SolidMolecular weight:370.1Ref: TM-TNU0784
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireN1-Ethylpseudouridine
CAS:N1-Ethylpseudouridine is a Nucleoside Derivative - C-nucleoside; N-Methylated nucleoside.Formula:C11H16N2O6Color and Shape:SolidMolecular weight:272.25Ref: TM-TNU0062
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire2'-Deoxy-O6-[2-(4-nitrophenylethyl)]guanosine
CAS:2'-Deoxy-O6-[2-(4-nitrophenylethyl)]guanosine is a Nucleoside Derivative - 6-Modified purine nucleoside.Formula:C18H20N6O6Color and Shape:SolidMolecular weight:416.39Ref: TM-TNU1005
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireKS15
CAS:KS15 is a cryptochrome (CRY) inhibitor that promotes G1 cell cycle arrest, enhances drug sensitivity in MCF-7 cells, antitumour against human breast cancer.Formula:C20H22BrNO4Color and Shape:SolidMolecular weight:420.33'-O-DMTr-thymidine 5'-CE phosphoramidite
CAS:3'-O-DMTr-thymidine 5'-CE phosphoramidite (2'-OMe-U Phosphoramidite) is a purine nucleoside analog and phosphoramidite derivative .Formula:C40H49N4O8PPurity:99.42%Color and Shape:SolidMolecular weight:744.81Lifitegrast sodium
CAS:Lifitegrast sodium (SAR-1118-023 sodium) is an integrin antagonist that reduces ocular surface inflammation and can be used to study dry eye.Formula:C29H23Cl2N2NaO7SPurity:99.33%Color and Shape:SolidMolecular weight:637.46GP-82996
CAS:GP-82996 (CINK4) inhibits CDK4/6; IC50s: 1.5 μM (CDK4/D1), 5.6 μM (CDK6/D1), 25 μM (Cdk5/p35); triggers U2OS cancer cell apoptosis.Formula:C27H32N6OPurity:99.94%Color and Shape:SolidMolecular weight:456.58HDGFRP2/PSIP1-IN-1
CAS:Compound BPP (HDGFRP2/PSIP1-IN-1) is a dual inhibitor targeting the PWWP domains of Hepatoma-derived Growth Factor Related Protein 2 (HDGFRP2) and its homologue PSIP1. This compound effectively hinders the occurrence and progression of Diffuse Intrinsic Pontine Glioma (DIPG). It demonstrates binding affinity with a Kd value of 7 μM for HDGFRP2, indicative of its efficient ligand efficacy at 0.47. Additionally, Compound BPP exhibits a Kd value of 27 μM when binding to the PSIP1 PWWP domain, and a Kd value of 14 μM against HDGFRP3, confirming its potency as an inhibitor within the HDGFRP2 PWWP subfamily.Formula:C8H6BrN3Color and Shape:SolidMolecular weight:224.06Napropamide
CAS:Napropamide is an acetamide herbicide that inhibits root growth to control annual grasses and broadleaf weeds.Formula:C17H21NO2Purity:99.14%Color and Shape:Colorless Crystals; (Tech Brown Solid) White-Like CrystalMolecular weight:271.35N-6-Furfurylguanosine
CAS:N-6-Furfurylguanosine (kinetin riboside) is a purine nucleoside analog with cytotoxicity, inhibiting the growth of cancer cells.Formula:C15H18N6O5Purity:99.58%Color and Shape:SolidMolecular weight:362.345,6-Dihydrothymidine
CAS:2'-Deoxy-N2-methylguanosine is a purine nucleoside analog that can be used as a chemical probe to study DNA-protein interactions.Formula:C10H16N2O5Purity:99.90%Color and Shape:SolidMolecular weight:244.24(S)-GNA-T-phosphoramidite
CAS:(S)-GNA-T-phosphoramidite is a nucleoside analog commonly used in the synthesis of other active compounds.Formula:C38H47N4O7PPurity:97.08%Color and Shape:SolidMolecular weight:702.782'-O-Methyl-5-methyl uridine
CAS:2'-O-Methyl-5-methyl uridine is a 2'-O-Methyl nucleoside.Formula:C11H16N2O6Color and Shape:SolidMolecular weight:272.25Ref: TM-TNU0716
