Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
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Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
BGB-102
CAS:807640-87-5
BGB-102 (JNJ-26483327) is a kinase inhibitor targeting FLT3 and YES1 and an antagonist targeting EGFR …
Formula:
C22H25BrN4O2
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
457.36
Ref: TM-T10531
| 1mg | 305.00 € | ||
| 5mg | 759.00 € | ||
| 10mg | 1,002.00 € | ||
| 25mg | 1,512.00 € | ||
| 50mg | 2,032.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
AKB-6899
CAS:1007377-55-0
AKB-6899 is an inhibitor of prolyl hydroxylase domain 3 (PHD3) and increases the soluble form …
Formula:
C14H11FN2O4
Purity:
97.11%
Color and Shape:
Solid
Molecular weight:
290.25
Ref: TM-T29797
| 1mg | 45.00 € | ||
| 1ml | 107.00 € | ||
| 2mg | 62.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 377.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
KER047
CAS:2248154-85-8
ALK2-IN-4, a highly effective ALK2 inhibitor.
Formula:
C26H30FN7O
Purity:
100% - 98.49%
Color and Shape:
Solid
Molecular weight:
475.56
Ref: TM-T39764
| 1mg | 94.00 € | ||
| 1ml | 246.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 739.00 € | ||
| 50mg | 1,053.00 € | ||
| 100mg | 1,613.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
EGFR-IN-1 hydrochloride
CAS:2227455-78-7
EGFR-IN-1 HCl targets L858R/T790M EGFR mutants over wild-type; IC50: 4 nM in H1975, 28 nM …
Formula:
C28H31ClN6O4
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
551.04
Ref: TM-T11157L
| 1mg | 95.00 € | ||
| 1ml | 335.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 737.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,033.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Canlitinib
CAS:2222730-78-9
Canlitinib, a tyrosine kinase inhibitor, holds potential for cancer research.
Formula:
C33H31F2N3O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
619.61
Ref: TM-T78206
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
TRK-IN-24
CAS:2937544-01-7
TRK-IN-24 (compound 10g) is a selective inhibitor of Trk receptors, effectively targeting TRKA, TRKC, and …
Formula:
C39H45N7O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
659.82
Ref: TM-T79706
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
TrkB-IN-1
CAS:1609067-49-3
TrkB-IN-1 is a potent, orally active agonist of the TrkB receptor, with favorable pharmacokinetic (PK) …
Formula:
C19H16N2O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
368.34
Ref: TM-T79011
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
WAY-600
CAS:1062159-35-6
WAY-600 is a potent, ATP-competitive and selective inhibitor of mTOR with IC50 of 9 nM; …
Formula:
C28H30N8O
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
494.59
Ref: TM-T6730
| 1mg | 38.00 € | ||
| 1ml | 111.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 355.00 € | ||
| 100mg | 495.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
CH6953755
CAS:2055918-71-1
CH6953755: oral YES1 kinase inhibitor, IC50 1.8 nM, potent, selective, anticancer, halts cell proliferation.
Formula:
C26H22F2N6O4S
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
552.55
Ref: TM-T10784
| 1mg | 57.00 € | ||
| 1ml | 149.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 576.00 € | ||
| 100mg | 924.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
CG 428
CAS:2412055-93-5
CG 428 is a potent tropomyosin receptor Kinase (TRK) Degrader (uSMITETM) with a DC50 of …
Formula:
C43H43FN10O6
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
814.86
Ref: TM-T41224
| 1mg | 172.00 € | ||
| 1ml | 434.00 € | ||
| 5mg | 415.00 € | ||
| 10mg | 609.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,753.00 € | ||
| 500mg | 3,511.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
UniPR1447
CAS:1809170-68-0
UniPR1447 is a dual antagonist for both EphA2 and EphB2 receptors, exhibiting an IC50 value …
Formula:
C36H50N2O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
574.79
Ref: TM-T80897
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
DYRKs-IN-2
CAS:1386980-04-6
DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM …
