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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1045 products of "Proteases/Proteasome"

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  • Avatrombopag

    CAS:
    <p>Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiation</p>
    Formula:C29H34Cl2N6O3S2
    Purity:99.01% - 99.63%
    Color and Shape:Solid
    Molecular weight:649.65
  • Velpatasvir

    CAS:
    <p>Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.</p>
    Formula:C49H54N8O8
    Purity:99.17% - 99.83%
    Color and Shape:Solid
    Molecular weight:883
  • Grazoprevir

    CAS:
    <p>Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.</p>
    Formula:C38H50N6O9S
    Purity:99.36% - >99.99%
    Color and Shape:Solid
    Molecular weight:766.9
  • Ditiocarb sodium

    CAS:
    <p>Ditiocarb sodium (Sodium diethyldithiocarbamate) (sodium diethiocarbamate) is a copper reagent, which reacts with Cu2 + solution to form a complex and improves</p>
    Formula:C5H10NNaS2
    Purity:98.04%
    Color and Shape:White Solid Crystalline
    Molecular weight:171.26
  • KGP94

    CAS:
    <p>KGP94 is a potent, selective, and competitive inhibitor of the lysosomal endopeptidase enzyme.</p>
    Formula:C14H12BrN3OS
    Purity:99.6%
    Color and Shape:Solid
    Molecular weight:350.23
  • Dabigatran Etexilate Mesylate

    CAS:
    <p>Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor.</p>
    Formula:C34H41N7O5·CH4O3S
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:723.84
  • ML281

    CAS:
    <p>ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.</p>
    Formula:C22H19N3O2S
    Purity:99.12% - 99.87%
    Color and Shape:Solid
    Molecular weight:389.47
  • Daclatasvir dihydrochloride

    CAS:
    <p>Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.</p>
    Formula:C40H52Cl2N8O6
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:811.8
  • (S,S)-TAPI-1

    CAS:
    <p>"(S,S)-TAPI-1, an isomer of TAPI-1, inhibits MMPs and TACE (ADAM17), reducing cell surface protein shedding."</p>
    Formula:C26H37N5O5
    Color and Shape:Solid
    Molecular weight:499.6
  • Anagliptin hydrochloride

    CAS:
    <p>Anagliptin (SK-0403) hydrochloride: potent, selective oral DPP-4 inhibitor; IC50: DPP-4 3.8 nM, DPP-8 68 nM, DPP-9 60 nM.</p>
    Formula:C19H26ClN7O2
    Color and Shape:Solid
    Molecular weight:419.91
  • Ixazomib citrate

    CAS:
    <p>Ixazomib citrate (MLN9708), a prodrug of Ixazomib (MMLN-2238), is an oral 2nd-gen proteasome inhibitor with anti-cancer potential (IC50: 3.4 nM).</p>
    Formula:C20H23BCl2N2O9
    Purity:98.37% - >99.99%
    Color and Shape:Solid
    Molecular weight:517.12
  • Darunavir

    CAS:
    <p>Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.</p>
    Formula:C27H37N3O7S
    Purity:99.67% - 99.76%
    Color and Shape:White Amorphous Solid
    Molecular weight:547.66
  • Coblopasvir dihydrochloride

    CAS:
    <p>Coblopasvir dihydrochloride can be used to study chronic HCV infection and is a pan-genotypic nonstructural protein 5A (NS5A) inhibitor.</p>
    Formula:C41H52Cl2N8O8
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:855.81
  • 4-Butylresorcinol

    CAS:
    <p>4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.</p>
    Formula:C10H14O2
    Purity:98.64% - ≥95%
    Color and Shape:Light Beige Solid Powder
    Molecular weight:166.22
  • XMD8-87

    CAS:
    <p>XMD8-87 (ACK1-B19), a TNK2 inhibitor, strongly blocks TNK2 phosphorylation and mutations in tumors.</p>
    Formula:C24H27N7O2
    Purity:98.05% - 99.89%
    Color and Shape:Solid
    Molecular weight:445.52
  • Paritaprevir

    CAS:
    <p>Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂,对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 1.31 μM。</p>
    Formula:C40H43N7O7S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:765.88
  • Bemnifosbuvir

    CAS:
    <p>Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.</p>
    Formula:C24H33FN7O7P
    Purity:99.35% - 99.54%
    Color and Shape:Solid
    Molecular weight:581.53
  • 7-Amino-4-methylcoumarin-3-acetic acid

    CAS:
    <p>7-Amino-4-methylcoumarin-3-acetic acid (7-Amino-4-methylcoumarin) is more suitable as a substrate for enteropeptidase than GD(4)K-NA.</p>
    Formula:C12H11NO4
    Purity:98.38%
    Color and Shape:Solid
    Molecular weight:233.22
  • Letermovir

    CAS:
    <p>Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.</p>
    Formula:C29H28F4N4O4
    Purity:99.85% - 99.87%
    Color and Shape:Solid
    Molecular weight:572.55
  • LY 3000328

    CAS:
    <p>LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.</p>
    Formula:C25H29FN4O5
    Purity:97.83% - 99.54%
    Color and Shape:Solid
    Molecular weight:484.52