AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 574 products of "AChR"
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Orphenadrine Citrate
CAS:<p>Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.</p>Formula:C18H23NO·C6H8O7Purity:98% - 99.58%Color and Shape:White SolidMolecular weight:461.5Ipratropium bromide monohydrate
CAS:<p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>Formula:C20H32BrNO4Purity:97.85%Color and Shape:SolidMolecular weight:430.38Gallamine triethiodide
CAS:<p>Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.</p>Formula:C30H60I3N3O3Purity:98.90%Color and Shape:White Amorphous Powder SolidMolecular weight:891.53Nicardipine hydrochloride
CAS:<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Formula:C26H30ClN3O6Purity:99.58% - 99.89%Color and Shape:Yellow SolidMolecular weight:515.99Bambuterol hydrochloride
CAS:<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Formula:C18H30ClN3O5Purity:99.53% - 99.61%Color and Shape:White SolidMolecular weight:403.91Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formula:C22H22FN3O2Purity:97.16% - 98%Color and Shape:SolidMolecular weight:379.43DL-trihexyphenidyl hydrochloride
CAS:<p>DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.</p>Formula:C20H32ClNOPurity:99.63% - 99.71%Color and Shape:SolidMolecular weight:337.93Dicyclomine hydrochloride
CAS:<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Formula:C19H36ClNO2Purity:99.81%Color and Shape:SolidMolecular weight:345.95Nebracetam hydrochloride
CAS:<p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>Formula:C12H17ClN2OPurity:99.23%Color and Shape:SolidMolecular weight:240.729MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formula:C25H25N3O2Purity:99.77% - 99.8%Color and Shape:SolidMolecular weight:399.48Homatropine Methylbromide
CAS:<p>Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.</p>Formula:C17H24BrNO3Purity:98.97%Color and Shape:SolidMolecular weight:370.29Acetamiprid
CAS:<p>Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.</p>Formula:C10H11ClN4Purity:99.66%Color and Shape:White PowderMolecular weight:222.67Temephos
CAS:<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Formula:C16H20O6P2S3Purity:≥95%Color and Shape:White Crystalline Solid Or LiquidMolecular weight:466.47Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purity:98.41% - 99.96%Color and Shape:White Crystalline Powder; Odourless Or Almost OdourlessMolecular weight:403.53Methscopolamine
CAS:<p>Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.</p>Formula:C18H24BrNO4Purity:99.12% - ≥98%Color and Shape:SolidMolecular weight:398.29Valethamate bromide
CAS:<p>Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.</p>Formula:C19H32BrNO2Purity:>99.99%Color and Shape:SolidMolecular weight:386.37Carbetapentane citrate
CAS:<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Formula:C20H31NO3·C6H8O7Purity:99.46%Color and Shape:White To Off-White SolidMolecular weight:525.59Diphenmanil methylsulfate
CAS:<p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>Formula:C20H24N·CH3O4SPurity:98% - 99.27%Color and Shape:SolidMolecular weight:389.51Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formula:C14H18N2O2Purity:97.37%Color and Shape:White To Off-White Crystalline PowderMolecular weight:246.3Procainamide hydrochloride
CAS:<p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>Formula:C13H21N3O·HClPurity:99.83% - 99.97%Color and Shape:White To Slightly Yellow PowderMolecular weight:271.79Trospium chloride
CAS:<p>Trospium chloride treats urinary incontinence without causing liver damage.</p>Formula:C25H30ClNO3Purity:99.84% - >99.99%Color and Shape:White To Off-White PowderMolecular weight:427.964Neostigmine methyl sulfate
CAS:<p>Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of myasthenia gravis.</p>Formula:C13H22N2O6SPurity:99.34% - 99.53%Color and Shape:Crystalline SolidMolecular weight:334.39Dipivefrin hydrochloride
CAS:<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Formula:C19H27NO5·HClPurity:99.22% - 99.92%Color and Shape:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorMolecular weight:387.9Methacholine Chloride
CAS:<p>Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of acetylcholine.</p>Formula:C8H18ClNO2Purity:99.37% - 99.74%Color and Shape:White Hygroscopic Crystals With Slight Odor Of Dead FishMolecular weight:195.69PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formula:C36H51Cl3N4O7SPurity:99.85%Color and Shape:SolidMolecular weight:790.24Adiphenine hydrochloride
