CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 985 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • MK-3281

    CAS:
    MK-3281: Oral, potent HCV NS5B inhibitor with promising properties and efficacy in replication trials, suitable for clinical use.
    Formula:C29H37N3O3
    Color and Shape:Solid
    Molecular weight:475.62

    Ref: TM-T33432

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • Cipemastat

    CAS:
    Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).
    Formula:C22H36N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.55

    Ref: TM-T10817

    25mg
    1,251.00€
    50mg
    1,629.00€
    100mg
    2,475.00€
  • Collagen proline hydroxylase inhibitor

    CAS:
    Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.
    Formula:C18H18N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:354.36

    Ref: TM-T10862

    25mg
    690.00€
    50mg
    897.00€
    100mg
    1,378.00€
  • Z-PDLDA-NHOH

    CAS:
    Z-PDLDA-NHOH is a potent, specific vertebrate collagenase inhibitor [1].
    Formula:C22H32N4O6
    Color and Shape:Solid
    Molecular weight:448.51

    Ref: TM-T80719

    5mg
    To inquire
    50mg
    To inquire
  • Petesicatib

    CAS:
    Petesicatib is an inhibitor of cathepsin S. Petesicatib used in the research of immune diseases.
    Formula:C25H23F6N5O4S
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:603.54

    Ref: TM-T16474

    1mg
    100.00€
    5mg
    236.00€
    10mg
    371.00€
    25mg
    735.00€
    50mg
    1,134.00€
    100mg
    1,468.00€
    200mg
    1,972.00€
    1mL*10mM (DMSO)
    314.00€
  • MMP13-IN-3

    CAS:
    MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.
    Formula:C24H22N4O5
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:446.46

    Ref: TM-T16124

    1mg
    93.00€
    5mg
    205.00€
    10mg
    334.00€
    25mg
    587.00€
    50mg
    802.00€
    100mg
    1,108.00€
    1mL*10mM (DMSO)
    227.00€
  • FK706

    CAS:
    FK706, a human neutrophil elastase inhibitor (IC50: 83 nM, Ki: 4.2 nM), also blocks mouse and porcine elastases. Anti-inflammatory.
    Formula:C26H33F3N4NaO7
    Color and Shape:Solid
    Molecular weight:593.556

    Ref: TM-T15285

    25mg
    1,378.00€
    50mg
    1,791.00€
    100mg
    2,872.00€
  • XL-784

    CAS:
    XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.
    Formula:C42H42Cl2F4MgN6O16S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1122.15

    Ref: TM-T13358

    2mg
    359.00€
    1mL*10mM (DMSO)
    33.00€
  • GSK-2485852

    CAS:
    GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.
    Formula:C27H25BF2N2O6S
    Color and Shape:Solid
    Molecular weight:554.37

    Ref: TM-T27463

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • XL-784 free base

    CAS:
    XL-784 free base selectively inhibits MMPs with IC50: MMP-1 (1.9µM), MMP-2 (0.81nM), MMP-3 (120nM), MMP-8 (10.8nM), MMP-9 (18nM), MMP-13 (0.56nM).
    Formula:C21H22ClF2N3O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:549.93

    Ref: TM-T13357

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • MDL-101146, (R)-

    CAS:
    MDL-101146, (R)- is an effective orally active inhibitor of human neutrophil elastase.
    Formula:C29H37F5N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:632.62

    Ref: TM-T25784

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • SSR 69071

    CAS:
    SSR69071: selective neutrophil elastase inhibitor, stronger for humans (Ki=0.0168 nM), may treat COPD, asthma, and reduce heart injury.
    Formula:C27H32N4O7S
    Color and Shape:Solid
    Molecular weight:556.63

    Ref: TM-T21989

    1mg
    105.00€
    5mg
    388.00€
    10mg
    750.00€
  • NK3201

    CAS:
    NK3201, a specific chymase inhibitor, suppresses bleomycin-induced pulmonary fibrosis in hamsters.
    Formula:C31H29N5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:567.59

    Ref: TM-T28177

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • Phe-Pro-Ala-pNA

    CAS:
    Phe-Pro-Ala-pNA is a chromogenic substrate utilized for assessing tripeptidyl peptidase activity.
    Formula:C23H27N5O5
    Color and Shape:Solid
    Molecular weight:453.49

    Ref: TM-T84840

    10mg
    To inquire
    50mg
    To inquire
  • DS-1040 Tosylate

    CAS:
    DS-1040 Tosylate is a thrombin-activated fibrinolysis inhibitor (TAFI) inhibitor and a fibrinolysis enhancer, used for researching thromboembolic diseases.
    Formula:C23H35N3O5S
    Color and Shape:Solid
    Molecular weight:465.61

    Ref: TM-T11100

    2mg
    111.00€
    25mg
    552.00€
    50mg
    718.00€
    100mg
    1,224.00€
  • MDL 27324

    CAS:
    MDL 27324 is an inhibitor of human neutrophil elastase.
    Formula:C29H38F3N5O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:641.7

    Ref: TM-T25782

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • BAY-678

    CAS:
    BAY-678: Oral selective human neutrophil elastase inhibitor; IC50: 20 nM; SGC-approved chemical probe.
    Formula:C20H15F3N4O2
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:400.35

    Ref: TM-T10473

    5mg
    37.00€
    10mg
    60.00€
    25mg
    119.00€
    50mg
    173.00€
    100mg
    264.00€
    200mg
    374.00€
    1mL*10mM (DMSO)
    42.00€
  • Z-FG-NHO-BzOME

    CAS:
    Z-FG-NHO-BzOME is a chemical compound functioning as a cysteine protease inhibitor, selectively targeting and inhibiting cathepsin B, cathepsin L, cathepsin S,
    Formula:C27H27N3O7
    Color and Shape:Solid
    Molecular weight:505.52

    Ref: TM-T80739

    5mg
    To inquire
    50mg
    To inquire
  • KB-R7785

    CAS:
    KB-R7785 is a novel ADAM12/MMP inhibitor improving heart function and insulin sensitivity by blocking HB-EGF and TNF-alpha.
    Formula:C18H27N3O4
    Color and Shape:Solid
    Molecular weight:349.42

    Ref: TM-T70280

    25mg
    4,483.00€
  • MDL 101146

    CAS:
    MDL 101146 is an orally active neutrophil elastase inhibitor.
    Formula:C29H37F5N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:632.62

    Ref: TM-T25781

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€