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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 990 products of "Proteases/Proteasome"

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  • TS-021

    CAS:
    TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.
    Formula:C17H24FN3O5S
    Purity:>99.99% - >99.99%
    Color and Shape:Solid
    Molecular weight:401.45

    Ref: TM-T29019

    1mg
    164.00€
    2mg
    234.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • Etarotene

    CAS:
    Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is a
    Formula:C25H32O2S
    Purity:99.58% - 99.98%
    Color and Shape:Solid
    Molecular weight:396.59

    Ref: TM-T25393

    1mg
    144.00€
    5mg
    346.00€
    10mg
    494.00€
    25mg
    740.00€
  • Cyclotheonellazole A

    CAS:
    Cyclotheonellazole A inhibits elastase (IC50=0.034nM) & chymotrypsin (IC50=0.62nM), a natural macrocyclic peptide.
    Formula:C44H54N9NaO14S2
    Color and Shape:Solid
    Molecular weight:1020.07

    Ref: TM-T76231

    5mg
    To inquire
    50mg
    To inquire
  • Inogatran

    CAS:
    Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.
    Formula:C21H38N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.56

    Ref: TM-T11659

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • AZD-9819

    CAS:
    AZD-9819 is a neutrophil elastase (HNE) inhibitor applicable for research into chronic obstructive pulmonary disease (COPD).
    Formula:C25H19F3N6O2
    Purity:100% - 99.18%
    Color and Shape:Solid
    Molecular weight:492.45

    Ref: TM-T68240

    1mg
    411.00€
    5mg
    954.00€
    10mg
    1,279.00€
    25mg
    1,873.00€
    50mg
    2,547.00€
  • NS5A-IN-2

    CAS:
    NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.
    Formula:C46H45N7O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:807.89

    Ref: TM-T73834

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • MMP-9-IN-8

    CAS:
    MMP-9-IN-8 (Compound 3), an MMP-9 inhibitor, exhibits inhibitory activities of 42.16% at 10 μM and 58.28% at 50 μM.
    Formula:C20H21F4N7O
    Color and Shape:Solid
    Molecular weight:451.42

    Ref: TM-T81777

    5mg
    To inquire
    50mg
    To inquire
  • Petesicatib

    CAS:
    Petesicatib is an inhibitor of cathepsin S. Petesicatib used in the research of immune diseases.
    Formula:C25H23F6N5O4S
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:603.54

    Ref: TM-T16474

    1mg
    100.00€
    5mg
    236.00€
    10mg
    371.00€
    25mg
    735.00€
    50mg
    1,134.00€
    100mg
    1,468.00€
    200mg
    1,972.00€
    1mL*10mM (DMSO)
    314.00€
  • LY52

    CAS:
    LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.
    Formula:C22H24N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.45

    Ref: TM-T25765

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • Ro 31-9790

    CAS:
    Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).
    Formula:C15H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.41

    Ref: TM-T12762

    25mg
    1,730.00€
    50mg
    2,262.00€
    100mg
    2,945.00€
  • FK706

    CAS:
    FK706, a human neutrophil elastase inhibitor (IC50: 83 nM, Ki: 4.2 nM), also blocks mouse and porcine elastases. Anti-inflammatory.
    Formula:C26H33F3N4NaO7
    Color and Shape:Solid
    Molecular weight:593.556

    Ref: TM-T15285

    25mg
    1,378.00€
    50mg
    1,791.00€
    100mg
    2,872.00€
  • XL-784

    CAS:
    XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.
    Formula:C42H42Cl2F4MgN6O16S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1122.15

    Ref: TM-T13358

    2mg
    359.00€
    1mL*10mM (DMSO)
    33.00€
  • KCC009

    CAS:
    KCC009 is a potent and selective Transglutaminase 2 Inhibitor.
    Formula:C21H22BrN3O5
    Color and Shape:Solid
    Molecular weight:476.32

    Ref: TM-T27717

    25mg
    690.00€
    50mg
    897.00€
    100mg
    1,341.00€
  • TP0556351

    CAS:
    TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.
    Formula:C50H70N10O16
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1067.15

    Ref: TM-T74632

    5mg
    To inquire
    50mg
    To inquire
  • JTK-853

    CAS:
    JTK-853: novel non-nucleoside HCV polymerase inhibitor with strong antiviral activity (EC50: 0.38 μM genotype 1a, 0.035 μM 1b).
    Formula:C28H23F7N6O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:704.64

    Ref: TM-T15631

    25mg
    4,374.00€
    50mg
    5,686.00€
    100mg
    7,397.00€
  • LU-005i

    CAS:
    LU-005i is a powerful inhibitor targeting the β5i subunit of immunoproteasomes, displaying a high potency with an IC 50 value of 6.6 nM, and exhibits selectivity by preferring β5i over the β5c subunit, which has an IC 50 value of 287 nM [1].
    Formula:C31H46N4O7
    Color and Shape:Solid
    Molecular weight:586.72

    Ref: TM-T84755

    10mg
    To inquire
    50mg
    To inquire
  • PTC725

    CAS:
    PTC725 is a selective HCV 1b replicons inhibitor. It has been shown to target the nonstructural protein 4B.
    Formula:C23H18F4N6O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.49

    Ref: TM-T24682

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • ONO 4817

    CAS:
    ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.
    Formula:C22H28N2O6
    Color and Shape:Solid
    Molecular weight:416.47

    Ref: TM-T21814

    1mg
    239.00€
    5mg
    1,044.00€
  • Thrombin inhibitor 1

    CAS:
    Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).
    Formula:C22H20Cl2F2N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.32

    Ref: TM-T10081

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • MK-3281

    CAS:
    MK-3281: Oral, potent HCV NS5B inhibitor with promising properties and efficacy in replication trials, suitable for clinical use.
    Formula:C29H37N3O3
    Color and Shape:Solid
    Molecular weight:475.62

    Ref: TM-T33432

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€