Formula:
C32H38ClN9O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
632.16
Ref: TM-T11133
| 25mg | 1,967.00 € | ||
| 50mg | 2,592.00 € | ||
| 100mg | 3,450.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
FIIN-1
CAS:1256152-35-8
FIIN-1 (FGFR irreversible inhibitor-1) is an irreversible and selective FGFR inhibitor with Kd of 2.8, …
Formula:
C32H39Cl2N7O4
Purity:
97.30%
Color and Shape:
Solid
Molecular weight:
656.6
Ref: TM-T37426
| 1mg | 78.00 € | ||
| 2mg | 101.00 € | ||
| 5mg | 198.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 766.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,077.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
c-Fms-IN-14
CAS:1898210-99-5
c-Fms-IN-14 (Example 76) is a potent inhibitor of the c-Fms kinase with an IC50 of …
Formula:
C26H24N6O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
436.51
Ref: TM-T79815
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
JND3229
CAS:2260886-64-2
JND3229 inhibits EGFRC797S; IC50: 5.8-30.5 nM; halts cell growth; effective in non-small cell lung cancer …
Formula:
C33H41ClN8O2
Purity:
97.35%
Color and Shape:
Solid
Molecular weight:
617.18
Ref: TM-T15615
| 1mg | 123.00 € | ||
| 1ml | 419.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 456.00 € | ||
| 25mg | 754.00 € | ||
| 50mg | 1,049.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
BMX-IN-1
CAS:1431525-23-3
BMX-IN-1 (BMX kinase inhibitor) is a selective inhibitor of bone marrow tyrosine kinase on chromosome …
Formula:
C29H24N4O4S
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
524.59
Ref: TM-T14692
| 1mg | 34.00 € | ||
| 1ml | 90.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 228.00 € | ||
| 50mg | 318.00 € | ||
| 100mg | 436.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
EGFR-IN-1
CAS:1625677-63-5
EGFR-IN-1: an oral, irreversible EGFR inhibitor targeting L858R/T790M mutations with high selectivity, showing potent antitumor …
Formula:
C28H30N6O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
514.58
Ref: TM-T11157
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Tyrphostin AG 538
CAS:133550-18-2
Tyrphostin AG 538 is a chalcone compound, an IGF-1 receptor kinase inhibitor (IC₅0 : for …
Formula:
C16H11NO5
Purity:
99.73%
Color and Shape:
Soild
Molecular weight:
297.26
Ref: TM-T67707
| 1mg | 96.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 604.00 € | ||
| 50mg | 825.00 € | ||
| 100mg | 1,091.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Syk-IN-8
CAS:2568963-01-7
Syk-IN-8 (compound 19q) functions as a Syk inhibitor with demonstrated antiproliferative effects on a variety …
Formula:
C23H26N10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
442.52
Ref: TM-T79443
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
TG 100572 Hydrochloride
CAS:867331-64-4
TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and …
Formula:
C26H27Cl2N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
512.43
Ref: TM-T13156L
| 1mg | 370.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
VEGFR-2-IN-9
CAS:408502-06-7
VEGFR-2-IN-9 (KDR-in-4) is a potent KDR/VEGFR2 inhibitor (IC50: 7 nM). It can be used to …
Formula:
C23H25N3O3
Purity:
97.19%
Color and Shape:
Solid
Molecular weight:
391.46
Ref: TM-T10123
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Brolucizumab
CAS:1531589-13-5
Brolucizumab (DLX1008) is a single-chain anti-VEGF-A antibody fragment exhibiting low picomolar affinity (K D = …
Purity:
98%
Color and Shape:
Solid
Ref: TM-T80593
| 1mg | 233.00 € | ||
| 5mg | 607.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,439.00 € | ||
| 50mg | 1,862.00 € | ||
| 100mg | 2,623.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
BT424
CAS:2755180-37-9
BT424, a specific HCK inhibitor, modulates macrophage activation and autophagy in vitro, and mitigates inflammation …
Formula:
C22H15BCl2N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
421.08
Ref: TM-T79516
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
JGK-068S
CAS:2490431-16-6
Compound I (JGK-068S) is a potent inhibitor of the epidermal growth factor receptor (EGFR) [1].
