5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 1025 products of "5-HT Receptor"
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Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Formula:C20H20NO4Purity:97.18% - 99.06%Color and Shape:SolidMolecular weight:338.38Urapidil
CAS:Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formula:C20H29N5O3Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:387.48RS-127445 hydrochloride
CAS:RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formula:C17H17ClFN3Purity:99.48%Color and Shape:SolidMolecular weight:317.79Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Ref: TM-T5336
1mg34.00€5mg71.00€10mg99.00€25mg212.00€50mg385.00€100mg618.00€200mg859.00€1mL*10mM (DMSO)79.00€8-Hydroxy-DPAT hydrobromide
CAS:8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.Formula:C16H26BrNOPurity:98.90% - 99.99%Color and Shape:SolidMolecular weight:328.29SB-203186 hydrochloride
CAS:SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFormula:C16H20N2O2·HClPurity:99.64%Color and Shape:SolidMolecular weight:308.81Myristicin
CAS:Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formula:C11H12O3Purity:99.828%Color and Shape:LiquidMolecular weight:192.21Hypidone hydrochloride
CAS:Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitorFormula:C18H23ClN2O2Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:334.84Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formula:C18H22N2SPurity:99.34% - 99.34%Color and Shape:SolidMolecular weight:298.45Ref: TM-T2395
1g477.00€10mg48.00€25mg65.00€50mg90.00€100mg117.00€200mg203.00€500mg333.00€1mL*10mM (DMSO)46.00€BRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formula:C14H18N2OPurity:98.07%Color and Shape:SolidMolecular weight:230.316-fluoro-DL-Tryptophan
CAS:6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formula:C11H11FN2O2Purity:99.25%Color and Shape:Off-White PowderMolecular weight:222.22Serotonin
CAS:Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Formula:C10H12N2OPurity:97.47% - 99.92%Color and Shape:SolidMolecular weight:176.22Ref: TM-TN2437
2mg34.00€5mg52.00€10mg85.00€25mg157.00€50mg250.00€100mg404.00€200mg585.00€1mL*10mM (DMSO)46.00€NAN-190 hydrobromide
CAS:NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formula:C23H28BrN3O3Purity:95.20%Color and Shape:SolidMolecular weight:474.39Perospirone hydrochloride
CAS:Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formula:C23H31ClN4O2SPurity:99.37%Color and Shape:White SolidMolecular weight:4633-AQC
CAS:3-AQC is a competitive antagonist of 5-HT3.Formula:C20H21N5O4Purity:99.45%Color and Shape:SolidMolecular weight:395.41AVN-101
CAS:AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formula:C21H25ClN2Purity:99.61%Color and Shape:SolidMolecular weight:340.89Ref: TM-T26690
1mg34.00€5mg75.00€10mg114.00€25mg205.00€50mg334.00€100mg557.00€200mg790.00€1mL*10mM (DMSO)92.00€SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurity:98% - 99.83%Color and Shape:SolidMolecular weight:324.24Ref: TM-T4369
1mg39.00€2mg50.00€5mg78.00€10mg97.00€25mg195.00€50mg369.00€100mg550.00€1mL*10mM (DMSO)78.00€Mosapride
CAS:Mosapride (AS-4370) is a selective 5HT4 agonistFormula:C21H25ClFN3O3Purity:99.56%Color and Shape:White To Off-White Crystalline SolidMolecular weight:421.89Tianeptine sodium salt
CAS:Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formula:C21H24ClN2NaO4SPurity:99.82%Color and Shape:SolidMolecular weight:458.93Vilazodone Hydrochloride
CAS:Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormula:C26H27N5O2·HClPurity:99.56% - >99.99%Color and Shape:SolidMolecular weight:477.99Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formula:C24H23ClF3NPurity:99.99%Color and Shape:SolidMolecular weight:417.89Ref: TM-T9272
1mg38.00€5mg80.00€10mg114.00€25mg222.00€50mg356.00€100mg512.00€200mg735.00€1mL*10mM (DMSO)92.00€lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formula:C31H36FN3O4SPurity:95.83% - 99.95%Color and Shape:SolidMolecular weight:565.7Cerlapirdine
CAS:Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Formula:C22H23N3O3SPurity:98.77%Color and Shape:SolidMolecular weight:409.5Ref: TM-T30798
