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JAK/STAT signaling
Products of "JAK/STAT signaling"
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Ilginatinib
CAS:1239358-86-1
Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H20FN7
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
389.43
Ref: TM-T12266
1mg | 93.00 € | ||
1ml | 213.00 € | ||
2mg | 133.00 € | ||
5mg | 218.00 € | ||
10mg | 303.00 € | ||
25mg | 444.00 € | ||
50mg | 639.00 € | ||
100mg | 916.00 € | ||
500mg | 1,838.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
JAK2 Inhibitor V
CAS:195371-52-9
JAK2 Inhibitor V (JAK2 Inhibitor V Z3) is a novel specific inhibitor of Jak2, inhibiting …
Formula:
C23H24N2O
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
344.45
Ref: TM-T3042
1ml | 63.00 € | ||
2mg | 39.00 € | ||
5mg | 56.00 € | ||
10mg | 83.00 € | ||
25mg | 153.00 € | ||
50mg | 268.00 € | ||
100mg | 494.00 € | ||
500mg | 1,100.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Ilginatinib maleate
CAS:1354799-87-3
Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C25H24FN7O4
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
505.5
Ref: TM-T12266L
1mg | 93.00 € | ||
1ml | 245.00 € | ||
2mg | 134.00 € | ||
5mg | 217.00 € | ||
10mg | 303.00 € | ||
25mg | 444.00 € | ||
50mg | 642.00 € | ||
100mg | 917.00 € | ||
500mg | 1,839.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Uzansertib phosphate
CAS:2088852-47-3
Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase, inhibiting PIM1, …
Formula:
C26H29F3N5O7P
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
611.51
Ref: TM-T12477
1mg | 94.00 € | ||
5mg | 275.00 € | ||
10mg | 410.00 € | ||
25mg | 677.00 € | ||
50mg | 922.00 € | ||
100mg | 1,290.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Ilginatinib hydrochloride
CAS:1239358-85-0
Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H21ClFN7
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
425.89
Ref: TM-T12266L2
1mg | 91.00 € | ||
1ml | 207.00 € | ||
5mg | 217.00 € | ||
10mg | 304.00 € | ||
25mg | 447.00 € | ||
50mg | 639.00 € | ||
100mg | 916.00 € | ||
500mg | 1,845.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Brepocitinib P-Tosylate
CAS:2140301-96-6
Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and …
Formula:
C25H29F2N7O4S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
561.6
Ref: TM-T12427
1mg | 35.00 € | ||
1ml | 87.00 € | ||
5mg | 69.00 € | ||
10mg | 102.00 € | ||
25mg | 212.00 € | ||
50mg | 384.00 € | ||
100mg | 616.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Delgocitinib
CAS:1263774-59-9
Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the …
Formula:
C16H18N6O
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
310.35
Ref: TM-T15096
1mg | 167.00 € | ||
1ml | 347.00 € | ||
5mg | 500.00 € | ||
10mg | 722.00 € | ||
25mg | 1,096.00 € | ||
50mg | 1,486.00 € | ||
100mg | 2,016.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Golidocitinib
CAS:2091134-68-6
Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: …
Formula:
C25H31N9O2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
489.57
Ref: TM-T10431
1ml | 168.00 € | ||
2mg | 94.00 € | ||
5mg | 160.00 € | ||
10mg | 262.00 € | ||
25mg | 457.00 € | ||
50mg | 605.00 € | ||
100mg | 861.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Gusacitinib
CAS:1425381-60-7
Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 …
Formula:
C24H28N8O2
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
460.53
Ref: TM-T14331
1mg | 47.00 € | ||
1ml | 116.00 € | ||
5mg | 94.00 € | ||
10mg | 121.00 € | ||
25mg | 185.00 € | ||
50mg | 343.00 € | ||
100mg | 510.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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JAK1-IN-10
CAS:2416858-88-1
JAK1-IN-10 (compound 9), a cyano-substituted cyclic hydrazine derivative, functions as a potent and selective inhibitor …
Formula:
C15H17N7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
295.34
Ref: TM-T79078
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-34
CAS:2068766-90-3
JAK-IN-34 (compound 11n) is a potent inhibitor of Janus kinases (JAKs), demonstrating IC50 values of …
Formula:
C27H26N6O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
450.53
Ref: TM-T82017
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-29
JAK-IN-29 (Compound 3) is a potent inhibitor of Janus kinases (JAK) [1].
Formula:
C17H14ClN5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
355.78
Ref: TM-T79222
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-25
CAS:2127110-22-7
JAK-IN-25 (compound 19), a potent JAK inhibitor, exhibits IC50 values of 6 nM for TYK2, …
Formula:
C19H17N5O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
379.37
Ref: TM-T78175
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-33
JAK-IN-33 (Compound 3 (R)) is a selective inhibitor of the Janus kinase (JAK) family [1].
Purity:
98%
Ref: TM-T82018
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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WDR5-IN-6
CAS:326901-92-2
WDR5-IN-6 is a WDR5 inhibitor targeting the WBM locus.WDR5-IN-6 is highly synergistic with OICR-9429, a …
Formula:
C13H8Cl2N2O2S
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
327.19
Ref: TM-T77495
1mg | 45.00 € | ||
5mg | 96.00 € | ||
10mg | 142.00 € | ||
25mg | 275.00 € | ||
50mg | 447.00 € | ||
100mg | 708.00 € | ||
500mg | 1,439.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK/HDAC-IN-2
JAK/HDAC-IN-2, a potent 2-amino-4-phenylaminopyrimidine dual-target inhibitor, effectively suppresses JAK1/2 and HDAC3/6 at nanomolar concentrations.