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire5-Aza-7-deazaguanine
CAS:5-Aza-7-deazaguanine is a non-natural substituted nucleobase with potential antiviral activity, used in cancer and bacterial infection research.Formula:C5H5N5OPurity:98.87%Color and Shape:SolidMolecular weight:151.13Yuanhuacine
CAS:Gnidilatidin is a biochemical.Formula:C37H44O10Color and Shape:SolidMolecular weight:648.7492'-O-Methyl isocytidine
CAS:Isocytidine derivative; 2’-O-Methyl nucleosideFormula:C10H15N3O5Color and Shape:SolidMolecular weight:257.24Ref: TM-TNU0050
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire6-Methylmercaptopurine riboside
CAS:6-Methylmercaptopurine riboside is a purine nucleoside analogue applicable to biochemical experiments and drug synthesis studies.Formula:C11H14N4O4SColor and Shape:SolidMolecular weight:298.32TCRS-417
CAS:TCRS-417 (T417) inhibits PBX1-DNA interaction in mammalian cells or cell clusters, used in autoimmune and neurodegenerative disease research.Formula:C25H19FN2O5Color and Shape:SolidMolecular weight:446.43N4-Benzoyl-5'-O-(4,4'-dimethoxytrityl)-2'-O-(2-methoxyethyl)-5-methylcytidine
CAS:Nucleoside Derivatives - 2’-Modified nucleoside, Protected nucleosides with NH2/OH open; Ready for phosphorylationFormula:C41H43N3O9Color and Shape:SolidMolecular weight:721.79Ref: TM-TNU1115
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquire(S)-GNA-G(iBu) phosphoramidite
CAS:(S)-GNA-G(iBu) phosphoramidite is a Nucleoside Derivative - Acyclic nucleoside;Nucleoside Phosphoramidite.Formula:C42H52N7O7PColor and Shape:SolidMolecular weight:797.88Ref: TM-TNU1440
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireX5050
CAS:X5050 is a REST inhibitor, with an EC 50 of 2.1 μM.Formula:C17H15N3O3Color and Shape:SolidMolecular weight:309.325Cytidine (Standard)
CAS:Cytidine (Standard) is the standard substance of Cytidine, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Cytidine (Cytosine-1-β-D-ribofuranoside) is a pyrimidine nucleoside comprised of a cytosine bound to ribose via a beta-N1-glycosidic bond. Cytidine is a precursor for uridine. Both cytidine and uridine are utilized in RNA synthesis.Formula:C9H13N3O5Color and Shape:Physical Description White Crystalline Powder (Ntp 1992)Molecular weight:243.225-Bromocytidine
CAS:5-Bromocytidine is a nucleoside analog that is a key disinfection by-product of drinking water and may interfere with nucleic acid synthesis.Formula:C9H12BrN3O5Purity:99.63%Color and Shape:SolidMolecular weight:322.115'-O-(4,4'-Dimethoxytrityl)-2'-O-(2-methoxyethyl)-5-methyluridine
CAS:5'-O-(4,4'-Dimethoxytrityl)-2'-O-(2-methoxyethyl)-5-methyluridine is a Nucleoside Derivative - 2'-Modified nucleoside; Protected nucleoside with NH2/OH open;Formula:C34H38N2O9Color and Shape:SolidMolecular weight:618.67Ref: TM-TNU1094
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireCeftriaxone Sodium
CAS:Ceftriaxone Sodium is a sporotaxin antibiotic that inhibits GSK3β and Aurora B. It is used in the study of sepsis and infective endocarditis.Formula:C18H17N8NaO7S3Color and Shape:SolidMolecular weight:576.5622'-Amino-2'-deoxy-b-D-arabino-5-methyl uridine
CAS:2'-Amino-2'-deoxy-b-D-arabino-5-methyl uridine is a purine nucleoside analog with potential antitumor activity.Formula:C10H15N3O5Purity:96.76%Color and Shape:SolidMolecular weight:257.24VP-U-6