Formula:
C22H23BrFN5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
488.35
Ref: TM-T79124
| 5mg | 1,290.00 € | ||
| 50mg | 2,618.00 € | ||
| 100mg | 3,484.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
FGFR4-IN-8
CAS:2765240-52-4
FGFR4-IN-8 is a selective, ATP-competitive FGFR4 inhibitor with IC50s as low as 0.25 nM, halting …
Formula:
C32H34Cl2FN7O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
654.56
Ref: TM-T73121
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
EGFR-IN-61
CAS:2890261-81-9
EGFR-IN-61 inhibits EGFR kinase (IC50: 42 nM L858R/T790M, 137 nM L858R/T790M/C797S, 743 nM WT) and …
Formula:
C33H37ClN8O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
629.15
Ref: TM-T73128
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
EGFR-IN-85
CAS:1956378-29-2
EGFR-IN-85 (Compound 1), an EGFR inhibitor, exhibits potent activity with an IC50 of 0.19 μM …
Formula:
C26H30N8O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
486.57
Ref: TM-T78574
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
KB SRC 4
CAS:1380088-03-8
KB SRC 4 is a selective and potent c-Src inhibitor with antitumour activity that inhibits …
Formula:
C32H23ClN8
Purity:
99.66% - 99.66%
Color and Shape:
Solid
Molecular weight:
555.03
Ref: TM-T11745
| 1mg | 147.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Type II TRK inhibitor 1
CAS:2937543-72-9
Type II TRK Inhibitor 1 is a potent inhibitor targeting multiple tropomyosin receptor kinase (TRK) …
Formula:
C35H33F3N8O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
670.68
Ref: TM-T72289
| 5mg | 1,290.00 € | ||
| 50mg | 2,618.00 € | ||
| 100mg | 3,484.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
FGFR-IN-11
CAS:2658488-68-5
FGFR-IN-11 (compound I-5) is an orally active, covalent inhibitor of FGFR, exhibiting IC50 values of …
Formula:
C28H29ClN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
521.01
Ref: TM-T79257
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
EGFR/ErbB-2 inhibitor-1
CAS:1135150-79-6
EGFR/ErbB-2 inhibitor-1 is a selective ErbB2/HER2 inhibitor that effectively blocks ErbB2 and HER2 signaling.
Formula:
C23H15ClFN3OS2
Purity:
97.55%
Color and Shape:
Solid
Molecular weight:
467.97
Ref: TM-T79861
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,004.00 € | ||
| 50mg | 1,385.00 € | ||
| 100mg | 1,831.00 € | ||
| 500mg | 3,652.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
ENT-C225
CAS:2919962-53-9
ENT-C225 is a potent TrkB neurotrophin receptor (TrkBR) activator with neuroprotective activity for the study …
Formula:
C26H40N4O5
Purity:
99.16% - 99.16%
Color and Shape:
Solid
Molecular weight:
488.62
Ref: TM-T73397
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,392.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
EGFR/CSC-IN-1
CAS:2820447-02-5
EGFR/CSC-IN-1 is a dual inhibitor targeting both the epidermal growth factor receptor (EGFR [IC50 10.52 …
Formula:
C54H54Cl2FN7O7S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1067.08
Ref: TM-T73995
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
ALK/EGFR-IN-1
CAS:2730430-08-5
ALK/EGFR-IN-1 (Compound 8l) is a dual inhibitor targeting both ALK and EGFR, effectively blocking their …
Formula:
C27H34ClN7O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
572.12
Ref: TM-T79392
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
YK-029A
CAS:2064269-82-3
YK-029A, an orally active EGFR mutant inhibitor, targets both EGFR T790M and EGFRex20ins mutations.
Formula:
C27H32N8O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.6
Ref: TM-T79461
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Tyrosine kinase-IN-6
CAS:2377507-01-0
Tyrosine kinase-IN-6 is a potent inhibitor of RON splice variants, demonstrating significant anticancer and antineoplastic …
Formula:
C37H31F2N5O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
695.73
Ref: TM-T79612
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Pirtobrutinib
CAS:2101700-15-4
Pirtobrutinib: a selective, non-covalent BTK inhibitor effective against BTK C481 mutations, causing tumor regression in …
Formula:
C22H21F4N5O3
Purity:
99.76% - 99.89%
Color and Shape:
Solid
Molecular weight:
479.43
Ref: TM-T36287
| 1mg | 37.00 € | ||
| 1ml | 83.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 628.00 € | ||
| 500mg | 1,336.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
2′-Thioadenosine
CAS:136904-69-3
2'-Thioadenosine (PD157432) serves as a selective and irreversible inhibitor of ErbB-1 and ErbB-2 tyrosine kinases, …
Formula:
C10H13N5O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
283.31
Ref: TM-T78634
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
TAK-020
CAS:1627603-21-7
TAK-020 is a potent covalent inhibitor of Btk with potential antitumor activity for the study …
Formula:
C18H17N5O3
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
351.36
Ref: TM-T9529
| 1mg | 143.00 € | ||
| 1ml | 375.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 616.00 € | ||
| 25mg | 1,277.00 € | ||
| 50mg | 1,977.00 € | ||
| 100mg | 3,044.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Brepocitinib
CAS:1883299-62-4
Brepocitinib (PF-06700841) is a potent dual JAK1/TYK2 inhibitor (IC50s: 17 nM/23 nM). Brepocitinib also inhibits …
Formula:
C18H21F2N7O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
389.4
Ref: TM-TQ0010
| 1mg | 35.00 € | ||
| 1ml | 117.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 383.00 € | ||
| 100mg | 614.00 € | ||
| 200mg | 859.00 € | ||
| 500mg | 1,270.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
DZD1516
CAS:2387570-00-3
DZD1516, a potent and selective HER2 inhibitor (IC50 = 0.56 nM), demonstrates good blood-brain barrier …
Formula:
C28H27F2N7O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
547.56
Ref: TM-T79297
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
BEBT-109
CAS:2050906-40-4
BEBT-109 is a potent selective inhibitor of pan-mutant EGFR with enhanced pharmacokinetic properties, suitable for …
Formula:
C27H32N8O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
516.59
Ref: TM-T80643
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
TIE-2/VEGFR-2 kinase-IN-5
CAS:1014407-83-0
TIE-2/VEGFR-2 kinase-IN-5 is a TIE-2 and VEGFR-2 tyrosine kinase receptor inhibitor commonly used in biomedical …
Formula:
C21H13F6N5O2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
481.35
Ref: TM-T79860
| 1mg | 181.00 € | ||
| 5mg | 447.00 € | ||
| 10mg | 639.00 € | ||
| 25mg | 998.00 € | ||
| 50mg | 1,376.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
EGFR-IN-8
CAS:2407957-87-1
EGFR-IN-8, a dual inhibitor targeting both EGFR and c-Met, shows potential as a promising candidate …
Formula:
C32H23ClF3N7O4
Purity:
97.45%
Color and Shape:
Solid
Molecular weight:
662.02
Ref: TM-T11162
| 1mg | 74.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 266.00 € | ||
| 25mg | 440.00 € | ||
| 50mg | 602.00 € | ||
| 100mg | 825.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
AZ-23
CAS:915720-21-7
AZ-23 is an inhibitor of ATP-competitive and Trk kinase A/B/C.
Formula:
C17H19ClFN7O
Purity:
99.4%
Color and Shape:
Solid
Molecular weight:
391.83
Ref: TM-T14363
| 1mg | 96.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Src Inhibitor 3
CAS:2380027-49-4
Src Inhibitor 3 blocks c-Src kinase (IC50 <3 nM CSK HTRF, <4 nM Caliper), boosting …
Formula:
C34H32ClFN8O4
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
671.12
Ref: TM-T13000
| 1mg | 90.00 € | ||
| 1ml | 277.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 315.00 € | ||
| 25mg | 499.00 € | ||
| 50mg | 690.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 27 Dec 2024
HM43239
CAS:2294874-49-8
HM43239: oral FLT3 inhibitor; IC50: FLT3 WT 1.1nM, ITD 1.8nM, D835Y 1.0nM; blocks p-STAT5/p-ERK; affects …
Formula:
C29H33ClN6
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
501.07
Ref: TM-T9428
| 1mg | 69.00 € | ||
| 1ml | 186.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 221.00 € | ||
| 25mg | 434.00 € | ||
| 50mg | 620.00 € | ||
| 100mg | 862.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
c-Met-IN-2
CAS:1635406-73-3
c-Met-IN-2 is a selective and orally available c-Met inhibitor (IC50: 0.6 nM) with antitumor activity.
Formula:
C24H21FN10O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
484.49
Ref: TM-T10654
| 25mg | 2,106.00 € | ||
| 50mg | 2,785.00 € | ||
| 100mg | 3,739.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
AMG-25
CAS:1003311-62-3
AMG-25 (c-Kit-IN-5-1) is a c-Kit inhibitor that inhibits c-Kit, KDR, p38, Lck, and Src, and …
Formula:
C23H17N5O2
Purity:
98.16%
Color and Shape:
Solid
Molecular weight:
395.41
Ref: TM-T22256
| 2mg | 466.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
DYRKs-IN-1
CAS:1387090-01-8
DYRKs-IN-1 has antitumor activity.
Formula:
C30H30ClN7O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
588.06
Ref: TM-T11132
| 25mg | 2,662.00 € | ||
| 50mg | 3,533.00 € | ||
| 100mg | 4,860.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Tyk2-IN-3
CAS:1779493-12-7
Tyk2-IN-3 is an inhibitor of Tyk2 pseudokinase (IC50: 485 nM).