Formula:
C28H38N6O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
570.7
Ref: TM-T78708
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK kinase-IN-1
CAS:2698389-43-2
JAK kinase-IN-1 (Example 1) functions as a potent inhibitor targeting the JAK family, which includes …
Formula:
C17H19F2N7OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
407.44
Ref: TM-T79807
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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Pumecitinib
CAS:2401057-12-1
Pumecitinib is a Janus kinase (JAK) inhibitor. Pumecitinib exhibits anti-inflammatory activity.
Formula:
C17H20N8O2S
Purity:
99.89%
Color and Shape:
Soild
Molecular weight:
400.46
Ref: TM-T67758
1mg | 35.00 € | ||
1ml | 96.00 € | ||
5mg | 79.00 € | ||
10mg | 114.00 € | ||
25mg | 202.00 € | ||
50mg | 322.00 € | ||
100mg | 459.00 € | ||
500mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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FD1024
CAS:1422456-47-0
FD1024 is a potent PIM inhibitor, displaying inhibitory concentrations (IC50s) of 1.96 nM, 38.9 nM, …
Formula:
C21H20F2N4O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
430.47
Ref: TM-T79456
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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TAK-901
CAS:934541-31-8
TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid …
Formula:
C28H32N4O3S
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
504.64
Ref: TM-T2709
5mg | 76.00 € | ||
25mg | 209.00 € | ||
50mg | 363.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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HS94
CAS:1892594-93-2
HS94 (DAPK3 inhibitor HS94) is a selective and potent DAPK3 inhibitor with a Ki value …
Formula:
C15H15N5O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.38
Ref: TM-T77777
1mg | 40.00 € | ||
5mg | 85.00 € | ||
10mg | 116.00 € | ||
25mg | 224.00 € | ||
50mg | 333.00 € | ||
100mg | 494.00 € | ||
500mg | 1,058.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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Pim-1 kinase inhibitor 8
CAS:916038-47-6
Pim-1 kinase inhibitor 8 is a Pim-1 kinase inhibitor with anticancer activity that inhibits cell …
Formula:
C14H17N3O3
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
275.3
Ref: TM-T83627
1mg | 61.00 € | ||
5mg | 133.00 € | ||
10mg | 206.00 € | ||
25mg | 414.00 € | ||
50mg | 664.00 € | ||
100mg | 1,045.00 € | ||
500mg | 2,116.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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S-Ruxolitinib
CAS:1160597-27-2
S-Ruxolitinib can be used in related research in the field of life sciences. Its product …
Formula:
C17H18N6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
306.37
Ref: TM-T3066
2mg | 48.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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Povorcitinib phosphate
CAS:1637677-33-8
Povorcitinib phosphate is a selective JAK1 inhibitor and can be used in studies about the …
Formula:
C23H25F5N7O5P
Purity:
97.71%
Color and Shape:
Solid
Molecular weight:
605.45
Ref: TM-T39113L
1mg | 95.00 € | ||
1ml | 313.00 € | ||
5mg | 231.00 € | ||
10mg | 346.00 € | ||
25mg | 587.00 € | ||
50mg | 833.00 € | ||
100mg | 1,133.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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ABBV-712
CAS:2368945-27-9
ABBV-712 is a selective Tyrosine Kinase 2 (TYK2) inhibitor, demonstrating an IC50 value of 0.195 …
Formula:
C24H28N4O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
452.5
Ref: TM-T83218
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK2-IN-6
CAS:353512-04-6
JAK2-IN-6: A potent JAK2-specific inhibitor (IC50=22.86μg/mL), blocks JAK2 signaling, has anticancer properties, and is inactive …
Formula:
C14H10ClN3OS2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
335.83
Ref: TM-T40443
1mg | 46.00 € | ||
5mg | 96.00 € | ||
10mg | 123.00 € | ||
25mg | 204.00 € | ||
50mg | 305.00 € | ||
100mg | 454.00 € | ||
500mg | 985.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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PIM-IN-2
CAS:1006699-45-1
PIM-IN-2 (Pim-2) is a potent inhibitor of Pim kinases, demonstrating an inhibition concentration half-maximal (IC50) …
Formula:
C19H22N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
338.4
Ref: TM-T81460
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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Lepzacitinib
CAS:2321488-47-3
Lepzacitinib, a Janus kinase inhibitor, specifically targets JAK 1/3.