CAS:VP-U-6 is a Nucleoside Phosphoramidite; Nucleoside Derivative - Phosphorus-containing nucleotide; 5'-Modified nucleoside.Formula:C24H40N4O9P2Color and Shape:SolidMolecular weight:590.54Ref: TM-TNU1009
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire500mgTo inquireDOTA-cyclo(RGDfK)
CAS:DOTA-cyclo(RGDfK) is a and DOTA-like chelator peptide,the αvβ3 integrin receptor ,radionuclide coupled compounds RDCs cancer diagnostics and therapy.Formula:C43H67N13O14Color and Shape:SoildMolecular weight:990.078-Hydroxyadenosine
CAS:8-Hydroxyadenosine (8-Oxoadenosine) is a purine nucleoside found in Torula yeast RNA.Formula:C10H13N5O5Purity:99.71%Color and Shape:SolidMolecular weight:283.24Verosudil
CAS:Verosudil (AR-12286), a ROCK1/2 inhibitor (Ki: 2 nM), lowers intraocular pressure in mice by enhancing aqueous outflow.Formula:C17H17N3O2SPurity:99.68%Color and Shape:SolidMolecular weight:327.4Ref: TM-T60924
1mg55.00€5mg147.00€1mL*10mM (DMSO)161.00€10mg231.00€25mg370.00€50mg522.00€100mg692.00€A-674563
CAS:A-674563 is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC.Formula:C22H22N4OPurity:99.21%Color and Shape:SolidMolecular weight:358.44GSK269962A hydrochloride
CAS:GSK269962A hydrochloride (GSK 269962 hydrochloride) is a ROCK inhibitor with anti-inflammatory and vasodilatory effects and inhibits ROCK1 and ROCK2.Formula:C29H31ClN8O5Color and Shape:SolidMolecular weight:607.06TG-693
CAS:TG-693, Oral CLK1 inhibitor, promotes exon 31 skipping of dystrophin gene, inhibits CLK1 substrate phosphorylation, for Duchenne muscular dystrophy.Formula:C12H9N3Purity:99.81%Color and Shape:SolidMolecular weight:195.23GPRP
CAS:GPRP (Gly-Pro-Arg-Pro) is a fibrin polymerization inhibitor.Formula:C18H31N7O5Color and Shape:White To Off-White PowderMolecular weight:425.48STD1T
CAS:STD1T is a USP2a inhibitor with anticancer activity that reduces levels of the cell cycle protein D1 protein in HCT116 colon cancer cells.Formula:C19H19N3O4S2Purity:98.77%Color and Shape:SolidMolecular weight:417.5PROTAC CDK9 Degrader-1
CAS:PROTAC CDK9 Degrader-1 is a selective PROTAC-based CDK9 degrader, composed of a Cereblon ligand and a CDK ligand.Formula:C33H35N5O7Purity:95.1%Color and Shape:SolidMolecular weight:613.66USP8-IN-1
CAS:USP8-IN-1 is an inhibitor of USP8 with an IC 50 of 1.9 μM. USP8-IN-1 inhibits H1975 cell growth with a GI 50 of 82.04 μM [1].Formula:C18H21N5O3SPurity:99.07%Color and Shape:SoildMolecular weight:387.46Ref: TM-T60146
1mg84.00€5mg177.00€1mL*10mM (DMSO)195.00€10mg250.00€25mg439.00€50mg620.00€100mg893.00€Belumosudil mesylate
CAS:Belumosudil mesylate (KD025 mesylate) is a ROCK2 inhibitor with antifibrotic activity, and can be used in chronic graft-versus-host disease research.Formula:C27H28N6O5SPurity:98.73%Color and Shape:SolidMolecular weight:548.61Ref: TM-T39555
1mg34.00€2mg46.00€5mg71.00€1mL*10mM (DMSO)85.00€10mg96.00€25mg155.00€50mg230.00€100mg353.00€200mg517.00€Cotosudil
CAS:Cotosudil is a ROCK kinase inhibitor with antihypertensive activity used to treat or prevent neurodegenerative diseases.Formula:C16H21N3O2SPurity:98.41%Color and Shape:SolidMolecular weight:319.42Maleic hydrazide
CAS:Maleic hydrazide is a plant germination inhibitor that participates in nucleic acid metabolism pathways ,inhibiting cell division in the apical meristem.Formula:C4H4N2O2Purity:98.4%Color and Shape:Crystals From Water Maleic Hydrazide Is An Odorless White Solid Sinks In Water (Uscg 1999)Molecular weight:112.09N6-Bz-5'-O-DMTr-3'-deoxyadenosine-2'-O-CED-phosphoramidite