CAS:<p>Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.</p>Formula:C20H25NO2·HClPurity:97.76% - 99.53%Color and Shape:White Or Almost White PowderMolecular weight:347.88Benzethonium chloride
CAS:<p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>Formula:C27H42ClNO2Purity:99.91%Color and Shape:White To Off-White Solid Solid Particulate/PowderMolecular weight:448.09VU 0365114
CAS:<p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>Formula:C22H14F3NO3Purity:99.86%Color and Shape:SolidMolecular weight:397.35Rivastigmine tartrate
CAS:<p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>Formula:C14H22N2O2·C4H6O6Purity:98% - 99.66%Color and Shape:White To Off-White PowderMolecular weight:400.43Zelminemab
CAS:<p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>Purity:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Color and Shape:LiquidPyrantel tartrate
CAS:<p>Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.</p>Formula:C15H20N2O6SPurity:99.96%Color and Shape:White CrystalsMolecular weight:356.39Pirenzepine dihydrochloride
CAS:<p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>Formula:C19H21N5O2·2HClPurity:99.48% - 99.62%Color and Shape:White PowderMolecular weight:424.32Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Formula:C17H20N2S·HClPurity:99.85%Color and Shape:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Molecular weight:320.88Bethanechol chloride
CAS:<p>Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.</p>Formula:C7H17N2O2·ClPurity:95% - 99.73%Color and Shape:White CrystallineMolecular weight:196.68Deschloroclozapine
CAS:<p>Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist.</p>Formula:C18H20N4Purity:99.61% - 99.98%Color and Shape:SolidMolecular weight:292.38Lysipressin acetate(50-57-7(fb_acetate))
CAS:<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Formula:C48H69N13O14S2Purity:98.08%Color and Shape:SolidMolecular weight:1116.28Fesoterodine fumarate
CAS:<p>Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.</p>Formula:C26H37NO3·C4H4O4Purity:99.16%Color and Shape:White SolidMolecular weight:527.65Vecuronium bromide
CAS:<p>Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscle</p>Formula:C34H57BrN2O4Purity:99.63% - 99.92%Color and Shape:White PowderMolecular weight:637.73Pancuronium dibromide
CAS:<p>Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.</p>Formula:C35H60Br2N2O4Purity:99.86%Color and Shape:solidMolecular weight:732.67Rocuronium bromide
CAS:<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Formula:C32H53BrN2O4Purity:99.77% - >99.99%Color and Shape:White Or Off-White PowderMolecular weight:609.68TAK-071
CAS:<p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>Formula:C24H24FN3O3Purity:98.02%Color and Shape:SolidMolecular weight:421.46nAChR agonist 1
CAS:<p>nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.</p>Formula:C20H18ClNO3S2Purity:97.59%Color and Shape:SolidMolecular weight:419.94Pyrantel pamoate
CAS:<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Formula:C34H30N2O6SPurity:99.71%Molecular weight:594.699-Cyclopentyladenine
CAS:<p>9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signaling</p>Formula:C10H13N5Purity:99.98%Color and Shape:SolidMolecular weight:203.24Clidinium bromide
CAS:<p>Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.</p>Formula:C22H26BrNO3Purity:98.89% - 99.86%Color and Shape:White Crystalline SolidMolecular weight:432.35Hexamethonium Bromide
CAS:<p>Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.</p>Formula:C12H30Br2N2Purity:99.76%Color and Shape:White Crystalline Powder And AgglomeratesMolecular weight:362.19Oxybutynin
CAS:<p>Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.</p>Formula:C22H31NO3Purity:97.81% - 99.57%Color and Shape:White To Off-White Crystalline PowderMolecular weight:357.49Benactyzine hydrochloride
CAS:<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Formula:C20H26ClNO3Purity:99.03% - 99.94%Color and Shape:SolidMolecular weight:363.88Flavoxate hydrochloride
CAS:<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Formula:C24H26ClNO4Purity:99.78%Color and Shape:White SolidMolecular weight:427.922',5'-Dideoxyadenosine
CAS:<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Formula:C10H13N5O2Purity:99.55%Color and Shape:White SolidMolecular weight:235.24Fipexide