Formula:
C18H21N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
355.39
Ref: TM-T78207
2mg | 91.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Nimucitinib
CAS:2740557-24-6
Nimucitinib is a Janus kinase (JAK) inhibitor that can be used to treat dry eye …
Formula:
C25H26F2N6O2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
480.51
Ref: TM-T67907
1mg | 95.00 € | ||
2mg | 139.00 € | ||
5mg | 226.00 € | ||
10mg | 351.00 € | ||
25mg | 649.00 € | ||
50mg | 931.00 € | ||
100mg | 1,443.00 € | ||
500mg | 2,801.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
JAK1-IN-11
CAS:2427608-43-1
JAK1-IN-11 (compound 11) serves as a potent inhibitor of Janus kinases, exhibiting nanomolar inhibitory concentrations …
Formula:
C26H36N6O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
528.67
Ref: TM-T79079
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-26
CAS:2417134-93-9
JAK-IN-26 (compound 2) is an orally active inhibitor of the Janus kinase (JAK) enzyme with …
Formula:
C22H24N6O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
420.46
Ref: TM-T78189
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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Pim-1 kinase inhibitor 5
CAS:2928606-67-9
Pim-1 kinase inhibitor 5 (Compound 4c), with an IC50 of 0.61 μM, exhibits cytotoxicity against …
Formula:
C22H13Cl2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
406.26
Ref: TM-T78980
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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STAT3-IN-18
CAS:2668267-41-0
STAT3-IN-18 (compound SPP), a platinum (IV) complex featuring an axial ligand from sandalwood, suppresses the …
Formula:
C18H24Cl2N2O6Pt
Purity:
98%
Color and Shape:
Solid
Molecular weight:
630.38
Ref: TM-T79609
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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QL-1200186
CAS:2848664-42-4
QL-1200186 is an orally active, selective TYK2 inhibitor that, upon dose-dependent oral administration, suppresses interferon-γ …
Formula:
C26H27N7O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
485.54
Ref: TM-T81331
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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DPP
CAS:2668267-47-6
DPP, a Platinum(IV) complex with a pterostilbene-derived axial ligand, inhibits the JAK2-STAT3 pathway in breast …
Formula:
C36H40Cl2N2O10Pt
Purity:
98%
Color and Shape:
Solid
Molecular weight:
926.7
Ref: TM-T79608
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-27
CAS:2673176-36-6
JAK-IN-27, also known as compound 1, is an orally active, potent inhibitor of the JAKS …
Formula:
C20H21F2N7O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
413.42
Ref: TM-T79110
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-31
CAS:2597016-88-9
JAK-IN-31 (Example 75), a JAK inhibitor, demonstrates IC50 values of ≤0.01 µM for JAK1, ≤0.01 …
Formula:
C21H19N7O2S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
465.55
Ref: TM-T79882
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JI069
CAS:850019-35-1
JI069 (WAY-354189) is a potent STAT3 inhibitor that inhibits gp130 signaling by inducing dissociation between …
Formula:
C15H12Cl2N2O4S
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
387.24
Ref: TM-T77672
1mg | 182.00 € | ||
5mg | 449.00 € | ||
10mg | 643.00 € | ||
25mg | 1,009.00 € | ||
50mg | 1,384.00 € | ||
100mg | 1,841.00 € | ||
500mg | 3,650.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Pim-1/2 kinase inhibitor 1
CAS:6320-51-0
Orally active Pim-1/2 inhibitor blocks kinase phosphorylation; used in prostate cancer research.
Formula:
C11H9NO3S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
235.26
Ref: TM-T9229
1mg | 40.00 € | ||
2mg | 95.00 € | ||
5mg | 83.00 € | ||
10mg | 122.00 € | ||
25mg | 237.00 € | ||
50mg | 369.00 € | ||
100mg | 553.00 € | ||
500mg | 1,160.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
(2R)-Octyl-α-hydroxyglutarate
CAS:1391194-67-4
(2R)-Octyl-α-hydroxyglutarate ((2R)-Octyl-2-HG) is a D-isomer 2-Hydroxyglutarate modified form.
Formula:
C13H24O5
Color and Shape:
Solid
Molecular weight:
260.33
Ref: TM-T19611
1ml | 130.00 € | ||
2mg | 91.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
CHZ868
CAS:1895895-38-1
CHZ868 is a type II JAK inhibitor with potential antitumor activity that reverses the persistence …
Formula:
C22H19F2N5O2
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
423.42
Ref: TM-TQ0061
2mg | 72.00 € | ||
5mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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DTP3
CAS:1809784-29-9
DTP3 is a selective MKK7/GADD45β inhibitor, which inhibits cancer-selective NF-κB survival pathway.
Formula:
C26H35N7O5
Color and Shape:
Solid
Molecular weight:
525.6
Ref: TM-T22319
2mg | 82.00 € | ||
5mg | 124.00 € | ||
10mg | 214.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
CX-6258 hydrochloride
CAS:1353859-00-3
CX-6258 hydrochloride (Pim-Kinase Inhibitor X) is an effective, orally efficacious Pim1/2/3 kinase inhibitor (IC50: 5/25/16 …
Formula:
C26H24ClN3O3·HCl
Purity:
97.98%
Color and Shape:
Solid
Molecular weight:
498.4
Ref: TM-T6148
1mg | 42.00 € | ||
1ml | 87.00 € | ||
2mg | 55.00 € | ||
5mg | 87.00 € | ||
10mg | 142.00 € | ||
25mg | 249.00 € | ||
50mg | 415.00 € | ||
100mg | 601.00 € | ||
500mg | 1,236.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
GS-829845
CAS:1257705-09-1
GS-829845 is a JAK1 inhibitor, the main component of the active metabolite of Filgotinib, which …
Formula:
C17H19N5O2S
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
357.43
Ref: TM-T67905
5mg | 46.00 € | ||
10mg | 62.00 € | ||
25mg | 87.00 € | ||
50mg | 123.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Momelotinib sulfate
CAS:1056636-06-6
Momelotinib sulfate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity …
Formula:
C23H26N6O10S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
610.62
Ref: TM-T15038
1ml | 110.00 € | ||
2mg | 50.00 € | ||
5mg | 84.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Cerdulatinib hydrochloride
CAS:1369761-01-2
Cerdulatinib hydrochloride is an oral tyrosine kinase inhibitor targeting JAK1/2/3, TYK2, Syk, and 19 others …
Formula:
C20H28ClN7O3S
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
482
Ref: TM-T6104
1mg | 44.00 € | ||
1ml | 89.00 € | ||
2mg | 57.00 € | ||
5mg | 94.00 € | ||
10mg | 114.00 € | ||
25mg | 187.00 € | ||
50mg | 280.00 € | ||
100mg | 429.00 € | ||
500mg | 931.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ifidancitinib
CAS:1236667-40-5
Ifidancitinib (ATI-50002) is a specific JAK kinase 1/3 inhibitor that induces hair growth in AA-affected …
Formula:
C20H18FN5O3
Color and Shape:
Solid
Molecular weight:
395.39
Ref: TM-T38623
1mg | 143.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SC99
CAS:882290-02-0
SC99 inhibits JAK2-STAT3, reducing STAT3 genes, platelet activity, and has anti-myeloma, anti-thrombotic effects.