CAS:N6-Bz-5'-O-DMTr-3'-deoxyadenosine-2'-O-CED-phosphoramidite is an adenine nucleoside analog with potential vasodilator activity and anticancer activity.Formula:C47H52N7O7PPurity:97.36%Color and Shape:SolidMolecular weight:857.932'-O-Methylinosine
CAS:2'-O-Methylinosine (2'-(o-Methyl)-inosine) is an orally bioavailable purine nucleoside analog with antihypertensive activity.Formula:C11H14N4O5Purity:99.88%Color and Shape:SolidMolecular weight:282.252',5-Difluoro-2'-deoxy-1-arabinosyluracil
CAS:2',5-Difluoro-2'-deoxy-1-arabinosyluracil (2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine) is a urinary pyrimidine nucleoside analogue with potential antiepilepticFormula:C9H10F2N2O5Purity:99.99%Color and Shape:SolidMolecular weight:264.18NU6102
CAS:NU6102 is a CDK2 inhibitor with antitumor activity against CDK1/cyclinB, CDK1/CDK2, CDK4, DYRK1A , PDK1, and ROCKII, and it can be used to study rectal cancer.Formula:C18H22N6O3SPurity:99.76%Color and Shape:SolidMolecular weight:402.47LDC4297
CAS:LDC4297 (LDC044297) is a potent and selective CDK7 inhibitor.Formula:C23H28N8OPurity:98.25%Color and Shape:SolidMolecular weight:432.52GW406108X
CAS:GW406108X is a Kif15 and ULK1 inhibitor; IC50: 0.82 µM (ATPase), pIC50: 6.37; blocks autophagy.Formula:C20H11Cl2NO4Purity:98%Color and Shape:SolidMolecular weight:400.21IRES-C11
CAS:IRES-C11 is a specific inhibitor of translation that targets the internal ribosome entry site (IRES) of the c-MYC gene. It functions by blocking the interaction between heterogeneous nuclear ribonucleoprotein A1, a trans-acting factor required for c-MYC IRES activity, and its corresponding IRES. Notably, IRES-C11 does not inhibit the IRES activity of BAG-1, XIAP, and p53.Formula:C13H11Cl2NO4Purity:99.89%Color and Shape:SolidMolecular weight:316.14Ref: TM-T40419
1mg94.00€5mg222.00€1mL*10mM (DMSO)245.00€10mg356.00€25mg708.00€50mg1,063.00€100mg1,674.00€200mg2,242.00€Poloxime
CAS:Poloxime is a hydrolysis product of poloxin and is a non-ATP-competitive Plk1 inhibitor. It also has moderate Plk1 inhibitory activity.Formula:C10H13NO2Purity:98%Color and Shape:SolidMolecular weight:179.22TAME
CAS:Tosyl-L-Arginine Methyl Ester (TAME (N-4-Tosyl-L-arginine methyl ester)) is an APC inhibitor.Formula:C14H22N4O4SPurity:98%Color and Shape:SolidMolecular weight:342.41Cilengitide TFA
CAS:Cilengitide, αvβ3/αvβ5 inhibitor, IC50: 4.1/79 nM in vitro. 10x selectivity vs. gpIIbIIIa. Phase 2.Formula:C29H41F3N8O9Color and Shape:SolidMolecular weight:702.68Nolatrexed dihydrochloride
CAS:Nolatrexed dihydrochloride (Thymitaq) is a soluble, lipophilic cancer drug that inhibits DNA replication, causing cell cycle arrest and apoptosis.Formula:C14H14Cl2N4OSPurity:97.02%Color and Shape:Tan SolidMolecular weight:357.26CCT244747
CAS:CCT244747 is a potent and selective CHK1 inhibitor oral, ATP-competitive, and cytotoxic, abrogating drug-induced S and G2 blockade and inducing apoptosis .Formula:C20H24N8O2Purity:99.17%Color and Shape:SolidMolecular weight:408.46Ribociclib hydrochloride
CAS:Ribociclib hydrochloride (LEE011 HCl) is a selective, orally active cyclin-dependent kinase CDK4/6 inhibitor (IC50=10/39 nM) that inhibits proliferation.Formula:C23H31ClN8OPurity:99.87%Color and Shape:SolidMolecular weight:471sAJM589
