
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(37 products)
- Cysteine Protease(111 products)
- DPP-4(24 products)
- Glutaminase(44 products)
- HIV Protease(502 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(89 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 992 products of "Proteases/Proteasome"
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2-MPPA
CAS:2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.Formula:C8H14O4SPurity:99.81%Color and Shape:SolidMolecular weight:206.26Ref: TM-T22497
1mg50.00€5mg99.00€10mg160.00€25mg358.00€50mg620.00€100mg1,108.00€200mg1,504.00€1mL*10mM (DMSO)109.00€Cofrogliptin
CAS:Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).Formula:C18H19F5N4O3SColor and Shape:SolidMolecular weight:466.43Gosogliptin
CAS:Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.Formula:C17H24F2N6OPurity:99.74%Color and Shape:SolidMolecular weight:366.41Efegatran sulfate
CAS:Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.Formula:C21H34N6O7SPurity:≥98% - ≥98%Color and Shape:SolidMolecular weight:514.6ZD-0892
CAS:ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).Formula:C24H32F3N3O5Purity:95% - 99.53%Color and Shape:SolidMolecular weight:499.52Calpain Inhibitor XII
CAS:Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.
Formula:C26H34N4O5Color and Shape:SolidMolecular weight:482.57MMP2-IN-2
CAS:MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.Formula:C13H8N4O4Purity:98.09%Color and Shape:SolidMolecular weight:284.23Etarotene
CAS:Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is aFormula:C25H32O2SPurity:99.58% - 99.98%Color and Shape:SolidMolecular weight:396.59Gemigliptin
CAS:Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)Formula:C18H19F8N5O2Purity:99.72%Color and Shape:SolidMolecular weight:489.36Ref: TM-T7369
2mg38.00€5mg57.00€10mg93.00€25mg148.00€50mg245.00€100mg385.00€500mg873.00€1mL*10mM (DMSO)84.00€Sirpiglenastat
CAS:Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.Formula:C22H27N5O5Purity:98.01% - 98.37%Color and Shape:SolidMolecular weight:441.48MMP2-IN-3
CAS:MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).Formula:C23H21N3OPurity:99.38%Color and Shape:SolidMolecular weight:355.43Ref: TM-T61271
1mg64.00€5mg132.00€10mg195.00€25mg315.00€50mg439.00€100mg590.00€200mg793.00€1mL*10mM (DMSO)140.00€TY-51469
CAS:TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).Formula:C20H15FN2O6S4Purity:99.65%Color and Shape:SolidMolecular weight:526.6Melagatran
CAS:Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.Formula:C22H31N5O4Purity:98.29% - >99.99%Color and Shape:SolidMolecular weight:429.51Ref: TM-T11994
1mg487.00€5mg1,134.00€10mg1,468.00€25mg2,215.00€50mg2,962.00€100mg4,024.00€1mL*10mM (DMSO)1,071.00€Sovaprevir
CAS:Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.Formula:C43H53N5O8SPurity:99.89%Color and Shape:SolidMolecular weight:799.97Ref: TM-T28830
1mg253.00€5mg620.00€10mg884.00€25mg1,314.00€50mg1,773.00€100mg2,385.00€1mL*10mM (DMSO)982.00€UK-396082
CAS:UK-396082 is a TAFI inhibitor that inhibits Carboxypeptidase B and can be used in the study of thrombosis, atherosclerosis, cancer and fibrotic conditions.Formula:C12H21N3O2Purity:99.89%Color and Shape:SolidMolecular weight:239.31P32/98 hemifumarate
CAS:P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.Formula:C22H40N4O6S2Purity:99.46%Color and Shape:SolidMolecular weight:520.71TG2-IN-3h
CAS:TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitorFormula:C21H26N4O4SPurity:99.34% - 99.76%Color and Shape:SolidMolecular weight:430.52Lenacapavir
CAS:Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.Formula:C39H32ClF10N7O5S2Purity:99.61% - 99.87%Color and Shape:SolidMolecular weight:968.28Ref: TM-T11465
1mg187.00€5mg376.00€10mg565.00€25mg998.00€50mg1,388.00€100mg1,882.00€200mg2,622.00€1mL*10mM (DMSO)615.00€PG-116800
CAS:PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.Formula:C24H27N3O7SPurity:98.03% - 99.66%Color and Shape:SolidMolecular weight:501.5520S Proteasome activator 1
CAS:20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.Formula:C27H19ClF2N2OSPurity:99.82%Color and Shape:SolidMolecular weight:492.97