Formula:
C15H8Cl2FN3O
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
336.15
Ref: TM-T8719
1mg | 69.00 € | ||
1ml | 165.00 € | ||
5mg | 150.00 € | ||
10mg | 222.00 € | ||
25mg | 393.00 € | ||
50mg | 591.00 € | ||
100mg | 735.00 € | ||
500mg | 1,511.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WP1066
CAS:857064-38-1
WP1066 is a inhibitor of JAK2 (IC50: 2.30 μM) and STAT3 (IC50: 2.43 μM) in …
Formula:
C17H14BrN3O
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
356.22
Ref: TM-T2156
1ml | 53.00 € | ||
5mg | 52.00 € | ||
10mg | 80.00 € | ||
25mg | 129.00 € | ||
50mg | 209.00 € | ||
100mg | 293.00 € | ||
500mg | 714.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AZ960
CAS:905586-69-8
AZ960 is an effective ATP competitive JAK2 inhibitor (IC50/Ki: <3 nM and0.45 nM).
Formula:
C18H16F2N6
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
354.36
Ref: TM-T6309
1mg | 77.00 € | ||
1ml | 96.00 € | ||
2mg | 94.00 € | ||
5mg | 127.00 € | ||
10mg | 198.00 € | ||
25mg | 360.00 € | ||
50mg | 534.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WDR5-0103 hydrochloride[890190-22-4(free base)]
WDR5-0103 hydrochloride[890190-22-4(free base)] (WD-Repeat Protein 5-0103) is an effective and specific WD repeat-containing protein 5 …
Formula:
C21H26ClN3O4
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
419.9
Ref: TM-T5140
1mg | 43.00 € | ||
2mg | 54.00 € | ||
5mg | 73.00 € | ||
10mg | 117.00 € | ||
25mg | 204.00 € | ||
50mg | 352.00 € | ||
100mg | 441.00 € | ||
200mg | 650.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Brevilin A
CAS:16503-32-5
Brevilin A, a sesquiterpene from Centipeda minima, hinders JAK and blocks STAT3 (IC50=10.6μM), inducing apoptosis …
Formula:
C20H26O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
346.42
Ref: TM-T4672
1mg | 94.00 € | ||
1ml | 235.00 € | ||
5mg | 212.00 € | ||
10mg | 362.00 € | ||
25mg | 601.00 € | ||
50mg | 822.00 € | ||
100mg | 1,112.00 € | ||
500mg | 2,265.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Hispidulin
CAS:1447-88-7
Hispidulin, a natural flavone with a broad spectrum of biological activities, is a Pim-1 inhibitor …
Formula:
C16H12O6
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
300.26
Ref: TM-TQ0201
1ml | 69.00 € | ||
10mg | 88.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AMG-47a
CAS:882663-88-9
AMG-47a inhibits Lck, T cell growth, and degrades KRAS oncoprotein, affecting EGFP-KRASG12V but not EGFP.
Formula:
C29H28F3N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
535.56
Ref: TM-T7123
1mg | 45.00 € | ||
1ml | 95.00 € | ||
5mg | 96.00 € | ||
10mg | 149.00 € | ||
25mg | 244.00 € | ||
50mg | 362.00 € | ||
100mg | 532.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Decernotinib
CAS:944842-54-0
Decernotinib (VRT-831509)(VX-509; VRT-831509) is a potent and selective Janus kinase 3 (JAK3) inhibitor with Ki …
Formula:
C18H19F3N6O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
392.38
Ref: TM-T2636
1mg | 52.00 € | ||
1ml | 89.00 € | ||
2mg | 68.00 € | ||
5mg | 93.00 € | ||
10mg | 130.00 € | ||
25mg | 257.00 € | ||
50mg | 456.00 € | ||
100mg | 639.00 € | ||
500mg | 1,327.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Fedratinib hydrochloride hydrate
CAS:1374744-69-0
Fedratinib hydrochloride hydrate (SAR 302503 hydrochloride hydrate) is a potent, selective, ATP-competitive and orally active …
Formula:
C27H40Cl2N6O4S
Purity:
98.96%
Color and Shape:
Solid
Molecular weight:
615.61
Ref: TM-T9251
1ml | 67.00 € | ||
5mg | 46.00 € | ||
10mg | 60.00 € | ||
25mg | 84.00 € | ||
50mg | 98.00 € | ||
100mg | 118.00 € | ||
200mg | 184.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
G5-7
CAS:939681-36-4
G5-7 is an oral JAK2 inhibitor targeting EGFR/STAT3 phosphorylation with potential for glioma research.