CAS:<p>Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.</p>Formula:C20H21ClN2O4Purity:97.6% - 99.95%Color and Shape:SolidMolecular weight:388.84(Rac)-ABT-202 dihydrochloride
CAS:<p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>Formula:C9H15Cl2N3Purity:97.4%Color and Shape:SolidMolecular weight:236.142Carbachol
CAS:<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Formula:C6H15ClN2O2Purity:>99.99%Color and Shape:SolidMolecular weight:182.65Tolterodine tartrate
CAS:<p>Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.</p>Formula:C22H31NO·C4H6O6Purity:99.95%Color and Shape:White-To-Off-White Crystalline PowderMolecular weight:475.58Propantheline bromide
CAS:<p>Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on smooth muscle</p>Formula:C23H30BrNO3Purity:98% - ≥98%Molecular weight:448.4Primidone
CAS:<p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>Formula:C12H14N2O2Purity:99.91%Color and Shape:Crystals (Ntp 1992)Molecular weight:218.25Dequalinium chloride
CAS:<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Formula:C30H40Cl2N4Purity:99.79% - 99.9%Color and Shape:SolidMolecular weight:527.59Solifenacin succinate
CAS:<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Formula:C23H26N2O2·C4H6O4Purity:99.85% - 99.98%Color and Shape:SolidMolecular weight:480.56Darifenacin hydrobromide
CAS:<p>Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome.</p>Formula:C28H31BrN2O2Purity:99.75% - >99.99%Color and Shape:SolidMolecular weight:505.45SSR 180
CAS:<p>SSR 180 is a potent and subtype-selective α7 agonist with applications in the study of Alzheimer;s disease and schizophrenia.</p>Formula:C14H17BrN2O2Purity:98.82%Color and Shape:SoildMolecular weight:325.20Atropine methyl bromide
CAS:<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Formula:C18H26BrNO3Purity:99.7%Color and Shape:SolidMolecular weight:384.308Tazomeline
CAS:<p>Tazomeline is a muscarinic M1 receptor agonist with neuroprotective activity.</p>Formula:C14H23N3S2Purity:99.63%Color and Shape:SolidMolecular weight:297.48V-11-0711 HCl
<p>V-11-0711 HCl is a selective and highly effective choline kinase α (ChoKα) inhibitor that inhibits the catalytic activity of Chk.</p>Formula:C27H36ClNO3Purity:99.87%Color and Shape:SolidMolecular weight:458.03(Rac)-Sabcomeline HCl
CAS:<p>Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.</p>Formula:C10H16ClN3OPurity:99.58%Color and Shape:SoildMolecular weight:229.71Cotinine
CAS:<p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>Formula:C10H12N2OPurity:98% - 99.89%Color and Shape:Viscous Oil SolidMolecular weight:176.22Ribavirin
CAS:<p>Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.</p>Formula:C8H12N4O5Purity:99.09% - 99.83%Color and Shape:Less Solid Colourless SolidMolecular weight:244.20Tiotropium bromide
CAS:<p>Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).</p>Formula:C19H22BrNO4S2Purity:96.82% - 99.97%Color and Shape:White SolidMolecular weight:472.42DSPE-PEG1000-RVG29
<p>DSPE-PEG1000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 can specifically bind to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and cross the BBB.</p>Color and Shape:Odour SolidMK-0969
CAS:<p>MK-0969 (J-104135) is a possible M3 antagonist for the treatment of chronic obstructive pulmonary disease.</p>Formula:C24H30F2N4O2Color and Shape:SolidMolecular weight:444.52nAChR modulator-2
CAS:<p>nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Formula:C12H8ClN3O2Color and Shape:SolidMolecular weight:261.66α-Muricholic acid
CAS:<p>α-Muricholic acid is the most abundant primary bile acid in rodents.</p>Formula:C24H40O5Purity:98%Color and Shape:SolidMolecular weight:408.57α-Conotoxin EI
CAS:<p>Selective antagonist of neuromuscular nicotinic receptors α1β1γδ</p>Formula:C83H125N27O27S5Purity:98%Color and Shape:SolidMolecular weight:2093.37Octamylamine
CAS:<p>Octamylamine is a bioactive chemical.</p>Formula:C13H29NColor and Shape:SolidMolecular weight:199.3761Bencycloquidium Bromide
CAS:<p>Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.</p>Formula:C21H32BrNO2Color and Shape:SolidMolecular weight:410.39nAChR agonist CMPI hydrochloride
CAS:<p>CMPI hydrochloride: Potent α4:α4 nAChR PAM; EC50 0.26 μM for (α4)3(β2)2 response to ACh; may aid nicotine dependence, neuropsychiatric research.</p>Formula:C18H20Cl2N4OColor and Shape:SolidMolecular weight:379.29(S)-Dinotefuran
