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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 993 products of "Proteases/Proteasome"

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  • Diethyl pyimDC

    CAS:
    Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).
    Formula:C14H15N3O4
    Color and Shape:Solid
    Molecular weight:289.29

    Ref: TM-T27170

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tyrosinase-IN-6

    CAS:
    Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.
    Formula:C24H31N3O2
    Color and Shape:Solid
    Molecular weight:393.52

    Ref: TM-T61817

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Aldumastat

    CAS:
    Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.
    Formula:C20H24F2N4O3
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:406.43

    Ref: TM-T35859

    1mg
    269.00€
  • Garvagliptin

    CAS:
    Garvagliptin has antidiabetic activity.
    Formula:C18H23F2N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.46

    Ref: TM-T27402

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alicapistat

    CAS:
    Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).
    Formula:C25H27N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.5

    Ref: TM-T14178

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • ZM223 hydrochloride (2031177-48-5 free base)


    ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.
    Formula:C23H18ClF3N4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:538.99

    Ref: TM-T13412L

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • NNGH

    CAS:
    NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.
    Formula:C13H20N2O5S
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:316.37

    Ref: TM-T21735

    1mg
    71.00€
    5mg
    105.00€
    10mg
    178.00€
    25mg
    313.00€
    50mg
    464.00€
    100mg
    660.00€
  • VEL-0230

    CAS:
    VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.
    Formula:C14H24NNaO5
    Color and Shape:Solid
    Molecular weight:309.33

    Ref: TM-T69793

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MK-4882

    CAS:
    MK-4882 is an effective inhibitor of HCV NS5A.
    Formula:C42H50N8O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:778.9

    Ref: TM-T24475

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • PK44 phosphate

    CAS:
    PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).
    Formula:C17H19F5N7O5P
    Color and Shape:Solid
    Molecular weight:527.349

    Ref: TM-T63698

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • BAY8040

    CAS:
    BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.
    Formula:C21H16F3N5O2
    Color and Shape:Solid
    Molecular weight:427.38

    Ref: TM-T30303

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SA 152

    CAS:
    SA 152 is an organophosphoric inhibitor.
    Formula:C19H12F12NO2P
    Color and Shape:Solid
    Molecular weight:545.26

    Ref: TM-T70705

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AA10 TG2 inhibitor

    CAS:
    AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).
    Formula:C32H36N4O5
    Color and Shape:Solid
    Molecular weight:556.65

    Ref: TM-T26494

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DPP-4-IN-1

    CAS:
    DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.
    Formula:C19H19ClN6
    Color and Shape:Solid
    Molecular weight:366.85

    Ref: TM-T61422

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ACH-806

    CAS:
    ACH-806 is an NS4A antagonist. It can inhibit Hepatitis C Virus (HCV) replication with an EC50 of 14 nM.
    Formula:C19H20F3N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.44

    Ref: TM-T14095

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • CAY10704

    CAS:
    CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.
    Formula:C18H20Cl2N2
    Color and Shape:Solid
    Molecular weight:335.27

    Ref: TM-T37463

    1mg
    166.00€
    5mg
    705.00€
    10mg
    1,234.00€
  • ASPER-29

    CAS:
    ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.
    Formula:C31H29BrN2O5S
    Color and Shape:Solid
    Molecular weight:621.54

    Ref: TM-T73395

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Sortin1

    CAS:
    Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.
    Formula:C26H19NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.43

    Ref: TM-T16912

    25mg
    2,570.00€
    50mg
    3,352.00€
    100mg
    5,089.00€
  • MDK7677

    CAS:
    MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.
    Formula:C12H10N4O3
    Color and Shape:Solid
    Molecular weight:258.23

    Ref: TM-T28003

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Furaprofen

    CAS:
    Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.
    Formula:C17H14O3
    Purity:98.49% - 99.52%
    Color and Shape:Solid
    Molecular weight:266.29

    Ref: TM-T16715

    1mg
    274.00€
    5mg
    655.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€