Formula:
C22H19F2NO3
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
383.39
Ref: TM-T8742
1mg | 82.00 € | ||
1ml | 168.00 € | ||
5mg | 158.00 € | ||
10mg | 230.00 € | ||
25mg | 424.00 € | ||
50mg | 613.00 € | ||
100mg | 856.00 € | ||
500mg | 1,700.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
(E/Z)-Zotiraciclib
CAS:937270-47-8
(E/Z)-Zotiraciclib ((E/Z)-TG02) inhibits CDK2, JAK2, and FLT3 effectively with IC50s of 13, 73, and 56 …
Formula:
C23H24N4O
Purity:
97.75%
Color and Shape:
Solid
Molecular weight:
372.46
Ref: TM-T21503
1mg | 45.00 € | ||
1ml | 95.00 € | ||
2mg | 58.00 € | ||
5mg | 96.00 € | ||
10mg | 118.00 € | ||
25mg | 207.00 € | ||
50mg | 343.00 € | ||
100mg | 495.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TG101209
CAS:936091-14-4
TG101209 is a selective JAK2 inhibitor with IC50 of 6 nM.
Formula:
C26H35N7O2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
509.67
Ref: TM-T3065
1ml | 73.00 € | ||
2mg | 47.00 € | ||
5mg | 66.00 € | ||
10mg | 92.00 € | ||
25mg | 104.00 € | ||
50mg | 122.00 € | ||
100mg | 193.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
GDC-0214
CAS:1831144-46-7
GDC-0214 is an inhaled small-molecule JAK1 inhibitor and reduces fractional exhaled nitric oxide (Feno).
Formula:
C28H28ClF2N9O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
612.03
Ref: TM-T9826
1mg | 143.00 € | ||
1ml | 428.00 € | ||
5mg | 312.00 € | ||
10mg | 462.00 € | ||
25mg | 737.00 € | ||
50mg | 1,054.00 € | ||
100mg | 1,420.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Baricitinib
CAS:1187594-09-7
Baricitinib (INCB028050) is an orally bioavailable inhibitor of Janus kinases 1 and 2 (JAK1/2), with …
Formula:
C16H17N7O2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
371.42
Ref: TM-T2485
1ml | 69.00 € | ||
5mg | 50.00 € | ||
10mg | 73.00 € | ||
25mg | 89.00 € | ||
50mg | 113.00 € | ||
100mg | 142.00 € | ||
200mg | 184.00 € | ||
500mg | 306.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TCS PIM-1 1
CAS:491871-58-0
TCS PIM-1 1 (SC 204330) is a potent ATP-competitive inhibitor of Pim-1 kinase with an …
Formula:
C18H11BrN2O2
Purity:
97%
Color and Shape:
Solid
Molecular weight:
367.2
Ref: TM-T2253
1ml | 96.00 € | ||
2mg | 45.00 € | ||
5mg | 63.00 € | ||
10mg | 87.00 € | ||
25mg | 184.00 € | ||
50mg | 339.00 € | ||
100mg | 501.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Pyridone 6
CAS:457081-03-7
Pyridone 6, a selective JAK1/2/3 and Tyk2 inhibitor with IC50s: JAK1=15 nM, JAK2=1 nM, JAK3 …
Formula:
C18H16FN3O
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
309.34
Ref: TM-T3080
1mg | 81.00 € | ||
1ml | 176.00 € | ||
2mg | 105.00 € | ||
5mg | 159.00 € | ||
10mg | 218.00 € | ||
25mg | 441.00 € | ||
50mg | 648.00 € | ||
100mg | 918.00 € | ||
500mg | 1,838.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WHI-P97
CAS:211555-05-4
WHI-P97 is a rationally designed potent inhibitor of JAK-3.
Formula:
C16H13Br2N3O3
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
455.1
Ref: TM-T4657
1mg | 38.00 € | ||
1ml | 88.00 € | ||
2mg | 49.00 € | ||
5mg | 80.00 € | ||
10mg | 116.00 € | ||
25mg | 210.00 € | ||
50mg | 314.00 € | ||
100mg | 468.00 € | ||
500mg | 1,009.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SGI-1776
CAS:1025065-69-3
SGI-1776 (Pim-Kinase Inhibitor IX) has been used in trials studying the treatment of Prostate Cancer, …
Formula:
C20H22F3N5O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
405.42
Ref: TM-T3078
1ml | 98.00 € | ||
2mg | 52.00 € | ||
5mg | 95.00 € | ||
10mg | 169.00 € | ||
25mg | 299.00 € | ||
50mg | 428.00 € | ||
100mg | 549.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Itacitinib
CAS:1334298-90-6
Itacitinib (INCB039110) is an orally bioavailable inhibitor of Janus-associated kinase 1 (JAK1) with potential antineoplastic …
Formula:
C26H23F4N9O
Purity:
96.4%
Color and Shape:
Solid
Molecular weight:
553.51
Ref: TM-T3998
1mg | 49.00 € | ||
1ml | 136.00 € | ||
2mg | 70.00 € | ||
5mg | 109.00 € | ||
10mg | 177.00 € | ||
25mg | 320.00 € | ||
50mg | 534.00 € | ||
100mg | 763.00 € | ||
500mg | 1,523.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tofacitinib
CAS:477600-75-2
Tofacitinib (Tasocitinib) is an oral, small molecule inhibitor of Janus kinases that is used to …
Formula:
C16H20N6O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
312.37
Ref: TM-T6321
1ml | 57.00 € | ||
5mg | 35.00 € | ||
10mg | 51.00 € | ||
25mg | 64.00 € | ||
50mg | 83.00 € | ||
100mg | 95.00 € | ||
200mg | 142.00 € | ||
500mg | 257.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Abrocitinib
CAS:1622902-68-4
Abrocitinib (PF-04965842) (PF-04965842) is a potent, specific and orally-active JAK1 inhibitor (IC50s: 29/803 nM for …
Formula:
C14H21N5O2S
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
323.41
Ref: TM-TQ0037
1mg | 83.00 € | ||
1ml | 187.00 € | ||
2mg | 106.00 € | ||
5mg | 164.00 € | ||
10mg | 278.00 € | ||
25mg | 456.00 € | ||
50mg | 677.00 € | ||
100mg | 920.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
2,6-Dichloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)benzamide
CAS:1258292-64-6
2,6-Dichloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)benzamide (GDC046), a potent lead analog, has good kinase selectivity and physicochemical properties.