CAS:<p>(S)-Dinotefuran, a neonicotinoid, more toxic to bees than its R-isomer, targets α8 nAChR.</p>Formula:C7H14N4O3Color and Shape:SolidMolecular weight:202.21Angiopeptin TFA
CAS:<p>Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.</p>Formula:C58H73F6N11O14S2Color and Shape:SolidMolecular weight:1326.39[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS:<p>[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.</p>Formula:C82H120N20O25Color and Shape:SolidMolecular weight:1785.95LtIA-F
<p>LtIA-F, a fluorescent LtIA derivative, aids study of α3β2 nAChR's structure, distribution, and binding domain.</p>Formula:C86H121N25O22S4Color and Shape:SolidMolecular weight:1985.31α-Conotoxin PIA TFA
<p>α-Conotoxin PIA TFA, targeting nicotinic acetylcholine receptor (nAChR) subtypes with α6 and α3 subunits, acts as an antagonist.</p>Formula:C81H126F3N27O27S4Purity:98.81%Color and Shape:SolidMolecular weight:2095.3Muscarinic toxin 3
CAS:<p>Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57</p>Formula:C319H489N89O97S8Purity:98%Color and Shape:SolidMolecular weight:7379.35DSPE-PEG5000-RVG29
<p>DSPE-PEG5000-RVG29 is a PEG compound comprised of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and facilitates passage through the BBB.</p>Color and Shape:Odour Solid(-)-Coclaurine hydrochloride
CAS:<p>(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.</p>Formula:C17H20ClNO3Purity:99.07%Color and Shape:SoildMolecular weight:321.8Perlapine
CAS:<p>Perlapine is an effective and selective HM3DQ DREADD agonist (EC50 = 2.8 nM).</p>Formula:C19H21N3Color and Shape:SolidMolecular weight:291.39Atracurium
CAS:<p>Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.</p>Formula:C53H72N2O122Color and Shape:SolidMolecular weight:929.14Anagyrine hydrochloride
CAS:<p>Anagyrine hydrochloride, a quinolizidine from Lupinus albus, targets muscarinic/nicotinic receptors; IC50: 132/2096 µM. It desensitizes nAChR directly.</p>Formula:C15H21ClN2OColor and Shape:SolidMolecular weight:280.798-Aminoadenine
CAS:<p>8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.</p>Formula:C5H6N6Purity:99.82%Color and Shape:SolidMolecular weight:150.14rac-Desethyl Oxybutynin (hydrochloride)
CAS:<p>rac-Desethyl oxybutynin, active oxybutynin metabolite, binds to mAChRs; K_i values 3.12-16 nM; lowers rat micturition pressure.</p>Formula:C20H28ClNO3Color and Shape:SolidMolecular weight:365.89TMPH
CAS:<p>TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.</p>Formula:C16H31NO2Purity:99.78%Color and Shape:SoildMolecular weight:269.42Guanylyl Imidodiphosphate (lithium salt)
CAS:<p>Guanylyl Imidodiphosphate (lithium salt) is a non-hydrolyzable GTP analog that increases adenylate cyclase activity.</p>Formula:C10H13Li4N6O13P3Color and Shape:SolidMolecular weight:545.93Doxacurium Chloride
CAS:<p>Doxacurium Chloride is a muscarinic acetylcholine receptor M2 antagonist.</p>Formula:C56H78ClN2O16Purity:98%Color and Shape:SolidMolecular weight:1070.69Epiboxidine hydrochloride
CAS:<p>Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.</p>Formula:C10H15ClN2OColor and Shape:SolidMolecular weight:214.69VU6028418
CAS:<p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>Color and Shape:SolidPF-4348235 HCl
<p>PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).</p>Formula:C36H50Cl2N4O7SPurity:98.81%Color and Shape:SolidMolecular weight:753.78R-(+)-Cotinine
CAS:<p>R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.</p>Formula:C10H12N2OColor and Shape:SolidMolecular weight:176.22Cisatracurium besylate
CAS:<p>Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.</p>Formula:C53H72N2O12·2C6H5O3SPurity:97.89% - 99.85%Color and Shape:White Or White Powder CategoryMolecular weight:1243.48Cyclodrine
CAS:<p>Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.</p>Formula:C19H29NO3Purity:97.62%Color and Shape:SoildMolecular weight:319.44Angiopeptin
CAS:<p>Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.</p>Formula:C54H71N11O10S2Color and Shape:SolidMolecular weight:1098.34Albanin A
<p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>Formula:C20H18O6Color and Shape:SolidMolecular weight:354.358α-Bungarotoxin
CAS:<p>Neurotoxin that blocks neuromuscular transmission via irreversible inhibition of nicotinic ACh receptors (nAChRs).</p>Formula:C338H529N97O105S11Purity:98%Color and Shape:SolidMolecular weight:7984.14Cevimeline hydrochloride hemihydrate
CAS:<p>Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.</p>Formula:C20H38Cl2N2O3S2Purity:97.00%Color and Shape:SolidMolecular weight:489.55AC1-IN-1