Formula:
C25H24N6O3S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
520.63
Ref: TM-T13233
| 25mg | 2,384.00 € | ||
| 50mg | 3,159.00 € | ||
| 100mg | 4,299.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
(-)-Cevimeline hydrochloride hemihydrate
(-)-Cevimeline HCl hemihydrate, a muscarinic agonist, treats Sjogren's xerostomia. Quick absorption, species-dependent metabolism.
Formula:
C10H19ClNO1·5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
244.78
Ref: TM-T13421
| 25mg | 3,673.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
G-744
CAS:1346669-54-2
G-744 is a selective and orally active inhibitor of Btk (IC50: 2 nM).
Formula:
C29H29N5O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
527.64
Ref: TM-T15365
| 25mg | 2,662.00 € | ||
| 50mg | 3,533.00 € | ||
| 100mg | 4,860.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
BTK-IN-16
CAS:2883232-92-4
BTK-IN-16 is a potential inhibitor of wild-type BTK and C481S mutants.BTK-IN-16 can be used to …
Formula:
C15H14N4O2
Purity:
99.04%
Color and Shape:
Soild
Molecular weight:
282.3
Ref: TM-T60542
| 1mg | 326.00 € | ||
| 5mg | 902.00 € | ||
| 10mg | 1,115.00 € | ||
| 25mg | 1,478.00 € | ||
| 50mg | 1,840.00 € | ||
| 100mg | 2,323.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
VEGFR2-IN-1
CAS:2765224-55-1
VEGFR2-IN-1 is a VEGFR2 inhibitor with antitumor activity used in the study of breast cancer.
Formula:
C22H18N6S
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
398.48
Ref: TM-T61899
| 1mg | 277.00 € | ||
| 5mg | 683.00 € | ||
| 10mg | 933.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 1,878.00 € | ||
| 100mg | 2,371.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
AZD-5672
CAS:780750-65-4
AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.
Formula:
C32H38F2N2O5S2
Purity:
95.58%
Color and Shape:
Solid
Molecular weight:
632.78
Ref: TM-T30260
| 1mg | 198.00 € | ||
| 1ml | 547.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 628.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,744.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
PF-06273340
CAS:1402438-74-7
PF-06273340: selective pan-Trk inhibitor (IC50: Trk-A 6 nM, B 4 nM, C 3 nM), low …
Formula:
C23H22ClN7O3
Purity:
98% - 98.00%
Color and Shape:
Solid
Molecular weight:
479.92
Ref: TM-T19649
| 1mg | 170.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
FGFR4-IN-4
CAS:2230973-67-6
FGFR4-IN-4 is a FGFR4 inhibitor with anti-tumor activity.
Formula:
C28H32Cl2N6O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
603.5
Ref: TM-T11280
| 25mg | 2,801.00 € | ||
| 50mg | 3,720.00 € | ||
| 100mg | 5,140.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
GENZ-882706
CAS:2070864-35-4
GENZ-882706 is a potent colony stimulating factor-1 receptor (CSF-1R) Inhibitor.
Formula:
C26H25N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
455.51
Ref: TM-T11390
| 25mg | 1,976.00 € | ||
| 50mg | 2,588.00 € | ||
| 100mg | 4,152.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Tarloxotinib bromide
CAS:1636180-98-7
Tarloxotinib bromide (TH-4000) is an irreversible inhibitor of EGFR/HER2.
Formula:
C24H24Br2ClN9O3
Purity:
97.15%
Color and Shape:
Solid
Molecular weight:
681.77
Ref: TM-T13088
| 1mg | 136.00 € | ||
| 1ml | 420.00 € | ||
| 5mg | 272.00 € | ||
| 10mg | 416.00 € | ||
| 25mg | 681.00 € | ||
| 50mg | 902.00 € | ||
| 100mg | 1,261.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Enbezotinib
CAS:2359649-81-1
Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.
Formula:
C21H21FN6O3
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
424.43
Ref: TM-T62285
| 1mg | 119.00 € | ||
| 1ml | 312.00 € | ||
| 5mg | 276.00 € | ||
| 10mg | 436.00 € | ||
| 25mg | 713.00 € | ||
| 50mg | 974.00 € | ||
| 100mg | 1,281.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
AZ12601011
CAS:2748337-86-0
AZ12601011 is a TGFBR1 kinase inhibitor that inhibits the growth of breast tumors.