Formula:
C16H13Cl2N3O2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
350.2
Ref: TM-T22338
1mg | 60.00 € | ||
5mg | 118.00 € | ||
10mg | 184.00 € | ||
25mg | 423.00 € | ||
50mg | 611.00 € | ||
100mg | 852.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Gandotinib
CAS:1229236-86-5
LY2784544(Gandotinib (LY2784544)) is a potent JAK2 inhibitor (IC50: 3 nM), effective in JAK2V617F(Ki: 0.245 nM).
Formula:
C23H25ClFN7O
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
469.94
Ref: TM-T2638
1ml | 57.00 € | ||
5mg | 51.00 € | ||
10mg | 86.00 € | ||
25mg | 158.00 € | ||
50mg | 290.00 € | ||
100mg | 460.00 € | ||
500mg | 1,012.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Filgotinib
CAS:1206161-97-8
Filgotinib (GLPG0634) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and …
Formula:
C21H23N5O3S
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
425.5
Ref: TM-T1929
1ml | 78.00 € | ||
2mg | 54.00 € | ||
5mg | 77.00 € | ||
10mg | 109.00 € | ||
25mg | 161.00 € | ||
50mg | 291.00 € | ||
100mg | 480.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Fedratinib
CAS:936091-26-8
Fedratinib (TG-101348) (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less …
Formula:
C27H36N6O3S
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
524.68
Ref: TM-T1995
1g | 613.00 € | ||
1ml | 57.00 € | ||
5mg | 49.00 € | ||
10mg | 68.00 € | ||
50mg | 111.00 € | ||
100mg | 132.00 € | ||
200mg | 213.00 € | ||
500mg | 463.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tofacitinib Citrate
CAS:540737-29-9
Tofacitinib Citrate (CP-690550 citrate) is a a potent, cell-permeable inhibitor of JAK1/2/3 (IC50s: 1/20/112 nM).
Formula:
C22H28N6O8
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
504.49
Ref: TM-T2398
1ml | 55.00 € | ||
5mg | 38.00 € | ||
10mg | 54.00 € | ||
50mg | 69.00 € | ||
100mg | 90.00 € | ||
200mg | 124.00 € | ||
500mg | 204.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ruxolitinib (S enantiomer)
CAS:941685-37-6
Ruxolitinib S enantiomer (INCB18424) is the S-enantiomer of Ruxolitinib. Ruxolitinib is the first potent, selective …
Formula:
C17H18N6
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
306.36
Ref: TM-T6156
1ml | 64.00 € | ||
5mg | 63.00 € | ||
10mg | 74.00 € | ||
50mg | 113.00 € | ||
100mg | 151.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SAR-20347
CAS:1450881-55-6
SAR-20347 is an inhibitor of TYK2, JAK1/2/3 (IC50: 0.6/23/26/41 nM).
Formula:
C21H18ClFN4O4
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
444.84
Ref: TM-T4210
1mg | 37.00 € | ||
1ml | 86.00 € | ||
5mg | 78.00 € | ||
10mg | 113.00 € | ||
25mg | 221.00 € | ||
50mg | 344.00 € | ||
100mg | 573.00 € | ||
500mg | 1,183.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ritlecitinib
CAS:1792180-81-4
Ritlecitinib (PF-06651600) is a potent JAK3-selective inhibitor (IC50: 33.1 nM).
Formula:
C15H19N5O
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
285.34
Ref: TM-T5382
1ml | 76.00 € | ||
2mg | 46.00 € | ||
5mg | 69.00 € | ||
10mg | 109.00 € | ||
25mg | 212.00 € | ||
50mg | 325.00 € | ||
100mg | 485.00 € | ||
200mg | 690.00 € | ||
500mg | 1,047.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Cucurbitacin I
CAS:2222-07-3
Cucurbitacin I (JSI-124), a natural compound, is a selective inhibitor of JAK2/STAT3 with anti-cancer activity.
Formula:
C30H42O7
Purity:
96.69%
Color and Shape:
Solid
Molecular weight:
514.65
Ref: TM-TQ0196
1mg | 83.00 € | ||
1ml | 184.00 € | ||
5mg | 172.00 € | ||
10mg | 222.00 € | ||
25mg | 367.00 € | ||
50mg | 546.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ruxolitinib phosphate
CAS:1092939-17-7
Ruxolitinib phosphate is a potent JAK1/2 inhibitor, selective with IC50s 3.3/2.8 nM, and >130x more …
Formula:
C17H21N6O4P
Purity:
100%
Color and Shape:
Solid
Molecular weight:
404.36
Ref: TM-T3043
1g | 604.00 € | ||
1ml | 59.00 € | ||
5mg | 52.00 € | ||
10mg | 64.00 € | ||
25mg | 81.00 € | ||
50mg | 95.00 € | ||
100mg | 144.00 € | ||
200mg | 223.00 € | ||
500mg | 408.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
GLPG0634 analog
CAS:1206101-20-3
GLPG0634 analog (GLPG0634 analogue) is a specific JAK1 inhibitor with IC50 of 10/28/810/116 nM for …
Formula:
C23H18N6O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
410.43
Ref: TM-T3076
1mg | 40.00 € | ||
1ml | 87.00 € | ||
2mg | 52.00 € | ||
5mg | 87.00 € | ||
10mg | 142.00 € | ||
25mg | 258.00 € | ||
50mg | 455.00 € | ||
100mg | 646.00 € | ||
500mg | 1,352.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
RO8191
CAS:691868-88-9
RO8191 (CDM-3008) (CDM-3008) is an agonist of interferon (IFN) receptor.