CAS:<p>AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).</p>Formula:C18H18FN5O2Purity:99.89%Color and Shape:SolidMolecular weight:355.37ANQ-9040
CAS:<p>ANQ-9040 is a nondepolarizing neuromuscular relaxant of the steroid class.</p>Formula:C36H58N2O5SColor and Shape:SolidMolecular weight:630.92Biperiden Hydrochloride
CAS:<p>Biperiden HCl is an anti-Parkinson's drug, blocks M1 receptors, manages all Parkinson's types, and is FDA-approved. Non-toxic at 0.11 mg/kg to rats' cognition.</p>Formula:C21H30ClNOPurity:98%Color and Shape:SolidMolecular weight:347.92nAChR agonist 2
CAS:<p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>Formula:C11H16N2Color and Shape:SolidMolecular weight:176.263Emraclidine
CAS:<p>Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.</p>Formula:C20H21F3N4OPurity:99.96%Color and Shape:SolidMolecular weight:390.4TIP 39, Tuberoinfundibular Neuropeptide
CAS:<p>TIP39 is a synthetic neuropeptide agonist for human and rat PTH2 receptors from the hypothalamus.</p>Formula:C202H325N61O54SPurity:98%Color and Shape:SolidMolecular weight:4504.2Lupanine hydrochloride
CAS:<p>Lupanine hydrochloride, a Sparteine derivative, binds to nAChR with a Ki of 500 nM and has ganglioplegic properties.</p>Formula:C15H25ClN2OColor and Shape:SolidMolecular weight:284.83Pozanicline hydrochloride
<p>Pozanicline hydrochloride is an oral α4β2 nAChR agonist with a 16.7 nM Ki, insignificantly binding to α7 nAChR.</p>Formula:C11H17ClN2OPurity:97.13% - 99.81%Color and Shape:SolidMolecular weight:228.72PDE4-IN-4
CAS:<p>PDE4-IN-4 is a compound acting as both a potent M3 antagonist (p IC 50 = 10.2) and a PDE4 inhibitor (p IC 50 = 8.8), designed for inhalation-based treatment of</p>Formula:C36H37Cl2N3O7SColor and Shape:SolidMolecular weight:726.67Methylatropine (nitrate)
CAS:<p>Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.</p>Formula:C18H26N2O6Color and Shape:SolidMolecular weight:366.414nAChR modulator-1
CAS:<p>nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Formula:C12H8ClN3O2Color and Shape:SolidMolecular weight:261.66Heliosupine N-oxide
<p>Heliosupine N-oxide is a useful organic compound for research related to life sciences and the catalog number is T125058.</p>Formula:C20H31NO8Color and Shape:SolidMolecular weight:413.467Small Cardioactive Peptide B (SCPB)
CAS:<p>SCPB: neurally active peptide, boosts adenylate cyclase in heart/gills, EC50s: 0.1 μM (heart), 1.0 μM (gills).</p>Formula:C52H80N14O11S2Purity:98%Color and Shape:SolidMolecular weight:1141.41Epiboxidine
CAS:<p>Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.</p>Formula:C10H14N2OColor and Shape:SolidMolecular weight:178.23M 8218
CAS:<p>M 8218 is a bioactive chemical.</p>Formula:C20H29NO2Color and Shape:SolidMolecular weight:315.45Desfesoterodine
CAS:<p>Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.</p>Formula:C22H31NO2Purity:99.77%Color and Shape:SolidMolecular weight:341.49α-Conotoxin AuIB
CAS:<p>Selective antagonist of α3β4 nicotinic acetylcholine receptors.</p>Formula:C65H89N17O21S4Purity:98%Color and Shape:SolidMolecular weight:1572.76Flupyradifurone
CAS:<p>Flupyradifurone (flupyradifurone) is a systemic insecticide and nicotinic acetylcholine receptor (nAChR) agonist interfer nervous system of insects.</p>Formula:C12H11ClF2N2O2Purity:99.83%Color and Shape:SolidMolecular weight:288.68α-Conotoxin imi
CAS:<p>alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.</p>Formula:C52H78N20O15S4Purity:98%Color and Shape:SolidMolecular weight:1351.56Tiquizium
CAS:<p>Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.</p>Formula:C19H24NS2Purity:99.82%Color and Shape:SolidMolecular weight:330.53CVN417
<p>CVN417 is an orally active antagonist of nAChR containing the α6 subunit, modulating phasic dopaminergic neurotransmission in an impulse-dependent fashion.</p>Color and Shape:Odour SolidPerindoprilat
CAS:<p>Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.</p>Formula:C17H28N2O5Purity:99.48%Color and Shape:SolidMolecular weight:340.41Dicloromezotiaz
CAS:<p>Dicloromezotiaz: Potent insecticide targeting nAChRs, controls various lepidoptera.</p>Formula:C19H12Cl3N3O2SColor and Shape:SolidMolecular weight:452.74[D-Trp7,9,10]-Substance P
CAS:<p>Substance P analog that inhibits activation of Gq/11 by M1 muscarinic ACh receptors. Does not inhibit Gi/o activation by M2 ACh receptors.</p>Formula:C79H105N21O13SPurity:98%Color and Shape:SolidMolecular weight:1588.89SIB 1553A