Formula:
C19H15N5
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
313.36
Ref: TM-T10426
| 1mg | 97.00 € | ||
| 1ml | 254.00 € | ||
| 5mg | 231.00 € | ||
| 10mg | 370.00 € | ||
| 25mg | 716.00 € | ||
| 50mg | 1,074.00 € | ||
| 100mg | 1,484.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Vecabrutinib
CAS:1510829-06-7
Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and …
Formula:
C22H24ClF4N7O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
529.92
Ref: TM-T17220
| 1mg | 85.00 € | ||
| 1ml | 218.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 487.00 € | ||
| 50mg | 646.00 € | ||
| 100mg | 905.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
TAS05567
CAS:1429038-15-2
TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).
Formula:
C21H29N9O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
439.51
Ref: TM-T16995
| 25mg | 2,106.00 € | ||
| 50mg | 2,785.00 € | ||
| 100mg | 3,739.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Protopine hydrochloride
CAS:6164-47-2
Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.
Formula:
C20H20ClNO5
Purity:
98%
Color and Shape:
Prisms From Alc Solid
Molecular weight:
389.83
Ref: TM-TMA1944
| 1mg | 394.00 € | ||
| 500µg | 221.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
NVP-BHG712
CAS:940310-85-0
Formula:
C26H20F3N7O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
503.4785
Ref: IN-DA00GU50
| 5mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
Pelitinib
CAS:257933-82-7
Formula:
C24H23ClFN5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
467.9231
Ref: IN-DA007LZB
| 5mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
4-Quinazolinamine, N-(3-bromophenyl)-6,7-dimethoxy-, hydrochloride (1:1)
CAS:183322-45-4
Formula:
C16H15BrClN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
396.6662
Ref: IN-DA0027IO
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 250mg | Discontinued | Request information |
Unii-33Y9anm545
CAS:635702-64-6
Formula:
C21H24ClN7O2S
Purity:
99%
Color and Shape:
Solid
Molecular weight:
473.9790
Ref: IN-DA00E9EW
| 1g | Discontinued | Request information | |
| 5g | Discontinued | Request information | |
| 10g | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 250mg | Discontinued | Request information |
Ref: IN-DA007R3D
| 1g | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 250mg | Discontinued | Request information |
![Propanedinitrile,2-[(3,4-dihydroxyphenyl)methylene]-](https://static.cymitquimica.com/products/IN/thumb/DA007QB5.jpg)
Propanedinitrile,2-[(3,4-dihydroxyphenyl)methylene]-
CAS:118409-57-7
Formula:
C10H6N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
186.1668
Ref: IN-DA007QB5
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 250mg | Discontinued | Request information |
CHMFL-KIT-033
CAS:2351801-41-5
CHMFL-KIT-033 is an effective and selective c-KIT inhibitor with an IC50 value of 45 nM …
Formula:
C23H18FN5O2
Purity:
97.26%
Color and Shape:
Solid
Molecular weight:
415.42
Ref: TM-T10803
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
CHMFL-ABL-121
CAS:2270879-07-5
CHMFL-ABL-121 is a highly potent inhibitor of type II ABL kinase (IC50s: 2 nM and …
Formula:
C30H31F3N6OS
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
580.67
Ref: TM-T10800
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
CHMFL-FLT3-122
CAS:1839150-56-9
CHMFL-FLT3-122 is a potent and orally available FLT3 kinase inhibitor used to treat FLT3-ITD positive …
Formula:
C26H29N7O2
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
471.55
Ref: TM-T27011
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
Bosutinib D8
Bosutinib D8 is a deuterium-labeled Bosutinib. Bosutinib (SKI-606) is a dual Src/Abl inhibitor (IC50s: 1.2 …
Formula:
C26H21D8Cl2N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.5
Ref: TM-T10583
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
CHMFL-ABL-039
CAS:2304344-56-5
CHMFL-ABL-039 is a type II native ABL kinase and drug-resistant V299L mutant BCR-ABL inhibitor (IC50s: …
Formula:
C31H33F3N6O3
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
594.63
Ref: TM-T10799
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Keap1-Nrf2-IN-1
CAS:2232112-72-8
Keap1-Nrf2 IN-1, a protein interaction inhibitor with 43 nM IC50, boosts Nrf2 cytoprotection and counters …
Formula:
C24H24N2O7S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
484.52
Ref: TM-T11752
| 5mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information |