Formula:
C14H5F6N5O
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
373.21
Ref: TM-T22142
1mg | 45.00 € | ||
2mg | 58.00 € | ||
5mg | 96.00 € | ||
10mg | 142.00 € | ||
25mg | 301.00 € | ||
50mg | 478.00 € | ||
100mg | 698.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
JAK3-IN-6
CAS:1443235-95-7
JAK3-IN-6 is irreversible Janus Associated Kinase 3 (JAK3) inhibitor, with an IC50 of 0.15 nM
Formula:
C19H18N4O3
Purity:
97.34%
Color and Shape:
Solid
Molecular weight:
350.37
Ref: TM-T5492
1ml | 67.00 € | ||
2mg | 40.00 € | ||
5mg | 59.00 € | ||
10mg | 93.00 € | ||
25mg | 153.00 € | ||
50mg | 237.00 € | ||
100mg | 370.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
RGB-286638 free base
CAS:784210-88-4
RGB-286638 free base inhibits CDKs (1-5 nM), weaker on CDK7/6.
Formula:
C29H35N7O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
545.63
Ref: TM-T2378
1mg | 46.00 € | ||
2mg | 60.00 € | ||
5mg | 87.00 € | ||
10mg | 144.00 € | ||
25mg | 263.00 € | ||
50mg | 396.00 € | ||
100mg | 554.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
FLLL32
CAS:1226895-15-3
FLLL32 is an effective JAK2/STAT3 inhibitor (IC50 of <5 μM).
Formula:
C28H32O6
Purity:
96.39%
Color and Shape:
Solid
Molecular weight:
464.55
Ref: TM-T6838
1ml | 72.00 € | ||
2mg | 45.00 € | ||
5mg | 66.00 € | ||
10mg | 92.00 € | ||
25mg | 122.00 € | ||
50mg | 193.00 € | ||
100mg | 343.00 € | ||
500mg | 822.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
JANEX-1
CAS:202475-60-3
JANEX-1: cell-permeable, reversible Jak3 inhibitor (IC50: 78 μM), ATP-competitive, selective; weak on JAK1/2, Zap/Syk, SRC.
Formula:
C16H15N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
297.31
Ref: TM-T2045
1mg | 44.00 € | ||
1ml | 92.00 € | ||
2mg | 54.00 € | ||
5mg | 90.00 € | ||
10mg | 147.00 € | ||
25mg | 243.00 € | ||
50mg | 435.00 € | ||
100mg | 637.00 € | ||
500mg | 1,347.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TP-3654
CAS:1361951-15-6
TP-3654 is a second-generation Pim kinase inhibitor (Ki values against Pim-1/3: 5/42 nM).
Formula:
C22H25F3N4O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
418.46
Ref: TM-T4523
1ml | 57.00 € | ||
5mg | 56.00 € | ||
10mg | 83.00 € | ||
25mg | 148.00 € | ||
50mg | 231.00 € | ||
100mg | 345.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Cerdulatinib
CAS:1198300-79-6
Cerdulatinib (PRT2070) is an novel oral dual Syk/JAK inhibitor.
Formula:
C20H27N7O3S
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
445.54
Ref: TM-T2487
1mg | 44.00 € | ||
1ml | 85.00 € | ||
2mg | 54.00 € | ||
5mg | 78.00 € | ||
10mg | 104.00 € | ||
25mg | 181.00 € | ||
50mg | 280.00 € | ||
100mg | 429.00 € | ||
200mg | 601.00 € | ||
500mg | 931.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Upadacitinib
CAS:1310726-60-3
Upadacitinib (ABT-494), a selective JAK1 inhibitor, is researched for autoimmune diseases; IC50: 43 nM.
Formula:
C17H19F3N6O
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
380.37
Ref: TM-T7503
1mg | 46.00 € | ||
1ml | 49.00 € | ||
2mg | 61.00 € | ||
5mg | 88.00 € | ||
10mg | 127.00 € | ||
25mg | 217.00 € | ||
50mg | 302.00 € | ||
100mg | 427.00 € | ||
200mg | 650.00 € | ||
500mg | 1,142.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
BD750
CAS:892686-59-8
BD750 is an effective immunosuppressant and a JAK3/STAT5 inhibitor, inhibits IL-2-induced JAK3/STAT5-dependent T cell proliferation(IC50 …
Formula:
C14H13N3OS
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
271.34
Ref: TM-T8546
1ml | 57.00 € | ||
5mg | 51.00 € | ||
10mg | 86.00 € | ||
25mg | 142.00 € | ||
50mg | 231.00 € | ||
100mg | 382.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SMI-16a
CAS:587852-28-6
SMI-16a (PIM1/2 Kinase Inhibitor VI) , a cell-permeable thiazolidinedione compound, acts as an effective, ATP-competitive …
Formula:
C13H13NO3S
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
263.31
Ref: TM-T3989
1mg | 35.00 € | ||
1ml | 92.00 € | ||
2mg | 47.00 € | ||
5mg | 69.00 € | ||
10mg | 96.00 € | ||
25mg | 158.00 € | ||
50mg | 231.00 € | ||
100mg | 346.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
HJ-PI01
CAS:6192-43-4
HJ-PI01 (HJ-PI01) is a Pim-2 inhibitor. HJ-PI01 (HJ-PI01) induces apoptosis and autophagic cell death in …
Formula:
C14H11NO2
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
225.24
Ref: TM-T9583
1mg | 52.00 € | ||
1ml | 114.00 € | ||
5mg | 118.00 € | ||
10mg | 184.00 € | ||
25mg | 424.00 € | ||
50mg | 626.00 € | ||
100mg | 891.00 € | ||
500mg | 1,789.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WHI-P97 HCl
WHI-P97 HCl is a potent and selective JAK-3 inhibitor.