1mg81.00€5mg170.00€10mg274.00€25mg543.00€50mg780.00€100mg1,074.00€1mL*10mM (DMSO)198.00€Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurity:99.78% - >99.99%Color and Shape:SolidMolecular weight:463.87Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formula:C18H20N4Purity:99.15% - 99.82%Color and Shape:SolidMolecular weight:292.38Indophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formula:C19H15BrClF3N2O3SPurity:99.76%Color and Shape:SolidMolecular weight:523.75Amperozide
CAS:Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formula:C23H29F2N3OPurity:99.68%Color and Shape:SolidMolecular weight:401.49Ref: TM-T23733
1mg87.00€5mg178.00€10mg295.00€25mg497.00€50mg708.00€100mg964.00€500mg1,918.00€1mL*10mM (DMSO)321.00€Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purity:99.33%Color and Shape:SolidMolecular weight:354.27Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Vortioxetine hydrobromide
CAS:Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formula:C18H22N2S·HBrPurity:98.85% - 99.98%Color and Shape:SolidMolecular weight:379.36Azaphen dihydrochloride monohydrate
CAS:Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Formula:C16H23Cl2N5O2Purity:99.85%Color and Shape:SolidMolecular weight:388.29RS-67333
CAS:RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.Formula:C19H29ClN2O2Purity:99.24%Color and Shape:SolidMolecular weight:352.9SB 243213
CAS:SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formula:C22H19F3N4O2Purity:98.78% - 99.86%Color and Shape:SolidMolecular weight:428.41Jatrorrhizine chloride
CAS:Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Formula:C20H20ClNO4Purity:99.79%Color and Shape:SolidMolecular weight:373.8Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purity:99.68%Color and Shape:SolidMolecular weight:545.51Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurity:98.45%Color and Shape:SolidMolecular weight:392.37LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purity:98%Color and Shape:SolidMolecular weight:562.94Rizatriptan
CAS:Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formula:C15H19N5Purity:99.74%Color and Shape:SolidMolecular weight:269.35Setiptiline
CAS:Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formula:C19H19NPurity:98.05% - 98.07%Color and Shape:SolidMolecular weight:261.36Citalopram
CAS:Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formula:C20H21FN2OPurity:99.78% - 99.89%Color and Shape:SolidMolecular weight:324.39(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formula:C17H19N3Purity:99.37%Color and Shape:SolidMolecular weight:265.35Rotigotine
CAS:Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formula:C19H25NOSPurity:99.04% - 99.88%Color and Shape:SolidMolecular weight:315.47Tandospirone
CAS:Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formula:C21H29N5O2Purity:99.94%Color and Shape:SolidMolecular weight:383.49Ref: TM-TQ0315
2mg34.00€5mg50.00€10mg80.00€25mg130.00€50mg178.00€100mg284.00€200mg408.00€1mL*10mM (DMSO)55.00€Renzapride
CAS:Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formula:C16H22ClN3O2Purity:98.97% - 99.09%Color and Shape:SolidMolecular weight:323.82Ref: TM-T38507
1mg93.00€2mg124.00€5mg200.00€10mg359.00€25mg692.00€50mg945.00€100mg1,279.00€200mg1,701.00€WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formula:C25H34N4O2·xC4H4O4Purity:99.96%Color and Shape:White SolidMolecular weight:538.645Ref: TM-T3453
2mg43.00€5mg63.00€10mg89.00€25mg150.00€50mg215.00€100mg316.00€500mg765.00€1mL*10mM (DMSO)74.00€(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formula:C17H19N3Purity:99.75%Color and Shape:SolidMolecular weight:265.35S1RA
CAS:S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formula:C20H23N3O2Purity:99.45%Color and Shape:SolidMolecular weight:337.42Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurity:97.63%Color and Shape:SolidMolecular weight:340.3R 59-022
CAS:R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formula:C27H26FN3OSPurity:98.55%Color and Shape:SolidMolecular weight:459.58Ref: TM-T16709
1mg35.00€5mg74.00€10mg119.00€25mg269.00€50mg447.00€100mg733.00€200mg973.00€1mL*10mM (DMSO)75.00€Cyproheptadine hydrochloride
CAS:Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
Formula:C21H21N·HClPurity:99.88% - 99.97%Color and Shape:SolidMolecular weight:323.86