CAS:<p>SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to study diseases associated with neurodegeneration.</p>Formula:C13H19NOSPurity:99.79%Color and Shape:SoildMolecular weight:237.36(+)-Coclaurine hydrochloride
CAS:<p>(+)-Coclaurine hydrochloride, also known as (+)-(R)-Coclaurine, is a benzyltetrahydroisoquinoline alkaloid extracted from multiple plant species.</p>Formula:C17H20ClNO3Purity:98%Color and Shape:SolidMolecular weight:321.8Destomycin A
CAS:<p>Destomycin A, an aminoglycoside antibiotic, exhibits activity against bacterial (Gram-positive and Gram-negative), antifungal, and anthelmintic agents. It inhibits peptide synthesis in Escherichia coli cells and stimulates adenylate cyclase in animal tissues.</p>Formula:C20H37N3O13Color and Shape:SolidMolecular weight:527.52CDD0102 HCl
CAS:<p>CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.</p>Formula:C8H13ClN4OPurity:99.7%Color and Shape:SoildMolecular weight:216.67Mant-GTPγS
CAS:<p>Mant-GTPγS, an effective GTP analog, displays strong competitive inhibition of adenylyl cyclase (AC). Additionally, it acts as a potent inhibitor of YdeH.</p>Formula:C18H23N6O14P3SColor and Shape:SolidMolecular weight:672.39Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Formula:C45H47N7O9S3Color and Shape:SolidMolecular weight:926.09Thiothixene
CAS:<p>Thiothixene has a wide range of applications in life science related research.</p>Formula:C23H29N3O2S2Color and Shape:SolidMolecular weight:443.62Fentonium bromide
CAS:<p>Fentonium bromide is a biochemical.</p>Formula:C31H34BrNO4Color and Shape:SolidMolecular weight:564.51(S)-UFR2709 hydrochloride
CAS:<p>(S)-UFR2709 HCl: competitive nAChR blocker, prefers α4β2 over α7, lessens anxiety & alcohol intake in rats, studies nicotine addiction.</p>Formula:C13H18ClNO2Purity:98.94%Color and Shape:SolidMolecular weight:255.74PF-06827443
<p>PF-06827443 is a orally bioavailable, CNS-penetrant M1-selective PAM with minimal agonist activity.</p>Formula:C24H24N2O4Color and Shape:SolidMolecular weight:404.475-Hydroxymethyl tolterodine formate
CAS:<p>5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine and Fesoterodine. It is synthesized by the cytochrome P450 (CYP) isoenzyme CYP2D6 and plasma esterases.</p>Formula:C23H33NO4Color and Shape:SolidMolecular weight:387.51(Rac)-5-Carboxy tolterodine
CAS:<p>(Rac)-5-Carboxy tolterodine is an inactive metabolite of Tolterodine, which acts as a muscarinic acetylcholine receptor antagonist.</p>Formula:C22H29NO3Color and Shape:SolidMolecular weight:355.47RuBi-Nicotine
CAS:<p>Nicotinic receptor agonist</p>Formula:C40H44Cl2N8RuPurity:98%Color and Shape:SolidMolecular weight:808.81(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
CAS:<p>(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.</p>Formula:C22H32ClNO2Color and Shape:SolidMolecular weight:377.95NNC 11-1607
CAS:<p>NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.</p>Formula:C30H32N6O2S2Color and Shape:SolidMolecular weight:572.74N,N-Dicyclohexylcarbodiimide
CAS:<p>N,N-Dicyclohexylcarbodiimide (Dicyclohexylcarbodiimide) is a cross-linking agent used in the synthesis of active ester-containing reagents.</p>Formula:C13H22N2Purity:98.28% - 99.73%Color and Shape:SolidMolecular weight:206.33bPiDDB
CAS:<p>bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.</p>Formula:C24H38Br2N2Purity:98.72%Color and Shape:SolidMolecular weight:514.38TC-2216
CAS:<p>TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.</p>Formula:C12H17N3Purity:99.33%Color and Shape:SolidMolecular weight:203.28Irsogladine maleate
CAS:<p>Compound PDK0375, with CAS No. 84504-69-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0375 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formula:C9H7Cl2N5Color and Shape:SolidMolecular weight:256.09trans-Cevimeline hydrochloride
CAS:<p>AF 102A hydrochloride is a biochemical.</p>Formula:C10H18ClNOSColor and Shape:SolidMolecular weight:235.77Lobeline sulfate
CAS:<p>Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.</p>Formula:C22H29NO6SPurity:98%Color and Shape:White PowderMolecular weight:435.54Hydroxybupropion
CAS:<p>Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).</p>Formula:C13H18ClNO2Purity:99.73%Color and Shape:Off-White SolidMolecular weight:255.74Oxotremorine