Formula:
C16H14Br2ClN3O3
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
491.56
Ref: TM-T4657L
1mg | 63.00 € | ||
1ml | 164.00 € | ||
2mg | 88.00 € | ||
5mg | 98.00 € | ||
10mg | 182.00 € | ||
25mg | 328.00 € | ||
50mg | 453.00 € | ||
100mg | 644.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WHI-P154
CAS:211555-04-3
WHI-P154 (Jak3 inhibitor ii) is a potent JAK3 inhibitor.
Formula:
C16H14BrN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
376.2
Ref: TM-T1985
1ml | 64.00 € | ||
2mg | 46.00 € | ||
5mg | 65.00 € | ||
10mg | 100.00 € | ||
25mg | 178.00 € | ||
50mg | 331.00 € | ||
100mg | 534.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AZD1208
CAS:1204144-28-4
AZD1208 is a novel, orally bioavailable, highly selective PIM kinase inhibitor with single nanomolar potency …
Formula:
C21H21N3O2S
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
379.48
Ref: TM-T2300
1ml | 57.00 € | ||
2mg | 38.00 € | ||
5mg | 51.00 € | ||
10mg | 74.00 € | ||
25mg | 117.00 € | ||
50mg | 210.00 € | ||
100mg | 370.00 € | ||
200mg | 487.00 € | ||
500mg | 778.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Atractylenolide I
CAS:73069-13-3
Atractylenolide-I reduces inflammation, improves sepsis, liver, and kidney function, and enhances EOC cell sensitivity to …
Formula:
C15H18O2
Purity:
97.55%
Color and Shape:
Solid
Molecular weight:
230.3
Ref: TM-T5S0167
1mg | 42.00 € | ||
1ml | 94.00 € | ||
5mg | 85.00 € | ||
10mg | 128.00 € | ||
25mg | 237.00 € | ||
50mg | 414.00 € | ||
100mg | 579.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
XL019
CAS:945755-56-6
XL019 is a potent and selective JAK2 inhibitor with IC50 of 2.2 nM, 100 fold …
Formula:
C25H28N6O2
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
444.53
Ref: TM-T3072
1ml | 82.00 € | ||
5mg | 73.00 € | ||
10mg | 118.00 € | ||
25mg | 208.00 € | ||
50mg | 343.00 € | ||
100mg | 510.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TCS-PIM-1-4a
CAS:327033-36-3
SMI-4a, a Pim inhibitor, activates AMPK, halts mTORC1, and kills various myeloid/lymphoid cells (IC50=0.8-40μM).
Formula:
C11H6F3NO2S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
273.23
Ref: TM-T4215
1ml | 55.00 € | ||
5mg | 51.00 € | ||
10mg | 75.00 € | ||
25mg | 122.00 € | ||
50mg | 210.00 € | ||
100mg | 315.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SHR0302
CAS:1445987-21-2
SHR0302 (ARQ252) is a JAK inhibitor that binds JAK1 with stronger affinity than others (Selectivity …
Formula:
C18H22N8O2S
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
414.48
Ref: TM-T9195
1mg | 157.00 € | ||
1ml | 445.00 € | ||
2mg | 259.00 € | ||
5mg | 384.00 € | ||
10mg | 606.00 € | ||
25mg | 1,012.00 € | ||
50mg | 1,447.00 € | ||
100mg | 1,837.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
ZM39923 hydrochloride
CAS:1021868-92-7
ZM39923 hydrochloride (JAK3 Inhibitor IV) is an JAK1/3 inhibitor, almost no activity to JAK2 and …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
367.91
Ref: TM-T6145
1ml | 95.00 € | ||
5mg | 58.00 € | ||
10mg | 93.00 € | ||
25mg | 168.00 € | ||
50mg | 304.00 € | ||
100mg | 455.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Peficitinib
CAS:944118-01-8
Peficitinib (ASP015K) (ASP015K, JNJ-54781532) is an orally bioavailable JAK inhibitor. Phase 3.
Formula:
C18H22N4O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
326.39
Ref: TM-T6933
1mg | 65.00 € | ||
5mg | 78.00 € | ||
10mg | 124.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Protosappanin A
CAS:102036-28-2
Protosappanin A combats brain inflammation, suppresses rat heart transplant rejection, fights MRSA, and inhibits HIV …
Formula:
C15H12O5
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
272.25
Ref: TM-TJS1779
1mg | 96.00 € | ||
1ml | 193.00 € | ||
5mg | 212.00 € | ||
10mg | 346.00 € | ||
25mg | 569.00 € | ||
50mg | 807.00 € | ||
100mg | 1,086.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024