CymitQuimica logo
Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

Show 13 more subcategories

Found 2280 products of "Membrane Transporter/Ion Channel"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • 3,4,5-Trimethoxycinnamic acid

    CAS:
    <p>3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the</p>
    Formula:C12H14O5
    Purity:98.91%
    Color and Shape:Solid
    Molecular weight:238.24
  • ML418

    CAS:
    <p>ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.</p>
    Formula:C19H24ClN3O3
    Purity:99.3%
    Color and Shape:Solid
    Molecular weight:377.87
  • Prilocaine hydrochloride

    CAS:
    <p>Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.</p>
    Formula:C13H21ClN2O
    Purity:99.97%
    Color and Shape:Needles White Or Off White Crystalline Powder
    Molecular weight:256.77
  • Flumazenil

    CAS:
    <p>Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous</p>
    Formula:C15H14FN3O3
    Purity:99.72% - 99.98%
    Color and Shape:Less Crystals Colourless Crystals
    Molecular weight:303.29
  • Dooku1

    CAS:
    Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.
    Formula:C13H9Cl2N3OS
    Purity:98.87% - 99.74%
    Color and Shape:Solid
    Molecular weight:326.2
  • Fluxametamide

    CAS:
    <p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>
    Formula:C20H16Cl2F3N3O3
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:474.26
  • NS13001

    CAS:
    <p>NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).</p>
    Formula:C17H16ClN7
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:353.81
  • Phenformin hydrochloride

    CAS:
    <p>Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.</p>
    Formula:C10H16ClN5
    Purity:97.11% - 99.80%
    Color and Shape:Lactic Acidosis
    Molecular weight:241.72
  • VU0134992 hydrochloride

    CAS:
    <p>VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).</p>
    Formula:C20H32BrClN2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:447.84
  • Pramocaine hydrochloride

    CAS:
    <p>Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.</p>
    Formula:C17H27NO3·HCl
    Purity:99.15% - 99.61%
    Color and Shape:Crystals White Or Off White Crystalline Powder
    Molecular weight:329.86
  • Flindokalner

    CAS:
    <p>Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.</p>
    Formula:C16H10ClF4NO2
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:359.7
  • TPC2-A1-P

    CAS:
    <p>TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).</p>
    Formula:C20H21BrF3NO3
    Purity:98.49%
    Color and Shape:Solid
    Molecular weight:460.29
  • Glipizide

    CAS:
    <p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>
    Formula:C21H27N5O4S
    Purity:99.67% - 99.75%
    Color and Shape:Solid
    Molecular weight:445.54
  • Manidipine dihydrochloride

    CAS:
    <p>Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).</p>
    Formula:C35H40Cl2N4O6
    Purity:99.76% - 99.86%
    Color and Shape:Solid
    Molecular weight:683.62
  • γ-Aminobutyric acid

    CAS:
    <p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>
    Formula:C4H9NO2
    Purity:99.95%
    Color and Shape:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid Powder
    Molecular weight:103.12
  • Baclofen

    CAS:
    <p>Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.</p>
    Formula:C10H12ClNO2
    Purity:98% - >99.99%
    Color and Shape:1992)
    Molecular weight:213.66
  • VU6036720


    <p>VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit</p>
    Formula:C20H22ClFN4O2S
    Purity:98.1%
    Color and Shape:Soild
    Molecular weight:436.93
  • DSP-2230

    CAS:
    <p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>
    Formula:C20H20F3N5O2
    Purity:97.14%
    Color and Shape:Solid
    Molecular weight:419.4
  • Methocarbamol

    CAS:
    <p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>
    Formula:C11H15NO5
    Purity:99.96%
    Color and Shape:Crystals From Benzene Solid
    Molecular weight:241.24
  • Celivarone

    CAS:
    <p>Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and atrial fibrillation.</p>
    Formula:C34H47NO4
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:533.74