CAS:<p>Oxotremorine acts as an agonist of mAChR, specifically activating the M1 and M3 acetylcholine receptors. In drug discrimination experiments with macaques, it exhibits effects similar to nicotine.</p>Formula:C12H18N2OColor and Shape:SolidMolecular weight:206.28Methyllycaconitine citrate
CAS:<p>Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.</p>Formula:C43H58N2O17Purity:98.03% - 98.91%Color and Shape:SolidMolecular weight:874.92G-Protein antagonist peptide
CAS:<p>Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.</p>Formula:C57H64N12O9SPurity:98%Color and Shape:SolidMolecular weight:1093.27M4 mAChR agonist-1
CAS:<p>M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).</p>Formula:C14H18N4OSPurity:99.14%Color and Shape:SolidMolecular weight:290.38Muscarine
CAS:<p>Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>Formula:C9H20NO2Purity:98%Color and Shape:SolidMolecular weight:174.26M3/PDE4 modulator-1
<p>M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor.</p>Formula:C38H41Cl2N3O8SColor and Shape:SolidMolecular weight:770.725-AMAM-2-CP
CAS:<p>5-AMAM-2-CP, a significant metabolite of Acetamiprid, serves as a global insecticide within the neonicotinoid class and acts as an nAChR agonist [1] [2].</p>Formula:C9H11ClN2OColor and Shape:SolidMolecular weight:198.65(R)-Dinotefuran
CAS:<p>(R)-Dinotefuran, a neonicotinoid, is 1.7-2.4x more effective against pests like Aphis gossypii and safer for bees.</p>Formula:C7H14N4O3Color and Shape:SolidMolecular weight:202.21Ebiratide TFA
<p>Ebiratide (HOE-427) TFA is a derivative of ACTH4-9 that exerts its effect directly on the central nervous system, enhancing memory. Ebiratide TFA also promotes the metabolism of acetylcholine (ACh) in the rat brain.</p>Formula:C48H73N11O10S·xC2HF3O2Color and Shape:SolidMolecular weight:996.23 (free base)TDI-10229
CAS:<p>TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.</p>Formula:C16H16ClN5Purity:99.85% - 99.89%Color and Shape:SoildMolecular weight:313.78BTMPS
CAS:<p>BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.</p>Formula:C28H52N2O4Purity:98.1%Color and Shape:SolidMolecular weight:480.72Anabaseine
CAS:<p>Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.</p>Formula:C10H12N2Color and Shape:SolidMolecular weight:160.22N-Ethyl-N-(3-pyridylmethyl)amine
CAS:<p>N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.</p>Formula:C8H12N2Purity:99.65%Color and Shape:SolidMolecular weight:136.19Soclenicant
CAS:<p>Soclenicant is a negative-altering modulator of α 7 -nAChR for anxiety, depression, and PTSD, due to its high selectivity, oral availability</p>Formula:C24H26N4O3Purity:99.57%Color and Shape:SoildMolecular weight:418.49Rivanicline 2HCl
<p>Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.</p>Formula:C10H16Cl2N2Purity:99.4%Color and Shape:SoildMolecular weight:235.15Proadrenomedullin (1-20), human
CAS:<p>Endogenous peptide; agonist of MRGPRX2 (EC50=251 nM); noncompetitive inhibitor of nicotinic receptors; reduces catecholamine secretion; antihypertensive.</p>Formula:C112H178N36O27Purity:98%Color and Shape:SolidMolecular weight:2460.84TC-2559 difumarate
CAS:<p>TC-2559 difumarate: Oral α4β2 nAChR partial agonist, CNS-selective, EC50 0.18 μM, prefers α4β2 over α2β4/α4β4/α3β4, antinociceptive.</p>Formula:C20H26N2O9Color and Shape:SolidMolecular weight:438.43Bensultap
CAS:<p>Bensultap is an agricultural chemical typically used as a pesticide.</p>Formula:C17H21NO4S4Purity:98%Color and Shape:SolidMolecular weight:431.61Ebiratide
CAS:<p>Ebiratide is an analog of ACTH 4-9.</p>Formula:C48H73N11O10SPurity:98%Color and Shape:SolidMolecular weight:996.23GeX-2
CAS:<p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>Formula:C103H169N43O27Color and Shape:SolidMolecular weight:2441.72Aceclidine (hydrochloride)
CAS:<p>agonist of muscarinic receptors</p>Formula:C9H16ClNO2Purity:98%Color and Shape:SolidMolecular weight:205.68Tropicamide
CAS:<p>Tropicamide (Ro 1-7683), a synthetic atropine-like muscarinic antagonist, dilates pupils and paralyzes eye muscles for diagnostic use.</p>Formula:C17H20N2O2Purity:99.78% - 99.94%Color and Shape:White PowderMolecular weight:284.35Navafenterol
CAS:<p>AZD-8871, a potential COPD and asthma treatment, may work well with ICS.</p>Formula:C38H42N6O6S2Color and Shape:SolidMolecular weight:742.91α-Conotoxin PIA
CAS:<p>Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM</p>Formula:C79H125N27O25S4Purity:98%Color and Shape:SolidMolecular weight:1981.3(-)-OPC-51803