CAS:sAJM589 is a Myc inhibitor that dose-dependently disrupts Myc-Max heterodimers, thereby decreasing Myc protein levels and inhibiting the cellular proliferation.Formula:C16H10N2OPurity:98%Color and Shape:SolidMolecular weight:246.26Synucleozid hydrochloride
CAS:Synucleozid hydrochloride inhibits the translation of the intrinsically disordered protein α-synuclein by targeting its structured mRNA.Formula:C22H21ClN6Purity:98.13%Color and Shape:SolidMolecular weight:404.9N,N-Dimethyl-2'-O-methylcytidine
CAS:N,N-Dimethyl-2'-O-methylcytidine (N4, N4, 2'-O-Trimethylcytidine) is a purine nucleoside analogue with anti-cancer activity.Formula:C12H19N3O5Purity:99.62%Color and Shape:SolidMolecular weight:285.38-Chloroinosine
CAS:8-Chloroinosine is a purine nucleoside analog and a metabolite of the anticancer compound 8-chloro-adenosine.Formula:C10H11ClN4O5Purity:99.37% - 99.56%Color and Shape:SolidMolecular weight:302.67Kinesore
CAS:Kinesore is a cell-permeable modulator that binds to the microtubule motor protein kinesin-1, thereby inhibiting the interaction between KLC2 and SKIP.Formula:C20H16Br2N4O4Purity:97.24%Color and Shape:SolidMolecular weight:536.17Ref: TM-T15663
2mg39.00€5mg58.00€1mL*10mM (DMSO)70.00€10mg93.00€25mg150.00€50mg219.00€100mg329.00€200mg494.00€5'-O-DMT-N2-ibu-dG
CAS:5'-O-DMT-N2-ibu-dG is a deoxynucleoside served as a building block in oligonucleotide synthesis, with protecting groups to prevent unwanted reactions.Formula:C35H37N5O7Purity:98.71%Color and Shape:SolidMolecular weight:639.78-Bromoadenosine
CAS:8-Bromoadenosine is an adenosine derivative. 8-Br-Adenosine inhibitis mitochondrial membrane potential, cytoplasmic Ca²⁺ levels, and RNA and protein synthesis.Formula:C10H12BrN5O4Purity:99.11%Color and Shape:SolidMolecular weight:346.14NSC 23766
CAS:NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.Formula:C24H35N7Purity:99.49%Color and Shape:SolidMolecular weight:421.58N2-Isobutyryl-2-deoxyguanosine
CAS:N2-Isobutyryl-2-deoxyguanosine(iBu-dG) is a nucleoside analog that can be used to synthesize oligonucleotides.Formula:C14H19N5O5Purity:97.03%Color and Shape:SolidMolecular weight:337.33APE1-IN-1
CAS:APE1-IN-1 is a purine/pyrimidine-free endonuclease 1 inhibitor with potential antitumor activity that enhances the toxicity of alkylating agents on cancer cellsFormula:C19H21N3OS2Purity:98.5%Color and Shape:SolidMolecular weight:371.52PD 407824
CAS:PD 407824 is a chemical BMP sensitiser that promotes increased cellular sensitivity to subthreshold amounts of BMP4.PD 407824 is a potent inhibitor of the checkpoint kinases Chk1 and WEE1 (IC50s: 47 and 97 nM, respectively).Formula:C20H12N2O3Purity:98.02%Color and Shape:SolidMolecular weight:328.322'-O-Methyl-5-iodouridine
CAS:2'-O-Methyl-5-iodouridine (5-Iodo-2'-O-methyluridine) is a purine nucleoside analog that targets malignant tumors of the inert lymphatic system and possesses a
Formula:C10H13IN2O6Purity:99.89%Color and Shape:SolidMolecular weight:384.12TG003
CAS:TG003 is a Clk1/Sty inhibitor that inhibits Clk1 and Clk4, suppresses cancer cell growth, and induces apoptosis.Formula:C13H15NO2SPurity:99.46%Color and Shape:SolidMolecular weight:249.33Ref: TM-T60367
1mg48.00€5mg92.00€10mg150.00€1mL*10mM (DMSO)167.00€25mg266.00€50mg440.00€100mg530.00€200mg767.00€Palmatine chloride
CAS:Palmatine chloride an isoquinoline alkaloid, is an important medicinal herbal extract with diverse pharmacological and biological properties.Formula:C21H22ClNO4Purity:97.9% - 99.47%Color and Shape:SolidMolecular weight:387.86Trimethoprim sulfate
CAS:Trimethoprim sulfate, a dihydrofolate reductase inhibitor, treats bacterial infections and sometimes malaria; may depress hematopoiesis.Formula:C28H38N8O10SColor and Shape:SolidMolecular weight:678.72GNE-6776
CAS:GNE-6776 is a selective USP7 inhibitor.Formula:C20H20N4O2Purity:96.59% - 98.2%Color and Shape:SolidMolecular weight:348.4Vidofludimus
CAS:Vidofludimus (SC12267) (4SC-101, SC12267) is a novel small molecule inhibitor of dihydroorotate dehydrogenase (DHODH).Formula:C20H18FNO4Purity:98.33% - 99.58%Color and Shape:SolidMolecular weight:355.36PKD-IN-1
CAS:CRT0066101 is an inhibitor of PKD.Formula:C18H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:342.82GDC-0575
CAS:GDC-0575 (ARRY-575) is a highly-selective oral small-molecule Chk1 inhibitor(IC50 of 1.2 nM).Formula:C16H20BrN5OPurity:≥95%Color and Shape:SolidMolecular weight:378.27CYC-116
CAS:CYC116 is a potent inhibitor of Aurora A/B with Ki of 8.0 nM/9.2 nM, is less potent to VEGFR2 (Ki of 44 nM), with 50-fold greater potency than CDKs, not activeFormula:C18H20N6OSPurity:97.36% - 97.59%Color and Shape:SolidMolecular weight:368.46Acelarin
CAS:Acelarin (NUC-1031) (NUC-1031) is a ProTide enhancement and transformation of the nucleoside analog, gemcitabine.Formula:C25H27F2N4O8PPurity:99.26%Color and Shape:SolidMolecular weight:580.47Ref: TM-T4060
200mgTo inquire1mg43.00€2mg56.00€1mL*10mM (DMSO)92.00€5mg93.00€10mg137.00€25mg259.00€50mg398.00€100mg555.00€TH588
CAS:TH588 is nudix hydrolase family inhibitor that effectively and selectively engages and inhibits the MTH1(IC50: 5 nM) in cells.Formula:C13H12Cl2N4Purity:96.05% - 99.82%Color and Shape:SolidMolecular weight:295.17Phthalazinone pyrazole
CAS:Phthalazinone pyrazole: a potent, selective oral Aurora-A kinase inhibitor, overexpressed in tumors with oncogenic activity.Formula:C18H15N5OPurity:97.03%Color and Shape:SolidMolecular weight:317.34POL1-IN-1
CAS:POL1-IN-1 (Compound 3A) 是一种RNA 聚合酶 1 POL1抑制剂,IC50值低于 0.5 uM。 它能有效抑制A375恶性黑色素瘤细胞系中RNA 聚合酶I 的转录。
Formula:C21H20N6Purity:98% - 98.01%Color and Shape:SolidMolecular weight:356.42Fialuridine
CAS:Fialuridine (DRG-0098), a DNA polymerase inhibitor, shows strong anti-HBV effects both in vitro and in vivo.Formula:C9H10FIN2O5Purity:99.71% - 99.88%Color and Shape:Less Crystals Colourless CrystalsMolecular weight:372.09MLS-573151
CAS:MLS-573151 is a selective inhibitor of GTPase Cdc42(EC50 of 2 μM).Formula:C21H19N3O2SPurity:98.80%Color and Shape:SolidMolecular weight:377.46Ref: TM-T22106
2mg34.00€5mg50.00€1mL*10mM (DMSO)55.00€10mg86.00€25mg161.00€50mg245.00€100mg363.00€200mg515.00€HA-100
CAS:HA-100 is an inhibitor of protein kinaseFormula:C13H15N3O2SPurity:99.44%Color and Shape:Pale Yellow Crystalline SolidMolecular weight:277.34AI-10-49
CAS:AI-10-49 is a selective inhibitor of the binding of CBFβ-SMMHC to RUNX1 with IC50 of 260 nM.Formula:C30H22F6N6O5Purity:97.14%Color and Shape:SolidMolecular weight:660.52Ref: TM-T6753
2mg38.00€5mg57.00€1mL*10mM (DMSO)84.00€10mg92.00€25mg160.00€50mg231.00€100mg343.00€200mg485.00€Ibezapolstat
CAS:Ibezapolstat (ACX-362E) is an antibiotic with antibacterial activity that inhibits Clostridium difficile.Formula:C18H20Cl2N6O2Purity:98% - 99.429%Color and Shape:SolidMolecular weight:423.3Ref: TM-T10243
1mg50.00€5mg105.00€1mL*10mM (DMSO)117.00€10mg170.00€25mg340.00€50mg557.00€100mg893.00€