CAS:<p>(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.</p>Formula:C26H32ClN3O2Purity:98.73% - 99.59%Color and Shape:SoildMolecular weight:454(rel)-Asperparaline A
CAS:<p>Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.</p>Formula:C20H29N3O3Color and Shape:SolidMolecular weight:359.47sabcomeline
CAS:<p>Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.</p>Formula:C10H15N3OColor and Shape:SolidMolecular weight:193.25DSPE-PEG2000-RVG29
<p>DSPE-PEG2000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and can traverse the BBB.</p>Color and Shape:Odour SolidLu AE51090
CAS:<p>Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.</p>Formula:C24H29N3O3Purity:99.57%Color and Shape:SolidMolecular weight:407.515-AAM-2-CP
CAS:<p>5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.</p>Formula:C8H9ClN2OPurity:99.58%Color and Shape:SolidMolecular weight:184.62(R)-(+)-Anatabine
CAS:<p>(R)-(+)-Anatabine is an less active R-enantiomer of Anatabine. Anatabine is a potent agonist of α4β2 nAChR.</p>Formula:C10H12N2Purity:98%Color and Shape:SolidMolecular weight:160.22(Rac)-Sabcomeline
CAS:<p>(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.</p>Formula:C10H15N3OPurity:99.14%Color and Shape:SolidMolecular weight:193.25LAS190792
CAS:<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Formula:C39H43ClN4O9S2Color and Shape:SolidMolecular weight:811.36Br-PBTC
CAS:<p>Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.</p>Formula:C14H15BrN2OSColor and Shape:SolidMolecular weight:339.25β2AR/M-receptor agonist-1
CAS:<p>β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and</p>Formula:C43H56BrN3O7Color and Shape:SolidMolecular weight:806.82Dexetimide
CAS:<p>Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.</p>Formula:C23H26N2O2Color and Shape:SolidMolecular weight:362.46Metixene hydrochloride hydrate
CAS:<p>Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.</p>Formula:C20H26ClNOSPurity:99.88%Color and Shape:SolidMolecular weight:363.95Fipexide hydrochloride
CAS:<p>Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.</p>Formula:C20H22Cl2N2O4Color and Shape:SolidMolecular weight:425.31NKH477
CAS:<p>NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.</p>Formula:C27H44ClNO8Purity:98% - 98%Color and Shape:SolidMolecular weight:546.09Tolterodine
CAS:<p>Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.</p>Formula:C22H31NOPurity:99.71%Color and Shape:White Like Or Light Brown Crystalline PowderMolecular weight:325.49YM-58790 hydrochloride
CAS:<p>YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).</p>Formula:C27H32ClN3O2Purity:98%Color and Shape:SolidMolecular weight:466.02Palmatine hydroxide
CAS:<p>Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.</p>Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.41Cevimeline
CAS:<p>Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.</p>Formula:C10H17NOSColor and Shape:Off-White SolidMolecular weight:199.31Pirmenol hydrochloride
CAS:<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Formula:C22H31ClN2OColor and Shape:SolidMolecular weight:374.95Varenicline Hydrochloride
CAS:<p>Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).</p>Formula:C13H14ClN3Purity:99.854%Color and Shape:SolidMolecular weight:247.72Cevimeline hydrochloride
CAS:<p>Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.</p>Formula:C10H18ClOSColor and Shape:SolidMolecular weight:235.77Glycerophosphoinositol choline
CAS:<p>Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.</p>Formula:C14H32NO12PColor and Shape:SolidMolecular weight:437.38Ispronicline
CAS:<p>Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitive</p>Formula:C14H22N2OPurity:97.70% - 99.16%Color and Shape:SolidMolecular weight:234.34Sabcomeline hydrochloride
CAS:<p>Sabcomeline is a selective M1 receptor partial agonist.</p>Formula:C10H16ClN3OColor and Shape:SolidMolecular weight:229.71(±)-Darifenacin
CAS:<p>(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.</p>Formula:C28H30N2O2Color and Shape:SolidMolecular weight:426.55VU0467485
CAS:<p>VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.</p>Formula:C17H17FN4O2SPurity:98%Color and Shape:SolidMolecular weight:360.41Clorprenaline
CAS:<p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>Formula:C11H16ClNOPurity:98.9%Color and Shape:SolidMolecular weight:213.7ABT-107
CAS:<p>ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.</p>Formula:C19H20N4OColor and Shape:SolidMolecular weight:320.396
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